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—— (5R)-4-[(4-butoxy-3-methylphenyl)-hydroxymethylidene]-5-(4-ethylphenyl)-1-(2-methoxyethyl)pyrrolidine-2,3-dione —— C27H33NO5
(5R)-4-[(4-butoxy-3-methylphenyl)-hydroxymethylidene]-5-(4-ethylphenyl)-1-(2-methoxyethyl)pyrrolidine-2,3-dione
—— 5-methyl-3-phenyl-N-[[(1S,5R)-1,3,3-trimethyl-5-[(5-methyl-3-phenyl-1,2-oxazole-4-carbonyl)amino]cyclohexyl]methyl]-1,2-oxazole-4-carboxamide —— C32H36N4O4
5-methyl-3-phenyl-N-[[(1S,5R)-1,3,3-trimethyl-5-[(5-methyl-3-phenyl-1,2-oxazole-4-carbonyl)amino]cyclohexyl]methyl]-1,2-oxazole-4-carboxamide
—— (5R)-4-[(4-butoxy-2-methylphenyl)-hydroxymethylidene]-5-(4-methylphenyl)-1-(3-morpholin-4-ylpropyl)pyrrolidine-2,3-dione —— C30H38N2O5
(5R)-4-[(4-butoxy-2-methylphenyl)-hydroxymethylidene]-5-(4-methylphenyl)-1-(3-morpholin-4-ylpropyl)pyrrolidine-2,3-dione
—— 5-[[(4R)-4-ethyl-6,7-dihydro-4H-thieno[3,2-c]pyridin-5-yl]methyl]-3-(3-fluoro-4-methylphenyl)-1,2,4-oxadiazole —— C19H20FN3OS
5-[[(4R)-4-ethyl-6,7-dihydro-4H-thieno[3,2-c]pyridin-5-yl]methyl]-3-(3-fluoro-4-methylphenyl)-1,2,4-oxadiazole
—— 5-[[5-[(3R,5S)-3,5-dimethylpiperidin-1-yl]-4-(furan-2-ylmethyl)-1,2,4-triazol-3-yl]sulfanylmethyl]-3-thiophen-3-yl-1,2,4-oxadiazole —— C21H24N6O2S2
5-[[5-[(3R,5S)-3,5-dimethylpiperidin-1-yl]-4-(furan-2-ylmethyl)-1,2,4-triazol-3-yl]sulfanylmethyl]-3-thiophen-3-yl-1,2,4-oxadiazole
—— 5-[[(2S)-2-(2,4-dimethoxyphenyl)pyrrolidin-1-yl]methyl]-3-(3-fluoro-4-methylphenyl)-1,2,4-oxadiazole —— C22H24FN3O3
5-[[(2S)-2-(2,4-dimethoxyphenyl)pyrrolidin-1-yl]methyl]-3-(3-fluoro-4-methylphenyl)-1,2,4-oxadiazole
—— (5S)-5-(4-bromophenyl)-4-[hydroxy-(3-methyl-4-propoxyphenyl)methylidene]-1-(2-morpholin-4-ylethyl)pyrrolidine-2,3-dione —— C27H31BrN2O5
(5S)-5-(4-bromophenyl)-4-[hydroxy-(3-methyl-4-propoxyphenyl)methylidene]-1-(2-morpholin-4-ylethyl)pyrrolidine-2,3-dione
—— (5S)-4-[hydroxy-(4-methylphenyl)methylidene]-1-(2-methoxyethyl)-5-(3-phenoxyphenyl)pyrrolidine-2,3-dione —— C27H25NO5
(5S)-4-[hydroxy-(4-methylphenyl)methylidene]-1-(2-methoxyethyl)-5-(3-phenoxyphenyl)pyrrolidine-2,3-dione
—— (5R)-5-(4-tert-butylphenyl)-4-[hydroxy-(3-methyl-4-phenylmethoxyphenyl)methylidene]-1-(3-morpholin-4-ylpropyl)pyrrolidine-2,3-dione —— C36H42N2O5
(5R)-5-(4-tert-butylphenyl)-4-[hydroxy-(3-methyl-4-phenylmethoxyphenyl)methylidene]-1-(3-morpholin-4-ylpropyl)pyrrolidine-2,3-dione
—— (5S)-5-(4-chlorophenyl)-4-[hydroxy-(3-methyl-4-prop-2-enoxyphenyl)methylidene]-1-(2-morpholin-4-ium-4-ylethyl)pyrrolidine-2,3-dione —— C27H30ClN2O5+
