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—— methyl 2-[(5R)-4-[hydroxy-[(2S)-2-methyl-2,3-dihydro-1-benzofuran-5-yl]methylidene]-2,3-dioxo-5-(3-pentoxyphenyl)pyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate —— C31H32N2O7S
methyl 2-[(5R)-4-[hydroxy-[(2S)-2-methyl-2,3-dihydro-1-benzofuran-5-yl]methylidene]-2,3-dioxo-5-(3-pentoxyphenyl)pyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate
—— methyl 2-[(2S)-1-[3-[(Z)-(3-hexyl-4-oxo-2-sulfanylidene-1,3-thiazolidin-5-ylidene)methyl]-7-methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl]-3-oxopiperazin-2-yl]acetate —— C26H31N5O5S2
methyl 2-[(2S)-1-[3-[(Z)-(3-hexyl-4-oxo-2-sulfanylidene-1,3-thiazolidin-5-ylidene)methyl]-7-methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl]-3-oxopiperazin-2-yl]acetate
—— Methyl 4-[5-(4-carbamoylphenyl)-2-methylpyrazol-3-yl]benzoate —— C19H17N3O3
Methyl 4-[5-(4-carbamoylphenyl)-2-methylpyrazol-3-yl]benzoate
—— methyl 4-[(2R)-1-(5-benzylsulfanyl-1,3,4-thiadiazol-2-yl)-3-[hydroxy-[(2S)-2-methyl-2,3-dihydro-1-benzofuran-5-yl]methylidene]-4,5-dioxopyrrolidin-2-yl]benzoate —— C31H25N3O6S2
methyl 4-[(2R)-1-(5-benzylsulfanyl-1,3,4-thiadiazol-2-yl)-3-[hydroxy-[(2S)-2-methyl-2,3-dihydro-1-benzofuran-5-yl]methylidene]-4,5-dioxopyrrolidin-2-yl]benzoate
—— methyl 2-[(2R)-2-(4-ethoxyphenyl)-3-[hydroxy-(3-methyl-4-phenylmethoxyphenyl)methylidene]-4,5-dioxopyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate —— C33H30N2O7S
methyl 2-[(2R)-2-(4-ethoxyphenyl)-3-[hydroxy-(3-methyl-4-phenylmethoxyphenyl)methylidene]-4,5-dioxopyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate
—— methyl 4-[(2S)-1-(5-benzylsulfanyl-1,3,4-thiadiazol-2-yl)-3-[hydroxy-[(2R)-2-methyl-2,3-dihydro-1-benzofuran-5-yl]methylidene]-4,5-dioxopyrrolidin-2-yl]benzoate —— C31H25N3O6S2
methyl 4-[(2S)-1-(5-benzylsulfanyl-1,3,4-thiadiazol-2-yl)-3-[hydroxy-[(2R)-2-methyl-2,3-dihydro-1-benzofuran-5-yl]methylidene]-4,5-dioxopyrrolidin-2-yl]benzoate
—— methyl 2-[(5S)-4-[hydroxy-[(2S)-2-methyl-2,3-dihydro-1-benzofuran-5-yl]methylidene]-2,3-dioxo-5-(3-pentoxyphenyl)pyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate —— C31H32N2O7S
methyl 2-[(5S)-4-[hydroxy-[(2S)-2-methyl-2,3-dihydro-1-benzofuran-5-yl]methylidene]-2,3-dioxo-5-(3-pentoxyphenyl)pyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate
—— Methyl 2-[2-[(3-fluorophenyl)-methylcarbamoyl]indol-1-yl]acetate —— C19H17FN2O3
Methyl 2-[2-[(3-fluorophenyl)-methylcarbamoyl]indol-1-yl]acetate
—— methyl N-(2-benzoyl-6-chloro-1H-indol-3-yl)carbamate —— C17H13ClN2O3
methyl N-(2-benzoyl-6-chloro-1H-indol-3-yl)carbamate
—— Methyl 2-(benzenesulfonamido)-3-(4-cyanophenyl)propanoate —— C17H16N2O4S
Methyl 2-(benzenesulfonamido)-3-(4-cyanophenyl)propanoate
—— methyl 2-[(2S)-2-(4-ethoxyphenyl)-3-[hydroxy-(3-methyl-4-phenylmethoxyphenyl)methylidene]-4,5-dioxopyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate —— C33H30N2O7S
