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中文名称 英文名称 CAS号 化学式 结构式图片
—— Methyl 6-[(2,5-dimethylphenyl)sulfonylamino]hexanoate —— C15H23NO4S
Methyl 6-[(2,5-dimethylphenyl)sulfonylamino]hexanoate
—— methyl 5-[(2S)-2-[[(1R)-1-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]amino]propanoyl]-2,4-dimethyl-1H-pyrrole-3-carboxylate —— C20H30N2O3
methyl 5-[(2S)-2-[[(1R)-1-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]amino]propanoyl]-2,4-dimethyl-1H-pyrrole-3-carboxylate
—— methyl (3R)-3-[2-[2-(4-ethoxyanilino)-2-oxoethoxy]-2-oxoethyl]-5-methyl-2-oxo-1,3-dihydropyrrole-4-carboxylate —— C19H22N2O7
methyl (3R)-3-[2-[2-(4-ethoxyanilino)-2-oxoethoxy]-2-oxoethyl]-5-methyl-2-oxo-1,3-dihydropyrrole-4-carboxylate
—— methyl (3S)-3-[2-[(2-methoxyphenyl)methyl-methylamino]-2-oxoethyl]-5-methyl-2-oxo-1,3-dihydropyrrole-4-carboxylate —— C18H22N2O5
methyl (3S)-3-[2-[(2-methoxyphenyl)methyl-methylamino]-2-oxoethyl]-5-methyl-2-oxo-1,3-dihydropyrrole-4-carboxylate
—— methyl (2S)-4-(2,3-dihydro-1H-inden-5-ylsulfonyl)-2,3-dihydro-1,4-benzoxazine-2-carboxylate —— C19H19NO5S
methyl (2S)-4-(2,3-dihydro-1H-inden-5-ylsulfonyl)-2,3-dihydro-1,4-benzoxazine-2-carboxylate
—— methyl (3R)-3-[2-[(2-methoxyphenyl)methyl-methylamino]-2-oxoethyl]-5-methyl-2-oxo-1,3-dihydropyrrole-4-carboxylate —— C18H22N2O5
methyl (3R)-3-[2-[(2-methoxyphenyl)methyl-methylamino]-2-oxoethyl]-5-methyl-2-oxo-1,3-dihydropyrrole-4-carboxylate
—— methyl (2S)-4-(4-ethoxyphenyl)sulfonyl-2,3-dihydro-1,4-benzoxazine-2-carboxylate —— C18H19NO6S
methyl (2S)-4-(4-ethoxyphenyl)sulfonyl-2,3-dihydro-1,4-benzoxazine-2-carboxylate
—— methyl (5R)-5-(2,4-dimethylphenyl)-7-methyl-3-[2-(4-methylpiperazin-1-yl)-2-oxoethyl]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C24H30N4O3S
methyl (5R)-5-(2,4-dimethylphenyl)-7-methyl-3-[2-(4-methylpiperazin-1-yl)-2-oxoethyl]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— Methyl 6-[(4-cyclohexylphenyl)sulfonylamino]hexanoate —— C19H29NO4S
Methyl 6-[(4-cyclohexylphenyl)sulfonylamino]hexanoate
—— Methyl 4-[(4-bromo-3-methylphenyl)sulfonylamino]butanoate —— C12H16BrNO4S
Methyl 4-[(4-bromo-3-methylphenyl)sulfonylamino]butanoate
—— methyl (5R)-5-(3-chlorophenyl)-3-[2-[(3R)-3-(dimethylamino)pyrrolidin-1-yl]-2-oxoethyl]-7-methyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C23H27ClN4O3S
methyl (5R)-5-(3-chlorophenyl)-3-[2-[(3R)-3-(dimethylamino)pyrrolidin-1-yl]-2-oxoethyl]-7-methyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— methyl (5R)-7-ethyl-3-[2-(4-methyl-1,4-diazepan-1-yl)-2-oxoethyl]-5-(3-methylphenyl)-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C25H32N4O3S
methyl (5R)-7-ethyl-3-[2-(4-methyl-1,4-diazepan-1-yl)-2-oxoethyl]-5-(3-methylphenyl)-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— methyl (5R)-5-(4-chlorophenyl)-3-[2-[4-(dimethylamino)piperidin-1-yl]-2-oxoethyl]-7-methyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C24H29ClN4O3S