(5S)-5-(4-chlorophenyl)-4-[hydroxy-(3-methyl-4-prop-2-enoxyphenyl)methylidene]-1-(2-morpholin-4-ium-4-ylethyl)pyrrolidine-2,3-dione
—— 5-(2-methoxyethyl)-N-(2-methylpropyl)-6,6-dioxo-4H-imidazo[5,1-d][1,2,5]benzothiadiazepine-3-carboxamide —— C18H24N4O4S
5-(2-methoxyethyl)-N-(2-methylpropyl)-6,6-dioxo-4H-imidazo[5,1-d][1,2,5]benzothiadiazepine-3-carboxamide
—— 5-[2-(4-Chlorophenyl)-2-oxoethyl]sulfanyl-4-(4-methoxyphenyl)-11-propyl-8-thia-4,6-diaza-11-azoniatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one —— C27H27ClN3O3S2+
5-[2-(4-Chlorophenyl)-2-oxoethyl]sulfanyl-4-(4-methoxyphenyl)-11-propyl-8-thia-4,6-diaza-11-azoniatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
—— 5-[[5-[(3R,5R)-3,5-dimethylpiperidin-1-yl]-4-(furan-2-ylmethyl)-1,2,4-triazol-3-yl]sulfanylmethyl]-3-thiophen-3-yl-1,2,4-oxadiazole —— C21H24N6O2S2
5-[[5-[(3R,5R)-3,5-dimethylpiperidin-1-yl]-4-(furan-2-ylmethyl)-1,2,4-triazol-3-yl]sulfanylmethyl]-3-thiophen-3-yl-1,2,4-oxadiazole
—— (5R)-4-[(4-chlorophenyl)-hydroxymethylidene]-5-(3,4-dichlorophenyl)-1-(3-methoxypropyl)pyrrolidine-2,3-dione —— C21H18Cl3NO4
(5R)-4-[(4-chlorophenyl)-hydroxymethylidene]-5-(3,4-dichlorophenyl)-1-(3-methoxypropyl)pyrrolidine-2,3-dione
—— (5S)-4-[hydroxy-(3-methyl-4-phenylmethoxyphenyl)methylidene]-1-(3-morpholin-4-ium-4-ylpropyl)-5-(3-phenoxyphenyl)pyrrolidine-2,3-dione —— C38H39N2O6+
(5S)-4-[hydroxy-(3-methyl-4-phenylmethoxyphenyl)methylidene]-1-(3-morpholin-4-ium-4-ylpropyl)-5-(3-phenoxyphenyl)pyrrolidine-2,3-dione
—— 5-[2-(4-Chlorophenyl)-2-oxoethyl]sulfanyl-4-phenyl-11-propyl-8-thia-4,6-diaza-11-azoniatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one —— C26H25ClN3O2S2+
5-[2-(4-Chlorophenyl)-2-oxoethyl]sulfanyl-4-phenyl-11-propyl-8-thia-4,6-diaza-11-azoniatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
—— 5-(4-bromophenyl)-N-[(6R)-6-tert-butyl-3-cyano-4,5,6,7-tetrahydro-1-benzothiophen-2-yl]-3-chloro-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidine-2-carboxamide —— C27H22BrClF3N5OS
5-(4-bromophenyl)-N-[(6R)-6-tert-butyl-3-cyano-4,5,6,7-tetrahydro-1-benzothiophen-2-yl]-3-chloro-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidine-2-carboxamide
—— (5S,10bS)-2-(4-bromophenyl)-5-[4-(difluoromethoxy)phenyl]-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine —— C23H17BrF2N2O2
(5S,10bS)-2-(4-bromophenyl)-5-[4-(difluoromethoxy)phenyl]-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine
—— 5-[[5-[(3S,5S)-3,5-dimethylpiperidin-1-yl]-4-(furan-2-ylmethyl)-1,2,4-triazol-3-yl]sulfanylmethyl]-3-thiophen-3-yl-1,2,4-oxadiazole —— C21H24N6O2S2
5-[[5-[(3S,5S)-3,5-dimethylpiperidin-1-yl]-4-(furan-2-ylmethyl)-1,2,4-triazol-3-yl]sulfanylmethyl]-3-thiophen-3-yl-1,2,4-oxadiazole
—— 5-[(1S)-1-[4-(1-methylpyrazolo[3,4-d]pyrimidin-4-yl)piperazin-1-yl]ethyl]-3-[3-(trifluoromethyl)phenyl]-1,2,4-oxadiazole —— C21H21F3N8O
5-[(1S)-1-[4-(1-methylpyrazolo[3,4-d]pyrimidin-4-yl)piperazin-1-yl]ethyl]-3-[3-(trifluoromethyl)phenyl]-1,2,4-oxadiazole
—— 5-bromo-2-fluoro-N-[[4-(pyrrolidin-1-ylmethyl)phenyl]methyl]benzamide —— C19H20BrFN2O
5-bromo-2-fluoro-N-[[4-(pyrrolidin-1-ylmethyl)phenyl]methyl]benzamide
—— 5-(2-methoxyethyl)-6,6-dioxo-N-pentan-3-yl-4H-imidazo[5,1-d][1,2,5]benzothiadiazepine-3-carboxamide —— C19H26N4O4S
5-(2-methoxyethyl)-6,6-dioxo-N-pentan-3-yl-4H-imidazo[5,1-d][1,2,5]benzothiadiazepine-3-carboxamide
—— 5-methyl-3-phenyl-N-[[(1S,5S)-1,3,3-trimethyl-5-[(5-methyl-3-phenyl-1,2-oxazole-4-carbonyl)amino]cyclohexyl]methyl]-1,2-oxazole-4-carboxamide —— C32H36N4O4
5-methyl-3-phenyl-N-[[(1S,5S)-1,3,3-trimethyl-5-[(5-methyl-3-phenyl-1,2-oxazole-4-carbonyl)amino]cyclohexyl]methyl]-1,2-oxazole-4-carboxamide
—— 5-[(1R)-1-[4-(1-methylpyrazolo[3,4-d]pyrimidin-4-yl)piperazin-1-yl]ethyl]-3-[3-(trifluoromethyl)phenyl]-1,2,4-oxadiazole —— C21H21F3N8O
5-[(1R)-1-[4-(1-methylpyrazolo[3,4-d]pyrimidin-4-yl)piperazin-1-yl]ethyl]-3-[3-(trifluoromethyl)phenyl]-1,2,4-oxadiazole
—— 5-chloro-N-cyclopropyl-N-[(3S)-1,1-dioxothiolan-3-yl]-1-benzofuran-2-carboxamide —— C16H16ClNO4S
5-chloro-N-cyclopropyl-N-[(3S)-1,1-dioxothiolan-3-yl]-1-benzofuran-2-carboxamide
—— 5-[[(4S)-4-ethyl-6,7-dihydro-4H-thieno[3,2-c]pyridin-5-yl]methyl]-3-(3-fluoro-4-methylphenyl)-1,2,4-oxadiazole —— C19H20FN3OS
5-[[(4S)-4-ethyl-6,7-dihydro-4H-thieno[3,2-c]pyridin-5-yl]methyl]-3-(3-fluoro-4-methylphenyl)-1,2,4-oxadiazole
—— (5S,10bS)-2-(4-chlorophenyl)-5-[4-(difluoromethoxy)phenyl]-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine —— C23H17ClF2N2O2
(5S,10bS)-2-(4-chlorophenyl)-5-[4-(difluoromethoxy)phenyl]-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine
—— 5-chloro-N-cyclopropyl-N-[(3R)-1,1-dioxothiolan-3-yl]-1-benzofuran-2-carboxamide —— C16H16ClNO4S
5-chloro-N-cyclopropyl-N-[(3R)-1,1-dioxothiolan-3-yl]-1-benzofuran-2-carboxamide
—— (5-fluoro-2-methoxyphenyl)methyl (3R)-1-(4-chlorophenyl)sulfonylpiperidine-3-carboxylate —— C20H21ClFNO5S
