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—— methyl (5S)-7-methyl-5-(2-methylphenyl)-3-[2-oxo-2-[[(2R)-oxolan-2-yl]methylamino]ethyl]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C23H27N3O4S
methyl (5S)-7-methyl-5-(2-methylphenyl)-3-[2-oxo-2-[[(2R)-oxolan-2-yl]methylamino]ethyl]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— methyl 3-[[(2S)-2-[(2S,6S)-2,6-dimethylmorpholin-4-ium-4-yl]propanoyl]amino]-1H-indole-2-carboxylate —— C19H26N3O4+
methyl 3-[[(2S)-2-[(2S,6S)-2,6-dimethylmorpholin-4-ium-4-yl]propanoyl]amino]-1H-indole-2-carboxylate
—— methyl (5S)-5-(4-chlorophenyl)-7-methyl-3-[2-oxo-2-[[(2S)-oxolan-2-yl]methylamino]ethyl]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C22H24ClN3O4S
methyl (5S)-5-(4-chlorophenyl)-7-methyl-3-[2-oxo-2-[[(2S)-oxolan-2-yl]methylamino]ethyl]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— methyl (1S,2R,3R,8aS)-6-acetyl-3-carbamoyl-1-cyano-2-(2-fluorophenyl)-3,8a-dihydro-2H-indolizine-1-carboxylate —— C20H18FN3O4
methyl (1S,2R,3R,8aS)-6-acetyl-3-carbamoyl-1-cyano-2-(2-fluorophenyl)-3,8a-dihydro-2H-indolizine-1-carboxylate
—— methyl (5S)-3-[2-[[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]amino]-2-oxoethyl]-7-ethyl-5-(2-methoxyphenyl)-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C26H31N3O4S
methyl (5S)-3-[2-[[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]amino]-2-oxoethyl]-7-ethyl-5-(2-methoxyphenyl)-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— methyl (1S,9S,12R)-9,10-dimethyl-11-oxo-8-oxa-10-azatricyclo[7.3.1.02,7]trideca-2,4,6-triene-12-carboxylate —— C15H17NO4
methyl (1S,9S,12R)-9,10-dimethyl-11-oxo-8-oxa-10-azatricyclo[7.3.1.02,7]trideca-2,4,6-triene-12-carboxylate
—— methyl (5R)-3-[2-(tert-butylamino)-2-oxoethyl]-7-ethyl-5-(2-methoxyphenyl)-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C23H29N3O4S
methyl (5R)-3-[2-(tert-butylamino)-2-oxoethyl]-7-ethyl-5-(2-methoxyphenyl)-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— methyl (5S)-3-[2-(cyclohexylamino)-2-oxoethyl]-7-ethyl-5-(2-methoxyphenyl)-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C25H31N3O4S
methyl (5S)-3-[2-(cyclohexylamino)-2-oxoethyl]-7-ethyl-5-(2-methoxyphenyl)-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— methyl (5R)-7-methyl-5-(2-methylphenyl)-3-[2-oxo-2-[[(2R)-oxolan-2-yl]methylamino]ethyl]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C23H27N3O4S
methyl (5R)-7-methyl-5-(2-methylphenyl)-3-[2-oxo-2-[[(2R)-oxolan-2-yl]methylamino]ethyl]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— methyl (2E,5S)-5-[4-(diethylamino)phenyl]-2-[[4-(difluoromethoxy)-3-methoxyphenyl]methylidene]-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C28H29F2N3O5S
methyl (2E,5S)-5-[4-(diethylamino)phenyl]-2-[[4-(difluoromethoxy)-3-methoxyphenyl]methylidene]-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— methyl (5R)-7-ethyl-5-(2-methoxyphenyl)-3-[2-oxo-2-(2-phenylethylamino)ethyl]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C27H29N3O4S
methyl (5R)-7-ethyl-5-(2-methoxyphenyl)-3-[2-oxo-2-(2-phenylethylamino)ethyl]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— methyl (1S,9R,13Z,16S)-13-[[4-(difluoromethoxy)-3-methoxyphenyl]methylidene]-9-methyl-14-oxo-8-oxa-12-thia-10,15-diazatetracyclo[7.6.1.02,7.011,15]hexadeca-2,4,6,10-tetraene-16-carboxylate —— C24H20F2N2O6S
methyl (1S,9R,13Z,16S)-13-[[4-(difluoromethoxy)-3-methoxyphenyl]methylidene]-9-methyl-14-oxo-8-oxa-12-thia-10,15-diazatetracyclo[7.6.1.02,7.011,15]hexadeca-2,4,6,10-tetraene-16-carboxylate
