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—— methyl 2-[[(4S,7S)-7-(4-methoxyphenyl)-2-methyl-5-oxo-4-phenyl-4,6,7,8-tetrahydro-1H-quinoline-3-carbonyl]amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate —— C34H34N2O5S
methyl 2-[[(4S,7S)-7-(4-methoxyphenyl)-2-methyl-5-oxo-4-phenyl-4,6,7,8-tetrahydro-1H-quinoline-3-carbonyl]amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
—— Methyl 4-[3-[3-[3-[[3-(aminomethyl)phenyl]methylcarbamoyloxy]prop-1-ynyl]-5-(2-methoxy-2-oxoethyl)phenyl]prop-2-ynoxycarbonylamino]-1-[3-[3-(aminomethyl)phenyl]propanoyl]pyrrolidine-2-carboxylate —— C41H45N5O9
Methyl 4-[3-[3-[3-[[3-(aminomethyl)phenyl]methylcarbamoyloxy]prop-1-ynyl]-5-(2-methoxy-2-oxoethyl)phenyl]prop-2-ynoxycarbonylamino]-1-[3-[3-(aminomethyl)phenyl]propanoyl]pyrrolidine-2-carboxylate
—— methyl 2-[[(4S,7S)-2-methyl-5-oxo-4,7-diphenyl-4,6,7,8-tetrahydro-1H-quinoline-3-carbonyl]amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate —— C33H32N2O4S
methyl 2-[[(4S,7S)-2-methyl-5-oxo-4,7-diphenyl-4,6,7,8-tetrahydro-1H-quinoline-3-carbonyl]amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
—— methyl 2-[[(4R)-2,7,7-trimethyl-4-(4-methylsulfanylphenyl)-5-oxo-1,4,6,8-tetrahydroquinoline-3-carbonyl]amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate —— C30H34N2O4S2
methyl 2-[[(4R)-2,7,7-trimethyl-4-(4-methylsulfanylphenyl)-5-oxo-1,4,6,8-tetrahydroquinoline-3-carbonyl]amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
—— methyl 2-[[(4R,7S)-2-methyl-5-oxo-4,7-diphenyl-4,6,7,8-tetrahydro-1H-quinoline-3-carbonyl]amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate —— C33H32N2O4S
methyl 2-[[(4R,7S)-2-methyl-5-oxo-4,7-diphenyl-4,6,7,8-tetrahydro-1H-quinoline-3-carbonyl]amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
—— methyl 2-[[(4R,7S)-7-(4-methoxyphenyl)-2-methyl-5-oxo-4-phenyl-4,6,7,8-tetrahydro-1H-quinoline-3-carbonyl]amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate —— C34H34N2O5S
methyl 2-[[(4R,7S)-7-(4-methoxyphenyl)-2-methyl-5-oxo-4-phenyl-4,6,7,8-tetrahydro-1H-quinoline-3-carbonyl]amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
—— methyl 4-[[2-[(4S)-1-benzyl-5-oxo-2-sulfanylidene-3-[[4-(trifluoromethoxy)phenyl]methyl]imidazolidin-4-yl]acetyl]amino]benzoate —— C28H24F3N3O5S
methyl 4-[[2-[(4S)-1-benzyl-5-oxo-2-sulfanylidene-3-[[4-(trifluoromethoxy)phenyl]methyl]imidazolidin-4-yl]acetyl]amino]benzoate
—— methyl 2-[[(4R,7R)-7-(4-methoxyphenyl)-2-methyl-5-oxo-4-phenyl-4,6,7,8-tetrahydro-1H-quinoline-3-carbonyl]amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate —— C34H34N2O5S
