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—— (5S,7R)-3-chloro-N-[2-oxo-2-(prop-2-enylamino)ethyl]adamantane-1-carboxamide —— C16H23ClN2O2
(5S,7R)-3-chloro-N-[2-oxo-2-(prop-2-enylamino)ethyl]adamantane-1-carboxamide
—— (5S,7S)-3-bromo-N-[2-(2,6-dichloroanilino)-2-oxoethyl]-N-ethyladamantane-1-carboxamide —— C21H25BrCl2N2O2
(5S,7S)-3-bromo-N-[2-(2,6-dichloroanilino)-2-oxoethyl]-N-ethyladamantane-1-carboxamide
—— (5S,7S)-3-bromo-N-[(R)-(3-fluorophenyl)-(1-methylimidazol-2-yl)methyl]adamantane-1-carboxamide —— C22H25BrFN3O
(5S,7S)-3-bromo-N-[(R)-(3-fluorophenyl)-(1-methylimidazol-2-yl)methyl]adamantane-1-carboxamide
—— 5-[2-(furan-2-ylmethylimino)-3,6-dihydro-1,3,4-thiadiazin-5-yl]-1-methyl-3H-indol-2-one —— C17H16N4O2S
5-[2-(furan-2-ylmethylimino)-3,6-dihydro-1,3,4-thiadiazin-5-yl]-1-methyl-3H-indol-2-one
—— 5-bromo-N-[2-[[(R)-(2-methoxyphenyl)-(1-methylimidazol-2-yl)methyl]amino]-2-oxoethyl]furan-2-carboxamide —— C19H19BrN4O4
5-bromo-N-[2-[[(R)-(2-methoxyphenyl)-(1-methylimidazol-2-yl)methyl]amino]-2-oxoethyl]furan-2-carboxamide
—— 5-bromo-N-[2-[[(S)-(2-methoxyphenyl)-(1-methylimidazol-2-yl)methyl]amino]-2-oxoethyl]furan-2-carboxamide —— C19H19BrN4O4
5-bromo-N-[2-[[(S)-(2-methoxyphenyl)-(1-methylimidazol-2-yl)methyl]amino]-2-oxoethyl]furan-2-carboxamide
—— 5-(1,3-benzothiazol-2-yl)-N-[(2R)-2-(5-methylfuran-2-yl)-2-morpholin-4-ylethyl]pentanamide —— C23H29N3O3S
5-(1,3-benzothiazol-2-yl)-N-[(2R)-2-(5-methylfuran-2-yl)-2-morpholin-4-ylethyl]pentanamide
—— 5-cyclopropyl-2-phenyl-N-(2,2,2-trifluoroethyl)pyrazole-3-carboxamide —— C15H14F3N3O
5-cyclopropyl-2-phenyl-N-(2,2,2-trifluoroethyl)pyrazole-3-carboxamide
—— 5-(5-{2-[(2-{[5-(3-Carboxy-4-chlorophenyl)-2-furyl]methylene}hydrazino)(oxo)acetyl]carbohydrazonoyl}-2-furyl)-2-chlorobenzoic acid —— C26H16Cl2N4O8
5-(5-{2-[(2-{[5-(3-Carboxy-4-chlorophenyl)-2-furyl]methylene}hydrazino)(oxo)acetyl]carbohydrazonoyl}-2-furyl)-2-chlorobenzoic acid
—— 5-[anilino(hydroxy)methylidene]-1-benzyltriazol-4-one —— C16H14N4O2
5-[anilino(hydroxy)methylidene]-1-benzyltriazol-4-one
—— 5-(1,3-benzothiazol-2-yl)-N-[(2S)-2-(5-methylfuran-2-yl)-2-morpholin-4-ylethyl]pentanamide —— C23H29N3O3S
5-(1,3-benzothiazol-2-yl)-N-[(2S)-2-(5-methylfuran-2-yl)-2-morpholin-4-ylethyl]pentanamide
—— (5S,7S)-3-bromo-N-[(S)-(3-fluorophenyl)-(1-methylimidazol-2-yl)methyl]adamantane-1-carboxamide —— C22H25BrFN3O
(5S,7S)-3-bromo-N-[(S)-(3-fluorophenyl)-(1-methylimidazol-2-yl)methyl]adamantane-1-carboxamide
—— 5-(diethylsulfamoyl)-N-[(R)-(2-methoxyphenyl)-(1-methylimidazol-2-yl)methyl]-2-methylbenzamide —— C24H30N4O4S
5-(diethylsulfamoyl)-N-[(R)-(2-methoxyphenyl)-(1-methylimidazol-2-yl)methyl]-2-methylbenzamide
—— 5-(1,3-benzothiazol-2-yl)-N-[(R)-(2-methoxyphenyl)-(1-methylimidazol-2-yl)methyl]thiophene-2-carboxamide —— C24H20N4O2S2
