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—— methyl (5R)-5-(2-methoxyphenyl)-7-methyl-3-[2-oxo-2-(4-propan-2-ylanilino)ethyl]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C27H29N3O4S
methyl (5R)-5-(2-methoxyphenyl)-7-methyl-3-[2-oxo-2-(4-propan-2-ylanilino)ethyl]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— methyl (5R)-5-(3-methoxyphenyl)-7-methyl-3-[2-oxo-2-(3-phenylpropylamino)ethyl]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C27H29N3O4S
methyl (5R)-5-(3-methoxyphenyl)-7-methyl-3-[2-oxo-2-(3-phenylpropylamino)ethyl]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— methyl (5S)-7-ethyl-5-(2-fluorophenyl)-3-[2-(3-methoxyanilino)-2-oxoethyl]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C25H24FN3O4S
methyl (5S)-7-ethyl-5-(2-fluorophenyl)-3-[2-(3-methoxyanilino)-2-oxoethyl]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— methyl (5R)-7-ethyl-5-(3-methylphenyl)-3-[2-oxo-2-(2-phenoxyethylamino)ethyl]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C27H29N3O4S
methyl (5R)-7-ethyl-5-(3-methylphenyl)-3-[2-oxo-2-(2-phenoxyethylamino)ethyl]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— methyl (5R)-3-[2-(benzylamino)-2-oxoethyl]-7-ethyl-5-(2-methoxyphenyl)-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C26H27N3O4S
methyl (5R)-3-[2-(benzylamino)-2-oxoethyl]-7-ethyl-5-(2-methoxyphenyl)-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— methyl (3aS,6aR)-5-(4-bromophenyl)-4,6-dioxo-1-phenyl-3a,6a-dihydropyrrolo[3,4-c]pyrazole-3-carboxylate —— C19H14BrN3O4
methyl (3aS,6aR)-5-(4-bromophenyl)-4,6-dioxo-1-phenyl-3a,6a-dihydropyrrolo[3,4-c]pyrazole-3-carboxylate
—— methyl (5S)-3-[2-(cyclopropylamino)-2-oxoethyl]-7-ethyl-5-(2-methoxyphenyl)-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C22H25N3O4S
methyl (5S)-3-[2-(cyclopropylamino)-2-oxoethyl]-7-ethyl-5-(2-methoxyphenyl)-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— methyl (5R)-7-ethyl-5-(3-methoxyphenyl)-3-[2-oxo-2-[[(1R)-1-phenylethyl]amino]ethyl]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C27H29N3O4S
methyl (5R)-7-ethyl-5-(3-methoxyphenyl)-3-[2-oxo-2-[[(1R)-1-phenylethyl]amino]ethyl]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— methyl (5S)-3-[2-(benzylamino)-2-oxoethyl]-7-ethyl-5-(3-methoxyphenyl)-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C26H27N3O4S
methyl (5S)-3-[2-(benzylamino)-2-oxoethyl]-7-ethyl-5-(3-methoxyphenyl)-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— methyl (5S)-5-(3-chlorophenyl)-7-ethyl-3-[2-oxo-2-[[(2S)-oxolan-2-yl]methylamino]ethyl]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C23H26ClN3O4S
methyl (5S)-5-(3-chlorophenyl)-7-ethyl-3-[2-oxo-2-[[(2S)-oxolan-2-yl]methylamino]ethyl]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— methyl (5R)-3-[2-[(3-fluorophenyl)methylamino]-2-oxoethyl]-5-(2-methoxyphenyl)-7-methyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C25H24FN3O4S
methyl (5R)-3-[2-[(3-fluorophenyl)methylamino]-2-oxoethyl]-5-(2-methoxyphenyl)-7-methyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— methyl (5S)-7-ethyl-5-(2-fluorophenyl)-3-[2-(4-methoxyanilino)-2-oxoethyl]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C25H24FN3O4S
methyl (5S)-7-ethyl-5-(2-fluorophenyl)-3-[2-(4-methoxyanilino)-2-oxoethyl]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— methyl (5S)-3-[2-(cyclopropylamino)-2-oxoethyl]-7-ethyl-5-(3-methoxyphenyl)-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C22H25N3O4S
