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—— (E)-3-[4-(2-amino-2-oxoethoxy)-3-methoxyphenyl]-N-[(R)-cyclopentyl-(4-fluorophenyl)methyl]prop-2-enamide —— C24H27FN2O4
(E)-3-[4-(2-amino-2-oxoethoxy)-3-methoxyphenyl]-N-[(R)-cyclopentyl-(4-fluorophenyl)methyl]prop-2-enamide
—— (E)-N-[[4-[[(3R,5S)-3,5-dimethylpiperidin-1-yl]methyl]phenyl]methyl]-3-[4-(dimethylsulfamoyl)phenyl]prop-2-enamide —— C26H35N3O3S
(E)-N-[[4-[[(3R,5S)-3,5-dimethylpiperidin-1-yl]methyl]phenyl]methyl]-3-[4-(dimethylsulfamoyl)phenyl]prop-2-enamide
—— (E)-3-[4-(2-amino-2-oxoethoxy)-3-methoxyphenyl]-N-[(1S)-1-(4-fluorophenyl)-2,2-dimethylpropyl]prop-2-enamide —— C23H27FN2O4
(E)-3-[4-(2-amino-2-oxoethoxy)-3-methoxyphenyl]-N-[(1S)-1-(4-fluorophenyl)-2,2-dimethylpropyl]prop-2-enamide
—— ethyl N-[(2R)-1-[[1-(4-fluorophenyl)cyclopentyl]methylamino]-3-methyl-1-oxobutan-2-yl]carbamate —— C20H29FN2O3
ethyl N-[(2R)-1-[[1-(4-fluorophenyl)cyclopentyl]methylamino]-3-methyl-1-oxobutan-2-yl]carbamate
—— Ethyl 2-[2-[4-(dimethylamino)anilino]-2-oxoethyl]sulfanylacetate —— C14H20N2O3S
Ethyl 2-[2-[4-(dimethylamino)anilino]-2-oxoethyl]sulfanylacetate
—— (E)-N-[(1S)-1-(4-fluorophenyl)-2,2-dimethylpropyl]-3-[4-methoxy-3-(methylsulfamoyl)phenyl]prop-2-enamide —— C22H27FN2O4S
(E)-N-[(1S)-1-(4-fluorophenyl)-2,2-dimethylpropyl]-3-[4-methoxy-3-(methylsulfamoyl)phenyl]prop-2-enamide
—— ethyl 2-[[2-[(3aS,7aS)-1,3-dioxo-3a,4,7,7a-tetrahydroisoindol-2-yl]acetyl]amino]benzoate —— C19H20N2O5
ethyl 2-[[2-[(3aS,7aS)-1,3-dioxo-3a,4,7,7a-tetrahydroisoindol-2-yl]acetyl]amino]benzoate
—— (E)-N-[(R)-cyclopentyl-(4-fluorophenyl)methyl]-3-[4-methoxy-3-(methylsulfamoyl)phenyl]prop-2-enamide —— C23H27FN2O4S
(E)-N-[(R)-cyclopentyl-(4-fluorophenyl)methyl]-3-[4-methoxy-3-(methylsulfamoyl)phenyl]prop-2-enamide
—— ethyl N-[(2S)-3-methyl-1-oxo-1-(quinolin-6-ylamino)butan-2-yl]carbamate —— C17H21N3O3
ethyl N-[(2S)-3-methyl-1-oxo-1-(quinolin-6-ylamino)butan-2-yl]carbamate
—— Ethyl 2-[2-(2,5-diethoxy-4-morpholin-4-ylanilino)-2-oxoethyl]sulfanylacetate —— C20H30N2O6S
Ethyl 2-[2-(2,5-diethoxy-4-morpholin-4-ylanilino)-2-oxoethyl]sulfanylacetate
—— (E)-N-[(1R)-1-(4-fluorophenyl)-2,2-dimethylpropyl]-3-[4-methoxy-3-(methylsulfamoyl)phenyl]prop-2-enamide —— C22H27FN2O4S
