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—— 7-[(S)-(3-hydroxyphenyl)-[(4-methylpyridin-2-yl)amino]methyl]-2-methylquinolin-8-ol —— C23H21N3O2
7-[(S)-(3-hydroxyphenyl)-[(4-methylpyridin-2-yl)amino]methyl]-2-methylquinolin-8-ol
—— 7-[(R)-[(4-methylpyridin-1-ium-2-yl)amino]-(6-methylpyridin-2-yl)methyl]quinolin-8-olate —— C22H20N4O
7-[(R)-[(4-methylpyridin-1-ium-2-yl)amino]-(6-methylpyridin-2-yl)methyl]quinolin-8-olate
—— 7-(2-Pyridin-3-ylquinazolin-4-yl)oxychromen-2-one —— C22H13N3O3
7-(2-Pyridin-3-ylquinazolin-4-yl)oxychromen-2-one
—— 7-[(S)-(5-methylthiophen-2-yl)-(pyridin-2-ylamino)methyl]quinolin-8-ol —— C20H17N3OS
7-[(S)-(5-methylthiophen-2-yl)-(pyridin-2-ylamino)methyl]quinolin-8-ol
—— (7S)-7-methyl-N-(2-phenylethyl)-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-amine —— C19H21N3S
(7S)-7-methyl-N-(2-phenylethyl)-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-amine
—— 7-[5-(4-Methoxyphenyl)thieno[2,3-d]pyrimidin-4-yl]oxychromen-2-one —— C22H14N2O4S
7-[5-(4-Methoxyphenyl)thieno[2,3-d]pyrimidin-4-yl]oxychromen-2-one
—— 7-[(R)-1,3-benzodioxol-5-yl-(pyridin-2-ylamino)methyl]-2-methylquinolin-8-ol —— C23H19N3O3
7-[(R)-1,3-benzodioxol-5-yl-(pyridin-2-ylamino)methyl]-2-methylquinolin-8-ol
—— 7-[(S)-1,3-benzodioxol-5-yl-(pyridin-2-ylamino)methyl]-2-methylquinolin-8-ol —— C23H19N3O3
7-[(S)-1,3-benzodioxol-5-yl-(pyridin-2-ylamino)methyl]-2-methylquinolin-8-ol
—— 7-(difluoromethyl)-N-(3-methoxy-5-nitrophenyl)-5-(4-methylphenyl)pyrazolo[1,5-a]pyrimidine-3-carboxamide —— C22H17F2N5O4
7-(difluoromethyl)-N-(3-methoxy-5-nitrophenyl)-5-(4-methylphenyl)pyrazolo[1,5-a]pyrimidine-3-carboxamide
—— 7-(difluoromethyl)-5-(4-methylphenyl)-N-(3-nitro-5-phenoxyphenyl)pyrazolo[1,5-a]pyrimidine-3-carboxamide —— C27H19F2N5O4
7-(difluoromethyl)-5-(4-methylphenyl)-N-(3-nitro-5-phenoxyphenyl)pyrazolo[1,5-a]pyrimidine-3-carboxamide
—— 7-(difluoromethyl)-N-[3-nitro-5-(2,2,2-trifluoroethoxy)phenyl]-5-phenylpyrazolo[1,5-a]pyrimidine-3-carboxamide —— C22H14F5N5O4
7-(difluoromethyl)-N-[3-nitro-5-(2,2,2-trifluoroethoxy)phenyl]-5-phenylpyrazolo[1,5-a]pyrimidine-3-carboxamide
—— 7-(difluoromethyl)-N-(4-fluoro-3-nitrophenyl)-5-(4-methoxyphenyl)pyrazolo[1,5-a]pyrimidine-3-carboxamide —— C21H14F3N5O4
7-(difluoromethyl)-N-(4-fluoro-3-nitrophenyl)-5-(4-methoxyphenyl)pyrazolo[1,5-a]pyrimidine-3-carboxamide
—— 7-(difluoromethyl)-N-(3-methoxy-5-nitrophenyl)-5-phenylpyrazolo[1,5-a]pyrimidine-3-carboxamide —— C21H15F2N5O4
7-(difluoromethyl)-N-(3-methoxy-5-nitrophenyl)-5-phenylpyrazolo[1,5-a]pyrimidine-3-carboxamide
—— 7-(difluoromethyl)-N-[3-nitro-5-(pyridin-2-ylsulfanyl)phenyl]-5-phenylpyrazolo[1,5-a]pyrimidine-3-carboxamide —— C25H16F2N6O3S