methyl 2-[[(4R,7R)-7-(4-methoxyphenyl)-2-methyl-5-oxo-4-phenyl-4,6,7,8-tetrahydro-1H-quinoline-3-carbonyl]amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
—— methyl 2-[[(4R)-4-(2-methoxyphenyl)-2,7,7-trimethyl-5-oxo-1,4,6,8-tetrahydroquinoline-3-carbonyl]amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate —— C30H34N2O5S
methyl 2-[[(4R)-4-(2-methoxyphenyl)-2,7,7-trimethyl-5-oxo-1,4,6,8-tetrahydroquinoline-3-carbonyl]amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
—— methyl 2-[[(4S)-4-(2-methoxyphenyl)-2,7,7-trimethyl-5-oxo-1,4,6,8-tetrahydroquinoline-3-carbonyl]amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate —— C30H34N2O5S
methyl 2-[[(4S)-4-(2-methoxyphenyl)-2,7,7-trimethyl-5-oxo-1,4,6,8-tetrahydroquinoline-3-carbonyl]amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
—— methyl (Z)-3-[4-[4-(4-fluorobenzoyl)piperazin-1-yl]-3-nitrophenyl]prop-2-enoate —— C21H20FN3O5
methyl (Z)-3-[4-[4-(4-fluorobenzoyl)piperazin-1-yl]-3-nitrophenyl]prop-2-enoate
—— methyl 3-[3-[1-[(4Z)-5-[(3,5-dichlorobenzoyl)-methylamino]-3-(3,4-dichlorophenyl)-4-methoxyiminopentyl]piperidin-4-yl]-2-oxo-1,3-diazinan-1-yl]propanoate —— C33H41Cl4N5O5
methyl 3-[3-[1-[(4Z)-5-[(3,5-dichlorobenzoyl)-methylamino]-3-(3,4-dichlorophenyl)-4-methoxyiminopentyl]piperidin-4-yl]-2-oxo-1,3-diazinan-1-yl]propanoate
—— methyl 2-[[(4S,7R)-7-(4-methoxyphenyl)-2-methyl-5-oxo-4-phenyl-4,6,7,8-tetrahydro-1H-quinoline-3-carbonyl]amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate —— C34H34N2O5S
methyl 2-[[(4S,7R)-7-(4-methoxyphenyl)-2-methyl-5-oxo-4-phenyl-4,6,7,8-tetrahydro-1H-quinoline-3-carbonyl]amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
—— methyl 2-[[(4R,7R)-2-methyl-5-oxo-4,7-diphenyl-4,6,7,8-tetrahydro-1H-quinoline-3-carbonyl]amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate —— C33H32N2O4S
methyl 2-[[(4R,7R)-2-methyl-5-oxo-4,7-diphenyl-4,6,7,8-tetrahydro-1H-quinoline-3-carbonyl]amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
—— methyl 2-[[(4S)-2,7,7-trimethyl-4-(4-methylsulfanylphenyl)-5-oxo-1,4,6,8-tetrahydroquinoline-3-carbonyl]amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate —— C30H34N2O4S2
methyl 2-[[(4S)-2,7,7-trimethyl-4-(4-methylsulfanylphenyl)-5-oxo-1,4,6,8-tetrahydroquinoline-3-carbonyl]amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
—— methyl (Z)-3-[4-(2-ethoxy-2-oxoethoxy)-3-methoxyphenyl]prop-2-enoate —— C15H18O6
methyl (Z)-3-[4-(2-ethoxy-2-oxoethoxy)-3-methoxyphenyl]prop-2-enoate