—— methyl (5R)-5-(4-chlorophenyl)-7-methyl-3-[2-oxo-2-[[(2S)-oxolan-2-yl]methylamino]ethyl]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C22H24ClN3O4S
methyl (5R)-5-(4-chlorophenyl)-7-methyl-3-[2-oxo-2-[[(2S)-oxolan-2-yl]methylamino]ethyl]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— methyl (5R)-7-ethyl-3-[2-oxo-2-(2-phenoxyethylamino)ethyl]-5-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C26H27N3O4S
methyl (5R)-7-ethyl-3-[2-oxo-2-(2-phenoxyethylamino)ethyl]-5-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— methyl (5S)-3-[2-(tert-butylamino)-2-oxoethyl]-7-ethyl-5-(2-methoxyphenyl)-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C23H29N3O4S
methyl (5S)-3-[2-(tert-butylamino)-2-oxoethyl]-7-ethyl-5-(2-methoxyphenyl)-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— methyl (5S)-7-ethyl-5-(2-methoxyphenyl)-3-[2-oxo-2-(2-phenylethylamino)ethyl]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C27H29N3O4S
methyl (5S)-7-ethyl-5-(2-methoxyphenyl)-3-[2-oxo-2-(2-phenylethylamino)ethyl]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— methyl 5-chloro-3-[[(2S)-2-[(3S)-3-methylpiperidin-1-yl]propanoyl]amino]-1H-indole-2-carboxylate —— C19H24ClN3O3
methyl 5-chloro-3-[[(2S)-2-[(3S)-3-methylpiperidin-1-yl]propanoyl]amino]-1H-indole-2-carboxylate
—— methyl (5S)-3-[2-[[(1R,2S,4R)-2-bicyclo[2.2.1]heptanyl]amino]-2-oxoethyl]-7-ethyl-5-(2-methoxyphenyl)-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C26H31N3O4S
methyl (5S)-3-[2-[[(1R,2S,4R)-2-bicyclo[2.2.1]heptanyl]amino]-2-oxoethyl]-7-ethyl-5-(2-methoxyphenyl)-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— methyl (5S)-3-[2-[(4-fluorophenyl)methylamino]-2-oxoethyl]-7-methyl-5-(3-phenylmethoxyphenyl)-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C31H28FN3O4S
methyl (5S)-3-[2-[(4-fluorophenyl)methylamino]-2-oxoethyl]-7-methyl-5-(3-phenylmethoxyphenyl)-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— methyl (5S)-7-ethyl-3-[2-(3-methoxyanilino)-2-oxoethyl]-5-(3-methylphenyl)-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C26H27N3O4S
methyl (5S)-7-ethyl-3-[2-(3-methoxyanilino)-2-oxoethyl]-5-(3-methylphenyl)-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— methyl (5R)-3-[2-(benzylamino)-2-oxoethyl]-5-(4-methoxyphenyl)-7-methyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C25H25N3O4S
methyl (5R)-3-[2-(benzylamino)-2-oxoethyl]-5-(4-methoxyphenyl)-7-methyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— methyl (5R)-7-ethyl-3-[2-(3-methoxyanilino)-2-oxoethyl]-5-(3-methylphenyl)-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C26H27N3O4S
methyl (5R)-7-ethyl-3-[2-(3-methoxyanilino)-2-oxoethyl]-5-(3-methylphenyl)-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— methyl (5R)-3-[2-(cyclohexylamino)-2-oxoethyl]-7-ethyl-5-(2-methoxyphenyl)-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C25H31N3O4S
methyl (5R)-3-[2-(cyclohexylamino)-2-oxoethyl]-7-ethyl-5-(2-methoxyphenyl)-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— methyl (5S)-5-(2,4-dimethylphenyl)-7-methyl-3-[2-oxo-2-[[(2R)-oxolan-2-yl]methylamino]ethyl]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C24H29N3O4S
methyl (5S)-5-(2,4-dimethylphenyl)-7-methyl-3-[2-oxo-2-[[(2R)-oxolan-2-yl]methylamino]ethyl]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— methyl (5R)-7-ethyl-3-[2-[(3-fluorophenyl)methylamino]-2-oxoethyl]-5-(2-methoxyphenyl)-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C26H26FN3O4S