methyl 2-[(2S)-2-(4-ethoxyphenyl)-3-[hydroxy-(3-methyl-4-phenylmethoxyphenyl)methylidene]-4,5-dioxopyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate
—— methyl 4-[(2R)-1-(5-benzylsulfanyl-1,3,4-thiadiazol-2-yl)-3-[hydroxy-[(2R)-2-methyl-2,3-dihydro-1-benzofuran-5-yl]methylidene]-4,5-dioxopyrrolidin-2-yl]benzoate —— C31H25N3O6S2
methyl 4-[(2R)-1-(5-benzylsulfanyl-1,3,4-thiadiazol-2-yl)-3-[hydroxy-[(2R)-2-methyl-2,3-dihydro-1-benzofuran-5-yl]methylidene]-4,5-dioxopyrrolidin-2-yl]benzoate
—— methyl 2-[(5S)-4-[hydroxy-[(2R)-2-methyl-2,3-dihydro-1-benzofuran-5-yl]methylidene]-2,3-dioxo-5-(3-pentoxyphenyl)pyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate —— C31H32N2O7S
methyl 2-[(5S)-4-[hydroxy-[(2R)-2-methyl-2,3-dihydro-1-benzofuran-5-yl]methylidene]-2,3-dioxo-5-(3-pentoxyphenyl)pyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate
—— methyl 4-[(2S)-1-(5-benzylsulfanyl-1,3,4-thiadiazol-2-yl)-3-[hydroxy-[(2S)-2-methyl-2,3-dihydro-1-benzofuran-5-yl]methylidene]-4,5-dioxopyrrolidin-2-yl]benzoate —— C31H25N3O6S2
methyl 4-[(2S)-1-(5-benzylsulfanyl-1,3,4-thiadiazol-2-yl)-3-[hydroxy-[(2S)-2-methyl-2,3-dihydro-1-benzofuran-5-yl]methylidene]-4,5-dioxopyrrolidin-2-yl]benzoate
—— methyl 2-[(5R)-4-[hydroxy-[(2R)-2-methyl-2,3-dihydro-1-benzofuran-5-yl]methylidene]-2,3-dioxo-5-(3-pentoxyphenyl)pyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate —— C31H32N2O7S
methyl 2-[(5R)-4-[hydroxy-[(2R)-2-methyl-2,3-dihydro-1-benzofuran-5-yl]methylidene]-2,3-dioxo-5-(3-pentoxyphenyl)pyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate
—— methyl 2-[(2S)-2-(4-hydroxy-3-methoxyphenyl)-3-[hydroxy-(2-methyl-4-phenylmethoxyphenyl)methylidene]-4,5-dioxopyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate —— C32H28N2O8S
methyl 2-[(2S)-2-(4-hydroxy-3-methoxyphenyl)-3-[hydroxy-(2-methyl-4-phenylmethoxyphenyl)methylidene]-4,5-dioxopyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate
—— methyl 2-[(5S)-4-[hydroxy-[(2R)-2-methyl-2,3-dihydro-1-benzofuran-5-yl]methylidene]-2,3-dioxo-5-(3-phenylmethoxyphenyl)pyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate —— C33H28N2O7S
methyl 2-[(5S)-4-[hydroxy-[(2R)-2-methyl-2,3-dihydro-1-benzofuran-5-yl]methylidene]-2,3-dioxo-5-(3-phenylmethoxyphenyl)pyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate
—— methyl 4-[(2S)-3-[hydroxy-[(2S)-2-methyl-2,3-dihydro-1-benzofuran-5-yl]methylidene]-1-(6-methoxy-1,3-benzothiazol-2-yl)-4,5-dioxopyrrolidin-2-yl]benzoate —— C30H24N2O7S
methyl 4-[(2S)-3-[hydroxy-[(2S)-2-methyl-2,3-dihydro-1-benzofuran-5-yl]methylidene]-1-(6-methoxy-1,3-benzothiazol-2-yl)-4,5-dioxopyrrolidin-2-yl]benzoate
—— methyl 2-[(2R)-2-(3-ethoxy-4-hydroxyphenyl)-3-[hydroxy-(3-methyl-4-phenylmethoxyphenyl)methylidene]-4,5-dioxopyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate —— C33H30N2O8S
