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—— (E)-3-(3-chloro-4-ethoxy-5-methoxyphenyl)-N-[(2R)-1-(6,7-dihydro-4H-thieno[3,2-c]pyridin-5-yl)-1-oxopentan-2-yl]prop-2-enamide —— C24H29ClN2O4S
(E)-3-(3-chloro-4-ethoxy-5-methoxyphenyl)-N-[(2R)-1-(6,7-dihydro-4H-thieno[3,2-c]pyridin-5-yl)-1-oxopentan-2-yl]prop-2-enamide
—— (E)-N-[(2R)-1-(6,7-dihydro-4H-thieno[3,2-c]pyridin-5-yl)-1-oxopentan-2-yl]-3-(furan-2-yl)prop-2-enamide —— C19H22N2O3S
(E)-N-[(2R)-1-(6,7-dihydro-4H-thieno[3,2-c]pyridin-5-yl)-1-oxopentan-2-yl]-3-(furan-2-yl)prop-2-enamide
—— (E)-3-(3-chloro-4-ethoxy-5-methoxyphenyl)-N-[(2S)-1-(6,7-dihydro-4H-thieno[3,2-c]pyridin-5-yl)-1-oxopentan-2-yl]prop-2-enamide —— C24H29ClN2O4S
(E)-3-(3-chloro-4-ethoxy-5-methoxyphenyl)-N-[(2S)-1-(6,7-dihydro-4H-thieno[3,2-c]pyridin-5-yl)-1-oxopentan-2-yl]prop-2-enamide
—— (E)-N-[(2S)-1-(6,7-dihydro-4H-thieno[3,2-c]pyridin-5-yl)-1-oxopentan-2-yl]-3-(4-nitrophenyl)prop-2-enamide —— C21H23N3O4S
(E)-N-[(2S)-1-(6,7-dihydro-4H-thieno[3,2-c]pyridin-5-yl)-1-oxopentan-2-yl]-3-(4-nitrophenyl)prop-2-enamide
—— (E)-3-(4-ethylphenyl)-1-(3-nitrophenyl)prop-2-en-1-one —— C17H15NO3
(E)-3-(4-ethylphenyl)-1-(3-nitrophenyl)prop-2-en-1-one
—— (E)-N-[(2S)-1-(6,7-dihydro-4H-thieno[3,2-c]pyridin-5-yl)-1-oxopentan-2-yl]-3-[4-(trifluoromethyl)phenyl]prop-2-enamide —— C22H23F3N2O2S
(E)-N-[(2S)-1-(6,7-dihydro-4H-thieno[3,2-c]pyridin-5-yl)-1-oxopentan-2-yl]-3-[4-(trifluoromethyl)phenyl]prop-2-enamide
—— (E)-N-[(2R)-1-(6,7-dihydro-4H-thieno[3,2-c]pyridin-5-yl)-1-oxopentan-2-yl]-3-[4-(trifluoromethyl)phenyl]prop-2-enamide —— C22H23F3N2O2S
(E)-N-[(2R)-1-(6,7-dihydro-4H-thieno[3,2-c]pyridin-5-yl)-1-oxopentan-2-yl]-3-[4-(trifluoromethyl)phenyl]prop-2-enamide
—— (E)-N-[(2R)-1-(6,7-dihydro-4H-thieno[3,2-c]pyridin-5-yl)-1-oxopentan-2-yl]-3-(4-fluorophenyl)prop-2-enamide —— C21H23FN2O2S
(E)-N-[(2R)-1-(6,7-dihydro-4H-thieno[3,2-c]pyridin-5-yl)-1-oxopentan-2-yl]-3-(4-fluorophenyl)prop-2-enamide
—— (E)-N-[(2S)-1-(6,7-dihydro-4H-thieno[3,2-c]pyridin-5-yl)-1-oxopentan-2-yl]-3-(3-fluorophenyl)prop-2-enamide —— C21H23FN2O2S
(E)-N-[(2S)-1-(6,7-dihydro-4H-thieno[3,2-c]pyridin-5-yl)-1-oxopentan-2-yl]-3-(3-fluorophenyl)prop-2-enamide