methyl (5S)-3-[2-(cyclopropylamino)-2-oxoethyl]-7-ethyl-5-(3-methoxyphenyl)-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— methyl (3aR,6aS)-5-(4-bromophenyl)-4,6-dioxo-1-phenyl-3a,6a-dihydropyrrolo[3,4-c]pyrazole-3-carboxylate —— C19H14BrN3O4
methyl (3aR,6aS)-5-(4-bromophenyl)-4,6-dioxo-1-phenyl-3a,6a-dihydropyrrolo[3,4-c]pyrazole-3-carboxylate
—— methyl (5S)-7-ethyl-5-(3-methoxyphenyl)-3-[2-oxo-2-[[(1S)-1-phenylethyl]amino]ethyl]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C27H29N3O4S
methyl (5S)-7-ethyl-5-(3-methoxyphenyl)-3-[2-oxo-2-[[(1S)-1-phenylethyl]amino]ethyl]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— methyl (5R)-7-ethyl-5-(3-methoxyphenyl)-3-[2-oxo-2-[[(1S)-1-phenylethyl]amino]ethyl]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C27H29N3O4S
methyl (5R)-7-ethyl-5-(3-methoxyphenyl)-3-[2-oxo-2-[[(1S)-1-phenylethyl]amino]ethyl]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— methyl (5R)-7-ethyl-3-[2-[(4-fluorophenyl)methylamino]-2-oxoethyl]-5-(2-methoxyphenyl)-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C26H26FN3O4S
methyl (5R)-7-ethyl-3-[2-[(4-fluorophenyl)methylamino]-2-oxoethyl]-5-(2-methoxyphenyl)-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— methyl (5R)-5-(2-chlorophenyl)-3-[2-(3-methoxyanilino)-2-oxoethyl]-7-methyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C24H22ClN3O4S
methyl (5R)-5-(2-chlorophenyl)-3-[2-(3-methoxyanilino)-2-oxoethyl]-7-methyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— methyl (5S)-5-(4-methoxyphenyl)-7-methyl-3-[2-oxo-2-(3-phenylpropylamino)ethyl]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C27H29N3O4S
methyl (5S)-5-(4-methoxyphenyl)-7-methyl-3-[2-oxo-2-(3-phenylpropylamino)ethyl]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— methyl (5R)-5-(2,4-dimethylphenyl)-7-ethyl-3-[2-oxo-2-[[(2R)-oxolan-2-yl]methylamino]ethyl]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C25H31N3O4S
methyl (5R)-5-(2,4-dimethylphenyl)-7-ethyl-3-[2-oxo-2-[[(2R)-oxolan-2-yl]methylamino]ethyl]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— methyl (5R)-3-[2-[(3-fluorophenyl)methylamino]-2-oxoethyl]-5-(4-methoxyphenyl)-7-methyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C25H24FN3O4S
methyl (5R)-3-[2-[(3-fluorophenyl)methylamino]-2-oxoethyl]-5-(4-methoxyphenyl)-7-methyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— methyl (5S)-3-[2-[[(1R,2S,4R)-2-bicyclo[2.2.1]heptanyl]amino]-2-oxoethyl]-5-(4-methoxyphenyl)-7-methyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C25H29N3O4S
methyl (5S)-3-[2-[[(1R,2S,4R)-2-bicyclo[2.2.1]heptanyl]amino]-2-oxoethyl]-5-(4-methoxyphenyl)-7-methyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— methyl (5R)-7-ethyl-5-(3-fluorophenyl)-3-[2-(3-methoxyanilino)-2-oxoethyl]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C25H24FN3O4S
methyl (5R)-7-ethyl-5-(3-fluorophenyl)-3-[2-(3-methoxyanilino)-2-oxoethyl]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— methyl (5R)-5-(2-chlorophenyl)-3-[2-(4-methoxyanilino)-2-oxoethyl]-7-methyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C24H22ClN3O4S
methyl (5R)-5-(2-chlorophenyl)-3-[2-(4-methoxyanilino)-2-oxoethyl]-7-methyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— methyl (5R)-5-(4-methoxyphenyl)-7-methyl-3-[2-oxo-2-[[3-(trifluoromethyl)phenyl]methylamino]ethyl]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C26H24F3N3O4S