7-(difluoromethyl)-N-[3-nitro-5-(pyridin-2-ylsulfanyl)phenyl]-5-phenylpyrazolo[1,5-a]pyrimidine-3-carboxamide
—— 7-nitro-1H-2,1,3-benzothiadiazol-6-one —— C6H3N3O3S
7-nitro-1H-2,1,3-benzothiadiazol-6-one
—— 7-(difluoromethyl)-N-[3-(4-fluorophenoxy)-5-nitrophenyl]-5-phenylpyrazolo[1,5-a]pyrimidine-3-carboxamide —— C26H16F3N5O4
7-(difluoromethyl)-N-[3-(4-fluorophenoxy)-5-nitrophenyl]-5-phenylpyrazolo[1,5-a]pyrimidine-3-carboxamide
—— 7-(difluoromethyl)-N-(3-nitro-5-phenoxyphenyl)-5-phenylpyrazolo[1,5-a]pyrimidine-3-carboxamide —— C26H17F2N5O4
7-(difluoromethyl)-N-(3-nitro-5-phenoxyphenyl)-5-phenylpyrazolo[1,5-a]pyrimidine-3-carboxamide
—— 7-(difluoromethyl)-5-(4-methoxyphenyl)-N-(3-nitro-5-pyridin-2-ylsulfanylphenyl)pyrazolo[1,5-a]pyrimidine-3-carboxamide —— C26H18F2N6O4S
7-(difluoromethyl)-5-(4-methoxyphenyl)-N-(3-nitro-5-pyridin-2-ylsulfanylphenyl)pyrazolo[1,5-a]pyrimidine-3-carboxamide
—— 7-(difluoromethyl)-N-(4-fluoro-3-nitrophenyl)-5-methyl[1,2,4]triazolo[1,5-a]pyrimidine-2-carboxamide —— C14H9F3N6O3
7-(difluoromethyl)-N-(4-fluoro-3-nitrophenyl)-5-methyl[1,2,4]triazolo[1,5-a]pyrimidine-2-carboxamide
—— 7-(difluoromethyl)-N-[3-nitro-5-(2,2,3,3-tetrafluoropropoxy)phenyl]-5-phenylpyrazolo[1,5-a]pyrimidine-3-carboxamide —— C23H15F6N5O4
7-(difluoromethyl)-N-[3-nitro-5-(2,2,3,3-tetrafluoropropoxy)phenyl]-5-phenylpyrazolo[1,5-a]pyrimidine-3-carboxamide
—— 7-(difluoromethyl)-N-(3-methoxy-5-nitrophenyl)-5-(4-methoxyphenyl)pyrazolo[1,5-a]pyrimidine-3-carboxamide —— C22H17F2N5O5
7-(difluoromethyl)-N-(3-methoxy-5-nitrophenyl)-5-(4-methoxyphenyl)pyrazolo[1,5-a]pyrimidine-3-carboxamide
—— 7-(difluoromethyl)-N-(4-fluoro-3-nitrophenyl)-5-(4-methylphenyl)pyrazolo[1,5-a]pyrimidine-3-carboxamide —— C21H14F3N5O3
7-(difluoromethyl)-N-(4-fluoro-3-nitrophenyl)-5-(4-methylphenyl)pyrazolo[1,5-a]pyrimidine-3-carboxamide
—— 7-(difluoromethyl)-5-(4-methylphenyl)-N-[3-nitro-5-(2,2,2-trifluoroethoxy)phenyl]pyrazolo[1,5-a]pyrimidine-3-carboxamide —— C23H16F5N5O4
7-(difluoromethyl)-5-(4-methylphenyl)-N-[3-nitro-5-(2,2,2-trifluoroethoxy)phenyl]pyrazolo[1,5-a]pyrimidine-3-carboxamide
—— 7-[(2R)-2-hydroxy-3-(4-methoxyphenoxy)propyl]-3-methyl-8-(methylamino)purine-2,6-dione —— C17H21N5O5
7-[(2R)-2-hydroxy-3-(4-methoxyphenoxy)propyl]-3-methyl-8-(methylamino)purine-2,6-dione
—— 7-[(2S)-2-hydroxy-3-(4-methoxyphenoxy)propyl]-3-methyl-8-(methylamino)purine-2,6-dione —— C17H21N5O5
7-[(2S)-2-hydroxy-3-(4-methoxyphenoxy)propyl]-3-methyl-8-(methylamino)purine-2,6-dione
—— 7-Benzyl-8-[2-(4-fluorophenyl)ethylamino]-3-methylpurine-2,6-dione —— C21H20FN5O2
7-Benzyl-8-[2-(4-fluorophenyl)ethylamino]-3-methylpurine-2,6-dione
—— 7-(methoxymethyl)-3-(4-methylphenyl)-1H-[1,2,4]triazolo[4,3-a]pyrimidin-5-one —— C14H14N4O2
7-(methoxymethyl)-3-(4-methylphenyl)-1H-[1,2,4]triazolo[4,3-a]pyrimidin-5-one
—— 7-[(S)-(4-nitrophenyl)-(1,3-thiazol-2-ylamino)methyl]quinolin-8-ol —— C19H14N4O3S
7-[(S)-(4-nitrophenyl)-(1,3-thiazol-2-ylamino)methyl]quinolin-8-ol
—— 7-(difluoromethyl)-N-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]-5-(4-methoxyphenyl)-N-methylpyrazolo[1,5-a]pyrimidine-3-carboxamide —— C23H24F2N6O2
7-(difluoromethyl)-N-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]-5-(4-methoxyphenyl)-N-methylpyrazolo[1,5-a]pyrimidine-3-carboxamide
—— 7-[(R)-(4-nitrophenyl)-(1,3-thiazol-2-ylamino)methyl]quinolin-8-ol —— C19H14N4O3S
7-[(R)-(4-nitrophenyl)-(1,3-thiazol-2-ylamino)methyl]quinolin-8-ol
—— 7-(difluoromethyl)-5-phenyl-N-[3-(trifluoromethyl)phenyl]pyrazolo[1,5-a]pyrimidine-3-carboxamide —— C21H13F5N4O
7-(difluoromethyl)-5-phenyl-N-[3-(trifluoromethyl)phenyl]pyrazolo[1,5-a]pyrimidine-3-carboxamide
—— 7-[5-(4-Fluorophenyl)thieno[2,3-d]pyrimidin-4-yl]oxychromen-2-one —— C21H11FN2O3S
7-[5-(4-Fluorophenyl)thieno[2,3-d]pyrimidin-4-yl]oxychromen-2-one
—— (7S,8S)-1-benzyl-7,8-dimethyl-1-azaspiro[4.4]nonane —— C17H25N
(7S,8S)-1-benzyl-7,8-dimethyl-1-azaspiro[4.4]nonane
—— [7-(Difluoromethyl)-5-(4-methoxyphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]-[4-(2,3-dimethylphenyl)piperazin-1-yl]methanone —— C27H27F2N5O2
[7-(Difluoromethyl)-5-(4-methoxyphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]-[4-(2,3-dimethylphenyl)piperazin-1-yl]methanone
—— 7-(difluoromethyl)-N-[1-(2-methylbenzyl)-1H-pyrazol-4-yl]-5-(4-methylphenyl)pyrazolo[1,5-a]pyrimidine-3-carboxamide —— C26H22F2N6O
7-(difluoromethyl)-N-[1-(2-methylbenzyl)-1H-pyrazol-4-yl]-5-(4-methylphenyl)pyrazolo[1,5-a]pyrimidine-3-carboxamide
—— 7-(difluoromethyl)-N-[(1R)-1-(4-ethoxyphenyl)ethyl]-5-(4-methoxyphenyl)pyrazolo[1,5-a]pyrimidine-3-carboxamide —— C25H24F2N4O3
7-(difluoromethyl)-N-[(1R)-1-(4-ethoxyphenyl)ethyl]-5-(4-methoxyphenyl)pyrazolo[1,5-a]pyrimidine-3-carboxamide
—— [7-(Difluoromethyl)-5-(4-methylphenyl)pyrazolo[1,5-A]pyrimidin-3-YL][4-(4-fluorophenyl)piperazino]methanone —— C25H22F3N5O
[7-(Difluoromethyl)-5-(4-methylphenyl)pyrazolo[1,5-A]pyrimidin-3-YL][4-(4-fluorophenyl)piperazino]methanone
—— 7-(difluoromethyl)-N-(2-fluorobenzyl)-5-methylpyrazolo[1,5-a]pyrimidine-3-carboxamide —— C16H13F3N4O
7-(difluoromethyl)-N-(2-fluorobenzyl)-5-methylpyrazolo[1,5-a]pyrimidine-3-carboxamide
—— [7-(Difluoromethyl)-5-(4-methoxyphenyl)pyrazolo[1,5-A]pyrimidin-3-YL](4-phenylpiperazino)methanone —— C25H23F2N5O2