methyl (5R)-5-(4-chlorophenyl)-3-[2-[4-(dimethylamino)piperidin-1-yl]-2-oxoethyl]-7-methyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— methyl (5S)-5-(4-chlorophenyl)-3-[2-[4-(dimethylamino)piperidin-1-yl]-2-oxoethyl]-7-methyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C24H29ClN4O3S
methyl (5S)-5-(4-chlorophenyl)-3-[2-[4-(dimethylamino)piperidin-1-yl]-2-oxoethyl]-7-methyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— Methyl 6-[[4-(trifluoromethoxy)phenyl]sulfonylamino]hexanoate —— C14H18F3NO5S
Methyl 6-[[4-(trifluoromethoxy)phenyl]sulfonylamino]hexanoate
—— methyl (5R)-5-(3-chlorophenyl)-3-[2-[(3S)-3-(dimethylamino)pyrrolidin-1-yl]-2-oxoethyl]-7-methyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C23H27ClN4O3S
methyl (5R)-5-(3-chlorophenyl)-3-[2-[(3S)-3-(dimethylamino)pyrrolidin-1-yl]-2-oxoethyl]-7-methyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— methyl 4-[[(Z)-3-[4-(5-pentylpyridin-2-yl)phenyl]prop-2-enoyl]amino]benzoate —— C27H28N2O3
methyl 4-[[(Z)-3-[4-(5-pentylpyridin-2-yl)phenyl]prop-2-enoyl]amino]benzoate
—— methyl (3R)-3-[2-[1,3-benzodioxol-5-ylmethyl(ethyl)amino]-2-oxoethyl]-5-methyl-2-oxo-1,3-dihydropyrrole-4-carboxylate —— C19H22N2O6
methyl (3R)-3-[2-[1,3-benzodioxol-5-ylmethyl(ethyl)amino]-2-oxoethyl]-5-methyl-2-oxo-1,3-dihydropyrrole-4-carboxylate
—— methyl 5-[(2R)-2-[[(1R)-1-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]amino]propanoyl]-2,4-dimethyl-1H-pyrrole-3-carboxylate —— C20H30N2O3
methyl 5-[(2R)-2-[[(1R)-1-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]amino]propanoyl]-2,4-dimethyl-1H-pyrrole-3-carboxylate
—— methyl (5S)-7-ethyl-3-[2-(4-methyl-1,4-diazepan-1-yl)-2-oxoethyl]-5-(3-methylphenyl)-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C25H32N4O3S
methyl (5S)-7-ethyl-3-[2-(4-methyl-1,4-diazepan-1-yl)-2-oxoethyl]-5-(3-methylphenyl)-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— methyl (5S)-7-ethyl-5-(4-methylphenyl)-3-[2-(4-methylpiperazin-1-yl)-2-oxoethyl]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C24H30N4O3S
methyl (5S)-7-ethyl-5-(4-methylphenyl)-3-[2-(4-methylpiperazin-1-yl)-2-oxoethyl]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— methyl (5S)-5-(3-chlorophenyl)-3-[2-[(3S)-3-(dimethylamino)pyrrolidin-1-yl]-2-oxoethyl]-7-methyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C23H27ClN4O3S
methyl (5S)-5-(3-chlorophenyl)-3-[2-[(3S)-3-(dimethylamino)pyrrolidin-1-yl]-2-oxoethyl]-7-methyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— methyl (5R)-7-ethyl-3-[2-[methyl-(1-methylpiperidin-4-yl)amino]-2-oxoethyl]-5-(3-methylphenyl)-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C26H34N4O3S
methyl (5R)-7-ethyl-3-[2-[methyl-(1-methylpiperidin-4-yl)amino]-2-oxoethyl]-5-(3-methylphenyl)-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— methyl (5S)-7-ethyl-3-[2-(4-methylpiperazin-1-yl)-2-oxoethyl]-5-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C23H28N4O3S
