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—— (E)-3-(1-benzyl-3-thiophen-2-ylpyrazol-4-yl)-1-[(4R)-4-(pyrrolidine-1-carbonyl)-1,3-thiazolidin-3-yl]prop-2-en-1-one —— C25H26N4O2S2
(E)-3-(1-benzyl-3-thiophen-2-ylpyrazol-4-yl)-1-[(4R)-4-(pyrrolidine-1-carbonyl)-1,3-thiazolidin-3-yl]prop-2-en-1-one
—— (E)-3-(5-bromo-2-fluorophenyl)-1-[(4R)-4-(pyrrolidine-1-carbonyl)-1,3-thiazolidin-3-yl]prop-2-en-1-one —— C17H18BrFN2O2S
(E)-3-(5-bromo-2-fluorophenyl)-1-[(4R)-4-(pyrrolidine-1-carbonyl)-1,3-thiazolidin-3-yl]prop-2-en-1-one
—— ethyl N-[[4-[(2-phenylphenoxy)methyl]benzoyl]amino]carbamate —— C23H22N2O4
ethyl N-[[4-[(2-phenylphenoxy)methyl]benzoyl]amino]carbamate
—— (E)-3-(4-fluorophenyl)-1-[(4S)-4-(pyrrolidine-1-carbonyl)-1,3-thiazolidin-3-yl]prop-2-en-1-one —— C17H19FN2O2S
(E)-3-(4-fluorophenyl)-1-[(4S)-4-(pyrrolidine-1-carbonyl)-1,3-thiazolidin-3-yl]prop-2-en-1-one
—— (E)-3-[5-chloro-3-methyl-1-(2-methylpropyl)pyrazol-4-yl]-1-[(4S)-4-(pyrrolidine-1-carbonyl)-1,3-thiazolidin-3-yl]prop-2-en-1-one —— C19H27ClN4O2S
(E)-3-[5-chloro-3-methyl-1-(2-methylpropyl)pyrazol-4-yl]-1-[(4S)-4-(pyrrolidine-1-carbonyl)-1,3-thiazolidin-3-yl]prop-2-en-1-one
—— (E)-3-(1-phenyl-3-thiophen-2-ylpyrazol-4-yl)-1-[(4S)-4-(pyrrolidine-1-carbonyl)-1,3-thiazolidin-3-yl]prop-2-en-1-one —— C24H24N4O2S2
(E)-3-(1-phenyl-3-thiophen-2-ylpyrazol-4-yl)-1-[(4S)-4-(pyrrolidine-1-carbonyl)-1,3-thiazolidin-3-yl]prop-2-en-1-one
—— (E)-3-(1,3-benzothiazol-2-yl)-1-[(4S)-4-(pyrrolidine-1-carbonyl)-1,3-thiazolidin-3-yl]prop-2-en-1-one —— C18H19N3O2S2
(E)-3-(1,3-benzothiazol-2-yl)-1-[(4S)-4-(pyrrolidine-1-carbonyl)-1,3-thiazolidin-3-yl]prop-2-en-1-one
—— (E)-3-(2-nitrophenyl)-1-[(4R)-4-(pyrrolidine-1-carbonyl)-1,3-thiazolidin-3-yl]prop-2-en-1-one —— C17H19N3O4S
(E)-3-(2-nitrophenyl)-1-[(4R)-4-(pyrrolidine-1-carbonyl)-1,3-thiazolidin-3-yl]prop-2-en-1-one
—— (E)-3-(1-phenyl-3-thiophen-2-ylpyrazol-4-yl)-1-[(4R)-4-(pyrrolidine-1-carbonyl)-1,3-thiazolidin-3-yl]prop-2-en-1-one —— C24H24N4O2S2
(E)-3-(1-phenyl-3-thiophen-2-ylpyrazol-4-yl)-1-[(4R)-4-(pyrrolidine-1-carbonyl)-1,3-thiazolidin-3-yl]prop-2-en-1-one
—— (E)-3-(3,4-dichlorophenyl)-1-[(4R)-4-(pyrrolidine-1-carbonyl)-1,3-thiazolidin-3-yl]prop-2-en-1-one —— C17H18Cl2N2O2S
(E)-3-(3,4-dichlorophenyl)-1-[(4R)-4-(pyrrolidine-1-carbonyl)-1,3-thiazolidin-3-yl]prop-2-en-1-one
—— (E)-3-[4-chloro-3-(trifluoromethyl)phenyl]-1-[(4R)-4-(pyrrolidine-1-carbonyl)-1,3-thiazolidin-3-yl]prop-2-en-1-one —— C18H18ClF3N2O2S
(E)-3-[4-chloro-3-(trifluoromethyl)phenyl]-1-[(4R)-4-(pyrrolidine-1-carbonyl)-1,3-thiazolidin-3-yl]prop-2-en-1-one
—— ethyl (E)-3-[(5-chloropyridin-2-yl)amino]-2-cyanoprop-2-enoate —— C11H10ClN3O2
