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中文名称 英文名称 CAS号 化学式 结构式图片
—— 7-methyl-1-[2-(2-methyl-1H-indol-3-yl)ethyl]-5,5-bis(trifluoromethyl)-5,8-dihydropyrimido[4,5-d]pyrimidine-2,4(1H,3H)-dione —— C20H17F6N5O2
7-methyl-1-[2-(2-methyl-1H-indol-3-yl)ethyl]-5,5-bis(trifluoromethyl)-5,8-dihydropyrimido[4,5-d]pyrimidine-2,4(1H,3H)-dione
—— 7-(difluoromethyl)-5-(4-methoxyphenyl)-N-[4-(piperidine-1-carbonyl)phenyl]pyrazolo[1,5-a]pyrimidine-3-carboxamide 492433-51-9 C27H25F2N5O3
7-(difluoromethyl)-5-(4-methoxyphenyl)-N-[4-(piperidine-1-carbonyl)phenyl]pyrazolo[1,5-a]pyrimidine-3-carboxamide
—— 7-Benzyl-1,3-dimethyl-8-{[(1H-1,2,3,4-tetrazol-5-YL)methyl]sulfanyl}-2,3,6,7-tetrahydro-1H-purine-2,6-dione —— C16H16N8O2S
7-Benzyl-1,3-dimethyl-8-{[(1H-1,2,3,4-tetrazol-5-YL)methyl]sulfanyl}-2,3,6,7-tetrahydro-1H-purine-2,6-dione
—— 7-(difluoromethyl)-5-(4-methoxyphenyl)-N-[4-(4-morpholinylcarbonyl)phenyl]pyrazolo[1,5-a]pyrimidine-3-carboxamide —— C26H23F2N5O4
7-(difluoromethyl)-5-(4-methoxyphenyl)-N-[4-(4-morpholinylcarbonyl)phenyl]pyrazolo[1,5-a]pyrimidine-3-carboxamide
—— 7-O-ethyl 2-O-methyl (6S)-8-methyl-4-oxo-6-(3,4,5-trimethoxyphenyl)-6H-pyrimido[2,1-b][1,3]thiazine-2,7-dicarboxylate —— C22H24N2O8S
7-O-ethyl 2-O-methyl (6S)-8-methyl-4-oxo-6-(3,4,5-trimethoxyphenyl)-6H-pyrimido[2,1-b][1,3]thiazine-2,7-dicarboxylate
—— 7-(difluoromethyl)-5-methyl-N-[3-nitro-5-(2,2,2-trifluoroethoxy)phenyl][1,2,4]triazolo[1,5-a]pyrimidine-2-carboxamide —— C16H11F5N6O4
7-(difluoromethyl)-5-methyl-N-[3-nitro-5-(2,2,2-trifluoroethoxy)phenyl][1,2,4]triazolo[1,5-a]pyrimidine-2-carboxamide
—— 7-[2-(4-Chlorophenyl)-2-oxoethyl]-1,3-dimethyl-8-(4-methylpiperazin-1-YL)-2,3,6,7-tetrahydro-1H-purine-2,6-dione —— C20H23ClN6O3
7-[2-(4-Chlorophenyl)-2-oxoethyl]-1,3-dimethyl-8-(4-methylpiperazin-1-YL)-2,3,6,7-tetrahydro-1H-purine-2,6-dione
—— 7-[(2-Fluorophenyl)methyl]-8-{[(3-methoxyphenyl)methyl]sulfanyl}-1,3-dimethyl-2,3,6,7-tetrahydro-1H-purine-2,6-dione —— C22H21FN4O3S
7-[(2-Fluorophenyl)methyl]-8-{[(3-methoxyphenyl)methyl]sulfanyl}-1,3-dimethyl-2,3,6,7-tetrahydro-1H-purine-2,6-dione
—— 7-(difluoromethyl)-N-[(2-fluorophenyl)methyl]-5-phenylpyrazolo[1,5-a]pyrimidine-3-carboxamide —— C21H15F3N4O
7-(difluoromethyl)-N-[(2-fluorophenyl)methyl]-5-phenylpyrazolo[1,5-a]pyrimidine-3-carboxamide
