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—— (7R)-N-benzyl-7-(3-bromophenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C20H18BrN5O
(7R)-N-benzyl-7-(3-bromophenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— 7-[(S)-[4-(difluoromethoxy)phenyl]-(pyridin-2-ylamino)methyl]quinolin-8-ol —— C22H17F2N3O2
7-[(S)-[4-(difluoromethoxy)phenyl]-(pyridin-2-ylamino)methyl]quinolin-8-ol
—— (7S)-N-benzyl-5-methyl-7-(4-methylsulfanylphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C21H21N5OS
(7S)-N-benzyl-5-methyl-7-(4-methylsulfanylphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-N-benzyl-5-methyl-7-(4-methylsulfanylphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C21H21N5OS
(7R)-N-benzyl-5-methyl-7-(4-methylsulfanylphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— 7-methyl-2-oxo-4-propyl-2H-chromen-5-yl 3-methoxybenzoate —— C21H20O5
7-methyl-2-oxo-4-propyl-2H-chromen-5-yl 3-methoxybenzoate
—— (7S)-7-methyl-4-[3-(trifluoromethyl)phenoxy]-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidine —— C18H15F3N2OS
(7S)-7-methyl-4-[3-(trifluoromethyl)phenoxy]-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidine
—— 7-[(R)-(2-fluorophenyl)-[(4-methylpyridin-2-yl)amino]methyl]quinolin-8-ol —— C22H18FN3O
7-[(R)-(2-fluorophenyl)-[(4-methylpyridin-2-yl)amino]methyl]quinolin-8-ol
—— (7S)-5-(3-bromophenyl)-7-phenyl-1,7-dihydrotetrazolo[1,5-a]pyrimidine —— C16H12BrN5
(7S)-5-(3-bromophenyl)-7-phenyl-1,7-dihydrotetrazolo[1,5-a]pyrimidine
—— 7-[(S)-(2-fluorophenyl)-[(4-methylpyridin-2-yl)amino]methyl]quinolin-8-ol —— C22H18FN3O
7-[(S)-(2-fluorophenyl)-[(4-methylpyridin-2-yl)amino]methyl]quinolin-8-ol
—— 7-[(R)-(4-hydroxyphenyl)-[(4-methylpyridin-1-ium-2-yl)amino]methyl]quinolin-8-olate —— C22H19N3O2
7-[(R)-(4-hydroxyphenyl)-[(4-methylpyridin-1-ium-2-yl)amino]methyl]quinolin-8-olate
—— 7-bromo-2-{[1-(4-nitrophenyl)-1H-pyrrol-2-yl]methylene}[1,3]thiazolo[2',3':2,3]imidazo[4,5-b]pyridin-3(2H)-one —— C19H10BrN5O3S
7-bromo-2-{[1-(4-nitrophenyl)-1H-pyrrol-2-yl]methylene}[1,3]thiazolo[2',3':2,3]imidazo[4,5-b]pyridin-3(2H)-one
—— 7-[(S)-(4-hydroxyphenyl)-[(4-methylpyridin-1-ium-2-yl)amino]methyl]quinolin-8-olate —— C22H19N3O2
7-[(S)-(4-hydroxyphenyl)-[(4-methylpyridin-1-ium-2-yl)amino]methyl]quinolin-8-olate
—— 7-[(R)-(4-chlorophenyl)-[(4-methylpyridin-2-yl)amino]methyl]quinolin-8-ol —— C22H18ClN3O
7-[(R)-(4-chlorophenyl)-[(4-methylpyridin-2-yl)amino]methyl]quinolin-8-ol
—— (7R)-5-(3-bromophenyl)-7-phenyl-1,7-dihydrotetrazolo[1,5-a]pyrimidine —— C16H12BrN5
(7R)-5-(3-bromophenyl)-7-phenyl-1,7-dihydrotetrazolo[1,5-a]pyrimidine
—— 7-[(R)-[4-(difluoromethoxy)phenyl]-(pyridin-2-ylamino)methyl]quinolin-8-ol —— C22H17F2N3O2
7-[(R)-[4-(difluoromethoxy)phenyl]-(pyridin-2-ylamino)methyl]quinolin-8-ol
—— 7-((6,7-dihydro-5H-cyclopenta[4,5]thieno[2,3-d]pyrimidin-4-yl)oxy)-4-methyl-2H-chromen-2-one —— C19H14N2O3S
7-((6,7-dihydro-5H-cyclopenta[4,5]thieno[2,3-d]pyrimidin-4-yl)oxy)-4-methyl-2H-chromen-2-one
—— 7-[(S)-(4-chlorophenyl)-[(4-methylpyridin-2-yl)amino]methyl]quinolin-8-ol —— C22H18ClN3O
7-[(S)-(4-chlorophenyl)-[(4-methylpyridin-2-yl)amino]methyl]quinolin-8-ol
—— 7-Methyl-8,10-dihydrospiro[naphtho[1,2-F]isoindole-9,1'-pyrrolidine] —— C21H22N+
7-Methyl-8,10-dihydrospiro[naphtho[1,2-F]isoindole-9,1'-pyrrolidine]
—— (7S)-3,7-dimethyl-2-[(3-methylquinoxalin-2-yl)methylsulfanyl]-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C22H22N4OS2
