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—— ethyl (3R)-3-[[3-(difluoromethylsulfanyl)phenyl]carbamoyl]piperidine-1-carboxylate —— C16H20F2N2O3S
ethyl (3R)-3-[[3-(difluoromethylsulfanyl)phenyl]carbamoyl]piperidine-1-carboxylate
—— (E)-N-[[(3R)-2,3-dihydro-1,4-benzodioxin-3-yl]methyl]-3-(2-methoxyphenyl)prop-2-enamide —— C19H19NO4
(E)-N-[[(3R)-2,3-dihydro-1,4-benzodioxin-3-yl]methyl]-3-(2-methoxyphenyl)prop-2-enamide
—— Ethyl 5-ethyl-4-methyl-2-[[2-(2-methyl-4-oxoquinazolin-3-yl)acetyl]amino]thiophene-3-carboxylate —— C21H23N3O4S
Ethyl 5-ethyl-4-methyl-2-[[2-(2-methyl-4-oxoquinazolin-3-yl)acetyl]amino]thiophene-3-carboxylate
—— ethyl (3S)-3-[[3-(difluoromethylsulfanyl)phenyl]carbamoyl]piperidine-1-carboxylate —— C16H20F2N2O3S
ethyl (3S)-3-[[3-(difluoromethylsulfanyl)phenyl]carbamoyl]piperidine-1-carboxylate
—— ethyl (2Z,5S)-2-[[3-(4-chlorophenyl)-1-phenylpyrazol-4-yl]methylidene]-5-(4-methoxyphenyl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C33H27ClN4O4S
ethyl (2Z,5S)-2-[[3-(4-chlorophenyl)-1-phenylpyrazol-4-yl]methylidene]-5-(4-methoxyphenyl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— (E)-2-(4-acetyl-3,5-dimethyl-1H-pyrrole-2-carbonyl)-3-(2,3-dihydro-1,4-benzodioxin-6-yl)prop-2-enenitrile —— C20H18N2O4
(E)-2-(4-acetyl-3,5-dimethyl-1H-pyrrole-2-carbonyl)-3-(2,3-dihydro-1,4-benzodioxin-6-yl)prop-2-enenitrile
—— [(E)-3-phenylprop-2-enyl] 2-(4-oxoquinazolin-3-yl)acetate —— C19H16N2O3
[(E)-3-phenylprop-2-enyl] 2-(4-oxoquinazolin-3-yl)acetate
—— (E)-N-[6-amino-1-(2-methylpropyl)-2,4-dioxopyrimidin-5-yl]-N-(2-methoxyethyl)-3-phenylprop-2-enamide —— C20H26N4O4
(E)-N-[6-amino-1-(2-methylpropyl)-2,4-dioxopyrimidin-5-yl]-N-(2-methoxyethyl)-3-phenylprop-2-enamide
—— ethyl (3S)-3-[(2-methylquinolin-8-yl)carbamoyl]piperidine-1-carboxylate —— C19H23N3O3
ethyl (3S)-3-[(2-methylquinolin-8-yl)carbamoyl]piperidine-1-carboxylate
—— (E)-N-[[(3S)-2,3-dihydro-1,4-benzodioxin-3-yl]methyl]-3-(2,5-dimethoxyphenyl)prop-2-enamide —— C20H21NO5
(E)-N-[[(3S)-2,3-dihydro-1,4-benzodioxin-3-yl]methyl]-3-(2,5-dimethoxyphenyl)prop-2-enamide
—— ethyl (4S)-4-ethyl-2-oxo-6-[[2-(4-oxoquinazolin-3-yl)acetyl]oxymethyl]-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C20H22N4O6
ethyl (4S)-4-ethyl-2-oxo-6-[[2-(4-oxoquinazolin-3-yl)acetyl]oxymethyl]-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— ethyl (4R)-4-ethyl-2-oxo-6-[[2-(4-oxoquinazolin-3-yl)acetyl]oxymethyl]-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C20H22N4O6
ethyl (4R)-4-ethyl-2-oxo-6-[[2-(4-oxoquinazolin-3-yl)acetyl]oxymethyl]-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— (E)-N-[[(3S)-2,3-dihydro-1,4-benzodioxin-3-yl]methyl]-3-(2-methoxyphenyl)prop-2-enamide —— C19H19NO4