(E)-N-[(1R)-1-(4-fluorophenyl)-2,2-dimethylpropyl]-3-[4-methoxy-3-(methylsulfamoyl)phenyl]prop-2-enamide
—— (E)-N-[[4-[[(3R,5S)-3,5-dimethylpiperidin-1-yl]methyl]phenyl]methyl]-3-[4-(ethylsulfamoyl)phenyl]prop-2-enamide —— C26H35N3O3S
(E)-N-[[4-[[(3R,5S)-3,5-dimethylpiperidin-1-yl]methyl]phenyl]methyl]-3-[4-(ethylsulfamoyl)phenyl]prop-2-enamide
—— ethyl 2-[[2-[(3aR,7aS)-1,3-dioxo-3a,4,7,7a-tetrahydroisoindol-2-yl]acetyl]amino]-4-ethyl-5-methylthiophene-3-carboxylate —— C20H24N2O5S
ethyl 2-[[2-[(3aR,7aS)-1,3-dioxo-3a,4,7,7a-tetrahydroisoindol-2-yl]acetyl]amino]-4-ethyl-5-methylthiophene-3-carboxylate
—— (E)-N-[[4-[[(3R,5R)-3,5-dimethylpiperidin-1-yl]methyl]phenyl]methyl]-3-(2-methyl-1,3-thiazol-4-yl)prop-2-enamide —— C22H29N3OS
(E)-N-[[4-[[(3R,5R)-3,5-dimethylpiperidin-1-yl]methyl]phenyl]methyl]-3-(2-methyl-1,3-thiazol-4-yl)prop-2-enamide
—— (E)-N-[[4-[[(3R,5R)-3,5-dimethylpiperidin-1-yl]methyl]phenyl]methyl]-3-[4-(methanesulfonamido)phenyl]prop-2-enamide —— C25H33N3O3S
(E)-N-[[4-[[(3R,5R)-3,5-dimethylpiperidin-1-yl]methyl]phenyl]methyl]-3-[4-(methanesulfonamido)phenyl]prop-2-enamide
—— (E)-N-[[4-[[(3S,5S)-3,5-dimethylpiperidin-1-yl]methyl]phenyl]methyl]-3-[4-(methylsulfamoyl)phenyl]prop-2-enamide —— C25H33N3O3S
(E)-N-[[4-[[(3S,5S)-3,5-dimethylpiperidin-1-yl]methyl]phenyl]methyl]-3-[4-(methylsulfamoyl)phenyl]prop-2-enamide
—— (E)-N-[[4-[[(3R,5R)-3,5-dimethylpiperidin-1-yl]methyl]phenyl]methyl]-3-[4-(ethylsulfamoyl)phenyl]prop-2-enamide —— C26H35N3O3S
(E)-N-[[4-[[(3R,5R)-3,5-dimethylpiperidin-1-yl]methyl]phenyl]methyl]-3-[4-(ethylsulfamoyl)phenyl]prop-2-enamide
—— ethyl 2-[(2R)-1-(4-morpholin-4-ylanilino)-1-oxopropan-2-yl]sulfanylacetate —— C17H24N2O4S
ethyl 2-[(2R)-1-(4-morpholin-4-ylanilino)-1-oxopropan-2-yl]sulfanylacetate
—— (E)-N-[[4-[[(3R,5S)-3,5-dimethylpiperidin-1-yl]methyl]phenyl]methyl]-3-(2-methyl-1,3-thiazol-4-yl)prop-2-enamide —— C22H29N3OS
(E)-N-[[4-[[(3R,5S)-3,5-dimethylpiperidin-1-yl]methyl]phenyl]methyl]-3-(2-methyl-1,3-thiazol-4-yl)prop-2-enamide
—— (E)-3-(1,3-benzoxazol-2-yl)-N-[[4-[[(3R,5R)-3,5-dimethylpiperidin-1-yl]methyl]phenyl]methyl]prop-2-enamide —— C25H29N3O2
(E)-3-(1,3-benzoxazol-2-yl)-N-[[4-[[(3R,5R)-3,5-dimethylpiperidin-1-yl]methyl]phenyl]methyl]prop-2-enamide