—— Methyl 23-(ethylsulfanylmethyl)-16-hydroxy-15-methyl-3-oxo-10-[[3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]oxymethyl]-28-oxa-4,14,19-triazaoctacyclo[12.11.2.115,18.02,6.07,27.08,13.019,26.020,25]octacosa-1,6,8(13),9,11,20(25),21,23,26-nonaene-16-carboxylate —— C37H39N3O11S
Methyl 23-(ethylsulfanylmethyl)-16-hydroxy-15-methyl-3-oxo-10-[[3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]oxymethyl]-28-oxa-4,14,19-triazaoctacyclo[12.11.2.115,18.02,6.07,27.08,13.019,26.020,25]octacosa-1,6,8(13),9,11,20(25),21,23,26-nonaene-16-carboxylate
—— methyl 4-[[2-[(4R)-1-benzyl-5-oxo-2-sulfanylidene-3-[[4-(trifluoromethoxy)phenyl]methyl]imidazolidin-4-yl]acetyl]amino]benzoate —— C28H24F3N3O5S
methyl 4-[[2-[(4R)-1-benzyl-5-oxo-2-sulfanylidene-3-[[4-(trifluoromethoxy)phenyl]methyl]imidazolidin-4-yl]acetyl]amino]benzoate
—— methyl (2S)-2-[(6-bromo-1,3-benzothiazol-2-yl)amino]-2-[(2,4-dichlorobenzoyl)amino]-3,3,3-trifluoropropanoate —— C18H11BrCl2F3N3O3S
methyl (2S)-2-[(6-bromo-1,3-benzothiazol-2-yl)amino]-2-[(2,4-dichlorobenzoyl)amino]-3,3,3-trifluoropropanoate
—— methyl 2-[[[(2R,3S)-3-[[(2S)-4-amino-4-oxo-2-(phenylmethoxycarbonylamino)butanoyl]amino]-2-hydroxy-4-phenylbutyl]-(2-methylpropyl)sulfamoyl]amino]-2-methylpropanoate —— C31H45N5O9S
methyl 2-[[[(2R,3S)-3-[[(2S)-4-amino-4-oxo-2-(phenylmethoxycarbonylamino)butanoyl]amino]-2-hydroxy-4-phenylbutyl]-(2-methylpropyl)sulfamoyl]amino]-2-methylpropanoate
—— methyl 2-[[(4S,7R)-2-methyl-5-oxo-4,7-diphenyl-4,6,7,8-tetrahydro-1H-quinoline-3-carbonyl]amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate —— C33H32N2O4S
methyl 2-[[(4S,7R)-2-methyl-5-oxo-4,7-diphenyl-4,6,7,8-tetrahydro-1H-quinoline-3-carbonyl]amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
—— methyl 1-[[(Z)-3-[3-(3,4-dimethoxyphenyl)-1-phenylpyrazol-4-yl]prop-2-enoyl]amino]cyclopentane-1-carboxylate —— C27H29N3O5
methyl 1-[[(Z)-3-[3-(3,4-dimethoxyphenyl)-1-phenylpyrazol-4-yl]prop-2-enoyl]amino]cyclopentane-1-carboxylate
—— methyl 4-[[(2Z,4E)-hexa-2,4-dienoyl]amino]-3-methylbenzoate —— C15H17NO3
methyl 4-[[(2Z,4E)-hexa-2,4-dienoyl]amino]-3-methylbenzoate
—— methyl 2-methyl-3-[[(Z)-3-(3,4,5-trimethoxyphenyl)prop-2-enoyl]amino]benzoate —— C21H23NO6
methyl 2-methyl-3-[[(Z)-3-(3,4,5-trimethoxyphenyl)prop-2-enoyl]amino]benzoate
—— methyl (2R)-2-[4-[(Z)-3-(1,3-benzodioxol-5-yl)prop-2-enoyl]piperazin-1-yl]-2-(2-chlorophenyl)acetate —— C23H23ClN2O5
methyl (2R)-2-[4-[(Z)-3-(1,3-benzodioxol-5-yl)prop-2-enoyl]piperazin-1-yl]-2-(2-chlorophenyl)acetate
—— methyl 5-[[(Z)-3-(2-chlorophenyl)prop-2-enoyl]amino]-2,4-difluorobenzoate —— C17H12ClF2NO3
methyl 5-[[(Z)-3-(2-chlorophenyl)prop-2-enoyl]amino]-2,4-difluorobenzoate
—— methyl 8-(bromomethyl)-6-[(E)-3-(4-methoxyphenyl)prop-2-enoyl]-2-methyl-4-(4-methylpiperazine-1-carbonyl)oxy-7,8-dihydro-3H-pyrrolo[3,2-e]indole-1-carboxylate —— C30H33BrN4O6
methyl 8-(bromomethyl)-6-[(E)-3-(4-methoxyphenyl)prop-2-enoyl]-2-methyl-4-(4-methylpiperazine-1-carbonyl)oxy-7,8-dihydro-3H-pyrrolo[3,2-e]indole-1-carboxylate
—— Methyl 7-(4-aminophenyl)-2-[(2,5-dimethoxyphenyl)methoxy]-8-oxo-5-(3,4,5-trimethoxyphenyl)-1,7-naphthyridine-6-carboxylate —— C34H33N3O9
Methyl 7-(4-aminophenyl)-2-[(2,5-dimethoxyphenyl)methoxy]-8-oxo-5-(3,4,5-trimethoxyphenyl)-1,7-naphthyridine-6-carboxylate
—— Methyl 2-ethylsulfanyl-3-[4-[[6-[(6-hydroxy-2,5,7,8-tetramethyl-3,4-dihydrochromen-2-yl)methoxy]-1-methylbenzimidazol-2-yl]methoxy]phenyl]propanoate —— C35H42N2O6S
Methyl 2-ethylsulfanyl-3-[4-[[6-[(6-hydroxy-2,5,7,8-tetramethyl-3,4-dihydrochromen-2-yl)methoxy]-1-methylbenzimidazol-2-yl]methoxy]phenyl]propanoate
—— methyl 4-[[(2E,4Z)-hexa-2,4-dienoyl]amino]-3-methylbenzoate —— C15H17NO3
methyl 4-[[(2E,4Z)-hexa-2,4-dienoyl]amino]-3-methylbenzoate
—— methyl 4-[[(2Z,4Z)-hexa-2,4-dienoyl]amino]-3-methylbenzoate —— C15H17NO3
methyl 4-[[(2Z,4Z)-hexa-2,4-dienoyl]amino]-3-methylbenzoate
—— methyl (Z)-3-[3-methoxy-4-[2-[[(2S)-5-methylhexan-2-yl]amino]-2-oxoethoxy]phenyl]prop-2-enoate —— C20H29NO5
methyl (Z)-3-[3-methoxy-4-[2-[[(2S)-5-methylhexan-2-yl]amino]-2-oxoethoxy]phenyl]prop-2-enoate
—— methyl 2-methyl-3-[[(Z)-3-[4-[(2-methyl-1,3-thiazol-4-yl)methoxy]phenyl]prop-2-enoyl]amino]benzoate —— C23H22N2O4S
methyl 2-methyl-3-[[(Z)-3-[4-[(2-methyl-1,3-thiazol-4-yl)methoxy]phenyl]prop-2-enoyl]amino]benzoate
—— methyl (2S)-2-(2-chlorophenyl)-2-[4-[(Z)-3-thiophen-2-ylprop-2-enoyl]piperazin-1-yl]acetate —— C20H21ClN2O3S
methyl (2S)-2-(2-chlorophenyl)-2-[4-[(Z)-3-thiophen-2-ylprop-2-enoyl]piperazin-1-yl]acetate
—— methyl (Z)-3-[4-[2-[(3,4-dimethylphenyl)sulfonyl-methylamino]acetyl]oxy-3-methoxyphenyl]prop-2-enoate —— C22H25NO7S
methyl (Z)-3-[4-[2-[(3,4-dimethylphenyl)sulfonyl-methylamino]acetyl]oxy-3-methoxyphenyl]prop-2-enoate
—— methyl (Z)-3-[3-methoxy-4-[2-[[(2R)-5-methylhexan-2-yl]amino]-2-oxoethoxy]phenyl]prop-2-enoate —— C20H29NO5
methyl (Z)-3-[3-methoxy-4-[2-[[(2R)-5-methylhexan-2-yl]amino]-2-oxoethoxy]phenyl]prop-2-enoate
—— methyl 5-[[(Z)-3-(4-chlorophenyl)prop-2-enoyl]amino]-2,4-difluorobenzoate —— C17H12ClF2NO3
methyl 5-[[(Z)-3-(4-chlorophenyl)prop-2-enoyl]amino]-2,4-difluorobenzoate
—— methyl (Z)-3-[4-(2,6-dichlorophenyl)sulfonyloxy-3-methoxyphenyl]prop-2-enoate —— C17H14Cl2O6S
methyl (Z)-3-[4-(2,6-dichlorophenyl)sulfonyloxy-3-methoxyphenyl]prop-2-enoate