—— 7-[(2,4-Dichlorophenyl)methyl]-1,3-dimethyl-8-(2-morpholin-4-ylethylamino)purine-2,6-dione —— C20H24Cl2N6O3
7-[(2,4-Dichlorophenyl)methyl]-1,3-dimethyl-8-(2-morpholin-4-ylethylamino)purine-2,6-dione
—— 7-(Difluoromethyl)-N~3~-(4-ethylphenyl)-5-phenylpyrazolo[1,5-A]pyrimidine-3-carboxamide —— C22H18F2N4O
7-(Difluoromethyl)-N~3~-(4-ethylphenyl)-5-phenylpyrazolo[1,5-A]pyrimidine-3-carboxamide
—— 7-(4-Chlorophenyl)-8-cyclohexyl-1,3-dimethyl-1H,2H,3H,4H,8H-imidazo[1,2-G]purine-2,4-dione —— C21H22ClN5O2
7-(4-Chlorophenyl)-8-cyclohexyl-1,3-dimethyl-1H,2H,3H,4H,8H-imidazo[1,2-G]purine-2,4-dione
—— 7-(Difluoromethyl)-5-phenyl-N-[(thiophen-2-YL)methyl]pyrazolo[1,5-A]pyrimidine-3-carboxamide —— C19H14F2N4OS
7-(Difluoromethyl)-5-phenyl-N-[(thiophen-2-YL)methyl]pyrazolo[1,5-A]pyrimidine-3-carboxamide
—— 7-[(3-Bromophenyl)methyl]-8-{[2-(3,4-dimethoxyphenyl)ethyl]amino}-1,3-dimethyl-2,3,6,7-tetrahydro-1H-purine-2,6-dione —— C24H26BrN5O4
7-[(3-Bromophenyl)methyl]-8-{[2-(3,4-dimethoxyphenyl)ethyl]amino}-1,3-dimethyl-2,3,6,7-tetrahydro-1H-purine-2,6-dione
—— 7-(difluoromethyl)-N-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]-N-methyl-5-phenylpyrazolo[1,5-a]pyrimidine-3-carboxamide —— C22H22F2N6O
7-(difluoromethyl)-N-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]-N-methyl-5-phenylpyrazolo[1,5-a]pyrimidine-3-carboxamide
—— [7-(difluoromethyl)-5-phenylpyrazolo[1,5-a]pyrimidin-3-yl]-[(2R)-2-methyl-2,3-dihydroindol-1-yl]methanone —— C23H18F2N4O
[7-(difluoromethyl)-5-phenylpyrazolo[1,5-a]pyrimidin-3-yl]-[(2R)-2-methyl-2,3-dihydroindol-1-yl]methanone
—— 7-(4-bromobenzyl)-8-(3,4-dihydro-2(1H)-isoquinolinyl)-1,3-dimethyl-3,7-dihydro-1H-purine-2,6-dione —— C23H22BrN5O2
7-(4-bromobenzyl)-8-(3,4-dihydro-2(1H)-isoquinolinyl)-1,3-dimethyl-3,7-dihydro-1H-purine-2,6-dione
—— [7-(Difluoromethyl)-5-(4-methoxyphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]-(2-methylimidazol-1-yl)methanone —— C19H15F2N5O2
[7-(Difluoromethyl)-5-(4-methoxyphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]-(2-methylimidazol-1-yl)methanone
—— 7-(difluoromethyl)-N-(2-furylmethyl)-5-(4-methylphenyl)pyrazolo[1,5-a]pyrimidine-3-carboxamide —— C20H16F2N4O2
7-(difluoromethyl)-N-(2-furylmethyl)-5-(4-methylphenyl)pyrazolo[1,5-a]pyrimidine-3-carboxamide