—— [(E)-3-phenylprop-2-enyl] 2-chloro-5-sulfamoylbenzoate —— C16H14ClNO4S
[(E)-3-phenylprop-2-enyl] 2-chloro-5-sulfamoylbenzoate
—— (E)-3-(3-chloro-5-methoxy-4-propan-2-yloxyphenyl)-N-[(2R)-1-(6,7-dihydro-4H-thieno[3,2-c]pyridin-5-yl)-1-oxopentan-2-yl]prop-2-enamide —— C25H31ClN2O4S
(E)-3-(3-chloro-5-methoxy-4-propan-2-yloxyphenyl)-N-[(2R)-1-(6,7-dihydro-4H-thieno[3,2-c]pyridin-5-yl)-1-oxopentan-2-yl]prop-2-enamide
—— (E)-N-[(2R)-1-(6,7-dihydro-4H-thieno[3,2-c]pyridin-5-yl)-1-oxopentan-2-yl]-3-(3-methoxy-4-propan-2-yloxyphenyl)prop-2-enamide —— C25H32N2O4S
(E)-N-[(2R)-1-(6,7-dihydro-4H-thieno[3,2-c]pyridin-5-yl)-1-oxopentan-2-yl]-3-(3-methoxy-4-propan-2-yloxyphenyl)prop-2-enamide
—— (E)-3-(4-chlorophenyl)-N-[(2S)-1-(6,7-dihydro-4H-thieno[3,2-c]pyridin-5-yl)-1-oxopentan-2-yl]prop-2-enamide —— C21H23ClN2O2S
(E)-3-(4-chlorophenyl)-N-[(2S)-1-(6,7-dihydro-4H-thieno[3,2-c]pyridin-5-yl)-1-oxopentan-2-yl]prop-2-enamide
—— ethyl 5-[[(2R)-1-(6,7-dihydro-4H-thieno[3,2-c]pyridin-5-yl)-1-oxopentan-2-yl]carbamoyl]-2,4-dimethyl-1H-pyrrole-3-carboxylate —— C22H29N3O4S
ethyl 5-[[(2R)-1-(6,7-dihydro-4H-thieno[3,2-c]pyridin-5-yl)-1-oxopentan-2-yl]carbamoyl]-2,4-dimethyl-1H-pyrrole-3-carboxylate
—— (E)-3-(1,3-benzodioxol-5-yl)-N-[(2S)-1-(6,7-dihydro-4H-thieno[3,2-c]pyridin-5-yl)-1-oxopentan-2-yl]prop-2-enamide —— C22H24N2O4S
(E)-3-(1,3-benzodioxol-5-yl)-N-[(2S)-1-(6,7-dihydro-4H-thieno[3,2-c]pyridin-5-yl)-1-oxopentan-2-yl]prop-2-enamide
—— (E)-N-[(2S)-1-(6,7-dihydro-4H-thieno[3,2-c]pyridin-5-yl)-1-oxopentan-2-yl]-3-(2-nitrophenyl)prop-2-enamide —— C21H23N3O4S
(E)-N-[(2S)-1-(6,7-dihydro-4H-thieno[3,2-c]pyridin-5-yl)-1-oxopentan-2-yl]-3-(2-nitrophenyl)prop-2-enamide
—— (E)-3-(3-chloro-4,5-dimethoxyphenyl)-N-[(2S)-1-(6,7-dihydro-4H-thieno[3,2-c]pyridin-5-yl)-1-oxopentan-2-yl]prop-2-enamide —— C23H27ClN2O4S
(E)-3-(3-chloro-4,5-dimethoxyphenyl)-N-[(2S)-1-(6,7-dihydro-4H-thieno[3,2-c]pyridin-5-yl)-1-oxopentan-2-yl]prop-2-enamide
—— (E)-3-(3-chloro-5-methoxy-4-propan-2-yloxyphenyl)-N-[(2S)-1-(6,7-dihydro-4H-thieno[3,2-c]pyridin-5-yl)-1-oxopentan-2-yl]prop-2-enamide —— C25H31ClN2O4S
(E)-3-(3-chloro-5-methoxy-4-propan-2-yloxyphenyl)-N-[(2S)-1-(6,7-dihydro-4H-thieno[3,2-c]pyridin-5-yl)-1-oxopentan-2-yl]prop-2-enamide