methyl (5R)-7-ethyl-3-[2-[(3-fluorophenyl)methylamino]-2-oxoethyl]-5-(2-methoxyphenyl)-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— methyl (5S)-7-ethyl-3-[2-(4-methoxyanilino)-2-oxoethyl]-5-(3-methylphenyl)-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C26H27N3O4S
methyl (5S)-7-ethyl-3-[2-(4-methoxyanilino)-2-oxoethyl]-5-(3-methylphenyl)-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— methyl (5S)-5-(2,4-dimethylphenyl)-7-methyl-3-[2-oxo-2-[[(2S)-oxolan-2-yl]methylamino]ethyl]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C24H29N3O4S
methyl (5S)-5-(2,4-dimethylphenyl)-7-methyl-3-[2-oxo-2-[[(2S)-oxolan-2-yl]methylamino]ethyl]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— methyl 7-[[(2R,6R)-2,6-dimethylmorpholin-4-yl]methylideneamino]-2-oxo-1H-thieno[2,3-b][1,4]thiazine-6-carboxylate —— C15H19N3O4S2
methyl 7-[[(2R,6R)-2,6-dimethylmorpholin-4-yl]methylideneamino]-2-oxo-1H-thieno[2,3-b][1,4]thiazine-6-carboxylate
—— methyl (5R)-3-[2-[(4-fluorophenyl)methylamino]-2-oxoethyl]-7-methyl-5-(3-phenylmethoxyphenyl)-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C31H28FN3O4S
methyl (5R)-3-[2-[(4-fluorophenyl)methylamino]-2-oxoethyl]-7-methyl-5-(3-phenylmethoxyphenyl)-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— methyl (2R)-2-[4-[(3,4-dichlorophenyl)carbamoylamino]-3-methoxyphenyl]-3,3,3-trifluoro-2-hydroxypropanoate —— C18H15Cl2F3N2O5
methyl (2R)-2-[4-[(3,4-dichlorophenyl)carbamoylamino]-3-methoxyphenyl]-3,3,3-trifluoro-2-hydroxypropanoate
—— methyl (5R)-3-[2-(benzylamino)-2-oxoethyl]-7-ethyl-5-(4-methoxyphenyl)-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C26H27N3O4S
methyl (5R)-3-[2-(benzylamino)-2-oxoethyl]-7-ethyl-5-(4-methoxyphenyl)-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— methyl (5R)-3-[2-(cyclopropylmethylamino)-2-oxoethyl]-5-(2-methoxyphenyl)-7-methyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C22H25N3O4S
methyl (5R)-3-[2-(cyclopropylmethylamino)-2-oxoethyl]-5-(2-methoxyphenyl)-7-methyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— methyl (5S)-7-ethyl-3-[2-oxo-2-(2-phenoxyethylamino)ethyl]-5-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C26H27N3O4S
methyl (5S)-7-ethyl-3-[2-oxo-2-(2-phenoxyethylamino)ethyl]-5-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— methyl 7-[[(2S,6S)-2,6-dimethylmorpholin-4-yl]methylideneamino]-2-oxo-1H-thieno[2,3-b][1,4]thiazine-6-carboxylate —— C15H19N3O4S2
methyl 7-[[(2S,6S)-2,6-dimethylmorpholin-4-yl]methylideneamino]-2-oxo-1H-thieno[2,3-b][1,4]thiazine-6-carboxylate
—— methyl (5S)-3-[2-(cyclopropylmethylamino)-2-oxoethyl]-5-(4-methoxyphenyl)-7-methyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C22H25N3O4S
methyl (5S)-3-[2-(cyclopropylmethylamino)-2-oxoethyl]-5-(4-methoxyphenyl)-7-methyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— methyl (5R)-7-ethyl-3-[2-(4-methoxyanilino)-2-oxoethyl]-5-(3-methylphenyl)-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C26H27N3O4S
methyl (5R)-7-ethyl-3-[2-(4-methoxyanilino)-2-oxoethyl]-5-(3-methylphenyl)-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— methyl (1R,2R,3R,3aR)-1-(4-chlorobenzoyl)-3-cyano-2-[4-(dimethylamino)phenyl]-2,3a-dihydro-1H-pyrrolo[1,2-a]quinoline-3-carboxylate —— C30H26ClN3O3
methyl (1R,2R,3R,3aR)-1-(4-chlorobenzoyl)-3-cyano-2-[4-(dimethylamino)phenyl]-2,3a-dihydro-1H-pyrrolo[1,2-a]quinoline-3-carboxylate