—— (E)-N-[[4-[[(3R,5R)-3,5-dimethylpiperidin-1-yl]methyl]phenyl]methyl]-3-pyridin-3-ylprop-2-enamide —— C23H29N3O
(E)-N-[[4-[[(3R,5R)-3,5-dimethylpiperidin-1-yl]methyl]phenyl]methyl]-3-pyridin-3-ylprop-2-enamide
—— (E)-3-(1,3-benzoxazol-2-yl)-N-[[4-[[(3S,5R)-3,5-dimethylpiperidin-1-yl]methyl]phenyl]methyl]prop-2-enamide —— C25H29N3O2
(E)-3-(1,3-benzoxazol-2-yl)-N-[[4-[[(3S,5R)-3,5-dimethylpiperidin-1-yl]methyl]phenyl]methyl]prop-2-enamide
—— (E)-N-[[4-[[(3S,5R)-3,5-dimethylpiperidin-1-yl]methyl]phenyl]methyl]-3-[4-(methanesulfonamido)phenyl]prop-2-enamide —— C25H33N3O3S
(E)-N-[[4-[[(3S,5R)-3,5-dimethylpiperidin-1-yl]methyl]phenyl]methyl]-3-[4-(methanesulfonamido)phenyl]prop-2-enamide
—— (E)-N-[[4-[[(3R,5S)-3,5-dimethylpiperidin-1-yl]methyl]phenyl]methyl]-3-pyridin-3-ylprop-2-enamide —— C23H29N3O
(E)-N-[[4-[[(3R,5S)-3,5-dimethylpiperidin-1-yl]methyl]phenyl]methyl]-3-pyridin-3-ylprop-2-enamide
—— ethyl 2-[[2-[(3aS,7aR)-1,3-dioxo-3a,4,7,7a-tetrahydroisoindol-2-yl]acetyl]amino]benzoate —— C19H20N2O5
ethyl 2-[[2-[(3aS,7aR)-1,3-dioxo-3a,4,7,7a-tetrahydroisoindol-2-yl]acetyl]amino]benzoate
—— ethyl 2-[[2-[(3aR,7aR)-1,3-dioxo-3a,4,7,7a-tetrahydroisoindol-2-yl]acetyl]amino]benzoate —— C19H20N2O5
ethyl 2-[[2-[(3aR,7aR)-1,3-dioxo-3a,4,7,7a-tetrahydroisoindol-2-yl]acetyl]amino]benzoate
—— ethyl N-[2-[(3aR,7aR)-1,3-dioxo-3a,4,7,7a-tetrahydroisoindol-2-yl]acetyl]carbamate —— C13H16N2O5
ethyl N-[2-[(3aR,7aR)-1,3-dioxo-3a,4,7,7a-tetrahydroisoindol-2-yl]acetyl]carbamate
—— ethyl 2-[[2-[(3aR,7aS)-1,3-dioxo-3a,4,7,7a-tetrahydroisoindol-2-yl]acetyl]amino]-5-ethyl-4-methylthiophene-3-carboxylate —— C20H24N2O5S
ethyl 2-[[2-[(3aR,7aS)-1,3-dioxo-3a,4,7,7a-tetrahydroisoindol-2-yl]acetyl]amino]-5-ethyl-4-methylthiophene-3-carboxylate
—— ethyl 2-[[2-[(3aR,7aS)-1,3-dioxo-3a,4,7,7a-tetrahydroisoindol-2-yl]acetyl]amino]-5-ethylthiophene-3-carboxylate —— C19H22N2O5S
ethyl 2-[[2-[(3aR,7aS)-1,3-dioxo-3a,4,7,7a-tetrahydroisoindol-2-yl]acetyl]amino]-5-ethylthiophene-3-carboxylate
—— ethyl N-[2-[(3aS,7aS)-1,3-dioxo-3a,4,7,7a-tetrahydroisoindol-2-yl]acetyl]carbamate —— C13H16N2O5
ethyl N-[2-[(3aS,7aS)-1,3-dioxo-3a,4,7,7a-tetrahydroisoindol-2-yl]acetyl]carbamate
—— ethyl N-[2-[(3aS,7aR)-1,3-dioxo-3a,4,7,7a-tetrahydroisoindol-2-yl]acetyl]carbamate —— C13H16N2O5