(E)-N-[[(3S)-2,3-dihydro-1,4-benzodioxin-3-yl]methyl]-3-(2-methoxyphenyl)prop-2-enamide
—— ethyl (2S,6S,8R,12S)-1,14-dimethyl-3,5,9,11-tetraoxo-4,10-bis(4-propan-2-ylphenyl)-4,10-diazatetracyclo[5.5.2.02,6.08,12]tetradec-13-ene-13-carboxylate —— C35H38N2O6
ethyl (2S,6S,8R,12S)-1,14-dimethyl-3,5,9,11-tetraoxo-4,10-bis(4-propan-2-ylphenyl)-4,10-diazatetracyclo[5.5.2.02,6.08,12]tetradec-13-ene-13-carboxylate
—— ethyl (2R,6R,8R,12S)-1,14-dimethyl-3,5,9,11-tetraoxo-4,10-bis(4-propan-2-ylphenyl)-4,10-diazatetracyclo[5.5.2.02,6.08,12]tetradec-13-ene-13-carboxylate —— C35H38N2O6
ethyl (2R,6R,8R,12S)-1,14-dimethyl-3,5,9,11-tetraoxo-4,10-bis(4-propan-2-ylphenyl)-4,10-diazatetracyclo[5.5.2.02,6.08,12]tetradec-13-ene-13-carboxylate
—— ethyl (3S)-3-[[5-methyl-2-[5-(trifluoromethyl)pyridin-2-yl]pyrazol-3-yl]carbamoyl]piperidine-1-carboxylate —— C19H22F3N5O3
ethyl (3S)-3-[[5-methyl-2-[5-(trifluoromethyl)pyridin-2-yl]pyrazol-3-yl]carbamoyl]piperidine-1-carboxylate
—— Ethyl 2-[(5-benzyl-1,3,4-oxadiazol-2-yl)sulfanylmethyl]-4-methylquinoline-3-carboxylate —— C23H21N3O3S
Ethyl 2-[(5-benzyl-1,3,4-oxadiazol-2-yl)sulfanylmethyl]-4-methylquinoline-3-carboxylate
—— ethyl (3R)-3-[(2-methylquinolin-8-yl)carbamoyl]piperidine-1-carboxylate —— C19H23N3O3
ethyl (3R)-3-[(2-methylquinolin-8-yl)carbamoyl]piperidine-1-carboxylate
—— (E)-3-(6-chloro-3,4-dihydro-2H-1,5-benzodioxepin-8-yl)-N-phenylprop-2-enamide —— C18H16ClNO3
(E)-3-(6-chloro-3,4-dihydro-2H-1,5-benzodioxepin-8-yl)-N-phenylprop-2-enamide
—— ethyl 2-[2-[[2-[(1R,5R)-3,3,5-trimethylcyclohexyl]acetyl]amino]-1,3-thiazol-4-yl]acetate —— C18H28N2O3S
ethyl 2-[2-[[2-[(1R,5R)-3,3,5-trimethylcyclohexyl]acetyl]amino]-1,3-thiazol-4-yl]acetate
—— (E)-N-[(2R)-2-(4-chlorophenyl)-2-morpholin-4-ylethyl]-3-(2-methoxyphenyl)but-2-enamide —— C23H27ClN2O3
(E)-N-[(2R)-2-(4-chlorophenyl)-2-morpholin-4-ylethyl]-3-(2-methoxyphenyl)but-2-enamide
—— ethyl N-[2-[(5-benzyl-1,3,4-oxadiazol-2-yl)sulfanyl]acetyl]carbamate —— C14H15N3O4S
ethyl N-[2-[(5-benzyl-1,3,4-oxadiazol-2-yl)sulfanyl]acetyl]carbamate
—— ethyl 2-[2-[[2-[(1S,5R)-3,3,5-trimethylcyclohexyl]acetyl]amino]-1,3-thiazol-4-yl]acetate —— C18H28N2O3S
ethyl 2-[2-[[2-[(1S,5R)-3,3,5-trimethylcyclohexyl]acetyl]amino]-1,3-thiazol-4-yl]acetate
—— ethyl (4R)-6-[(5-benzyl-1,3,4-oxadiazol-2-yl)sulfanylmethyl]-4-ethyl-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C19H22N4O4S
ethyl (4R)-6-[(5-benzyl-1,3,4-oxadiazol-2-yl)sulfanylmethyl]-4-ethyl-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— (E)-N-[(2S)-2-(4-chlorophenyl)-2-morpholin-4-ylethyl]-3-(2-methoxyphenyl)but-2-enamide —— C23H27ClN2O3