—— (E)-N-[(2R)-1-(6,7-dihydro-4H-thieno[3,2-c]pyridin-5-yl)-1-oxopentan-2-yl]-3-(4-nitrophenyl)prop-2-enamide —— C21H23N3O4S
(E)-N-[(2R)-1-(6,7-dihydro-4H-thieno[3,2-c]pyridin-5-yl)-1-oxopentan-2-yl]-3-(4-nitrophenyl)prop-2-enamide
—— (E)-3-[4-(difluoromethoxy)-3-methoxyphenyl]-N-[(2R)-1-(6,7-dihydro-4H-thieno[3,2-c]pyridin-5-yl)-1-oxopentan-2-yl]prop-2-enamide —— C23H26F2N2O4S
(E)-3-[4-(difluoromethoxy)-3-methoxyphenyl]-N-[(2R)-1-(6,7-dihydro-4H-thieno[3,2-c]pyridin-5-yl)-1-oxopentan-2-yl]prop-2-enamide
—— (E)-3-(1,3-benzodioxol-5-yl)-N-[(2R)-1-(6,7-dihydro-4H-thieno[3,2-c]pyridin-5-yl)-1-oxopentan-2-yl]prop-2-enamide —— C22H24N2O4S
(E)-3-(1,3-benzodioxol-5-yl)-N-[(2R)-1-(6,7-dihydro-4H-thieno[3,2-c]pyridin-5-yl)-1-oxopentan-2-yl]prop-2-enamide
—— (E)-N-[(2S)-1-(6,7-dihydro-4H-thieno[3,2-c]pyridin-5-yl)-1-oxopentan-2-yl]-3-(4-fluorophenyl)prop-2-enamide —— C21H23FN2O2S
(E)-N-[(2S)-1-(6,7-dihydro-4H-thieno[3,2-c]pyridin-5-yl)-1-oxopentan-2-yl]-3-(4-fluorophenyl)prop-2-enamide
—— (E)-3-(3-chloro-5-ethoxy-4-methoxyphenyl)-N-[(2R)-1-(6,7-dihydro-4H-thieno[3,2-c]pyridin-5-yl)-1-oxopentan-2-yl]prop-2-enamide —— C24H29ClN2O4S
(E)-3-(3-chloro-5-ethoxy-4-methoxyphenyl)-N-[(2R)-1-(6,7-dihydro-4H-thieno[3,2-c]pyridin-5-yl)-1-oxopentan-2-yl]prop-2-enamide
—— ethyl 2-[2-[[(2S)-2-(3,5-dichlorophenoxy)propanoyl]amino]-1,3-thiazol-4-yl]acetate —— C16H16Cl2N2O4S
ethyl 2-[2-[[(2S)-2-(3,5-dichlorophenoxy)propanoyl]amino]-1,3-thiazol-4-yl]acetate
—— (E)-N-[(2R)-1-(6,7-dihydro-4H-thieno[3,2-c]pyridin-5-yl)-1-oxopentan-2-yl]-3-(3,4-dimethoxyphenyl)prop-2-enamide —— C23H28N2O4S
(E)-N-[(2R)-1-(6,7-dihydro-4H-thieno[3,2-c]pyridin-5-yl)-1-oxopentan-2-yl]-3-(3,4-dimethoxyphenyl)prop-2-enamide
—— (E)-N-[(2S)-1-(6,7-dihydro-4H-thieno[3,2-c]pyridin-5-yl)-1-oxopentan-2-yl]-3-(furan-2-yl)prop-2-enamide —— C19H22N2O3S
(E)-N-[(2S)-1-(6,7-dihydro-4H-thieno[3,2-c]pyridin-5-yl)-1-oxopentan-2-yl]-3-(furan-2-yl)prop-2-enamide
—— (E)-N-[(2S)-1-(6,7-dihydro-4H-thieno[3,2-c]pyridin-5-yl)-1-oxopentan-2-yl]-3-(3,4-dimethoxyphenyl)prop-2-enamide —— C23H28N2O4S
(E)-N-[(2S)-1-(6,7-dihydro-4H-thieno[3,2-c]pyridin-5-yl)-1-oxopentan-2-yl]-3-(3,4-dimethoxyphenyl)prop-2-enamide