ethyl N-[2-[(3aS,7aR)-1,3-dioxo-3a,4,7,7a-tetrahydroisoindol-2-yl]acetyl]carbamate
—— ethyl 2-[[2-[(3aS,7aS)-1,3-dioxo-3a,4,7,7a-tetrahydroisoindol-2-yl]acetyl]amino]-5-ethyl-4-methylthiophene-3-carboxylate —— C20H24N2O5S
ethyl 2-[[2-[(3aS,7aS)-1,3-dioxo-3a,4,7,7a-tetrahydroisoindol-2-yl]acetyl]amino]-5-ethyl-4-methylthiophene-3-carboxylate
—— ethyl 2-[[2-[(3aR,7aR)-1,3-dioxo-3a,4,7,7a-tetrahydroisoindol-2-yl]acetyl]amino]-5-ethylthiophene-3-carboxylate —— C19H22N2O5S
ethyl 2-[[2-[(3aR,7aR)-1,3-dioxo-3a,4,7,7a-tetrahydroisoindol-2-yl]acetyl]amino]-5-ethylthiophene-3-carboxylate
—— ethyl 2-[[2-[(3aR,7aS)-1,3-dioxo-3a,4,7,7a-tetrahydroisoindol-2-yl]acetyl]amino]-4,5-dimethylthiophene-3-carboxylate —— C19H22N2O5S
ethyl 2-[[2-[(3aR,7aS)-1,3-dioxo-3a,4,7,7a-tetrahydroisoindol-2-yl]acetyl]amino]-4,5-dimethylthiophene-3-carboxylate
—— ethyl 2-[[2-[(3aS,7aS)-1,3-dioxo-3a,4,7,7a-tetrahydroisoindol-2-yl]acetyl]amino]-4-ethyl-5-methylthiophene-3-carboxylate —— C20H24N2O5S
ethyl 2-[[2-[(3aS,7aS)-1,3-dioxo-3a,4,7,7a-tetrahydroisoindol-2-yl]acetyl]amino]-4-ethyl-5-methylthiophene-3-carboxylate
—— (E)-N-[[4-[[(3S)-3-methylpiperidin-1-yl]methyl]phenyl]methyl]-3-pyridin-3-ylprop-2-enamide —— C22H27N3O
(E)-N-[[4-[[(3S)-3-methylpiperidin-1-yl]methyl]phenyl]methyl]-3-pyridin-3-ylprop-2-enamide
—— ethyl 2-[[2-[(3aR,7aR)-1,3-dioxo-3a,4,7,7a-tetrahydroisoindol-2-yl]acetyl]amino]-5,6-dihydro-4H-cyclopenta[b]thiophene-3-carboxylate —— C20H22N2O5S
ethyl 2-[[2-[(3aR,7aR)-1,3-dioxo-3a,4,7,7a-tetrahydroisoindol-2-yl]acetyl]amino]-5,6-dihydro-4H-cyclopenta[b]thiophene-3-carboxylate
—— (E)-N-(3-ethyl-4-methoxy-1,3-benzothiazol-2-ylidene)-3-(5-nitrothiophen-2-yl)prop-2-enamide —— C17H15N3O4S2
(E)-N-(3-ethyl-4-methoxy-1,3-benzothiazol-2-ylidene)-3-(5-nitrothiophen-2-yl)prop-2-enamide
—— ethyl 2-[[2-[(3aS,7aR)-1,3-dioxo-3a,4,7,7a-tetrahydroisoindol-2-yl]acetyl]amino]-5,6-dihydro-4H-cyclopenta[b]thiophene-3-carboxylate —— C20H22N2O5S
ethyl 2-[[2-[(3aS,7aR)-1,3-dioxo-3a,4,7,7a-tetrahydroisoindol-2-yl]acetyl]amino]-5,6-dihydro-4H-cyclopenta[b]thiophene-3-carboxylate
—— (E)-N-[(1R)-1-[4-(carbamoylamino)phenyl]ethyl]-3-(4-nitrophenyl)prop-2-enamide —— C18H18N4O4
(E)-N-[(1R)-1-[4-(carbamoylamino)phenyl]ethyl]-3-(4-nitrophenyl)prop-2-enamide