(E)-N-[(2S)-2-(4-chlorophenyl)-2-morpholin-4-ylethyl]-3-(2-methoxyphenyl)but-2-enamide
—— ethyl 2-[2-[[2-[(1S,5S)-3,3,5-trimethylcyclohexyl]acetyl]amino]-1,3-thiazol-4-yl]acetate —— C18H28N2O3S
ethyl 2-[2-[[2-[(1S,5S)-3,3,5-trimethylcyclohexyl]acetyl]amino]-1,3-thiazol-4-yl]acetate
—— ethyl 2-[2-[[(2S)-2-benzylsulfanyl-3-methylbutanoyl]amino]-1,3-thiazol-4-yl]acetate —— C19H24N2O3S2
ethyl 2-[2-[[(2S)-2-benzylsulfanyl-3-methylbutanoyl]amino]-1,3-thiazol-4-yl]acetate
—— (E)-N-[3-chloro-4-[[(2R)-2-(3,5-dimethylpyrazol-1-yl)propanoyl]amino]phenyl]-3-(2-methoxyphenyl)but-2-enamide —— C25H27ClN4O3
(E)-N-[3-chloro-4-[[(2R)-2-(3,5-dimethylpyrazol-1-yl)propanoyl]amino]phenyl]-3-(2-methoxyphenyl)but-2-enamide
—— ethyl (3S)-3-[[2-[4-(pyrazol-1-ylmethyl)phenyl]phenyl]methylcarbamoyl]piperidine-1-carboxylate —— C26H30N4O3
ethyl (3S)-3-[[2-[4-(pyrazol-1-ylmethyl)phenyl]phenyl]methylcarbamoyl]piperidine-1-carboxylate
—— Ethyl 3-[(5-benzyl-1,3,4-oxadiazol-2-yl)sulfanylmethyl]-1-benzofuran-2-carboxylate —— C21H18N2O4S
Ethyl 3-[(5-benzyl-1,3,4-oxadiazol-2-yl)sulfanylmethyl]-1-benzofuran-2-carboxylate
—— ethyl 6-[(3R)-3-pyrrolidin-1-ylpyrrolidin-1-yl]pyridine-3-carboxylate —— C16H23N3O2
ethyl 6-[(3R)-3-pyrrolidin-1-ylpyrrolidin-1-yl]pyridine-3-carboxylate
—— (E)-N-[3-chloro-4-[[(2S)-2-(3,5-dimethylpyrazol-1-yl)propanoyl]amino]phenyl]-3-(2-methoxyphenyl)but-2-enamide —— C25H27ClN4O3
(E)-N-[3-chloro-4-[[(2S)-2-(3,5-dimethylpyrazol-1-yl)propanoyl]amino]phenyl]-3-(2-methoxyphenyl)but-2-enamide
—— ethyl 4-[(3R)-3-pyrrolidin-1-ylpyrrolidin-1-yl]quinoline-3-carboxylate —— C20H25N3O2
ethyl 4-[(3R)-3-pyrrolidin-1-ylpyrrolidin-1-yl]quinoline-3-carboxylate
—— ethyl 6-[(3S)-3-pyrrolidin-1-ylpyrrolidin-1-yl]pyridine-3-carboxylate —— C16H23N3O2
ethyl 6-[(3S)-3-pyrrolidin-1-ylpyrrolidin-1-yl]pyridine-3-carboxylate
—— ethyl 5-[[(2S)-1-(6,7-dihydro-4H-thieno[3,2-c]pyridin-5-yl)-1-oxopentan-2-yl]carbamoyl]-2,4-dimethyl-1H-pyrrole-3-carboxylate —— C22H29N3O4S
ethyl 5-[[(2S)-1-(6,7-dihydro-4H-thieno[3,2-c]pyridin-5-yl)-1-oxopentan-2-yl]carbamoyl]-2,4-dimethyl-1H-pyrrole-3-carboxylate
—— ethyl (2R)-2-benzyl-3-[(6-pyrrolidin-1-ylpyridine-3-carbonyl)amino]propanoate —— C22H27N3O3
ethyl (2R)-2-benzyl-3-[(6-pyrrolidin-1-ylpyridine-3-carbonyl)amino]propanoate
—— ethyl (2S)-2-benzyl-3-[(6-pyrrolidin-1-ylpyridine-3-carbonyl)amino]propanoate —— C22H27N3O3
ethyl (2S)-2-benzyl-3-[(6-pyrrolidin-1-ylpyridine-3-carbonyl)amino]propanoate
—— ethyl 4-[2-[(5-benzyl-1,3,4-oxadiazol-2-yl)sulfanyl]acetyl]-2,5-dimethyl-1H-pyrrole-3-carboxylate —— C20H21N3O4S