5-(1,3-benzothiazol-2-yl)-N-[(R)-(2-methoxyphenyl)-(1-methylimidazol-2-yl)methyl]thiophene-2-carboxamide
—— 5-bromo-N-[2-(4-butylanilino)-2-oxoethyl]furan-2-carboxamide —— C17H19BrN2O3
5-bromo-N-[2-(4-butylanilino)-2-oxoethyl]furan-2-carboxamide
—— 5-[2,5-dimethyl-1-(5-methyl-1,2-oxazol-3-yl)pyrrol-3-yl]-N-[[(2R)-oxolan-2-yl]methyl]-3,6-dihydro-1,3,4-thiadiazin-2-imine —— C18H23N5O2S
5-[2,5-dimethyl-1-(5-methyl-1,2-oxazol-3-yl)pyrrol-3-yl]-N-[[(2R)-oxolan-2-yl]methyl]-3,6-dihydro-1,3,4-thiadiazin-2-imine
—— 5-[(2S)-2-(1H-benzimidazol-2-yl)pyrrolidine-1-carbonyl]-2-benzylisoindole-1,3-dione —— C27H22N4O3
5-[(2S)-2-(1H-benzimidazol-2-yl)pyrrolidine-1-carbonyl]-2-benzylisoindole-1,3-dione
—— 5-[(2R)-2-(1H-benzimidazol-2-yl)pyrrolidine-1-carbonyl]-2-benzylisoindole-1,3-dione —— C27H22N4O3
5-[(2R)-2-(1H-benzimidazol-2-yl)pyrrolidine-1-carbonyl]-2-benzylisoindole-1,3-dione
—— 5-chloro-N-[(R)-(3-fluorophenyl)-(1-methylimidazol-2-yl)methyl]-3-methyl-1-[(4-methylphenyl)methyl]pyrazole-4-carboxamide —— C24H23ClFN5O
5-chloro-N-[(R)-(3-fluorophenyl)-(1-methylimidazol-2-yl)methyl]-3-methyl-1-[(4-methylphenyl)methyl]pyrazole-4-carboxamide
—— 5-(1,3-benzothiazol-2-yl)-N-[(S)-(2-methoxyphenyl)-(1-methylimidazol-2-yl)methyl]thiophene-2-carboxamide —— C24H20N4O2S2
5-(1,3-benzothiazol-2-yl)-N-[(S)-(2-methoxyphenyl)-(1-methylimidazol-2-yl)methyl]thiophene-2-carboxamide
—— 5-chloro-N-[(S)-(3-fluorophenyl)-(1-methylimidazol-2-yl)methyl]-3-methyl-1-[(4-methylphenyl)methyl]pyrazole-4-carboxamide —— C24H23ClFN5O
5-chloro-N-[(S)-(3-fluorophenyl)-(1-methylimidazol-2-yl)methyl]-3-methyl-1-[(4-methylphenyl)methyl]pyrazole-4-carboxamide
—— 5-[(2S)-2-(1,3-benzothiazol-2-yl)piperidine-1-carbonyl]-N,N-diethyl-1-methylpyrrole-3-sulfonamide —— C22H28N4O3S2
5-[(2S)-2-(1,3-benzothiazol-2-yl)piperidine-1-carbonyl]-N,N-diethyl-1-methylpyrrole-3-sulfonamide
—— 5-[(4-methoxyphenyl)sulfamoyl]-N,2-dimethyl-N-[(1S)-1-thiophen-2-ylethyl]benzamide —— C22H24N2O4S2
5-[(4-methoxyphenyl)sulfamoyl]-N,2-dimethyl-N-[(1S)-1-thiophen-2-ylethyl]benzamide
—— 5-[(2R)-2-(1,3-benzothiazol-2-yl)piperidine-1-carbonyl]-N,N-diethyl-1-methylpyrrole-3-sulfonamide —— C22H28N4O3S2
5-[(2R)-2-(1,3-benzothiazol-2-yl)piperidine-1-carbonyl]-N,N-diethyl-1-methylpyrrole-3-sulfonamide
—— 5-(1,3-benzothiazol-2-yl)-N-methyl-N-[(1S)-1-thiophen-2-ylethyl]furan-2-carboxamide —— C19H16N2O2S2
5-(1,3-benzothiazol-2-yl)-N-methyl-N-[(1S)-1-thiophen-2-ylethyl]furan-2-carboxamide
—— 5-(1,3-benzothiazol-2-yl)-N-methyl-N-[(1R)-1-thiophen-2-ylethyl]furan-2-carboxamide —— C19H16N2O2S2
5-(1,3-benzothiazol-2-yl)-N-methyl-N-[(1R)-1-thiophen-2-ylethyl]furan-2-carboxamide
—— 5-methyl-4-[1-[[(2S)-oxolan-2-yl]methyl]tetrazol-5-yl]sulfanyl-6-phenylthieno[2,3-d]pyrimidine —— C19H18N6OS2