—— methyl (1R,3R,4R)-2-(4-methylphenyl)sulfonyl-3-(trifluoromethyl)-2-azabicyclo[2.2.1]hept-5-ene-3-carboxylate —— C16H16F3NO4S
methyl (1R,3R,4R)-2-(4-methylphenyl)sulfonyl-3-(trifluoromethyl)-2-azabicyclo[2.2.1]hept-5-ene-3-carboxylate
—— methyl (5R)-5-(2,4-dimethylphenyl)-7-methyl-3-[2-oxo-2-[[(2R)-oxolan-2-yl]methylamino]ethyl]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C24H29N3O4S
methyl (5R)-5-(2,4-dimethylphenyl)-7-methyl-3-[2-oxo-2-[[(2R)-oxolan-2-yl]methylamino]ethyl]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— methyl (5S)-5-(2-chlorophenyl)-7-ethyl-3-[2-oxo-2-[[(2R)-oxolan-2-yl]methylamino]ethyl]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C23H26ClN3O4S
methyl (5S)-5-(2-chlorophenyl)-7-ethyl-3-[2-oxo-2-[[(2R)-oxolan-2-yl]methylamino]ethyl]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— methyl (5S)-3-[2-(benzylamino)-2-oxoethyl]-5-(4-methoxyphenyl)-7-methyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C25H25N3O4S
methyl (5S)-3-[2-(benzylamino)-2-oxoethyl]-5-(4-methoxyphenyl)-7-methyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— methyl (5R)-5-(2-chlorophenyl)-7-ethyl-3-[2-oxo-2-[[(2S)-oxolan-2-yl]methylamino]ethyl]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C23H26ClN3O4S
methyl (5R)-5-(2-chlorophenyl)-7-ethyl-3-[2-oxo-2-[[(2S)-oxolan-2-yl]methylamino]ethyl]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— methyl (5R)-7-ethyl-5-(2-methoxyphenyl)-3-[2-oxo-2-(2-thiophen-2-ylethylamino)ethyl]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C25H27N3O4S2
methyl (5R)-7-ethyl-5-(2-methoxyphenyl)-3-[2-oxo-2-(2-thiophen-2-ylethylamino)ethyl]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— methyl 7-[[(2R,6S)-2,6-dimethylmorpholin-4-yl]methylideneamino]-2-oxo-1H-thieno[2,3-b][1,4]thiazine-6-carboxylate —— C15H19N3O4S2
methyl 7-[[(2R,6S)-2,6-dimethylmorpholin-4-yl]methylideneamino]-2-oxo-1H-thieno[2,3-b][1,4]thiazine-6-carboxylate
—— methyl (5R)-5-(2-chlorophenyl)-7-ethyl-3-[2-oxo-2-[[(2R)-oxolan-2-yl]methylamino]ethyl]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C23H26ClN3O4S
methyl (5R)-5-(2-chlorophenyl)-7-ethyl-3-[2-oxo-2-[[(2R)-oxolan-2-yl]methylamino]ethyl]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— methyl (5S)-5-(2-chlorophenyl)-7-ethyl-3-[2-oxo-2-[[(2S)-oxolan-2-yl]methylamino]ethyl]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C23H26ClN3O4S
methyl (5S)-5-(2-chlorophenyl)-7-ethyl-3-[2-oxo-2-[[(2S)-oxolan-2-yl]methylamino]ethyl]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— methyl (5R)-3-[2-[[(1R,2S,4R)-2-bicyclo[2.2.1]heptanyl]amino]-2-oxoethyl]-7-ethyl-5-(2-methoxyphenyl)-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C26H31N3O4S
methyl (5R)-3-[2-[[(1R,2S,4R)-2-bicyclo[2.2.1]heptanyl]amino]-2-oxoethyl]-7-ethyl-5-(2-methoxyphenyl)-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— methyl 1-[(1S,4S)-4,7,7-trimethyl-3-oxobicyclo[2.2.1]heptane-1-carbonyl]piperidine-4-carboxylate —— C18H27NO4
methyl 1-[(1S,4S)-4,7,7-trimethyl-3-oxobicyclo[2.2.1]heptane-1-carbonyl]piperidine-4-carboxylate
—— methyl 2-[(6aR)-3-(4-chlorophenyl)-4,6-dioxo-2,6a-dihydropyrrolo[3,4-d][1,2]oxazol-5-yl]benzoate —— C19H13ClN2O5
methyl 2-[(6aR)-3-(4-chlorophenyl)-4,6-dioxo-2,6a-dihydropyrrolo[3,4-d][1,2]oxazol-5-yl]benzoate
—— methyl 3-[[(5S,7S)-3-bromoadamantane-1-carbonyl]amino]-5-chloro-1H-indole-2-carboxylate —— C21H22BrClN2O3
methyl 3-[[(5S,7S)-3-bromoadamantane-1-carbonyl]amino]-5-chloro-1H-indole-2-carboxylate