(7S)-3,7-dimethyl-2-[(3-methylquinoxalin-2-yl)methylsulfanyl]-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— (7R)-N-(4-chlorophenyl)-5-methyl-7-(4-methylsulfanylphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C20H18ClN5OS
(7R)-N-(4-chlorophenyl)-5-methyl-7-(4-methylsulfanylphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-3,7-dimethyl-2-[(3-methylquinoxalin-2-yl)methylsulfanyl]-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C22H22N4OS2
(7R)-3,7-dimethyl-2-[(3-methylquinoxalin-2-yl)methylsulfanyl]-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— (7S)-N-(4-chlorophenyl)-5-methyl-7-(4-methylsulfanylphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C20H18ClN5OS
(7S)-N-(4-chlorophenyl)-5-methyl-7-(4-methylsulfanylphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-N-benzyl-5-methyl-7-[2-(trifluoromethyl)phenyl]-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C21H18F3N5O
(7R)-N-benzyl-5-methyl-7-[2-(trifluoromethyl)phenyl]-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— 7-Amino-2-(phenoxymethyl)-3-phenylpyrazolo[1,5-a]pyrimidine-6-carbonitrile —— C20H15N5O
7-Amino-2-(phenoxymethyl)-3-phenylpyrazolo[1,5-a]pyrimidine-6-carbonitrile
—— 7-[chloro(difluoro)methyl]-N-[4-(morpholine-4-carbonyl)phenyl]-5-thiophen-2-ylpyrazolo[1,5-a]pyrimidine-2-carboxamide —— C23H18ClF2N5O3S
7-[chloro(difluoro)methyl]-N-[4-(morpholine-4-carbonyl)phenyl]-5-thiophen-2-ylpyrazolo[1,5-a]pyrimidine-2-carboxamide
—— (7S)-N-benzyl-5-methyl-7-[2-(trifluoromethyl)phenyl]-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C21H18F3N5O
(7S)-N-benzyl-5-methyl-7-[2-(trifluoromethyl)phenyl]-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-3,7-dimethyl-2-[(3-phenyl-1,2,4-oxadiazol-5-yl)methylsulfanyl]-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C21H20N4O2S2
(7R)-3,7-dimethyl-2-[(3-phenyl-1,2,4-oxadiazol-5-yl)methylsulfanyl]-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— (7S)-3,7-dimethyl-2-[(3-phenyl-1,2,4-oxadiazol-5-yl)methylsulfanyl]-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C21H20N4O2S2
(7S)-3,7-dimethyl-2-[(3-phenyl-1,2,4-oxadiazol-5-yl)methylsulfanyl]-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— [7-[Chloro(difluoro)methyl]-5-thiophen-2-ylpyrazolo[1,5-a]pyrimidin-2-yl]-piperidin-1-ylmethanone —— C17H15ClF2N4OS
[7-[Chloro(difluoro)methyl]-5-thiophen-2-ylpyrazolo[1,5-a]pyrimidin-2-yl]-piperidin-1-ylmethanone
—— 7-[Chloro(difluoro)methyl]-3-(4-chlorophenyl)-5-methylpyrazolo[1,5-a]pyrimidine —— C14H9Cl2F2N3
7-[Chloro(difluoro)methyl]-3-(4-chlorophenyl)-5-methylpyrazolo[1,5-a]pyrimidine
—— (7S)-N-(4-chloro-2,5-dimethoxyphenyl)-7-(2,4-dichlorophenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C21H18Cl3N5O3
(7S)-N-(4-chloro-2,5-dimethoxyphenyl)-7-(2,4-dichlorophenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-N-(4-chloro-2,5-dimethoxyphenyl)-7-(2,4-dichlorophenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C21H18Cl3N5O3
(7R)-N-(4-chloro-2,5-dimethoxyphenyl)-7-(2,4-dichlorophenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-N-(2,4-dimethoxyphenyl)-5-methyl-7-(4-phenylmethoxyphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C28H27N5O4
(7S)-N-(2,4-dimethoxyphenyl)-5-methyl-7-(4-phenylmethoxyphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-N-(2,4-dimethoxyphenyl)-5-methyl-7-(4-phenylmethoxyphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C28H27N5O4