5-methyl-4-[1-[[(2S)-oxolan-2-yl]methyl]tetrazol-5-yl]sulfanyl-6-phenylthieno[2,3-d]pyrimidine
—— 5-[(4-methoxyphenyl)sulfamoyl]-N,2-dimethyl-N-[(1R)-1-thiophen-2-ylethyl]benzamide —— C22H24N2O4S2
5-[(4-methoxyphenyl)sulfamoyl]-N,2-dimethyl-N-[(1R)-1-thiophen-2-ylethyl]benzamide
—— (5R,7R)-5-(4-fluorophenyl)-7-(trifluoromethyl)-N-[(E)-[(1R,4R)-1,7,7-trimethyl-2-bicyclo[2.2.1]heptanylidene]amino]-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide —— C24H27F4N5O
(5R,7R)-5-(4-fluorophenyl)-7-(trifluoromethyl)-N-[(E)-[(1R,4R)-1,7,7-trimethyl-2-bicyclo[2.2.1]heptanylidene]amino]-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide
—— 5-bromo-N-[2-(4-fluoroanilino)-2-oxoethyl]-N-methylpyridine-3-carboxamide —— C15H13BrFN3O2
5-bromo-N-[2-(4-fluoroanilino)-2-oxoethyl]-N-methylpyridine-3-carboxamide
—— (5S,7R)-5-(4-fluorophenyl)-7-(1,1,2,2,2-pentafluoroethyl)-N-[(E)-[(1R,4R)-1,7,7-trimethyl-2-bicyclo[2.2.1]heptanylidene]amino]-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide —— C25H27F6N5O
(5S,7R)-5-(4-fluorophenyl)-7-(1,1,2,2,2-pentafluoroethyl)-N-[(E)-[(1R,4R)-1,7,7-trimethyl-2-bicyclo[2.2.1]heptanylidene]amino]-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide
—— (5S,7S)-5-(4-fluorophenyl)-7-(trifluoromethyl)-N-[(E)-[(1R,4R)-1,7,7-trimethyl-2-bicyclo[2.2.1]heptanylidene]amino]-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide —— C24H27F4N5O
(5S,7S)-5-(4-fluorophenyl)-7-(trifluoromethyl)-N-[(E)-[(1R,4R)-1,7,7-trimethyl-2-bicyclo[2.2.1]heptanylidene]amino]-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide
—— 5-[2,5-dimethyl-1-(4-methyl-1,3-thiazol-2-yl)pyrrol-3-yl]-N-[[(2S)-oxolan-2-yl]methyl]-3,6-dihydro-1,3,4-thiadiazin-2-imine —— C18H23N5OS2
5-[2,5-dimethyl-1-(4-methyl-1,3-thiazol-2-yl)pyrrol-3-yl]-N-[[(2S)-oxolan-2-yl]methyl]-3,6-dihydro-1,3,4-thiadiazin-2-imine
—— 5,5-Bis(4-methoxyphenyl)-3-(2-methylpropyl)imidazolidine-2,4-dione —— C21H24N2O4
5,5-Bis(4-methoxyphenyl)-3-(2-methylpropyl)imidazolidine-2,4-dione
—— (5S,7S)-5-(4-fluorophenyl)-7-(1,1,2,2,2-pentafluoroethyl)-N-[(E)-[(1R,4R)-1,7,7-trimethyl-2-bicyclo[2.2.1]heptanylidene]amino]-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide —— C25H27F6N5O
(5S,7S)-5-(4-fluorophenyl)-7-(1,1,2,2,2-pentafluoroethyl)-N-[(E)-[(1R,4R)-1,7,7-trimethyl-2-bicyclo[2.2.1]heptanylidene]amino]-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide
—— 5-(1,3-benzothiazol-2-yl)-N-[(2S)-2-(5-methylfuran-2-yl)-2-morpholin-4-ylethyl]thiophene-2-carboxamide —— C23H23N3O3S2
5-(1,3-benzothiazol-2-yl)-N-[(2S)-2-(5-methylfuran-2-yl)-2-morpholin-4-ylethyl]thiophene-2-carboxamide
—— (5S,7R)-5-(4-fluorophenyl)-7-(trifluoromethyl)-N-[(E)-[(1R,4R)-1,7,7-trimethyl-2-bicyclo[2.2.1]heptanylidene]amino]-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide —— C24H27F4N5O