(5-fluoro-2-methoxyphenyl)methyl (3R)-1-(4-chlorophenyl)sulfonylpiperidine-3-carboxylate
—— 5-[[(2R)-2-(2,4-dimethoxyphenyl)pyrrolidin-1-yl]methyl]-3-(3-fluoro-4-methylphenyl)-1,2,4-oxadiazole —— C22H24FN3O3
5-[[(2R)-2-(2,4-dimethoxyphenyl)pyrrolidin-1-yl]methyl]-3-(3-fluoro-4-methylphenyl)-1,2,4-oxadiazole
—— 5-(dimethylsulfamoyl)-2-fluoro-N-[[4-(pyrrolidin-1-ylmethyl)phenyl]methyl]benzamide —— C21H26FN3O3S
5-(dimethylsulfamoyl)-2-fluoro-N-[[4-(pyrrolidin-1-ylmethyl)phenyl]methyl]benzamide
—— 5-chloro-N-[[4-[(dimethylamino)methyl]phenyl]methyl]-2-methoxybenzamide —— C18H21ClN2O2
5-chloro-N-[[4-[(dimethylamino)methyl]phenyl]methyl]-2-methoxybenzamide
—— (5R)-5-methyl-N-[[4-(2-methylpropanoylamino)phenyl]methyl]-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide —— C21H26N2O2S
(5R)-5-methyl-N-[[4-(2-methylpropanoylamino)phenyl]methyl]-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide
—— (5-Chloro-2-hydroxyphenyl)-[2-(3-hydroxypropyl)-[1,2,4]triazolo[1,5-a]pyrimidin-6-yl]methanone —— C15H13ClN4O3
(5-Chloro-2-hydroxyphenyl)-[2-(3-hydroxypropyl)-[1,2,4]triazolo[1,5-a]pyrimidin-6-yl]methanone
—— (5S)-5-methyl-N-[[4-(2-methylpropanoylamino)phenyl]methyl]-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide —— C21H26N2O2S
(5S)-5-methyl-N-[[4-(2-methylpropanoylamino)phenyl]methyl]-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide
—— [5-(1,3-benzothiazol-2-yl)furan-2-yl]methyl-[(1S,2R)-1-hydroxy-1-(4-hydroxyphenyl)propan-2-yl]azanium —— C21H21N2O3S+
[5-(1,3-benzothiazol-2-yl)furan-2-yl]methyl-[(1S,2R)-1-hydroxy-1-(4-hydroxyphenyl)propan-2-yl]azanium
—— (5S,7S)-N-(1,3-benzothiazol-2-yl)-3-bromo-N-methyladamantane-1-carboxamide —— C19H21BrN2OS
(5S,7S)-N-(1,3-benzothiazol-2-yl)-3-bromo-N-methyladamantane-1-carboxamide
—— 5-methyl-N-[[(15R)-15-tetracyclo[6.6.2.02,7.09,14]hexadeca-2,4,6,9,11,13-hexaenyl]methyl]-1-[5-(trifluoromethyl)pyridin-2-yl]pyrazole-4-carboxamide —— C28H23F3N4O
5-methyl-N-[[(15R)-15-tetracyclo[6.6.2.02,7.09,14]hexadeca-2,4,6,9,11,13-hexaenyl]methyl]-1-[5-(trifluoromethyl)pyridin-2-yl]pyrazole-4-carboxamide
—— 5-[(5-Chloro-2,3-dihydro-1,4-benzodioxin-7-yl)methylsulfanyl]-1-(3-fluorophenyl)tetrazole —— C16H12ClFN4O2S
5-[(5-Chloro-2,3-dihydro-1,4-benzodioxin-7-yl)methylsulfanyl]-1-(3-fluorophenyl)tetrazole
—— 5-methyl-N-[[(15S)-15-tetracyclo[6.6.2.02,7.09,14]hexadeca-2,4,6,9,11,13-hexaenyl]methyl]-1-[5-(trifluoromethyl)pyridin-2-yl]pyrazole-4-carboxamide —— C28H23F3N4O