ethyl (E)-3-[(5-chloropyridin-2-yl)amino]-2-cyanoprop-2-enoate
—— (E)-2-benzoyl-3-[4-(cyanomethoxy)-3-methoxyphenyl]prop-2-enenitrile —— C19H14N2O3
(E)-2-benzoyl-3-[4-(cyanomethoxy)-3-methoxyphenyl]prop-2-enenitrile
—— (E)-3-(1-benzyl-3-thiophen-2-ylpyrazol-4-yl)-1-[(4S)-4-(pyrrolidine-1-carbonyl)-1,3-thiazolidin-3-yl]prop-2-en-1-one —— C25H26N4O2S2
(E)-3-(1-benzyl-3-thiophen-2-ylpyrazol-4-yl)-1-[(4S)-4-(pyrrolidine-1-carbonyl)-1,3-thiazolidin-3-yl]prop-2-en-1-one
—— (E)-3-(5-bromo-2-fluorophenyl)-1-[(4S)-4-(pyrrolidine-1-carbonyl)-1,3-thiazolidin-3-yl]prop-2-en-1-one —— C17H18BrFN2O2S
(E)-3-(5-bromo-2-fluorophenyl)-1-[(4S)-4-(pyrrolidine-1-carbonyl)-1,3-thiazolidin-3-yl]prop-2-en-1-one
—— (E)-3-(furan-2-yl)-1-[(4R)-4-(pyrrolidine-1-carbonyl)-1,3-thiazolidin-3-yl]prop-2-en-1-one —— C15H18N2O3S
(E)-3-(furan-2-yl)-1-[(4R)-4-(pyrrolidine-1-carbonyl)-1,3-thiazolidin-3-yl]prop-2-en-1-one
—— (E)-3-(1,3-diphenylpyrazol-4-yl)-1-[(4R)-4-(pyrrolidine-1-carbonyl)-1,3-thiazolidin-3-yl]prop-2-en-1-one —— C26H26N4O2S
(E)-3-(1,3-diphenylpyrazol-4-yl)-1-[(4R)-4-(pyrrolidine-1-carbonyl)-1,3-thiazolidin-3-yl]prop-2-en-1-one
—— (E)-3-[5-chloro-3-methyl-1-[(4-methylphenyl)methyl]pyrazol-4-yl]-1-[(4R)-4-(pyrrolidine-1-carbonyl)-1,3-thiazolidin-3-yl]prop-2-en-1-one —— C23H27ClN4O2S
(E)-3-[5-chloro-3-methyl-1-[(4-methylphenyl)methyl]pyrazol-4-yl]-1-[(4R)-4-(pyrrolidine-1-carbonyl)-1,3-thiazolidin-3-yl]prop-2-en-1-one
—— (E)-3-(1,3-benzothiazol-2-yl)-1-[(4R)-4-(pyrrolidine-1-carbonyl)-1,3-thiazolidin-3-yl]prop-2-en-1-one —— C18H19N3O2S2
(E)-3-(1,3-benzothiazol-2-yl)-1-[(4R)-4-(pyrrolidine-1-carbonyl)-1,3-thiazolidin-3-yl]prop-2-en-1-one
—— (E)-N-[4-(4-methoxyphenyl)-1,3-thiazol-2-yl]-3-(2-nitrophenyl)prop-2-enamide —— C19H15N3O4S
(E)-N-[4-(4-methoxyphenyl)-1,3-thiazol-2-yl]-3-(2-nitrophenyl)prop-2-enamide
—— ethyl 4-[[2-(3,4-dihydro-2H-1,5-benzodioxepin-7-ylsulfanyl)acetyl]amino]benzoate —— C20H21NO5S
ethyl 4-[[2-(3,4-dihydro-2H-1,5-benzodioxepin-7-ylsulfanyl)acetyl]amino]benzoate
—— ethyl (4R)-6-(3,4-dihydro-2H-1,5-benzodioxepin-7-ylsulfanylmethyl)-4-ethyl-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C19H24N2O5S
ethyl (4R)-6-(3,4-dihydro-2H-1,5-benzodioxepin-7-ylsulfanylmethyl)-4-ethyl-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— (E)-2-cyano-N-(3-methoxypropyl)-3-[3-(trifluoromethyl)phenyl]prop-2-enamide —— C15H15F3N2O2
(E)-2-cyano-N-(3-methoxypropyl)-3-[3-(trifluoromethyl)phenyl]prop-2-enamide
—— ethyl 2-[[2-(3,4-dihydro-2H-1,5-benzodioxepin-7-ylsulfanyl)acetyl]amino]-4,5-dimethylthiophene-3-carboxylate —— C20H23NO5S2
ethyl 2-[[2-(3,4-dihydro-2H-1,5-benzodioxepin-7-ylsulfanyl)acetyl]amino]-4,5-dimethylthiophene-3-carboxylate