methyl 2-[(2R)-2-(3-ethoxy-4-hydroxyphenyl)-3-[hydroxy-(3-methyl-4-phenylmethoxyphenyl)methylidene]-4,5-dioxopyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate
—— methyl 4-[(2R)-3-[hydroxy-[(2S)-2-methyl-2,3-dihydro-1-benzofuran-5-yl]methylidene]-1-(6-methoxy-1,3-benzothiazol-2-yl)-4,5-dioxopyrrolidin-2-yl]benzoate —— C30H24N2O7S
methyl 4-[(2R)-3-[hydroxy-[(2S)-2-methyl-2,3-dihydro-1-benzofuran-5-yl]methylidene]-1-(6-methoxy-1,3-benzothiazol-2-yl)-4,5-dioxopyrrolidin-2-yl]benzoate
—— methyl 2-[(2S)-2-(4-ethoxy-3-methoxyphenyl)-3-[hydroxy-(3-methyl-4-phenylmethoxyphenyl)methylidene]-4,5-dioxopyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate —— C34H32N2O8S
methyl 2-[(2S)-2-(4-ethoxy-3-methoxyphenyl)-3-[hydroxy-(3-methyl-4-phenylmethoxyphenyl)methylidene]-4,5-dioxopyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate
—— methyl 2-[(2S)-2-(3-bromophenyl)-3-[hydroxy-(4-methoxy-3-methylphenyl)methylidene]-4,5-dioxopyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate —— C25H21BrN2O6S
methyl 2-[(2S)-2-(3-bromophenyl)-3-[hydroxy-(4-methoxy-3-methylphenyl)methylidene]-4,5-dioxopyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate
—— methyl (1S,4S,9R,12R)-5,8-dimethyl-3,10-dioxotetracyclo[10.2.1.02,11.04,9]pentadec-6-ene-4-carboxylate —— C19H24O4
methyl (1S,4S,9R,12R)-5,8-dimethyl-3,10-dioxotetracyclo[10.2.1.02,11.04,9]pentadec-6-ene-4-carboxylate
—— methyl 4-[hydroxy-[(2R)-1-(3-morpholin-4-ylpropyl)-4,5-dioxo-2-(3,4,5-trimethoxyphenyl)pyrrolidin-3-ylidene]methyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate —— C29H37N3O9
methyl 4-[hydroxy-[(2R)-1-(3-morpholin-4-ylpropyl)-4,5-dioxo-2-(3,4,5-trimethoxyphenyl)pyrrolidin-3-ylidene]methyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate
—— methyl 2-[(2S)-2-(3-ethoxy-4-hydroxyphenyl)-3-[hydroxy-(3-methyl-4-phenylmethoxyphenyl)methylidene]-4,5-dioxopyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate —— C33H30N2O8S
methyl 2-[(2S)-2-(3-ethoxy-4-hydroxyphenyl)-3-[hydroxy-(3-methyl-4-phenylmethoxyphenyl)methylidene]-4,5-dioxopyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate
—— methyl 2-[(2R)-2-(3-bromophenyl)-3-[hydroxy-(4-methoxy-3-methylphenyl)methylidene]-4,5-dioxopyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate —— C25H21BrN2O6S
methyl 2-[(2R)-2-(3-bromophenyl)-3-[hydroxy-(4-methoxy-3-methylphenyl)methylidene]-4,5-dioxopyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate
—— methyl 4-[(5Z)-5-[(4-methoxyphenyl)methylidene]-2,4-dioxo-1,3-oxazolidin-3-yl]butanoate —— C16H17NO6
methyl 4-[(5Z)-5-[(4-methoxyphenyl)methylidene]-2,4-dioxo-1,3-oxazolidin-3-yl]butanoate
—— methyl 2-[(5R)-4-[hydroxy-[(2R)-2-methyl-2,3-dihydro-1-benzofuran-5-yl]methylidene]-2,3-dioxo-5-(3-phenylmethoxyphenyl)pyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate —— C33H28N2O7S