methyl (5S)-7-ethyl-3-[2-(4-methylpiperazin-1-yl)-2-oxoethyl]-5-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— methyl (5S)-7-ethyl-3-[2-[methyl-(1-methylpiperidin-4-yl)amino]-2-oxoethyl]-5-(3-methylphenyl)-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C26H34N4O3S
methyl (5S)-7-ethyl-3-[2-[methyl-(1-methylpiperidin-4-yl)amino]-2-oxoethyl]-5-(3-methylphenyl)-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— methyl (5S)-5-(3-chlorophenyl)-3-[2-[(3R)-3-(dimethylamino)pyrrolidin-1-yl]-2-oxoethyl]-7-methyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C23H27ClN4O3S
methyl (5S)-5-(3-chlorophenyl)-3-[2-[(3R)-3-(dimethylamino)pyrrolidin-1-yl]-2-oxoethyl]-7-methyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— methyl (5S)-7-ethyl-3-[2-(4-methylpiperazin-1-yl)-2-oxoethyl]-5-(4-propan-2-ylphenyl)-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C26H34N4O3S
methyl (5S)-7-ethyl-3-[2-(4-methylpiperazin-1-yl)-2-oxoethyl]-5-(4-propan-2-ylphenyl)-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— methyl (5R)-7-ethyl-3-[2-(4-methylpiperazin-1-yl)-2-oxoethyl]-5-(4-propan-2-ylphenyl)-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C26H34N4O3S
methyl (5R)-7-ethyl-3-[2-(4-methylpiperazin-1-yl)-2-oxoethyl]-5-(4-propan-2-ylphenyl)-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— methyl (5R)-7-ethyl-3-[2-(4-methylpiperazin-1-yl)-2-oxoethyl]-5-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C23H28N4O3S
methyl (5R)-7-ethyl-3-[2-(4-methylpiperazin-1-yl)-2-oxoethyl]-5-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— methyl (13R,14R,15S)-14-ethyl-14-(4-methylbenzoyl)-12-oxo-11-oxatetracyclo[8.5.0.02,7.013,15]pentadeca-1(10),2,4,6,8-pentaene-13-carboxylate —— C26H22O5
methyl (13R,14R,15S)-14-ethyl-14-(4-methylbenzoyl)-12-oxo-11-oxatetracyclo[8.5.0.02,7.013,15]pentadeca-1(10),2,4,6,8-pentaene-13-carboxylate
—— methyl (5R)-7-methyl-3-[2-(4-methyl-1,4-diazepan-1-yl)-2-oxoethyl]-5-(4-propan-2-ylphenyl)-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C26H34N4O3S
methyl (5R)-7-methyl-3-[2-(4-methyl-1,4-diazepan-1-yl)-2-oxoethyl]-5-(4-propan-2-ylphenyl)-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— methyl (5S)-7-methyl-3-[2-(4-methyl-1,4-diazepan-1-yl)-2-oxoethyl]-5-(4-propan-2-ylphenyl)-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C26H34N4O3S
methyl (5S)-7-methyl-3-[2-(4-methyl-1,4-diazepan-1-yl)-2-oxoethyl]-5-(4-propan-2-ylphenyl)-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— methyl (2R)-4-(4-bromophenyl)sulfonyl-2,3-dihydro-1,4-benzoxazine-2-carboxylate —— C16H14BrNO5S
methyl (2R)-4-(4-bromophenyl)sulfonyl-2,3-dihydro-1,4-benzoxazine-2-carboxylate
—— methyl (2R)-4-(4-methoxyphenyl)sulfonyl-2,3-dihydro-1,4-benzoxazine-2-carboxylate —— C17H17NO6S
methyl (2R)-4-(4-methoxyphenyl)sulfonyl-2,3-dihydro-1,4-benzoxazine-2-carboxylate
—— Methyl 4-[(2,3,5,6-tetramethylphenyl)sulfonylamino]butanoate —— C15H23NO4S
