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—— 7-methoxy-3-[[[(1R)-2-methyl-1-[1-(2-methylbutan-2-yl)tetrazol-5-yl]propyl]-(thiophen-2-ylmethyl)amino]methyl]-1H-quinolin-2-one —— C26H34N6O2S
7-methoxy-3-[[[(1R)-2-methyl-1-[1-(2-methylbutan-2-yl)tetrazol-5-yl]propyl]-(thiophen-2-ylmethyl)amino]methyl]-1H-quinolin-2-one
—— 7-methyl-3-[[[(1S)-2-methyl-1-[1-[[(2S)-oxolan-2-yl]methyl]tetrazol-5-yl]propyl]-(thiophen-2-ylmethyl)amino]methyl]-1H-quinolin-2-one —— C26H32N6O2S
7-methyl-3-[[[(1S)-2-methyl-1-[1-[[(2S)-oxolan-2-yl]methyl]tetrazol-5-yl]propyl]-(thiophen-2-ylmethyl)amino]methyl]-1H-quinolin-2-one
—— 7-methyl-3-[[[(1R)-2-methyl-1-[1-(2-methylbutan-2-yl)tetrazol-5-yl]propyl]-(thiophen-2-ylmethyl)amino]methyl]-1H-quinolin-2-one —— C26H34N6OS
7-methyl-3-[[[(1R)-2-methyl-1-[1-(2-methylbutan-2-yl)tetrazol-5-yl]propyl]-(thiophen-2-ylmethyl)amino]methyl]-1H-quinolin-2-one
—— 7-methoxy-3-[[[(1R)-2-methyl-1-[1-(2-phenylethyl)tetrazol-5-yl]propyl]-(thiophen-2-ylmethyl)amino]methyl]-1H-quinolin-2-one —— C29H32N6O2S
7-methoxy-3-[[[(1R)-2-methyl-1-[1-(2-phenylethyl)tetrazol-5-yl]propyl]-(thiophen-2-ylmethyl)amino]methyl]-1H-quinolin-2-one
—— 7-methoxy-3-[[[(1S)-2-methyl-1-[1-(2-phenylethyl)tetrazol-5-yl]propyl]-(thiophen-2-ylmethyl)amino]methyl]-1H-quinolin-2-one —— C29H32N6O2S
7-methoxy-3-[[[(1S)-2-methyl-1-[1-(2-phenylethyl)tetrazol-5-yl]propyl]-(thiophen-2-ylmethyl)amino]methyl]-1H-quinolin-2-one
—— 7-methyl-3-[[[(1S)-2-methyl-1-[1-(2-methylbutan-2-yl)tetrazol-5-yl]propyl]-(thiophen-2-ylmethyl)amino]methyl]-1H-quinolin-2-one —— C26H34N6OS
7-methyl-3-[[[(1S)-2-methyl-1-[1-(2-methylbutan-2-yl)tetrazol-5-yl]propyl]-(thiophen-2-ylmethyl)amino]methyl]-1H-quinolin-2-one
—— (7R)-7-methyl-3-[2-[(2S)-2-methyl-2,3-dihydroindol-1-yl]-2-oxoethyl]-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]triazin-4-one —— C21H22N4O2S
(7R)-7-methyl-3-[2-[(2S)-2-methyl-2,3-dihydroindol-1-yl]-2-oxoethyl]-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]triazin-4-one
—— 7-[4-(4-Fluorophenyl)piperazin-1-yl]-5,6-dimethyl-2-thiophen-2-ylpyrazolo[1,5-a]pyrimidine —— C22H22FN5S
7-[4-(4-Fluorophenyl)piperazin-1-yl]-5,6-dimethyl-2-thiophen-2-ylpyrazolo[1,5-a]pyrimidine
—— 7-[4-(2-Methoxyphenyl)piperazin-1-yl]-5,6-dimethyl-2-thiophen-2-ylpyrazolo[1,5-a]pyrimidine —— C23H25N5OS
7-[4-(2-Methoxyphenyl)piperazin-1-yl]-5,6-dimethyl-2-thiophen-2-ylpyrazolo[1,5-a]pyrimidine
—— 7-[4-(3-Methoxyphenyl)piperazin-1-yl]-5,6-dimethyl-2-thiophen-2-ylpyrazolo[1,5-a]pyrimidine —— C23H25N5OS
7-[4-(3-Methoxyphenyl)piperazin-1-yl]-5,6-dimethyl-2-thiophen-2-ylpyrazolo[1,5-a]pyrimidine
—— (7R)-3-[2-(2,3-dihydroindol-1-yl)-2-oxoethyl]-7-methyl-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]triazin-4-one —— C20H20N4O2S
(7R)-3-[2-(2,3-dihydroindol-1-yl)-2-oxoethyl]-7-methyl-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]triazin-4-one
—— (7S)-7-tert-butyl-3-[2-(2,3-dihydroindol-1-yl)-2-oxoethyl]-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]triazin-4-one —— C23H26N4O2S
(7S)-7-tert-butyl-3-[2-(2,3-dihydroindol-1-yl)-2-oxoethyl]-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]triazin-4-one
—— (7R)-7-methyl-3-[2-[(2R)-2-methyl-2,3-dihydroindol-1-yl]-2-oxoethyl]-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]triazin-4-one —— C21H22N4O2S
(7R)-7-methyl-3-[2-[(2R)-2-methyl-2,3-dihydroindol-1-yl]-2-oxoethyl]-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]triazin-4-one
—— (7S)-7-methyl-3-[2-[(2R)-2-methyl-2,3-dihydroindol-1-yl]-2-oxoethyl]-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]triazin-4-one —— C21H22N4O2S
(7S)-7-methyl-3-[2-[(2R)-2-methyl-2,3-dihydroindol-1-yl]-2-oxoethyl]-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]triazin-4-one
—— (7S)-7-tert-butyl-3-[2-(3,4-dihydro-2H-quinolin-1-yl)-2-oxoethyl]-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]triazin-4-one —— C24H28N4O2S
(7S)-7-tert-butyl-3-[2-(3,4-dihydro-2H-quinolin-1-yl)-2-oxoethyl]-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]triazin-4-one
—— 7-[4-(2-Fluorophenyl)piperazin-1-yl]-5,6-dimethyl-2-thiophen-2-ylpyrazolo[1,5-a]pyrimidine —— C22H22FN5S
7-[4-(2-Fluorophenyl)piperazin-1-yl]-5,6-dimethyl-2-thiophen-2-ylpyrazolo[1,5-a]pyrimidine
—— (7S)-7-methyl-3-[2-[(2S)-2-methylpiperidin-1-yl]-2-oxoethyl]-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]triazin-4-one —— C18H24N4O2S
(7S)-7-methyl-3-[2-[(2S)-2-methylpiperidin-1-yl]-2-oxoethyl]-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]triazin-4-one
—— (7S)-7-methyl-3-[2-[(2S)-2-methyl-2,3-dihydroindol-1-yl]-2-oxoethyl]-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]triazin-4-one —— C21H22N4O2S
(7S)-7-methyl-3-[2-[(2S)-2-methyl-2,3-dihydroindol-1-yl]-2-oxoethyl]-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]triazin-4-one
—— (7S)-3-[2-(2,3-dihydroindol-1-yl)-2-oxoethyl]-7-methyl-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]triazin-4-one —— C20H20N4O2S
(7S)-3-[2-(2,3-dihydroindol-1-yl)-2-oxoethyl]-7-methyl-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]triazin-4-one
—— (7R)-7-tert-butyl-3-[2-[4-(furan-2-carbonyl)piperazin-1-yl]-2-oxoethyl]-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]triazin-4-one —— C24H29N5O4S
(7R)-7-tert-butyl-3-[2-[4-(furan-2-carbonyl)piperazin-1-yl]-2-oxoethyl]-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]triazin-4-one
—— (7S)-7-tert-butyl-3-[2-oxo-2-(3-oxo-2,4-dihydroquinoxalin-1-yl)ethyl]-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]triazin-4-one —— C23H25N5O3S
(7S)-7-tert-butyl-3-[2-oxo-2-(3-oxo-2,4-dihydroquinoxalin-1-yl)ethyl]-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]triazin-4-one
—— (7R)-3-[2-(azepan-1-yl)-2-oxoethyl]-7-methyl-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]triazin-4-one —— C18H24N4O2S
(7R)-3-[2-(azepan-1-yl)-2-oxoethyl]-7-methyl-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]triazin-4-one
—— (7S)-7-tert-butyl-3-[2-[4-(furan-2-carbonyl)piperazin-1-yl]-2-oxoethyl]-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]triazin-4-one —— C24H29N5O4S
(7S)-7-tert-butyl-3-[2-[4-(furan-2-carbonyl)piperazin-1-yl]-2-oxoethyl]-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]triazin-4-one