5-methyl-N-[[(15S)-15-tetracyclo[6.6.2.02,7.09,14]hexadeca-2,4,6,9,11,13-hexaenyl]methyl]-1-[5-(trifluoromethyl)pyridin-2-yl]pyrazole-4-carboxamide
—— (5R)-9-(3,5-dimethylbenzoyl)-13-(2-methoxyethyl)-3,9,13-triazadispiro[4.0.56.35]tetradecan-4-one —— C23H33N3O3
(5R)-9-(3,5-dimethylbenzoyl)-13-(2-methoxyethyl)-3,9,13-triazadispiro[4.0.56.35]tetradecan-4-one
—— 5,6-dimethyl-3-[3-[(6S)-6-methylspiro[2,3,6,8-tetrahydro-[1,4]dioxino[2,3-g]isoquinoline-9,1'-cyclopentane]-7-yl]-3-oxopropyl]thieno[2,3-d]pyrimidin-4-one —— C27H31N3O4S
5,6-dimethyl-3-[3-[(6S)-6-methylspiro[2,3,6,8-tetrahydro-[1,4]dioxino[2,3-g]isoquinoline-9,1'-cyclopentane]-7-yl]-3-oxopropyl]thieno[2,3-d]pyrimidin-4-one
—— 5,6-dimethyl-3-[3-[(6R)-6-methylspiro[2,3,6,8-tetrahydro-[1,4]dioxino[2,3-g]isoquinoline-9,1'-cyclopentane]-7-yl]-3-oxopropyl]thieno[2,3-d]pyrimidin-4-one —— C27H31N3O4S
5,6-dimethyl-3-[3-[(6R)-6-methylspiro[2,3,6,8-tetrahydro-[1,4]dioxino[2,3-g]isoquinoline-9,1'-cyclopentane]-7-yl]-3-oxopropyl]thieno[2,3-d]pyrimidin-4-one
—— [(5S,10bR)-9-chloro-2-thiophen-2-yl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazin-5-yl]-(4-chlorophenyl)methanone —— C21H14Cl2N2O2S
[(5S,10bR)-9-chloro-2-thiophen-2-yl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazin-5-yl]-(4-chlorophenyl)methanone
—— [5-(5-Methyl-3-phenyl-1,2-oxazol-4-yl)-1,3,4-oxadiazol-2-yl]methyl 3-methylthiophene-2-carboxylate —— C19H15N3O4S
[5-(5-Methyl-3-phenyl-1,2-oxazol-4-yl)-1,3,4-oxadiazol-2-yl]methyl 3-methylthiophene-2-carboxylate
—— 5-N-[(1S)-1-(1-adamantyl)ethyl]-6-N-(3,4-dichlorophenyl)-[1,2,5]oxadiazolo[3,4-b]pyrazine-5,6-diamine —— C22H24Cl2N6O
5-N-[(1S)-1-(1-adamantyl)ethyl]-6-N-(3,4-dichlorophenyl)-[1,2,5]oxadiazolo[3,4-b]pyrazine-5,6-diamine
—— 5-Chloro-1-methyl-2-[(5-methyl-2-nitrophenoxy)methyl]imidazole 879302-67-7 C12H12ClN3O3
5-Chloro-1-methyl-2-[(5-methyl-2-nitrophenoxy)methyl]imidazole
—— (5S,10bS)-9-bromo-2,5-bis(4-chlorophenyl)-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine —— C22H15BrCl2N2O
(5S,10bS)-9-bromo-2,5-bis(4-chlorophenyl)-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine
—— 5-chloro-N-[4-(4-methylpiperazin-4-ium-1-yl)phenyl]-2,3-dihydro-1,4-benzodioxine-7-carboxamide —— C20H23ClN3O3+
5-chloro-N-[4-(4-methylpiperazin-4-ium-1-yl)phenyl]-2,3-dihydro-1,4-benzodioxine-7-carboxamide
—— (5S,7S)-3-(2-amino-2-oxoethyl)-5,7-dimethyladamantane-1-carboxamide —— C15H24N2O2
(5S,7S)-3-(2-amino-2-oxoethyl)-5,7-dimethyladamantane-1-carboxamide