Methyl 4-[(2,3,5,6-tetramethylphenyl)sulfonylamino]butanoate
—— methyl (2S)-4-(4-methylphenyl)sulfonyl-2,3-dihydro-1,4-benzoxazine-2-carboxylate —— C17H17NO5S
methyl (2S)-4-(4-methylphenyl)sulfonyl-2,3-dihydro-1,4-benzoxazine-2-carboxylate
—— Methyl 4-[(2,6-dichlorophenyl)sulfonylamino]butanoate —— C11H13Cl2NO4S
Methyl 4-[(2,6-dichlorophenyl)sulfonylamino]butanoate
—— Methyl 4-[(2,3,4,5,6-pentamethylphenyl)sulfonylamino]butanoate —— C16H25NO4S
Methyl 4-[(2,3,4,5,6-pentamethylphenyl)sulfonylamino]butanoate
—— methyl 4-[[(5S)-5-(pyrrolidin-1-ylmethyl)-1,4-thiazepan-4-yl]sulfonyl]benzoate —— C18H26N2O4S2
methyl 4-[[(5S)-5-(pyrrolidin-1-ylmethyl)-1,4-thiazepan-4-yl]sulfonyl]benzoate
—— methyl (Z)-3-(thiophene-2-carbonylamino)but-2-enoate —— C10H11NO3S
methyl (Z)-3-(thiophene-2-carbonylamino)but-2-enoate
—— methyl N-[(2S)-2-[[5-(3,5-dimethoxyphenyl)-1,3,4-oxadiazol-2-yl]sulfanyl]propanoyl]carbamate —— C15H17N3O6S
methyl N-[(2S)-2-[[5-(3,5-dimethoxyphenyl)-1,3,4-oxadiazol-2-yl]sulfanyl]propanoyl]carbamate
—— methyl 4-[[(5R)-5-(pyrrolidin-1-ylmethyl)-1,4-thiazepan-4-yl]sulfonyl]benzoate —— C18H26N2O4S2
methyl 4-[[(5R)-5-(pyrrolidin-1-ylmethyl)-1,4-thiazepan-4-yl]sulfonyl]benzoate
—— methyl (5R)-5-(4-methoxyphenyl)-7-methyl-3-[2-(4-methylpiperazin-1-yl)-2-oxoethyl]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C23H28N4O4S
methyl (5R)-5-(4-methoxyphenyl)-7-methyl-3-[2-(4-methylpiperazin-1-yl)-2-oxoethyl]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— methyl (5S)-5-(4-methoxyphenyl)-7-methyl-3-[2-(4-methylpiperazin-1-yl)-2-oxoethyl]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C23H28N4O4S
methyl (5S)-5-(4-methoxyphenyl)-7-methyl-3-[2-(4-methylpiperazin-1-yl)-2-oxoethyl]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— methyl (5R)-5-(4-chlorophenyl)-7-ethyl-3-[2-(4-methylpiperazin-1-yl)-2-oxoethyl]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C23H27ClN4O3S
methyl (5R)-5-(4-chlorophenyl)-7-ethyl-3-[2-(4-methylpiperazin-1-yl)-2-oxoethyl]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— methyl 4-chloro-3-[[(2Z,4Z)-hexa-2,4-dienoyl]amino]benzoate —— C14H14ClNO3
methyl 4-chloro-3-[[(2Z,4Z)-hexa-2,4-dienoyl]amino]benzoate
—— methyl 4-chloro-3-[[(2Z,4E)-hexa-2,4-dienoyl]amino]benzoate —— C14H14ClNO3
methyl 4-chloro-3-[[(2Z,4E)-hexa-2,4-dienoyl]amino]benzoate
—— methyl 1-[(Z)-3-(4-fluorophenyl)prop-2-enoyl]piperidine-4-carboxylate —— C16H18FNO3
methyl 1-[(Z)-3-(4-fluorophenyl)prop-2-enoyl]piperidine-4-carboxylate
—— methyl 4-chloro-3-[[(2E,4Z)-hexa-2,4-dienoyl]amino]benzoate —— C14H14ClNO3
methyl 4-chloro-3-[[(2E,4Z)-hexa-2,4-dienoyl]amino]benzoate
—— methyl (5S)-5-(2,4-dimethylphenyl)-7-methyl-3-[2-oxo-2-(pyridin-2-ylmethylamino)ethyl]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C25H26N4O3S
methyl (5S)-5-(2,4-dimethylphenyl)-7-methyl-3-[2-oxo-2-(pyridin-2-ylmethylamino)ethyl]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate