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中文名称 英文名称 CAS号 化学式 结构式图片
—— 7-[[(1-benzyltetrazol-5-yl)methyl-cyclopentylamino]methyl]-5H-[1,3]dioxolo[4,5-g]quinolin-6-one —— C25H26N6O3
7-[[(1-benzyltetrazol-5-yl)methyl-cyclopentylamino]methyl]-5H-[1,3]dioxolo[4,5-g]quinolin-6-one
—— 7,8-dimethyl-3-[[[(1R)-1-[1-(2-phenylethyl)tetrazol-5-yl]propyl]-(thiophen-2-ylmethyl)amino]methyl]-1H-quinolin-2-one —— C29H32N6OS
7,8-dimethyl-3-[[[(1R)-1-[1-(2-phenylethyl)tetrazol-5-yl]propyl]-(thiophen-2-ylmethyl)amino]methyl]-1H-quinolin-2-one
—— 7-[[(1-cyclohexyltetrazol-5-yl)methyl-[[(2S)-oxolan-2-yl]methyl]amino]methyl]-5H-[1,3]dioxolo[4,5-g]quinolin-6-one —— C24H30N6O4
7-[[(1-cyclohexyltetrazol-5-yl)methyl-[[(2S)-oxolan-2-yl]methyl]amino]methyl]-5H-[1,3]dioxolo[4,5-g]quinolin-6-one
—— 7-[[[(1R)-1-[1-[(4-fluorophenyl)methyl]tetrazol-5-yl]propyl]-(thiophen-2-ylmethyl)amino]methyl]-5H-[1,3]dioxolo[4,5-g]quinolin-6-one —— C27H25FN6O3S
7-[[[(1R)-1-[1-[(4-fluorophenyl)methyl]tetrazol-5-yl]propyl]-(thiophen-2-ylmethyl)amino]methyl]-5H-[1,3]dioxolo[4,5-g]quinolin-6-one
—— 7-[[[(1S)-1-[1-[(4-fluorophenyl)methyl]tetrazol-5-yl]propyl]-(2-phenylethyl)amino]methyl]-5H-[1,3]dioxolo[4,5-g]quinolin-6-one —— C30H29FN6O3
7-[[[(1S)-1-[1-[(4-fluorophenyl)methyl]tetrazol-5-yl]propyl]-(2-phenylethyl)amino]methyl]-5H-[1,3]dioxolo[4,5-g]quinolin-6-one
—— 7-[[cyclopentyl-[(1-cyclopentyltetrazol-5-yl)methyl]amino]methyl]-5H-[1,3]dioxolo[4,5-g]quinolin-6-one —— C23H28N6O3
7-[[cyclopentyl-[(1-cyclopentyltetrazol-5-yl)methyl]amino]methyl]-5H-[1,3]dioxolo[4,5-g]quinolin-6-one
—— 7,8-dimethyl-3-[[[(1S)-1-[1-(2-methylbutan-2-yl)tetrazol-5-yl]propyl]-(pyridin-3-ylmethyl)amino]methyl]-1H-quinolin-2-one —— C27H35N7O
7,8-dimethyl-3-[[[(1S)-1-[1-(2-methylbutan-2-yl)tetrazol-5-yl]propyl]-(pyridin-3-ylmethyl)amino]methyl]-1H-quinolin-2-one
—— 7-[[(1-cyclohexyltetrazol-5-yl)methyl-[[(2R)-oxolan-2-yl]methyl]amino]methyl]-5H-[1,3]dioxolo[4,5-g]quinolin-6-one —— C24H30N6O4
7-[[(1-cyclohexyltetrazol-5-yl)methyl-[[(2R)-oxolan-2-yl]methyl]amino]methyl]-5H-[1,3]dioxolo[4,5-g]quinolin-6-one
—— 7-[[(1-benzyltetrazol-5-yl)methyl-[(4-methylphenyl)methyl]amino]methyl]-5H-[1,3]dioxolo[4,5-g]quinolin-6-one —— C28H26N6O3
7-[[(1-benzyltetrazol-5-yl)methyl-[(4-methylphenyl)methyl]amino]methyl]-5H-[1,3]dioxolo[4,5-g]quinolin-6-one
—— 7,8-dimethyl-3-[[[(1S)-1-[1-(2-phenylethyl)tetrazol-5-yl]propyl]-(thiophen-2-ylmethyl)amino]methyl]-1H-quinolin-2-one —— C29H32N6OS
7,8-dimethyl-3-[[[(1S)-1-[1-(2-phenylethyl)tetrazol-5-yl]propyl]-(thiophen-2-ylmethyl)amino]methyl]-1H-quinolin-2-one
—— 7,8-dimethyl-3-[[[(1R)-1-[1-(2-methylbutan-2-yl)tetrazol-5-yl]propyl]-[[(2S)-oxolan-2-yl]methyl]amino]methyl]-1H-quinolin-2-one —— C26H38N6O2
7,8-dimethyl-3-[[[(1R)-1-[1-(2-methylbutan-2-yl)tetrazol-5-yl]propyl]-[[(2S)-oxolan-2-yl]methyl]amino]methyl]-1H-quinolin-2-one
—— 7-[[(1-cyclopentyltetrazol-5-yl)methyl-(furan-2-ylmethyl)amino]methyl]-5H-[1,3]dioxolo[4,5-g]quinolin-6-one —— C23H24N6O4
7-[[(1-cyclopentyltetrazol-5-yl)methyl-(furan-2-ylmethyl)amino]methyl]-5H-[1,3]dioxolo[4,5-g]quinolin-6-one
—— 7,8-dimethyl-3-[[[(1S)-1-[1-(2-methylbutan-2-yl)tetrazol-5-yl]propyl]-(thiophen-2-ylmethyl)amino]methyl]-1H-quinolin-2-one —— C26H34N6OS
7,8-dimethyl-3-[[[(1S)-1-[1-(2-methylbutan-2-yl)tetrazol-5-yl]propyl]-(thiophen-2-ylmethyl)amino]methyl]-1H-quinolin-2-one
—— 7-methoxy-3-[[(4-methoxyphenyl)methyl-[(1R)-1-[1-(2-methylbutan-2-yl)tetrazol-5-yl]propyl]amino]methyl]-1H-quinolin-2-one —— C28H36N6O3
7-methoxy-3-[[(4-methoxyphenyl)methyl-[(1R)-1-[1-(2-methylbutan-2-yl)tetrazol-5-yl]propyl]amino]methyl]-1H-quinolin-2-one
—— 7-methoxy-3-[[[(1S)-1-[1-[(4-methoxyphenyl)methyl]tetrazol-5-yl]propyl]-(thiophen-2-ylmethyl)amino]methyl]-1H-quinolin-2-one —— C28H30N6O3S
7-methoxy-3-[[[(1S)-1-[1-[(4-methoxyphenyl)methyl]tetrazol-5-yl]propyl]-(thiophen-2-ylmethyl)amino]methyl]-1H-quinolin-2-one
—— 7-methyl-3-[[[(1R)-1-[1-(2-phenylethyl)tetrazol-5-yl]propyl]-(thiophen-2-ylmethyl)amino]methyl]-1H-quinolin-2-one —— C28H30N6OS
7-methyl-3-[[[(1R)-1-[1-(2-phenylethyl)tetrazol-5-yl]propyl]-(thiophen-2-ylmethyl)amino]methyl]-1H-quinolin-2-one
—— 7-methoxy-3-[[[(1R)-1-[1-(2-phenylethyl)tetrazol-5-yl]propyl]-(thiophen-2-ylmethyl)amino]methyl]-1H-quinolin-2-one —— C28H30N6O2S
7-methoxy-3-[[[(1R)-1-[1-(2-phenylethyl)tetrazol-5-yl]propyl]-(thiophen-2-ylmethyl)amino]methyl]-1H-quinolin-2-one
—— 7-methoxy-3-[[(4-methoxyphenyl)methyl-[(1S)-1-[1-(2-phenylethyl)tetrazol-5-yl]propyl]amino]methyl]-1H-quinolin-2-one —— C31H34N6O3
7-methoxy-3-[[(4-methoxyphenyl)methyl-[(1S)-1-[1-(2-phenylethyl)tetrazol-5-yl]propyl]amino]methyl]-1H-quinolin-2-one
—— 7-methoxy-3-[[(4-methoxyphenyl)methyl-[(1R)-1-[1-(2-phenylethyl)tetrazol-5-yl]propyl]amino]methyl]-1H-quinolin-2-one —— C31H34N6O3
7-methoxy-3-[[(4-methoxyphenyl)methyl-[(1R)-1-[1-(2-phenylethyl)tetrazol-5-yl]propyl]amino]methyl]-1H-quinolin-2-one
—— 7-methoxy-3-[[[(1S)-1-[1-(2-phenylethyl)tetrazol-5-yl]propyl]-(thiophen-2-ylmethyl)amino]methyl]-1H-quinolin-2-one —— C28H30N6O2S
7-methoxy-3-[[[(1S)-1-[1-(2-phenylethyl)tetrazol-5-yl]propyl]-(thiophen-2-ylmethyl)amino]methyl]-1H-quinolin-2-one
—— 7-methoxy-3-[[2-phenylethyl-[(1S)-1-[1-(2-phenylethyl)tetrazol-5-yl]propyl]amino]methyl]-1H-quinolin-2-one —— C31H34N6O2
7-methoxy-3-[[2-phenylethyl-[(1S)-1-[1-(2-phenylethyl)tetrazol-5-yl]propyl]amino]methyl]-1H-quinolin-2-one
—— 7-methoxy-3-[[(4-methoxyphenyl)methyl-[(1S)-1-[1-(2-methylbutan-2-yl)tetrazol-5-yl]propyl]amino]methyl]-1H-quinolin-2-one —— C28H36N6O3
7-methoxy-3-[[(4-methoxyphenyl)methyl-[(1S)-1-[1-(2-methylbutan-2-yl)tetrazol-5-yl]propyl]amino]methyl]-1H-quinolin-2-one
—— 7-methyl-3-[[[(1S)-1-[1-(2-methylbutan-2-yl)tetrazol-5-yl]propyl]-(thiophen-2-ylmethyl)amino]methyl]-1H-quinolin-2-one —— C25H32N6OS
7-methyl-3-[[[(1S)-1-[1-(2-methylbutan-2-yl)tetrazol-5-yl]propyl]-(thiophen-2-ylmethyl)amino]methyl]-1H-quinolin-2-one
—— 7-methoxy-3-[[[(1S)-1-[1-(2-methylbutan-2-yl)tetrazol-5-yl]propyl]-(thiophen-2-ylmethyl)amino]methyl]-1H-quinolin-2-one —— C25H32N6O2S
7-methoxy-3-[[[(1S)-1-[1-(2-methylbutan-2-yl)tetrazol-5-yl]propyl]-(thiophen-2-ylmethyl)amino]methyl]-1H-quinolin-2-one
—— 7-methoxy-3-[[2-phenylethyl-[(1R)-1-[1-(2-phenylethyl)tetrazol-5-yl]propyl]amino]methyl]-1H-quinolin-2-one —— C31H34N6O2
7-methoxy-3-[[2-phenylethyl-[(1R)-1-[1-(2-phenylethyl)tetrazol-5-yl]propyl]amino]methyl]-1H-quinolin-2-one
—— 7-methyl-3-[[(4-methylphenyl)methyl-[[1-[[(2S)-oxolan-2-yl]methyl]tetrazol-5-yl]methyl]amino]methyl]-1H-quinolin-2-one —— C26H30N6O2
7-methyl-3-[[(4-methylphenyl)methyl-[[1-[[(2S)-oxolan-2-yl]methyl]tetrazol-5-yl]methyl]amino]methyl]-1H-quinolin-2-one
—— 7,8-dimethyl-3-[[[1-(2-phenylethyl)tetrazol-5-yl]methyl-(thiophen-2-ylmethyl)amino]methyl]-1H-quinolin-2-one —— C27H28N6OS
7,8-dimethyl-3-[[[1-(2-phenylethyl)tetrazol-5-yl]methyl-(thiophen-2-ylmethyl)amino]methyl]-1H-quinolin-2-one
—— 7-methoxy-3-[[(4-methylphenyl)methyl-[[1-(2-phenylethyl)tetrazol-5-yl]methyl]amino]methyl]-1H-quinolin-2-one —— C29H30N6O2
7-methoxy-3-[[(4-methylphenyl)methyl-[[1-(2-phenylethyl)tetrazol-5-yl]methyl]amino]methyl]-1H-quinolin-2-one
—— 7-methoxy-3-[[(4-methoxyphenyl)methyl-[[1-(2-phenylethyl)tetrazol-5-yl]methyl]amino]methyl]-1H-quinolin-2-one —— C29H30N6O3
7-methoxy-3-[[(4-methoxyphenyl)methyl-[[1-(2-phenylethyl)tetrazol-5-yl]methyl]amino]methyl]-1H-quinolin-2-one
—— 7-methyl-3-[[(4-methylphenyl)methyl-[[1-(2-phenylethyl)tetrazol-5-yl]methyl]amino]methyl]-1H-quinolin-2-one —— C29H30N6O
7-methyl-3-[[(4-methylphenyl)methyl-[[1-(2-phenylethyl)tetrazol-5-yl]methyl]amino]methyl]-1H-quinolin-2-one
—— 7-methyl-3-[[[1-(2-methylbutan-2-yl)tetrazol-5-yl]methyl-[(4-methylphenyl)methyl]amino]methyl]-1H-quinolin-2-one —— C26H32N6O
7-methyl-3-[[[1-(2-methylbutan-2-yl)tetrazol-5-yl]methyl-[(4-methylphenyl)methyl]amino]methyl]-1H-quinolin-2-one
—— 7-methyl-3-[[2-phenylethyl-[[1-(2-phenylethyl)tetrazol-5-yl]methyl]amino]methyl]-1H-quinolin-2-one —— C29H30N6O
7-methyl-3-[[2-phenylethyl-[[1-(2-phenylethyl)tetrazol-5-yl]methyl]amino]methyl]-1H-quinolin-2-one
—— 7-methyl-3-[[(4-methylphenyl)methyl-[[1-[[(2R)-oxolan-2-yl]methyl]tetrazol-5-yl]methyl]amino]methyl]-1H-quinolin-2-one —— C26H30N6O2
7-methyl-3-[[(4-methylphenyl)methyl-[[1-[[(2R)-oxolan-2-yl]methyl]tetrazol-5-yl]methyl]amino]methyl]-1H-quinolin-2-one
—— 7-methoxy-3-[[[1-(2-phenylethyl)tetrazol-5-yl]methyl-(pyridin-3-ylmethyl)amino]methyl]-1H-quinolin-2-one —— C27H27N7O2
7-methoxy-3-[[[1-(2-phenylethyl)tetrazol-5-yl]methyl-(pyridin-3-ylmethyl)amino]methyl]-1H-quinolin-2-one
—— 7-methoxy-3-[[[1-[(4-methoxyphenyl)methyl]tetrazol-5-yl]methyl-[(4-methylphenyl)methyl]amino]methyl]-1H-quinolin-2-one —— C29H30N6O3
7-methoxy-3-[[[1-[(4-methoxyphenyl)methyl]tetrazol-5-yl]methyl-[(4-methylphenyl)methyl]amino]methyl]-1H-quinolin-2-one
—— 7,8-dimethyl-3-[[[1-(2-phenylethyl)tetrazol-5-yl]methyl-(pyridin-3-ylmethyl)amino]methyl]-1H-quinolin-2-one —— C28H29N7O
7,8-dimethyl-3-[[[1-(2-phenylethyl)tetrazol-5-yl]methyl-(pyridin-3-ylmethyl)amino]methyl]-1H-quinolin-2-one
—— 7-methoxy-3-[[(2-methoxyphenyl)methyl-[[1-(2-phenylethyl)tetrazol-5-yl]methyl]amino]methyl]-1H-quinolin-2-one —— C29H30N6O3
7-methoxy-3-[[(2-methoxyphenyl)methyl-[[1-(2-phenylethyl)tetrazol-5-yl]methyl]amino]methyl]-1H-quinolin-2-one
—— 7-methyl-3-[[[1-(2-phenylethyl)tetrazol-5-yl]methyl-(thiophen-2-ylmethyl)amino]methyl]-1H-quinolin-2-one —— C26H26N6OS
7-methyl-3-[[[1-(2-phenylethyl)tetrazol-5-yl]methyl-(thiophen-2-ylmethyl)amino]methyl]-1H-quinolin-2-one
—— 7-methoxy-3-[[2-phenylethyl-[[1-(2-phenylethyl)tetrazol-5-yl]methyl]amino]methyl]-1H-quinolin-2-one —— C29H30N6O2
7-methoxy-3-[[2-phenylethyl-[[1-(2-phenylethyl)tetrazol-5-yl]methyl]amino]methyl]-1H-quinolin-2-one
—— 7-methoxy-3-[[[1-(2-phenylethyl)tetrazol-5-yl]methyl-(thiophen-2-ylmethyl)amino]methyl]-1H-quinolin-2-one —— C26H26N6O2S
7-methoxy-3-[[[1-(2-phenylethyl)tetrazol-5-yl]methyl-(thiophen-2-ylmethyl)amino]methyl]-1H-quinolin-2-one
—— 7-methoxy-3-[[[1-(2-methylbutan-2-yl)tetrazol-5-yl]methyl-[(4-methylphenyl)methyl]amino]methyl]-1H-quinolin-2-one —— C26H32N6O2
7-methoxy-3-[[[1-(2-methylbutan-2-yl)tetrazol-5-yl]methyl-[(4-methylphenyl)methyl]amino]methyl]-1H-quinolin-2-one
—— 7-Methyl-5-(pyridin-2-ylmethylsulfanyl)-10-thia-3,4,6,8-tetrazatetracyclo[7.7.0.02,6.011,16]hexadeca-1(9),2,4,7,11(16)-pentaene —— C18H17N5S2
7-Methyl-5-(pyridin-2-ylmethylsulfanyl)-10-thia-3,4,6,8-tetrazatetracyclo[7.7.0.02,6.011,16]hexadeca-1(9),2,4,7,11(16)-pentaene
—— 7-[(2S)-2-methylpiperidin-1-yl]-3-(4-nitrophenyl)-[1,2]thiazolo[4,5-d]pyrimidine —— C17H17N5O2S
7-[(2S)-2-methylpiperidin-1-yl]-3-(4-nitrophenyl)-[1,2]thiazolo[4,5-d]pyrimidine
—— 7-[4-(3-Fluorophenyl)sulfonylpiperazin-1-yl]-3-(4-methoxyphenyl)-[1,2]thiazolo[4,5-d]pyrimidine —— C22H20FN5O3S2
7-[4-(3-Fluorophenyl)sulfonylpiperazin-1-yl]-3-(4-methoxyphenyl)-[1,2]thiazolo[4,5-d]pyrimidine
—— 7-(4-Ethylpiperazin-1-yl)-3-phenyl-[1,2]thiazolo[4,5-d]pyrimidine —— C17H19N5S
7-(4-Ethylpiperazin-1-yl)-3-phenyl-[1,2]thiazolo[4,5-d]pyrimidine
—— 7-(4-Benzylpiperazin-1-yl)-3-(4-chlorophenyl)-[1,2]thiazolo[4,5-d]pyrimidine —— C22H20ClN5S
7-(4-Benzylpiperazin-1-yl)-3-(4-chlorophenyl)-[1,2]thiazolo[4,5-d]pyrimidine
—— 7-(4-Benzylpiperazin-1-yl)-3-phenyl-[1,2]thiazolo[4,5-d]pyrimidine —— C22H21N5S
7-(4-Benzylpiperazin-1-yl)-3-phenyl-[1,2]thiazolo[4,5-d]pyrimidine
—— 7-[4-(4-Fluorophenyl)piperazin-1-yl]-3-phenyl-[1,2]thiazolo[4,5-d]pyrimidine —— C21H18FN5S
7-[4-(4-Fluorophenyl)piperazin-1-yl]-3-phenyl-[1,2]thiazolo[4,5-d]pyrimidine
—— 7-(Azepan-1-yl)-3-(4-methoxyphenyl)-[1,2]thiazolo[4,5-d]pyrimidine —— C18H20N4OS
7-(Azepan-1-yl)-3-(4-methoxyphenyl)-[1,2]thiazolo[4,5-d]pyrimidine
—— 7-[4-(2-Fluoro-benzenesulfonyl)-piperazin-1-yl]-3-(4-methoxy-phenyl)-isothiazolo[4,5-d]pyrimidine —— C22H20FN5O3S2
7-[4-(2-Fluoro-benzenesulfonyl)-piperazin-1-yl]-3-(4-methoxy-phenyl)-isothiazolo[4,5-d]pyrimidine