—— ethyl 4-[2-[[(2S)-butan-2-yl]amino]-2-oxoethyl]sulfanyl-2,5-dimethylthieno[2,3-d]pyrimidine-6-carboxylate —— C17H23N3O3S2
ethyl 4-[2-[[(2S)-butan-2-yl]amino]-2-oxoethyl]sulfanyl-2,5-dimethylthieno[2,3-d]pyrimidine-6-carboxylate
—— ethyl 2-[(2R)-4-benzylmorpholin-2-yl]-4-methyl-1,3-thiazole-5-carboxylate —— C18H22N2O3S
ethyl 2-[(2R)-4-benzylmorpholin-2-yl]-4-methyl-1,3-thiazole-5-carboxylate
—— ethyl (7R)-5-methyl-7-(3-methylthiophen-2-yl)-2-thiophen-2-yl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate —— C18H18N4O2S2
ethyl (7R)-5-methyl-7-(3-methylthiophen-2-yl)-2-thiophen-2-yl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate
—— ethyl 5-[2-[(2R)-4-benzylmorpholin-2-yl]-1,3-thiazol-4-yl]-2,4-dimethyl-1H-pyrrole-3-carboxylate —— C23H27N3O3S
ethyl 5-[2-[(2R)-4-benzylmorpholin-2-yl]-1,3-thiazol-4-yl]-2,4-dimethyl-1H-pyrrole-3-carboxylate
—— Ethyl 4-[[2-(4-chloro-2-propanoylphenoxy)acetyl]amino]benzoate —— C20H20ClNO5
Ethyl 4-[[2-(4-chloro-2-propanoylphenoxy)acetyl]amino]benzoate
—— ethyl 5-[2-[(2S)-4-benzylmorpholin-2-yl]-1,3-thiazol-4-yl]-2,4-dimethyl-1H-pyrrole-3-carboxylate —— C23H27N3O3S
ethyl 5-[2-[(2S)-4-benzylmorpholin-2-yl]-1,3-thiazol-4-yl]-2,4-dimethyl-1H-pyrrole-3-carboxylate
—— ethyl (3S)-3-[[1-(3-methylphenyl)cyclopentyl]methylcarbamoyl]piperidine-1-carboxylate —— C22H32N2O3
ethyl (3S)-3-[[1-(3-methylphenyl)cyclopentyl]methylcarbamoyl]piperidine-1-carboxylate
—— ethyl 4-[[(2S)-2-hydroxypropyl]amino]-2,5-dimethylthieno[2,3-d]pyrimidine-6-carboxylate —— C14H19N3O3S
ethyl 4-[[(2S)-2-hydroxypropyl]amino]-2,5-dimethylthieno[2,3-d]pyrimidine-6-carboxylate
—— Ethyl 2-[[5-(4-fluorophenyl)tetrazol-2-yl]methyl]-4-methylquinoline-3-carboxylate —— C21H18FN5O2
Ethyl 2-[[5-(4-fluorophenyl)tetrazol-2-yl]methyl]-4-methylquinoline-3-carboxylate
—— Ethyl 2-[[2-(4-chloro-2-propanoylphenoxy)acetyl]amino]benzoate —— C20H20ClNO5
Ethyl 2-[[2-(4-chloro-2-propanoylphenoxy)acetyl]amino]benzoate
—— ethyl 2-[(2S)-4-benzylmorpholin-2-yl]-4-methyl-1,3-thiazole-5-carboxylate —— C18H22N2O3S
ethyl 2-[(2S)-4-benzylmorpholin-2-yl]-4-methyl-1,3-thiazole-5-carboxylate