—— 7-O-ethyl 2-O-methyl (6R)-8-methyl-4-oxo-6-(3,4,5-trimethoxyphenyl)-6H-pyrimido[2,1-b][1,3]thiazine-2,7-dicarboxylate —— C22H24N2O8S
7-O-ethyl 2-O-methyl (6R)-8-methyl-4-oxo-6-(3,4,5-trimethoxyphenyl)-6H-pyrimido[2,1-b][1,3]thiazine-2,7-dicarboxylate
—— 7-(4-Chlorophenyl)-8-[2-(3,4-diethoxyphenyl)ethyl]-1,3-dimethyl-1H,2H,3H,4H,8H-imidazo[1,2-G]purine-2,4-dione —— C27H28ClN5O4
7-(4-Chlorophenyl)-8-[2-(3,4-diethoxyphenyl)ethyl]-1,3-dimethyl-1H,2H,3H,4H,8H-imidazo[1,2-G]purine-2,4-dione
—— 7-(4-Chlorophenyl)-8-[2-(3,4-dimethoxyphenyl)ethyl]-1,3-dimethyl-1H,2H,3H,4H,8H-imidazo[1,2-G]purine-2,4-dione —— C25H24ClN5O4
7-(4-Chlorophenyl)-8-[2-(3,4-dimethoxyphenyl)ethyl]-1,3-dimethyl-1H,2H,3H,4H,8H-imidazo[1,2-G]purine-2,4-dione
—— 7-(4-Fluorophenyl)-1,3-dimethyl-8-(2-phenylethyl)-1H,2H,3H,4H,8H-imidazo[1,2-G]purine-2,4-dione —— C23H20FN5O2
7-(4-Fluorophenyl)-1,3-dimethyl-8-(2-phenylethyl)-1H,2H,3H,4H,8H-imidazo[1,2-G]purine-2,4-dione
—— 7-[(2-Chlorophenyl)methyl]-8-{[2-(3,4-dimethoxyphenyl)ethyl]amino}-1,3-dimethyl-2,3,6,7-tetrahydro-1H-purine-2,6-dione —— C24H26ClN5O4
7-[(2-Chlorophenyl)methyl]-8-{[2-(3,4-dimethoxyphenyl)ethyl]amino}-1,3-dimethyl-2,3,6,7-tetrahydro-1H-purine-2,6-dione
—— 7-(4-fluorophenyl)-1,3-dimethyl-8-propyl-1H,2H,3H,4H,8H-imidazo[1,2-g]purine-2,4-dione —— C18H18FN5O2
7-(4-fluorophenyl)-1,3-dimethyl-8-propyl-1H,2H,3H,4H,8H-imidazo[1,2-g]purine-2,4-dione
—— 7-(3-chlorobenzyl)-1,3-dimethyl-8-(4-methylphenoxy)-3,7-dihydro-1H-purine-2,6-dione —— C21H19ClN4O3
7-(3-chlorobenzyl)-1,3-dimethyl-8-(4-methylphenoxy)-3,7-dihydro-1H-purine-2,6-dione
—— (7R)-5-amino-7-[4-[3,3-bis(ethylamino)-2-oxopropoxy]-3-methoxyphenyl]-2-(trifluoromethyl)-1,7-dihydropyrano[2,3-d]imidazole-6-carbonitrile —— C22H25F3N6O4
(7R)-5-amino-7-[4-[3,3-bis(ethylamino)-2-oxopropoxy]-3-methoxyphenyl]-2-(trifluoromethyl)-1,7-dihydropyrano[2,3-d]imidazole-6-carbonitrile
—— (7S)-5-amino-7-(3-hydroxyphenyl)-2,4-diphenyl-7H-[1,3]oxazolo[5,4-b]pyridine-6-carbonitrile —— C25H18N4O2
(7S)-5-amino-7-(3-hydroxyphenyl)-2,4-diphenyl-7H-[1,3]oxazolo[5,4-b]pyridine-6-carbonitrile
—— (7S)-5-amino-2-methyl-4-phenyl-7-(4-propan-2-yloxyphenyl)-7H-[1,3]oxazolo[5,4-b]pyridine-6-carbonitrile —— C23H22N4O2