(5S,7R)-5-(4-fluorophenyl)-7-(trifluoromethyl)-N-[(E)-[(1R,4R)-1,7,7-trimethyl-2-bicyclo[2.2.1]heptanylidene]amino]-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide
—— 5-(1,3-benzothiazol-2-yl)-N-[(2R)-2-(5-methylfuran-2-yl)-2-morpholin-4-ylethyl]thiophene-2-carboxamide —— C23H23N3O3S2
5-(1,3-benzothiazol-2-yl)-N-[(2R)-2-(5-methylfuran-2-yl)-2-morpholin-4-ylethyl]thiophene-2-carboxamide
—— 5-[2,5-dimethyl-1-(4-methyl-1,3-thiazol-2-yl)pyrrol-3-yl]-N-[[(2R)-oxolan-2-yl]methyl]-3,6-dihydro-1,3,4-thiadiazin-2-imine —— C18H23N5OS2
5-[2,5-dimethyl-1-(4-methyl-1,3-thiazol-2-yl)pyrrol-3-yl]-N-[[(2R)-oxolan-2-yl]methyl]-3,6-dihydro-1,3,4-thiadiazin-2-imine
—— 5-[(4-fluorophenoxy)methyl]-N-[(2S)-2-(5-methylfuran-2-yl)-2-morpholin-4-ylethyl]furan-2-carboxamide —— C23H25FN2O5
5-[(4-fluorophenoxy)methyl]-N-[(2S)-2-(5-methylfuran-2-yl)-2-morpholin-4-ylethyl]furan-2-carboxamide
—— 5-bromo-N-[2-(3-fluoroanilino)-2-oxoethyl]-N-methylpyridine-3-carboxamide —— C15H13BrFN3O2
5-bromo-N-[2-(3-fluoroanilino)-2-oxoethyl]-N-methylpyridine-3-carboxamide
—— 5-cyclopropyl-N-[(2,3-dimethoxyphenyl)methyl]-N-methyl-2-phenylpyrazole-3-carboxamide —— C23H25N3O3
5-cyclopropyl-N-[(2,3-dimethoxyphenyl)methyl]-N-methyl-2-phenylpyrazole-3-carboxamide
—— 5-(4-chlorophenyl)-N-[(3S)-1,1-dioxothiolan-3-yl]thieno[2,3-d]pyrimidin-4-amine —— C16H14ClN3O2S2
5-(4-chlorophenyl)-N-[(3S)-1,1-dioxothiolan-3-yl]thieno[2,3-d]pyrimidin-4-amine
—— 5-[(5-Chlorothiadiazol-4-yl)methyl]-1-phenylpyrazolo[3,4-d]pyrimidin-4-one —— C14H9ClN6OS
5-[(5-Chlorothiadiazol-4-yl)methyl]-1-phenylpyrazolo[3,4-d]pyrimidin-4-one
—— (5S)-5-ethyl-N-[2-(3-fluoroanilino)-2-oxoethyl]-N-methyl-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide —— C20H23FN2O2S
(5S)-5-ethyl-N-[2-(3-fluoroanilino)-2-oxoethyl]-N-methyl-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide
—— 5-cyclopropyl-N-[3-(ethylcarbamoyl)phenyl]-2-phenylpyrazole-3-carboxamide —— C22H22N4O2
5-cyclopropyl-N-[3-(ethylcarbamoyl)phenyl]-2-phenylpyrazole-3-carboxamide
—— 5-cyclopropyl-N-[2-(2-fluorophenyl)ethyl]-2-phenylpyrazole-3-carboxamide —— C21H20FN3O
5-cyclopropyl-N-[2-(2-fluorophenyl)ethyl]-2-phenylpyrazole-3-carboxamide
—— 5-chloro-N-[2-(5-chloro-2-methoxyanilino)-2-oxoethyl]-N-methylthiophene-2-carboxamide —— C15H14Cl2N2O3S
5-chloro-N-[2-(5-chloro-2-methoxyanilino)-2-oxoethyl]-N-methylthiophene-2-carboxamide
—— 5-chloro-N-[2-(4-methoxyanilino)-2-oxoethyl]-N-methylthiophene-2-carboxamide —— C15H15ClN2O3S
5-chloro-N-[2-(4-methoxyanilino)-2-oxoethyl]-N-methylthiophene-2-carboxamide
—— 5-bromo-N-[2-(5-chloro-2-methoxyanilino)-2-oxoethyl]-N-methylfuran-2-carboxamide —— C15H14BrClN2O4
5-bromo-N-[2-(5-chloro-2-methoxyanilino)-2-oxoethyl]-N-methylfuran-2-carboxamide