—— ethyl (3R)-3-[[2-(1-adamantylamino)phenyl]carbamoyl]piperidine-1-carboxylate —— C25H35N3O3
ethyl (3R)-3-[[2-(1-adamantylamino)phenyl]carbamoyl]piperidine-1-carboxylate
—— ethyl N-[2-(3,4-dihydro-2H-1,5-benzodioxepin-7-ylsulfanyl)acetyl]carbamate —— C14H17NO5S
ethyl N-[2-(3,4-dihydro-2H-1,5-benzodioxepin-7-ylsulfanyl)acetyl]carbamate
—— ethyl 2-[[2-(3,4-dihydro-2H-1,5-benzodioxepin-7-ylsulfanyl)acetyl]amino]benzoate —— C20H21NO5S
ethyl 2-[[2-(3,4-dihydro-2H-1,5-benzodioxepin-7-ylsulfanyl)acetyl]amino]benzoate
—— ethyl (2S)-2-(4-oxo-6-phenyl-3-prop-2-enylthieno[3,2-d]pyrimidin-2-yl)sulfanylpropanoate —— C20H20N2O3S2
ethyl (2S)-2-(4-oxo-6-phenyl-3-prop-2-enylthieno[3,2-d]pyrimidin-2-yl)sulfanylpropanoate
—— ethyl (3S)-3-[2-cyanoethyl(pyridin-3-ylmethyl)carbamoyl]piperidine-1-carboxylate —— C18H24N4O3
ethyl (3S)-3-[2-cyanoethyl(pyridin-3-ylmethyl)carbamoyl]piperidine-1-carboxylate
—— ethyl 5-[(2R)-2-(3,4-dihydro-2H-1,5-benzodioxepin-7-ylsulfanyl)propanoyl]-2,4-dimethyl-1H-pyrrole-3-carboxylate —— C21H25NO5S
ethyl 5-[(2R)-2-(3,4-dihydro-2H-1,5-benzodioxepin-7-ylsulfanyl)propanoyl]-2,4-dimethyl-1H-pyrrole-3-carboxylate
—— ethyl 5-amino-4-cyano-3-(3,4-dihydro-2H-1,5-benzodioxepin-7-ylsulfanylmethyl)thiophene-2-carboxylate —— C18H18N2O4S2
ethyl 5-amino-4-cyano-3-(3,4-dihydro-2H-1,5-benzodioxepin-7-ylsulfanylmethyl)thiophene-2-carboxylate
—— ethyl 5-[(2S)-2-(3,4-dihydro-2H-1,5-benzodioxepin-7-ylsulfanyl)propanoyl]-2,4-dimethyl-1H-pyrrole-3-carboxylate —— C21H25NO5S
ethyl 5-[(2S)-2-(3,4-dihydro-2H-1,5-benzodioxepin-7-ylsulfanyl)propanoyl]-2,4-dimethyl-1H-pyrrole-3-carboxylate
—— ethyl (3S)-3-[(3,4-dichlorophenyl)methyl-(pyridin-2-ylmethyl)carbamoyl]piperidine-1-carboxylate —— C22H25Cl2N3O3
ethyl (3S)-3-[(3,4-dichlorophenyl)methyl-(pyridin-2-ylmethyl)carbamoyl]piperidine-1-carboxylate
—— ethyl (2S)-2-[[5-(2-chlorophenyl)-4-(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)-1,2,4-triazol-3-yl]sulfanyl]propanoate —— C24H24ClN5O3S
ethyl (2S)-2-[[5-(2-chlorophenyl)-4-(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)-1,2,4-triazol-3-yl]sulfanyl]propanoate
—— ethyl (2S)-2-[[5-[(2R)-2-phenylpropyl]-1,3,4-oxadiazol-2-yl]sulfanyl]propanoate —— C16H20N2O3S
ethyl (2S)-2-[[5-[(2R)-2-phenylpropyl]-1,3,4-oxadiazol-2-yl]sulfanyl]propanoate
—— ethyl (2R)-2-(4-oxo-6-phenyl-3-prop-2-enylthieno[2,3-d]pyrimidin-2-yl)sulfanylpropanoate —— C20H20N2O3S2
ethyl (2R)-2-(4-oxo-6-phenyl-3-prop-2-enylthieno[2,3-d]pyrimidin-2-yl)sulfanylpropanoate
—— ethyl (2R)-2-[[5-oxo-4-(2-propan-2-ylphenyl)-[1,2,4]triazolo[4,3-a]quinazolin-1-yl]sulfanyl]propanoate —— C23H24N4O3S