methyl (5R)-5-(4-methoxyphenyl)-7-methyl-3-[2-oxo-2-[[3-(trifluoromethyl)phenyl]methylamino]ethyl]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— methyl (5S)-3-[2-(3-methoxyanilino)-2-oxoethyl]-7-methyl-5-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C24H23N3O4S
methyl (5S)-3-[2-(3-methoxyanilino)-2-oxoethyl]-7-methyl-5-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— methyl (5R)-5-(2,4-dimethylphenyl)-7-ethyl-3-[2-oxo-2-[[(2S)-oxolan-2-yl]methylamino]ethyl]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C25H31N3O4S
methyl (5R)-5-(2,4-dimethylphenyl)-7-ethyl-3-[2-oxo-2-[[(2S)-oxolan-2-yl]methylamino]ethyl]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— methyl (5S)-3-[2-(3,4-dimethylanilino)-2-oxoethyl]-7-ethyl-5-(3-methoxyphenyl)-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C27H29N3O4S
methyl (5S)-3-[2-(3,4-dimethylanilino)-2-oxoethyl]-7-ethyl-5-(3-methoxyphenyl)-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— methyl (5R)-3-[2-(cyclohexylamino)-2-oxoethyl]-5-(4-methoxyphenyl)-7-methyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C24H29N3O4S
methyl (5R)-3-[2-(cyclohexylamino)-2-oxoethyl]-5-(4-methoxyphenyl)-7-methyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— methyl (5S)-7-methyl-3-[2-oxo-2-(propan-2-ylamino)ethyl]-5-(3-phenoxyphenyl)-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C26H27N3O4S
methyl (5S)-7-methyl-3-[2-oxo-2-(propan-2-ylamino)ethyl]-5-(3-phenoxyphenyl)-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— methyl (5S)-5-(2-chlorophenyl)-3-[2-(4-methoxyanilino)-2-oxoethyl]-7-methyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C24H22ClN3O4S
methyl (5S)-5-(2-chlorophenyl)-3-[2-(4-methoxyanilino)-2-oxoethyl]-7-methyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— methyl (5S)-3-[2-(cyclohexylamino)-2-oxoethyl]-7-ethyl-5-(3-methoxyphenyl)-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C25H31N3O4S
methyl (5S)-3-[2-(cyclohexylamino)-2-oxoethyl]-7-ethyl-5-(3-methoxyphenyl)-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— methyl (5R)-3-[2-[[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]amino]-2-oxoethyl]-5-(4-methoxyphenyl)-7-methyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C25H29N3O4S
methyl (5R)-3-[2-[[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]amino]-2-oxoethyl]-5-(4-methoxyphenyl)-7-methyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— methyl (5S)-3-[2-[(3-fluorophenyl)methylamino]-2-oxoethyl]-5-(4-methoxyphenyl)-7-methyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C25H24FN3O4S
methyl (5S)-3-[2-[(3-fluorophenyl)methylamino]-2-oxoethyl]-5-(4-methoxyphenyl)-7-methyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— methyl (5R)-5-(4-methoxyphenyl)-7-methyl-3-[2-oxo-2-(3-phenylpropylamino)ethyl]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C27H29N3O4S
methyl (5R)-5-(4-methoxyphenyl)-7-methyl-3-[2-oxo-2-(3-phenylpropylamino)ethyl]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— methyl (5S)-3-[2-(4-methoxyanilino)-2-oxoethyl]-7-methyl-5-(4-methylphenyl)-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C25H25N3O4S
methyl (5S)-3-[2-(4-methoxyanilino)-2-oxoethyl]-7-methyl-5-(4-methylphenyl)-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— methyl (5R)-3-[2-(2-fluoroanilino)-2-oxoethyl]-5-(4-methoxyphenyl)-7-methyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C24H22FN3O4S
methyl (5R)-3-[2-(2-fluoroanilino)-2-oxoethyl]-5-(4-methoxyphenyl)-7-methyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— methyl (5S)-5-(2,4-dimethylphenyl)-7-ethyl-3-[2-oxo-2-[[(2S)-oxolan-2-yl]methylamino]ethyl]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C25H31N3O4S