—— (7R)-7-methyl-3-[2-[(2R)-2-methylpiperidin-1-yl]-2-oxoethyl]-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]triazin-4-one —— C18H24N4O2S
(7R)-7-methyl-3-[2-[(2R)-2-methylpiperidin-1-yl]-2-oxoethyl]-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]triazin-4-one
—— (7S)-3-[2-(3-methoxyphenyl)-2-oxoethyl]-7-methyl-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]triazin-4-one —— C19H19N3O3S
(7S)-3-[2-(3-methoxyphenyl)-2-oxoethyl]-7-methyl-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]triazin-4-one
—— (7S)-3-[2-(azepan-1-yl)-2-oxoethyl]-7-methyl-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]triazin-4-one —— C18H24N4O2S
(7S)-3-[2-(azepan-1-yl)-2-oxoethyl]-7-methyl-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]triazin-4-one
—— (7R)-7-tert-butyl-3-phenacyl-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]triazin-4-one —— C21H23N3O2S
(7R)-7-tert-butyl-3-phenacyl-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]triazin-4-one
—— (7S)-7-tert-butyl-3-phenacyl-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]triazin-4-one —— C21H23N3O2S
(7S)-7-tert-butyl-3-phenacyl-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]triazin-4-one
—— (7S)-7-tert-butyl-3-[(4-methoxyphenyl)methyl]-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]triazin-4-one —— C21H25N3O2S
(7S)-7-tert-butyl-3-[(4-methoxyphenyl)methyl]-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]triazin-4-one
—— (7R)-7-tert-butyl-3-[2-(3,4-dihydro-2H-quinolin-1-yl)-2-oxoethyl]-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]triazin-4-one —— C24H28N4O2S
(7R)-7-tert-butyl-3-[2-(3,4-dihydro-2H-quinolin-1-yl)-2-oxoethyl]-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]triazin-4-one
—— (7S)-7-methyl-3-[2-[(2R)-2-methylpiperidin-1-yl]-2-oxoethyl]-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]triazin-4-one —— C18H24N4O2S
(7S)-7-methyl-3-[2-[(2R)-2-methylpiperidin-1-yl]-2-oxoethyl]-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]triazin-4-one
—— (7R)-7-methyl-3-[2-[(2S)-2-methylpiperidin-1-yl]-2-oxoethyl]-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]triazin-4-one —— C18H24N4O2S
(7R)-7-methyl-3-[2-[(2S)-2-methylpiperidin-1-yl]-2-oxoethyl]-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]triazin-4-one
—— (7R)-7-tert-butyl-3-[(4-methoxyphenyl)methyl]-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]triazin-4-one —— C21H25N3O2S
(7R)-7-tert-butyl-3-[(4-methoxyphenyl)methyl]-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]triazin-4-one
—— 7-Propyl-3-(pyridin-2-ylmethylsulfanyl)-[1,2,4]triazolo[4,3-c]pyrimidin-5-amine —— C14H16N6S
7-Propyl-3-(pyridin-2-ylmethylsulfanyl)-[1,2,4]triazolo[4,3-c]pyrimidin-5-amine
—— 7-(2-Oxopropylsulfanyl)-2,3-dihydro-[1,4]dioxino[2,3-g]quinoline-8-carbonitrile —— C15H12N2O3S
7-(2-Oxopropylsulfanyl)-2,3-dihydro-[1,4]dioxino[2,3-g]quinoline-8-carbonitrile
—— 7-(Pyridin-3-ylmethylsulfanyl)-2,3-dihydro-[1,4]dioxino[2,3-g]quinoline-8-carbonitrile —— C18H13N3O2S
7-(Pyridin-3-ylmethylsulfanyl)-2,3-dihydro-[1,4]dioxino[2,3-g]quinoline-8-carbonitrile
—— 7-methoxy-3-[5-methyl-3-[[(2S)-oxolan-2-yl]methylamino]imidazo[1,2-a]pyridin-2-yl]-1H-quinolin-2-one —— C23H24N4O3
7-methoxy-3-[5-methyl-3-[[(2S)-oxolan-2-yl]methylamino]imidazo[1,2-a]pyridin-2-yl]-1H-quinolin-2-one
—— 7-methoxy-3-[3-(2-methylbutan-2-ylamino)imidazo[1,2-a]pyridin-2-yl]-1H-quinolin-2-one —— C22H24N4O2
7-methoxy-3-[3-(2-methylbutan-2-ylamino)imidazo[1,2-a]pyridin-2-yl]-1H-quinolin-2-one
—— 7-methoxy-3-[5-methyl-3-[[(2R)-oxolan-2-yl]methylamino]imidazo[1,2-a]pyridin-2-yl]-1H-quinolin-2-one —— C23H24N4O3
7-methoxy-3-[5-methyl-3-[[(2R)-oxolan-2-yl]methylamino]imidazo[1,2-a]pyridin-2-yl]-1H-quinolin-2-one
—— 7-methoxy-3-[3-[(4-methoxyphenyl)methylamino]-5-methylimidazo[1,2-a]pyridin-2-yl]-1H-quinolin-2-one —— C26H24N4O3
7-methoxy-3-[3-[(4-methoxyphenyl)methylamino]-5-methylimidazo[1,2-a]pyridin-2-yl]-1H-quinolin-2-one
—— 7,8-dimethyl-3-[6-methyl-3-[[(2R)-oxolan-2-yl]methylamino]imidazo[1,2-a]pyridin-2-yl]-1H-quinolin-2-one —— C24H26N4O2
7,8-dimethyl-3-[6-methyl-3-[[(2R)-oxolan-2-yl]methylamino]imidazo[1,2-a]pyridin-2-yl]-1H-quinolin-2-one
—— 7,8-dimethyl-3-[6-methyl-3-[[(2S)-oxolan-2-yl]methylamino]imidazo[1,2-a]pyridin-2-yl]-1H-quinolin-2-one —— C24H26N4O2
7,8-dimethyl-3-[6-methyl-3-[[(2S)-oxolan-2-yl]methylamino]imidazo[1,2-a]pyridin-2-yl]-1H-quinolin-2-one
—— 7,8-dimethyl-3-[3-(2-methylbutan-2-ylamino)imidazo[1,2-a]pyridin-2-yl]-1H-quinolin-2-one —— C23H26N4O
7,8-dimethyl-3-[3-(2-methylbutan-2-ylamino)imidazo[1,2-a]pyridin-2-yl]-1H-quinolin-2-one
—— 7,9-Dimethyl-1-(pyridin-3-ylmethylsulfanyl)-11-thia-2,4,10-triaza-benzo[b]fluorene —— C21H16N4S2
7,9-Dimethyl-1-(pyridin-3-ylmethylsulfanyl)-11-thia-2,4,10-triaza-benzo[b]fluorene
—— 7-[[(1-benzyltetrazol-5-yl)methyl-[(4-fluorophenyl)methyl]amino]methyl]-5H-[1,3]dioxolo[4,5-g]quinolin-6-one —— C27H23FN6O3
7-[[(1-benzyltetrazol-5-yl)methyl-[(4-fluorophenyl)methyl]amino]methyl]-5H-[1,3]dioxolo[4,5-g]quinolin-6-one
—— 7-[[(1-cyclopentyltetrazol-5-yl)methyl-[(4-fluorophenyl)methyl]amino]methyl]-5H-[1,3]dioxolo[4,5-g]quinolin-6-one —— C25H25FN6O3
7-[[(1-cyclopentyltetrazol-5-yl)methyl-[(4-fluorophenyl)methyl]amino]methyl]-5H-[1,3]dioxolo[4,5-g]quinolin-6-one
—— 7-[[benzyl-[(1-cyclopentyltetrazol-5-yl)methyl]amino]methyl]-5H-[1,3]dioxolo[4,5-g]quinolin-6-one —— C25H26N6O3
7-[[benzyl-[(1-cyclopentyltetrazol-5-yl)methyl]amino]methyl]-5H-[1,3]dioxolo[4,5-g]quinolin-6-one
—— 7-[[(1-benzyltetrazol-5-yl)methyl-[(4-methoxyphenyl)methyl]amino]methyl]-5H-[1,3]dioxolo[4,5-g]quinolin-6-one —— C28H26N6O4
7-[[(1-benzyltetrazol-5-yl)methyl-[(4-methoxyphenyl)methyl]amino]methyl]-5H-[1,3]dioxolo[4,5-g]quinolin-6-one
—— 7-[[(4-fluorophenyl)methyl-[[1-(2-methylbutan-2-yl)tetrazol-5-yl]methyl]amino]methyl]-5H-[1,3]dioxolo[4,5-g]quinolin-6-one —— C25H27FN6O3
7-[[(4-fluorophenyl)methyl-[[1-(2-methylbutan-2-yl)tetrazol-5-yl]methyl]amino]methyl]-5H-[1,3]dioxolo[4,5-g]quinolin-6-one
—— 7-[[(1-cyclohexyltetrazol-5-yl)methyl-[(4-methoxyphenyl)methyl]amino]methyl]-5H-[1,3]dioxolo[4,5-g]quinolin-6-one —— C27H30N6O4
7-[[(1-cyclohexyltetrazol-5-yl)methyl-[(4-methoxyphenyl)methyl]amino]methyl]-5H-[1,3]dioxolo[4,5-g]quinolin-6-one