ethyl (2R)-2-[[5-oxo-4-(2-propan-2-ylphenyl)-[1,2,4]triazolo[4,3-a]quinazolin-1-yl]sulfanyl]propanoate
—— ethyl (2S)-2-[[5-(4-tert-butylphenyl)-4-(furan-2-ylmethyl)-1,2,4-triazol-3-yl]sulfanyl]propanoate —— C22H27N3O3S
ethyl (2S)-2-[[5-(4-tert-butylphenyl)-4-(furan-2-ylmethyl)-1,2,4-triazol-3-yl]sulfanyl]propanoate
—— ethyl (2R)-2-[[5-(2-chlorophenyl)-4-(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)-1,2,4-triazol-3-yl]sulfanyl]propanoate —— C24H24ClN5O3S
ethyl (2R)-2-[[5-(2-chlorophenyl)-4-(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)-1,2,4-triazol-3-yl]sulfanyl]propanoate
—— ethyl (2R)-2-[[5-[(2-chlorophenoxy)methyl]-4-phenyl-1,2,4-triazol-3-yl]sulfanyl]propanoate —— C20H20ClN3O3S
ethyl (2R)-2-[[5-[(2-chlorophenoxy)methyl]-4-phenyl-1,2,4-triazol-3-yl]sulfanyl]propanoate
—— ethyl (2S)-2-(4-oxo-6-phenyl-3-prop-2-enylthieno[2,3-d]pyrimidin-2-yl)sulfanylpropanoate —— C20H20N2O3S2
ethyl (2S)-2-(4-oxo-6-phenyl-3-prop-2-enylthieno[2,3-d]pyrimidin-2-yl)sulfanylpropanoate
—— ethyl (2R)-2-(4-oxo-6-phenyl-3-prop-2-enylthieno[3,2-d]pyrimidin-2-yl)sulfanylpropanoate —— C20H20N2O3S2
ethyl (2R)-2-(4-oxo-6-phenyl-3-prop-2-enylthieno[3,2-d]pyrimidin-2-yl)sulfanylpropanoate
—— ethyl (2S)-2-[[5-[(2-chlorophenoxy)methyl]-4-phenyl-1,2,4-triazol-3-yl]sulfanyl]propanoate —— C20H20ClN3O3S
ethyl (2S)-2-[[5-[(2-chlorophenoxy)methyl]-4-phenyl-1,2,4-triazol-3-yl]sulfanyl]propanoate
—— ethyl (2R)-2-[[5-(4-tert-butylphenyl)-4-(furan-2-ylmethyl)-1,2,4-triazol-3-yl]sulfanyl]propanoate —— C22H27N3O3S
ethyl (2R)-2-[[5-(4-tert-butylphenyl)-4-(furan-2-ylmethyl)-1,2,4-triazol-3-yl]sulfanyl]propanoate
—— ethyl 4-[2-(3,4-dihydro-2H-1,5-benzodioxepin-7-ylsulfanyl)acetyl]-2,5-dimethyl-1H-pyrrole-3-carboxylate —— C20H23NO5S
ethyl 4-[2-(3,4-dihydro-2H-1,5-benzodioxepin-7-ylsulfanyl)acetyl]-2,5-dimethyl-1H-pyrrole-3-carboxylate
—— (E)-3-(3,4-dichlorophenyl)-N-[(1S,2S)-2-methylcyclohexyl]prop-2-enamide —— C16H19Cl2NO
(E)-3-(3,4-dichlorophenyl)-N-[(1S,2S)-2-methylcyclohexyl]prop-2-enamide
—— (E)-3-(3,4-dichlorophenyl)-N-[(1R,2S)-2-methylcyclohexyl]prop-2-enamide —— C16H19Cl2NO
(E)-3-(3,4-dichlorophenyl)-N-[(1R,2S)-2-methylcyclohexyl]prop-2-enamide
—— (E)-3-(3-bromophenyl)-N-[(1R,2S)-2-methylcyclohexyl]prop-2-enamide —— C16H20BrNO
(E)-3-(3-bromophenyl)-N-[(1R,2S)-2-methylcyclohexyl]prop-2-enamide
—— (E)-3-(2,4-dimethoxyphenyl)-N-[(1R,2R)-2-methylcyclohexyl]prop-2-enamide —— C18H25NO3
(E)-3-(2,4-dimethoxyphenyl)-N-[(1R,2R)-2-methylcyclohexyl]prop-2-enamide
—— (E)-3-[4-(furan-2-ylmethylsulfamoyl)phenyl]-N-[(1R,2S)-2-methylcyclohexyl]prop-2-enamide —— C21H26N2O4S
(E)-3-[4-(furan-2-ylmethylsulfamoyl)phenyl]-N-[(1R,2S)-2-methylcyclohexyl]prop-2-enamide