methyl 2-[(5R)-4-[hydroxy-[(2R)-2-methyl-2,3-dihydro-1-benzofuran-5-yl]methylidene]-2,3-dioxo-5-(3-phenylmethoxyphenyl)pyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate
—— methyl 2-[(5S)-4-[hydroxy-[(2S)-2-methyl-2,3-dihydro-1-benzofuran-5-yl]methylidene]-2,3-dioxo-5-(3-phenylmethoxyphenyl)pyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate —— C33H28N2O7S
methyl 2-[(5S)-4-[hydroxy-[(2S)-2-methyl-2,3-dihydro-1-benzofuran-5-yl]methylidene]-2,3-dioxo-5-(3-phenylmethoxyphenyl)pyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate
—— methyl 4-[[(2S)-2-(3-bromophenyl)-1-(3-morpholin-4-ylpropyl)-4,5-dioxopyrrolidin-3-ylidene]-hydroxymethyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate —— C26H30BrN3O6
methyl 4-[[(2S)-2-(3-bromophenyl)-1-(3-morpholin-4-ylpropyl)-4,5-dioxopyrrolidin-3-ylidene]-hydroxymethyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate
—— methyl 2-[(2R)-2-(3,4-dimethoxyphenyl)-3-[hydroxy-(2-methyl-4-phenylmethoxyphenyl)methylidene]-4,5-dioxopyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate —— C33H30N2O8S
methyl 2-[(2R)-2-(3,4-dimethoxyphenyl)-3-[hydroxy-(2-methyl-4-phenylmethoxyphenyl)methylidene]-4,5-dioxopyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate
—— methyl 2-[(5S)-4-[hydroxy-(4-methoxy-3-methylphenyl)methylidene]-2,3-dioxo-5-(3,4,5-trimethoxyphenyl)pyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate —— C28H28N2O9S
methyl 2-[(5S)-4-[hydroxy-(4-methoxy-3-methylphenyl)methylidene]-2,3-dioxo-5-(3,4,5-trimethoxyphenyl)pyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate
—— methyl 2-[(2R)-2-(4-hydroxy-3-methoxyphenyl)-3-[hydroxy-(2-methyl-4-phenylmethoxyphenyl)methylidene]-4,5-dioxopyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate —— C32H28N2O8S
methyl 2-[(2R)-2-(4-hydroxy-3-methoxyphenyl)-3-[hydroxy-(2-methyl-4-phenylmethoxyphenyl)methylidene]-4,5-dioxopyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate
—— methyl 2-[(2S)-2-(3,4-dimethoxyphenyl)-3-[hydroxy-(2-methyl-4-phenylmethoxyphenyl)methylidene]-4,5-dioxopyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate —— C33H30N2O8S
methyl 2-[(2S)-2-(3,4-dimethoxyphenyl)-3-[hydroxy-(2-methyl-4-phenylmethoxyphenyl)methylidene]-4,5-dioxopyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate
—— methyl 2-(4,6,7,7a-tetrahydro-3aH-thieno[3,2-c]pyridin-5-yl)-2-(2-chlorophenyl)acetate —— C16H18ClNO2S
methyl 2-(4,6,7,7a-tetrahydro-3aH-thieno[3,2-c]pyridin-5-yl)-2-(2-chlorophenyl)acetate
—— methyl 2-[(5R)-4-[hydroxy-(2-methyl-4-phenylmethoxyphenyl)methylidene]-2,3-dioxo-5-(3-phenoxyphenyl)pyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate —— C37H30N2O7S
methyl 2-[(5R)-4-[hydroxy-(2-methyl-4-phenylmethoxyphenyl)methylidene]-2,3-dioxo-5-(3-phenoxyphenyl)pyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate
—— methyl 2-[(5S)-4-[hydroxy-(2-methyl-4-phenylmethoxyphenyl)methylidene]-2,3-dioxo-5-(3-phenoxyphenyl)pyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate —— C37H30N2O7S
methyl 2-[(5S)-4-[hydroxy-(2-methyl-4-phenylmethoxyphenyl)methylidene]-2,3-dioxo-5-(3-phenoxyphenyl)pyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate
—— methyl 4-[[(2R)-2-(3-bromophenyl)-1-(3-morpholin-4-ylpropyl)-4,5-dioxopyrrolidin-3-ylidene]-hydroxymethyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate —— C26H30BrN3O6
methyl 4-[[(2R)-2-(3-bromophenyl)-1-(3-morpholin-4-ylpropyl)-4,5-dioxopyrrolidin-3-ylidene]-hydroxymethyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate
—— methyl 2-[(2S)-2-(3-ethoxy-4-hydroxyphenyl)-3-[hydroxy-(2-methyl-4-phenylmethoxyphenyl)methylidene]-4,5-dioxopyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate —— C33H30N2O8S
methyl 2-[(2S)-2-(3-ethoxy-4-hydroxyphenyl)-3-[hydroxy-(2-methyl-4-phenylmethoxyphenyl)methylidene]-4,5-dioxopyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate
—— methyl 2-[(2R)-2-(3-ethoxy-4-hydroxyphenyl)-3-[hydroxy-(2-methyl-4-phenylmethoxyphenyl)methylidene]-4,5-dioxopyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate —— C33H30N2O8S
methyl 2-[(2R)-2-(3-ethoxy-4-hydroxyphenyl)-3-[hydroxy-(2-methyl-4-phenylmethoxyphenyl)methylidene]-4,5-dioxopyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate
—— Methyl 8-(chloromethyl)-4-hydroxy-2-methyl-7,8-dihydrothieno[2,3-e]indole-6-carboxylate —— C14H14ClNO3S
Methyl 8-(chloromethyl)-4-hydroxy-2-methyl-7,8-dihydrothieno[2,3-e]indole-6-carboxylate
—— methyl (E)-2-acetamido-5-phenyl-2-propanoylpent-4-enoate —— C17H21NO4
methyl (E)-2-acetamido-5-phenyl-2-propanoylpent-4-enoate
—— methyl 2-[(5R)-4-[hydroxy-(4-methoxy-3-methylphenyl)methylidene]-2,3-dioxo-5-(3,4,5-trimethoxyphenyl)pyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate —— C28H28N2O9S
methyl 2-[(5R)-4-[hydroxy-(4-methoxy-3-methylphenyl)methylidene]-2,3-dioxo-5-(3,4,5-trimethoxyphenyl)pyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate
—— methyl (2R,3S)-3-(2,6-dimethylphenyl)-3-(ethoxycarbonylamino)-2-hydroxypropanoate —— C15H21NO5
methyl (2R,3S)-3-(2,6-dimethylphenyl)-3-(ethoxycarbonylamino)-2-hydroxypropanoate
—— Methyl 2-acetamido-2-benzoylpent-4-enoate —— C15H17NO4
Methyl 2-acetamido-2-benzoylpent-4-enoate
—— methyl (2S)-2-[[(2S)-2-amino-4-methylpentanethioyl]amino]-4-methylpentanoate —— C13H26N2O2S
methyl (2S)-2-[[(2S)-2-amino-4-methylpentanethioyl]amino]-4-methylpentanoate
—— methyl (3S)-6-diethoxyphosphoryl-3-hydroxyhex-5-ynoate —— C11H19O6P
methyl (3S)-6-diethoxyphosphoryl-3-hydroxyhex-5-ynoate
—— Methyl 2-[2-[4-(trifluoromethyl)pyridin-3-yl]-1,3-oxazol-4-yl]acetate —— C12H9F3N2O3
Methyl 2-[2-[4-(trifluoromethyl)pyridin-3-yl]-1,3-oxazol-4-yl]acetate
—— Met-Pro-Asp —— C14H23N3O6S
Met-Pro-Asp
—— methyl 2-[(4-oxocyclohexa-2,5-dien-1-ylidene)methylamino]-3-phenylpropanoate —— C17H17NO3
methyl 2-[(4-oxocyclohexa-2,5-dien-1-ylidene)methylamino]-3-phenylpropanoate