(7S)-5-amino-2-methyl-4-phenyl-7-(4-propan-2-yloxyphenyl)-7H-[1,3]oxazolo[5,4-b]pyridine-6-carbonitrile
—— (7S)-5-amino-7-(3-methoxy-4-propan-2-yloxyphenyl)-2-propyl-4,7-dihydro-[1,3]oxazolo[5,4-b]pyridine-6-carbonitrile —— C20H24N4O3
(7S)-5-amino-7-(3-methoxy-4-propan-2-yloxyphenyl)-2-propyl-4,7-dihydro-[1,3]oxazolo[5,4-b]pyridine-6-carbonitrile
—— (7S)-5-amino-2-methoxy-7-(3-methoxy-4-propan-2-yloxyphenyl)-1,7-dihydropyrano[2,3-d]imidazole-6-carbonitrile —— C18H20N4O4
(7S)-5-amino-2-methoxy-7-(3-methoxy-4-propan-2-yloxyphenyl)-1,7-dihydropyrano[2,3-d]imidazole-6-carbonitrile
—— (7R)-5-amino-2-methoxy-7-(3-methoxy-4-propan-2-yloxyphenyl)-1,7-dihydropyrano[2,3-d]imidazole-6-carbonitrile —— C18H20N4O4
(7R)-5-amino-2-methoxy-7-(3-methoxy-4-propan-2-yloxyphenyl)-1,7-dihydropyrano[2,3-d]imidazole-6-carbonitrile
—— (7S)-5-amino-7-[2-[(4-chlorophenoxy)methyl]phenyl]-2-(methoxymethyl)-1,7-dihydropyrano[2,3-d]imidazole-6-carbonitrile —— C22H19ClN4O3
(7S)-5-amino-7-[2-[(4-chlorophenoxy)methyl]phenyl]-2-(methoxymethyl)-1,7-dihydropyrano[2,3-d]imidazole-6-carbonitrile
—— (7R)-5-amino-7-[2-[(4-chlorophenoxy)methyl]phenyl]-2-(methoxymethyl)-1,7-dihydropyrano[2,3-d]imidazole-6-carbonitrile —— C22H19ClN4O3
(7R)-5-amino-7-[2-[(4-chlorophenoxy)methyl]phenyl]-2-(methoxymethyl)-1,7-dihydropyrano[2,3-d]imidazole-6-carbonitrile
—— (7S)-5-amino-7-[4-[3,3-bis(ethylamino)-2-oxopropoxy]-3-methoxyphenyl]-2-(trifluoromethyl)-1,7-dihydropyrano[2,3-d]imidazole-6-carbonitrile —— C22H25F3N6O4
(7S)-5-amino-7-[4-[3,3-bis(ethylamino)-2-oxopropoxy]-3-methoxyphenyl]-2-(trifluoromethyl)-1,7-dihydropyrano[2,3-d]imidazole-6-carbonitrile
—— (7R)-5-amino-2-methyl-4-phenyl-7-(4-propan-2-yloxyphenyl)-7H-[1,3]oxazolo[5,4-b]pyridine-6-carbonitrile —— C23H22N4O2
(7R)-5-amino-2-methyl-4-phenyl-7-(4-propan-2-yloxyphenyl)-7H-[1,3]oxazolo[5,4-b]pyridine-6-carbonitrile
—— 7-[(3-Fluorophenyl)methyl]-1,3-dimethyl-8-{[2-(morpholin-4-YL)ethyl]amino}-2,3,6,7-tetrahydro-1H-purine-2,6-dione —— C20H25FN6O3
7-[(3-Fluorophenyl)methyl]-1,3-dimethyl-8-{[2-(morpholin-4-YL)ethyl]amino}-2,3,6,7-tetrahydro-1H-purine-2,6-dione
—— 7-benzyl-2-(3-methoxyphenoxy)-1-methyl-1,7-dihydro-6H-purin-6-one —— C20H18N4O3
7-benzyl-2-(3-methoxyphenoxy)-1-methyl-1,7-dihydro-6H-purin-6-one