methyl (5S)-5-(2,4-dimethylphenyl)-7-ethyl-3-[2-oxo-2-[[(2S)-oxolan-2-yl]methylamino]ethyl]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— methyl (5R)-3-[2-(cyclopropylmethylamino)-2-oxoethyl]-7-ethyl-5-(3-methoxyphenyl)-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C23H27N3O4S
methyl (5R)-3-[2-(cyclopropylmethylamino)-2-oxoethyl]-7-ethyl-5-(3-methoxyphenyl)-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— methyl (5R)-3-[2-(4-methoxyanilino)-2-oxoethyl]-7-methyl-5-(4-methylphenyl)-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C25H25N3O4S
methyl (5R)-3-[2-(4-methoxyanilino)-2-oxoethyl]-7-methyl-5-(4-methylphenyl)-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— methyl (5S)-3-[2-(2-fluoroanilino)-2-oxoethyl]-5-(4-methoxyphenyl)-7-methyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C24H22FN3O4S
methyl (5S)-3-[2-(2-fluoroanilino)-2-oxoethyl]-5-(4-methoxyphenyl)-7-methyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— methyl (1S,2R,5S)-3-(3-methoxythiophene-2-carbonyl)-3-azabicyclo[3.1.0]hexane-2-carboxylate —— C13H15NO4S
methyl (1S,2R,5S)-3-(3-methoxythiophene-2-carbonyl)-3-azabicyclo[3.1.0]hexane-2-carboxylate
—— methyl (5S)-5-(2,4-dimethylphenyl)-7-ethyl-3-[2-oxo-2-[[(2R)-oxolan-2-yl]methylamino]ethyl]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C25H31N3O4S
methyl (5S)-5-(2,4-dimethylphenyl)-7-ethyl-3-[2-oxo-2-[[(2R)-oxolan-2-yl]methylamino]ethyl]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— methyl (5S)-3-[2-(cyclopropylmethylamino)-2-oxoethyl]-7-ethyl-5-(3-methoxyphenyl)-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C23H27N3O4S
methyl (5S)-3-[2-(cyclopropylmethylamino)-2-oxoethyl]-7-ethyl-5-(3-methoxyphenyl)-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— methyl (5S)-7-ethyl-5-(3-fluorophenyl)-3-[2-(3-methoxyanilino)-2-oxoethyl]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C25H24FN3O4S
methyl (5S)-7-ethyl-5-(3-fluorophenyl)-3-[2-(3-methoxyanilino)-2-oxoethyl]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— methyl (5R)-7-methyl-3-[2-oxo-2-(propan-2-ylamino)ethyl]-5-(3-phenoxyphenyl)-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C26H27N3O4S
methyl (5R)-7-methyl-3-[2-oxo-2-(propan-2-ylamino)ethyl]-5-(3-phenoxyphenyl)-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— methyl (5R)-3-[2-(cyclohexylamino)-2-oxoethyl]-7-ethyl-5-(3-methoxyphenyl)-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C25H31N3O4S
methyl (5R)-3-[2-(cyclohexylamino)-2-oxoethyl]-7-ethyl-5-(3-methoxyphenyl)-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— methyl (5S)-3-[2-(cyclohexylamino)-2-oxoethyl]-5-(4-methoxyphenyl)-7-methyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C24H29N3O4S
methyl (5S)-3-[2-(cyclohexylamino)-2-oxoethyl]-5-(4-methoxyphenyl)-7-methyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— methyl (5R)-3-[2-(3,4-dimethylanilino)-2-oxoethyl]-7-ethyl-5-(3-methoxyphenyl)-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C27H29N3O4S
methyl (5R)-3-[2-(3,4-dimethylanilino)-2-oxoethyl]-7-ethyl-5-(3-methoxyphenyl)-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— morpholin-4-yl-[(1R,12S)-12,15,15-trimethyl-3,10-diazatetracyclo[10.2.1.02,11.04,9]pentadeca-2,4,6,8,10-pentaen-1-yl]methanone —— C21H25N3O2
morpholin-4-yl-[(1R,12S)-12,15,15-trimethyl-3,10-diazatetracyclo[10.2.1.02,11.04,9]pentadeca-2,4,6,8,10-pentaen-1-yl]methanone