ethyl 4-[2-[(5-benzyl-1,3,4-oxadiazol-2-yl)sulfanyl]acetyl]-2,5-dimethyl-1H-pyrrole-3-carboxylate
—— ethyl 4-[(3S)-3-pyrrolidin-1-ylpyrrolidin-1-yl]quinoline-3-carboxylate —— C20H25N3O2
ethyl 4-[(3S)-3-pyrrolidin-1-ylpyrrolidin-1-yl]quinoline-3-carboxylate
—— ethyl 4-[(3,4-dimethoxybenzoyl)amino]-2-ethyl-1H-1,5-benzodiazepine-3-carboxylate —— C23H25N3O5
ethyl 4-[(3,4-dimethoxybenzoyl)amino]-2-ethyl-1H-1,5-benzodiazepine-3-carboxylate
—— ethyl N-[[(2R)-2-(3,5-dichlorophenoxy)propanoyl]amino]carbamate —— C12H14Cl2N2O4
ethyl N-[[(2R)-2-(3,5-dichlorophenoxy)propanoyl]amino]carbamate
—— ethyl (3S)-3-[[2-methyl-2-[3-(trifluoromethyl)phenyl]propyl]carbamoyl]piperidine-1-carboxylate —— C20H27F3N2O3
ethyl (3S)-3-[[2-methyl-2-[3-(trifluoromethyl)phenyl]propyl]carbamoyl]piperidine-1-carboxylate
—— (E)-3-(3-chloro-4,5-dimethoxyphenyl)-N-[(2R)-1-(6,7-dihydro-4H-thieno[3,2-c]pyridin-5-yl)-1-oxopentan-2-yl]prop-2-enamide —— C23H27ClN2O4S
(E)-3-(3-chloro-4,5-dimethoxyphenyl)-N-[(2R)-1-(6,7-dihydro-4H-thieno[3,2-c]pyridin-5-yl)-1-oxopentan-2-yl]prop-2-enamide
—— ethyl N-[[(2S)-2-(3,5-dichlorophenoxy)propanoyl]amino]carbamate —— C12H14Cl2N2O4
ethyl N-[[(2S)-2-(3,5-dichlorophenoxy)propanoyl]amino]carbamate
—— (E)-3-(4-chlorophenyl)-N-[(2R)-1-(6,7-dihydro-4H-thieno[3,2-c]pyridin-5-yl)-1-oxopentan-2-yl]prop-2-enamide —— C21H23ClN2O2S
(E)-3-(4-chlorophenyl)-N-[(2R)-1-(6,7-dihydro-4H-thieno[3,2-c]pyridin-5-yl)-1-oxopentan-2-yl]prop-2-enamide
—— (E)-N-[(2R)-1-(6,7-dihydro-4H-thieno[3,2-c]pyridin-5-yl)-1-oxopentan-2-yl]-3-(2-nitrophenyl)prop-2-enamide —— C21H23N3O4S
(E)-N-[(2R)-1-(6,7-dihydro-4H-thieno[3,2-c]pyridin-5-yl)-1-oxopentan-2-yl]-3-(2-nitrophenyl)prop-2-enamide
—— (E)-3-[4-(difluoromethoxy)-3-methoxyphenyl]-N-[(2S)-1-(6,7-dihydro-4H-thieno[3,2-c]pyridin-5-yl)-1-oxopentan-2-yl]prop-2-enamide —— C23H26F2N2O4S
(E)-3-[4-(difluoromethoxy)-3-methoxyphenyl]-N-[(2S)-1-(6,7-dihydro-4H-thieno[3,2-c]pyridin-5-yl)-1-oxopentan-2-yl]prop-2-enamide
—— ethyl (3R)-3-[[2-methyl-2-[3-(trifluoromethyl)phenyl]propyl]carbamoyl]piperidine-1-carboxylate —— C20H27F3N2O3
ethyl (3R)-3-[[2-methyl-2-[3-(trifluoromethyl)phenyl]propyl]carbamoyl]piperidine-1-carboxylate
—— (E)-N-[(2R)-1-(6,7-dihydro-4H-thieno[3,2-c]pyridin-5-yl)-1-oxopentan-2-yl]-3-(3-fluorophenyl)prop-2-enamide —— C21H23FN2O2S
(E)-N-[(2R)-1-(6,7-dihydro-4H-thieno[3,2-c]pyridin-5-yl)-1-oxopentan-2-yl]-3-(3-fluorophenyl)prop-2-enamide
—— (E)-N-[(2S)-1-(6,7-dihydro-4H-thieno[3,2-c]pyridin-5-yl)-1-oxopentan-2-yl]-3-(3-methoxy-4-propan-2-yloxyphenyl)prop-2-enamide —— C25H32N2O4S
(E)-N-[(2S)-1-(6,7-dihydro-4H-thieno[3,2-c]pyridin-5-yl)-1-oxopentan-2-yl]-3-(3-methoxy-4-propan-2-yloxyphenyl)prop-2-enamide