—— 7-(4-Bromophenyl)-8-[(furan-2-YL)methyl]-1,3-dimethyl-1H,2H,3H,4H,8H-imidazo[1,2-G]purine-2,4-dione —— C20H16BrN5O3
7-(4-Bromophenyl)-8-[(furan-2-YL)methyl]-1,3-dimethyl-1H,2H,3H,4H,8H-imidazo[1,2-G]purine-2,4-dione
—— 7-(difluoromethyl)-5-(4-methylphenyl)-N-pyridin-3-ylpyrazolo[1,5-a]pyrimidine-3-carboxamide —— C20H15F2N5O
7-(difluoromethyl)-5-(4-methylphenyl)-N-pyridin-3-ylpyrazolo[1,5-a]pyrimidine-3-carboxamide
—— (7R)-7-phenyl-4-pyrrolidin-1-yl-6,8-dihydro-5H-[1]benzothiolo[2,3-d]pyrimidine-7-carbonitrile —— C21H20N4S
(7R)-7-phenyl-4-pyrrolidin-1-yl-6,8-dihydro-5H-[1]benzothiolo[2,3-d]pyrimidine-7-carbonitrile
—— 7-benzyl-8-[(3S,5S)-3,5-dimethylpiperidin-1-yl]-1,3-dimethylpurine-2,6-dione —— C21H27N5O2
7-benzyl-8-[(3S,5S)-3,5-dimethylpiperidin-1-yl]-1,3-dimethylpurine-2,6-dione
—— 7-[(2-Chloro-6-fluorophenyl)methyl]-8-[2-(dimethylamino)ethylamino]-1,3-dimethylpurine-2,6-dione —— C18H22ClFN6O2
7-[(2-Chloro-6-fluorophenyl)methyl]-8-[2-(dimethylamino)ethylamino]-1,3-dimethylpurine-2,6-dione
—— 7-(2-chloro-5-methoxybenzyl)-1,3-dimethyl-8-[(2-pyridinylmethyl)amino]-3,7-dihydro-1H-purine-2,6-dione —— C21H21ClN6O3
7-(2-chloro-5-methoxybenzyl)-1,3-dimethyl-8-[(2-pyridinylmethyl)amino]-3,7-dihydro-1H-purine-2,6-dione
—— (7R)-2-methyl-3,5,7-triphenyl-6,7-dihydropyrazolo[1,5-a]pyrimidine —— C25H21N3
(7R)-2-methyl-3,5,7-triphenyl-6,7-dihydropyrazolo[1,5-a]pyrimidine
—— 7-(2-chloro-6-fluorobenzyl)-8-{[2-(1-cyclohexen-1-yl)ethyl]amino}-1,3-dimethyl-3,7-dihydro-1H-purine-2,6-dione —— C22H25ClFN5O2
7-(2-chloro-6-fluorobenzyl)-8-{[2-(1-cyclohexen-1-yl)ethyl]amino}-1,3-dimethyl-3,7-dihydro-1H-purine-2,6-dione
—— 7-benzyl-8-[(3R,5R)-3,5-dimethylpiperidin-1-yl]-1,3-dimethylpurine-2,6-dione —— C21H27N5O2
7-benzyl-8-[(3R,5R)-3,5-dimethylpiperidin-1-yl]-1,3-dimethylpurine-2,6-dione
—— (7S)-2-methyl-3,5,7-triphenyl-6,7-dihydropyrazolo[1,5-a]pyrimidine —— C25H21N3
(7S)-2-methyl-3,5,7-triphenyl-6,7-dihydropyrazolo[1,5-a]pyrimidine
—— 7-(1,3-Dimethylpyrazol-4-yl)pyrazolo[1,5-a]pyrimidine-2-carboxylic acid —— C12H11N5O2
7-(1,3-Dimethylpyrazol-4-yl)pyrazolo[1,5-a]pyrimidine-2-carboxylic acid
—— 7-benzyl-8-[(3R,5S)-3,5-dimethylpiperidin-1-yl]-1,3-dimethylpurine-2,6-dione —— C21H27N5O2
7-benzyl-8-[(3R,5S)-3,5-dimethylpiperidin-1-yl]-1,3-dimethylpurine-2,6-dione