—— methyl 10,23-bis[[(E)-but-2-enoyl]amino]-16-hydroxy-15-methyl-3-oxo-28-oxa-4,14,19-triazaoctacyclo[12.11.2.115,18.02,6.07,27.08,13.019,26.020,25]octacosa-1,6,8(13),9,11,20(25),21,23,26-nonaene-16-carboxylate —— C35H31N5O7
methyl 10,23-bis[[(E)-but-2-enoyl]amino]-16-hydroxy-15-methyl-3-oxo-28-oxa-4,14,19-triazaoctacyclo[12.11.2.115,18.02,6.07,27.08,13.019,26.020,25]octacosa-1,6,8(13),9,11,20(25),21,23,26-nonaene-16-carboxylate
—— methyl N-[4-[2-[(5E)-5-[(2-fluorophenyl)methylidene]-2,4-dioxo-1,3-thiazolidin-3-yl]ethylcarbamoyl]phenyl]carbamate —— C21H18FN3O5S
methyl N-[4-[2-[(5E)-5-[(2-fluorophenyl)methylidene]-2,4-dioxo-1,3-thiazolidin-3-yl]ethylcarbamoyl]phenyl]carbamate
—— methyl (Z)-3-[4-(4-acetamido-3-methylanilino)-3-nitrophenyl]prop-2-enoate —— C19H19N3O5
methyl (Z)-3-[4-(4-acetamido-3-methylanilino)-3-nitrophenyl]prop-2-enoate
—— methyl (Z)-3-[4-(3-fluorophenyl)sulfonyloxy-3-methoxyphenyl]prop-2-enoate —— C17H15FO6S
methyl (Z)-3-[4-(3-fluorophenyl)sulfonyloxy-3-methoxyphenyl]prop-2-enoate
—— methyl (2R)-2-[(6-bromo-1,3-benzothiazol-2-yl)amino]-2-[(2,4-dichlorobenzoyl)amino]-3,3,3-trifluoropropanoate —— C18H11BrCl2F3N3O3S
methyl (2R)-2-[(6-bromo-1,3-benzothiazol-2-yl)amino]-2-[(2,4-dichlorobenzoyl)amino]-3,3,3-trifluoropropanoate
—— methyl (Z)-3-[4-[4-(2-anilino-2-oxoethyl)piperazin-1-yl]-3-nitrophenyl]prop-2-enoate —— C22H24N4O5
methyl (Z)-3-[4-[4-(2-anilino-2-oxoethyl)piperazin-1-yl]-3-nitrophenyl]prop-2-enoate
—— methyl (2R)-2-[[(Z)-2-cyano-3-[4-(dimethylamino)phenyl]prop-2-enoyl]amino]-3-(1H-indol-3-yl)propanoate —— C24H24N4O3
methyl (2R)-2-[[(Z)-2-cyano-3-[4-(dimethylamino)phenyl]prop-2-enoyl]amino]-3-(1H-indol-3-yl)propanoate
—— methyl (E)-3-[3-methoxy-4-[(Z)-3-(3-methoxy-4-prop-2-enoxyphenyl)prop-2-enoyl]oxyphenyl]prop-2-enoate —— C24H24O7
methyl (E)-3-[3-methoxy-4-[(Z)-3-(3-methoxy-4-prop-2-enoxyphenyl)prop-2-enoyl]oxyphenyl]prop-2-enoate
—— methyl 5-[[(Z)-3-(3-chlorophenyl)prop-2-enoyl]amino]-2,4-difluorobenzoate —— C17H12ClF2NO3
methyl 5-[[(Z)-3-(3-chlorophenyl)prop-2-enoyl]amino]-2,4-difluorobenzoate
—— methyl 3-[2-[3-[[(Z)-3-(furan-2-yl)prop-2-enoyl]amino]phenyl]ethynyl]benzoate —— C23H17NO4
methyl 3-[2-[3-[[(Z)-3-(furan-2-yl)prop-2-enoyl]amino]phenyl]ethynyl]benzoate
—— methyl (2S)-2-[4-[(Z)-3-(1,3-benzodioxol-5-yl)prop-2-enoyl]piperazin-1-yl]-2-(2-chlorophenyl)acetate —— C23H23ClN2O5
methyl (2S)-2-[4-[(Z)-3-(1,3-benzodioxol-5-yl)prop-2-enoyl]piperazin-1-yl]-2-(2-chlorophenyl)acetate
—— methyl (2S)-2-[[(Z)-2-cyano-3-[4-(dimethylamino)phenyl]prop-2-enoyl]amino]-3-(1H-indol-3-yl)propanoate —— C24H24N4O3
methyl (2S)-2-[[(Z)-2-cyano-3-[4-(dimethylamino)phenyl]prop-2-enoyl]amino]-3-(1H-indol-3-yl)propanoate