—— (E)-N-[(1R)-1-[4-(carbamoylamino)phenyl]ethyl]-3-(1,3-diphenylpyrazol-4-yl)prop-2-enamide —— C27H25N5O2
(E)-N-[(1R)-1-[4-(carbamoylamino)phenyl]ethyl]-3-(1,3-diphenylpyrazol-4-yl)prop-2-enamide
—— ethyl 2-[[2-[(3aR,7aR)-1,3-dioxo-3a,4,7,7a-tetrahydroisoindol-2-yl]acetyl]amino]-4-ethyl-5-methylthiophene-3-carboxylate —— C20H24N2O5S
ethyl 2-[[2-[(3aR,7aR)-1,3-dioxo-3a,4,7,7a-tetrahydroisoindol-2-yl]acetyl]amino]-4-ethyl-5-methylthiophene-3-carboxylate
—— ethyl 2-[[2-[(3aS,7aS)-1,3-dioxo-3a,4,7,7a-tetrahydroisoindol-2-yl]acetyl]amino]-4,5-dimethylthiophene-3-carboxylate —— C19H22N2O5S
ethyl 2-[[2-[(3aS,7aS)-1,3-dioxo-3a,4,7,7a-tetrahydroisoindol-2-yl]acetyl]amino]-4,5-dimethylthiophene-3-carboxylate
—— (E)-N-[(2R)-2-(4-phenylpiperazin-1-yl)propyl]-3-[4-(pyridin-2-ylmethoxy)phenyl]prop-2-enamide —— C28H32N4O2
(E)-N-[(2R)-2-(4-phenylpiperazin-1-yl)propyl]-3-[4-(pyridin-2-ylmethoxy)phenyl]prop-2-enamide
—— (E)-N-[(1S)-1-[4-(carbamoylamino)phenyl]ethyl]-3-(1-phenyl-3-pyridin-3-ylpyrazol-4-yl)prop-2-enamide —— C26H24N6O2
(E)-N-[(1S)-1-[4-(carbamoylamino)phenyl]ethyl]-3-(1-phenyl-3-pyridin-3-ylpyrazol-4-yl)prop-2-enamide
—— (E)-N-[(2R)-2-(4-phenylpiperazin-1-yl)propyl]-3-[4-(pyridin-3-ylmethoxy)phenyl]prop-2-enamide —— C28H32N4O2
(E)-N-[(2R)-2-(4-phenylpiperazin-1-yl)propyl]-3-[4-(pyridin-3-ylmethoxy)phenyl]prop-2-enamide
—— ethyl 4-[2-[(3aR,7aS)-1,3-dioxo-3a,4,7,7a-tetrahydroisoindol-2-yl]acetyl]-2,5-dimethyl-1H-pyrrole-3-carboxylate —— C19H22N2O5
ethyl 4-[2-[(3aR,7aS)-1,3-dioxo-3a,4,7,7a-tetrahydroisoindol-2-yl]acetyl]-2,5-dimethyl-1H-pyrrole-3-carboxylate
—— ethyl 4-[2-[(3aS,7aS)-1,3-dioxo-3a,4,7,7a-tetrahydroisoindol-2-yl]acetyl]-2,5-dimethyl-1H-pyrrole-3-carboxylate —— C19H22N2O5
ethyl 4-[2-[(3aS,7aS)-1,3-dioxo-3a,4,7,7a-tetrahydroisoindol-2-yl]acetyl]-2,5-dimethyl-1H-pyrrole-3-carboxylate
—— ethyl 4-[2-[(3aR,7aR)-1,3-dioxo-3a,4,7,7a-tetrahydroisoindol-2-yl]acetyl]-2,5-dimethyl-1H-pyrrole-3-carboxylate —— C19H22N2O5
ethyl 4-[2-[(3aR,7aR)-1,3-dioxo-3a,4,7,7a-tetrahydroisoindol-2-yl]acetyl]-2,5-dimethyl-1H-pyrrole-3-carboxylate
—— (E)-N-[(1R)-1-[4-(carbamoylamino)phenyl]ethyl]-3-(2-methoxyphenyl)prop-2-enamide —— C19H21N3O3
(E)-N-[(1R)-1-[4-(carbamoylamino)phenyl]ethyl]-3-(2-methoxyphenyl)prop-2-enamide