[7-(Difluoromethyl)-5-(4-methoxyphenyl)pyrazolo[1,5-A]pyrimidin-3-YL](4-phenylpiperazino)methanone
—— 7-(difluoromethyl)-N-[(1S)-1-(4-ethoxyphenyl)ethyl]-5-(4-methoxyphenyl)pyrazolo[1,5-a]pyrimidine-3-carboxamide —— C25H24F2N4O3
7-(difluoromethyl)-N-[(1S)-1-(4-ethoxyphenyl)ethyl]-5-(4-methoxyphenyl)pyrazolo[1,5-a]pyrimidine-3-carboxamide
—— 7-(difluoromethyl)-N-(3-methoxyphenyl)-5-(4-methoxyphenyl)pyrazolo[1,5-a]pyrimidine-3-carboxamide —— C22H18F2N4O3
7-(difluoromethyl)-N-(3-methoxyphenyl)-5-(4-methoxyphenyl)pyrazolo[1,5-a]pyrimidine-3-carboxamide
—— 7-(difluoromethyl)-N-[1-(4-fluorobenzyl)-1H-pyrazol-4-yl]-5-(4-methylphenyl)pyrazolo[1,5-a]pyrimidine-3-carboxamide —— C25H19F3N6O
7-(difluoromethyl)-N-[1-(4-fluorobenzyl)-1H-pyrazol-4-yl]-5-(4-methylphenyl)pyrazolo[1,5-a]pyrimidine-3-carboxamide
—— [7-(Difluoromethyl)-5-methylpyrazolo[1,5-a]pyrimidin-3-yl]-[4-(4-methoxyphenyl)piperazin-1-yl]methanone —— C20H21F2N5O2
[7-(Difluoromethyl)-5-methylpyrazolo[1,5-a]pyrimidin-3-yl]-[4-(4-methoxyphenyl)piperazin-1-yl]methanone
—— 7-(difluoromethyl)-5-(4-methoxyphenyl)-N-[2-(2-methoxyphenyl)ethyl]pyrazolo[1,5-a]pyrimidine-3-carboxamide —— C24H22F2N4O3
7-(difluoromethyl)-5-(4-methoxyphenyl)-N-[2-(2-methoxyphenyl)ethyl]pyrazolo[1,5-a]pyrimidine-3-carboxamide
—— 7-(difluoromethyl)-N-(4-fluoro-2-methylphenyl)-5-(4-methylphenyl)pyrazolo[1,5-a]pyrimidine-3-carboxamide —— C22H17F3N4O
7-(difluoromethyl)-N-(4-fluoro-2-methylphenyl)-5-(4-methylphenyl)pyrazolo[1,5-a]pyrimidine-3-carboxamide
—— 7-(difluoromethyl)-N-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-5-(4-methoxyphenyl)pyrazolo[1,5-a]pyrimidine-3-carboxamide —— C21H20F2N6O2
7-(difluoromethyl)-N-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-5-(4-methoxyphenyl)pyrazolo[1,5-a]pyrimidine-3-carboxamide
—— 7-(difluoromethyl)-5-phenyl-N-[4-(trifluoromethyl)phenyl]pyrazolo[1,5-a]pyrimidine-3-carboxamide —— C21H13F5N4O
7-(difluoromethyl)-5-phenyl-N-[4-(trifluoromethyl)phenyl]pyrazolo[1,5-a]pyrimidine-3-carboxamide
—— 7-(Difluoromethyl)-N-{1-[(2-methylphenyl)methyl]-1H-pyrazol-4-YL}-5-phenylpyrazolo[1,5-A]pyrimidine-3-carboxamide —— C25H20F2N6O
7-(Difluoromethyl)-N-{1-[(2-methylphenyl)methyl]-1H-pyrazol-4-YL}-5-phenylpyrazolo[1,5-A]pyrimidine-3-carboxamide
—— 7-(Difluoromethyl)-N~3~-(2-fluorobenzyl)-5-(4-methoxyphenyl)pyrazolo[1,5-A]pyrimidine-3-carboxamide —— C22H17F3N4O2
7-(Difluoromethyl)-N~3~-(2-fluorobenzyl)-5-(4-methoxyphenyl)pyrazolo[1,5-A]pyrimidine-3-carboxamide
—— 7-(difluoromethyl)-N-(2,6-dimethylphenyl)-5-phenylpyrazolo[1,5-a]pyrimidine-3-carboxamide —— C22H18F2N4O
7-(difluoromethyl)-N-(2,6-dimethylphenyl)-5-phenylpyrazolo[1,5-a]pyrimidine-3-carboxamide