(7R)-N-(2,4-dimethoxyphenyl)-5-methyl-7-(4-phenylmethoxyphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-5-[4-chloro-2-(difluoromethoxy)phenyl]-7-(2,3-dimethoxyphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine —— C20H17ClF2N4O3
(7S)-5-[4-chloro-2-(difluoromethoxy)phenyl]-7-(2,3-dimethoxyphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine
—— (7R)-5-(4-bromophenyl)-7-(2,4-dimethoxyphenyl)-1,7-dihydrotetrazolo[1,5-a]pyrimidine —— C18H16BrN5O2
(7R)-5-(4-bromophenyl)-7-(2,4-dimethoxyphenyl)-1,7-dihydrotetrazolo[1,5-a]pyrimidine
—— (7R)-5-[4-chloro-2-(difluoromethoxy)phenyl]-7-(2,3-dimethoxyphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine —— C20H17ClF2N4O3
(7R)-5-[4-chloro-2-(difluoromethoxy)phenyl]-7-(2,3-dimethoxyphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine
—— (7S)-5-(4-bromophenyl)-7-(2,4-dimethoxyphenyl)-1,7-dihydrotetrazolo[1,5-a]pyrimidine —— C18H16BrN5O2
(7S)-5-(4-bromophenyl)-7-(2,4-dimethoxyphenyl)-1,7-dihydrotetrazolo[1,5-a]pyrimidine
—— 7-[(4aS)-1,3,4,4a,5,6,7,8-octahydropyrrolo[1,2-c]pyrimidin-8-ium-2-yl]-1-ethyl-6-fluoro-4-oxoquinoline-3-carboxylate —— C19H22FN3O3
7-[(4aS)-1,3,4,4a,5,6,7,8-octahydropyrrolo[1,2-c]pyrimidin-8-ium-2-yl]-1-ethyl-6-fluoro-4-oxoquinoline-3-carboxylate
—— (7R)-N-(4-chloro-2,5-dimethoxyphenyl)-5-methyl-7-(4-methylsulfanylphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C22H22ClN5O3S
(7R)-N-(4-chloro-2,5-dimethoxyphenyl)-5-methyl-7-(4-methylsulfanylphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-N-(4-chloro-2,5-dimethoxyphenyl)-5-methyl-7-(4-methylsulfanylphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C22H22ClN5O3S
(7S)-N-(4-chloro-2,5-dimethoxyphenyl)-5-methyl-7-(4-methylsulfanylphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-N-(4-chloro-2,5-dimethoxyphenyl)-7-(3-fluorophenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C21H19ClFN5O3
(7R)-N-(4-chloro-2,5-dimethoxyphenyl)-7-(3-fluorophenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— 7-nitro-1H-imidazo[1,2-b]pyrazole —— C5H4N4O2
7-nitro-1H-imidazo[1,2-b]pyrazole
—— (7S)-5-(3,4-dimethylphenyl)-7-(4-fluorophenyl)-1,7-dihydrotetrazolo[1,5-a]pyrimidine —— C18H16FN5
(7S)-5-(3,4-dimethylphenyl)-7-(4-fluorophenyl)-1,7-dihydrotetrazolo[1,5-a]pyrimidine
—— 7-{4-[(2,3-Dihydro-1,4-benzodioxin-6-ylamino)carbothioyl]piperazino}-1-ethyl-6-fluoro-4-oxo-1,4-dihydro-3-quinolinecarboxylic acid —— C25H25FN4O5S
7-{4-[(2,3-Dihydro-1,4-benzodioxin-6-ylamino)carbothioyl]piperazino}-1-ethyl-6-fluoro-4-oxo-1,4-dihydro-3-quinolinecarboxylic acid
—— (7R)-5-(3,4-dimethylphenyl)-7-(4-fluorophenyl)-1,7-dihydrotetrazolo[1,5-a]pyrimidine —— C18H16FN5
(7R)-5-(3,4-dimethylphenyl)-7-(4-fluorophenyl)-1,7-dihydrotetrazolo[1,5-a]pyrimidine
—— (7R)-3-(4-hydroxyphenyl)-7-methyl-2H-[1,3]thiazolo[2,3-c][1,2,4]triazin-6-one —— C12H11N3O2S
(7R)-3-(4-hydroxyphenyl)-7-methyl-2H-[1,3]thiazolo[2,3-c][1,2,4]triazin-6-one
—— (7S)-3-(3,4-dihydroxyphenyl)-7-methyl-2H-[1,3]thiazolo[2,3-c][1,2,4]triazin-6-one —— C12H11N3O3S
(7S)-3-(3,4-dihydroxyphenyl)-7-methyl-2H-[1,3]thiazolo[2,3-c][1,2,4]triazin-6-one
—— (7S)-3-(2,6-dichlorophenyl)-7-methyl-2H-[1,3]thiazolo[2,3-c][1,2,4]triazin-6-one —— C12H9Cl2N3OS
(7S)-3-(2,6-dichlorophenyl)-7-methyl-2H-[1,3]thiazolo[2,3-c][1,2,4]triazin-6-one
—— 7,7-Dimethyl-2-(4-methylphenyl)-1-(2-phenylethyl)-5,8-dihydropyrano[4,3-d]pyrimidine-4-thione —— C24H26N2OS
7,7-Dimethyl-2-(4-methylphenyl)-1-(2-phenylethyl)-5,8-dihydropyrano[4,3-d]pyrimidine-4-thione