—— ethyl 5-[2-(4-chloro-2-propanoylphenoxy)acetyl]-2,4-dimethyl-1H-pyrrole-3-carboxylate —— C20H22ClNO5
ethyl 5-[2-(4-chloro-2-propanoylphenoxy)acetyl]-2,4-dimethyl-1H-pyrrole-3-carboxylate
—— ethyl (5E)-5-[(2-chlorophenyl)methylidene]-3-methyl-4-oxo-6,7-dihydro-1H-indole-2-carboxylate —— C19H18ClNO3
ethyl (5E)-5-[(2-chlorophenyl)methylidene]-3-methyl-4-oxo-6,7-dihydro-1H-indole-2-carboxylate
—— ethyl (3R)-3-[[1-(3-methylphenyl)cyclopentyl]methylcarbamoyl]piperidine-1-carboxylate —— C22H32N2O3
ethyl (3R)-3-[[1-(3-methylphenyl)cyclopentyl]methylcarbamoyl]piperidine-1-carboxylate
—— (E)-2-cyano-3-ethoxybut-2-enoate —— C7H8NO3-
(E)-2-cyano-3-ethoxybut-2-enoate
—— ethyl 4-[[(2R)-2-hydroxypropyl]amino]-2,5-dimethylthieno[2,3-d]pyrimidine-6-carboxylate —— C14H19N3O3S
ethyl 4-[[(2R)-2-hydroxypropyl]amino]-2,5-dimethylthieno[2,3-d]pyrimidine-6-carboxylate
—— (E)-N-[2-[(2R)-butan-2-yl]phenyl]-3-(2-methoxyphenyl)prop-2-enamide —— C20H23NO2
(E)-N-[2-[(2R)-butan-2-yl]phenyl]-3-(2-methoxyphenyl)prop-2-enamide
—— (E)-3-phenyl-N-[(1R)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]prop-2-enamide —— C19H18N4O
(E)-3-phenyl-N-[(1R)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]prop-2-enamide
—— (E)-3-phenyl-N-[(1S)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]prop-2-enamide —— C19H18N4O
(E)-3-phenyl-N-[(1S)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]prop-2-enamide
—— ethyl 5-[(2R)-2-(4-cyano-2-ethoxyphenoxy)propanoyl]-2,4-dimethyl-1H-pyrrole-3-carboxylate —— C21H24N2O5
ethyl 5-[(2R)-2-(4-cyano-2-ethoxyphenoxy)propanoyl]-2,4-dimethyl-1H-pyrrole-3-carboxylate
—— ethyl 4-[2-[[(2R)-butan-2-yl]amino]-2-oxoethyl]sulfanyl-2,5-dimethylthieno[2,3-d]pyrimidine-6-carboxylate —— C17H23N3O3S2
ethyl 4-[2-[[(2R)-butan-2-yl]amino]-2-oxoethyl]sulfanyl-2,5-dimethylthieno[2,3-d]pyrimidine-6-carboxylate
—— Ethyl 2-[[2-(4-cyano-2-ethoxyphenoxy)acetyl]amino]-5-ethylthiophene-3-carboxylate —— C20H22N2O5S
Ethyl 2-[[2-(4-cyano-2-ethoxyphenoxy)acetyl]amino]-5-ethylthiophene-3-carboxylate
—— ethyl 5-[(2S)-2-(4-cyano-2-ethoxyphenoxy)propanoyl]-2,4-dimethyl-1H-pyrrole-3-carboxylate —— C21H24N2O5
ethyl 5-[(2S)-2-(4-cyano-2-ethoxyphenoxy)propanoyl]-2,4-dimethyl-1H-pyrrole-3-carboxylate