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—— 5-Benzyloxy-2-(4-benzyloxy-phenyl)-3-chloro-1-[4-(2-piperidin-1-yl-ethoxy)-benzyl]-1H-indole —— C42H41ClN2O3
5-Benzyloxy-2-(4-benzyloxy-phenyl)-3-chloro-1-[4-(2-piperidin-1-yl-ethoxy)-benzyl]-1H-indole
—— 5-(2-fluorophenyl)-N-[(1R,3R)-3-(trifluoromethyl)cyclohexyl]thiophene-2-carboxamide —— C18H17F4NOS
5-(2-fluorophenyl)-N-[(1R,3R)-3-(trifluoromethyl)cyclohexyl]thiophene-2-carboxamide
—— 5-benzylsulfonyl-N,N-diethyl-4-(1-phenylpiperidin-4-yl)-2-(2-pyrrolidin-1-ylethylamino)benzamide —— C35H46N4O3S
5-benzylsulfonyl-N,N-diethyl-4-(1-phenylpiperidin-4-yl)-2-(2-pyrrolidin-1-ylethylamino)benzamide
—— (5Z)-5-[[4-[[(2S)-1-[(2,2,4,6,7-pentamethyl-5-phenylmethoxy-3H-1-benzofuran-3-yl)methyl]pyrrolidin-2-yl]methoxy]phenyl]methylidene]-1,3-thiazolidine-2,4-dione —— C36H40N2O5S
(5Z)-5-[[4-[[(2S)-1-[(2,2,4,6,7-pentamethyl-5-phenylmethoxy-3H-1-benzofuran-3-yl)methyl]pyrrolidin-2-yl]methoxy]phenyl]methylidene]-1,3-thiazolidine-2,4-dione
—— (5-methoxy-2,3-dihydro-1,4-benzodioxin-7-yl)-[(2R)-2-(6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-a]azepin-3-yl)pyrrolidin-1-yl]methanone —— C21H26N4O4
(5-methoxy-2,3-dihydro-1,4-benzodioxin-7-yl)-[(2R)-2-(6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-a]azepin-3-yl)pyrrolidin-1-yl]methanone
—— [5-cyclopropyl-1-(2,4-dichlorophenyl)pyrazol-4-yl]-[(3R)-3-(6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-a]azepin-3-yl)piperidin-1-yl]methanone —— C25H28Cl2N6O
[5-cyclopropyl-1-(2,4-dichlorophenyl)pyrazol-4-yl]-[(3R)-3-(6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-a]azepin-3-yl)piperidin-1-yl]methanone
—— [5-[(1-methylimidazol-2-yl)sulfanylmethyl]furan-2-yl]-[(3R)-3-(6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-a]azepin-3-yl)piperidin-1-yl]methanone —— C22H28N6O2S
[5-[(1-methylimidazol-2-yl)sulfanylmethyl]furan-2-yl]-[(3R)-3-(6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-a]azepin-3-yl)piperidin-1-yl]methanone
—— [5-(2,3-dihydro-1,4-benzodioxin-6-yl)thiophen-2-yl]-[(2R)-2-(6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-a]azepin-3-yl)pyrrolidin-1-yl]methanone —— C24H26N4O3S
[5-(2,3-dihydro-1,4-benzodioxin-6-yl)thiophen-2-yl]-[(2R)-2-(6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-a]azepin-3-yl)pyrrolidin-1-yl]methanone
—— 5-[(3aS,4S,6aR)-2-oxo-1,3,3a,4,6,6a-hexahydrothieno[3,4-d]imidazol-4-yl]pentanoic acid;chromium;pyridine-2-carboxylic acid —— C28H31CrN5O9S
5-[(3aS,4S,6aR)-2-oxo-1,3,3a,4,6,6a-hexahydrothieno[3,4-d]imidazol-4-yl]pentanoic acid;chromium;pyridine-2-carboxylic acid
—— [5-(2,3-dihydro-1,4-benzodioxin-6-yl)thiophen-2-yl]-[(2S)-2-(6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-a]azepin-3-yl)pyrrolidin-1-yl]methanone —— C24H26N4O3S
[5-(2,3-dihydro-1,4-benzodioxin-6-yl)thiophen-2-yl]-[(2S)-2-(6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-a]azepin-3-yl)pyrrolidin-1-yl]methanone
—— 5-bromo-2-[3-oxo-3-[(2R)-2-(6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-a]azepin-3-yl)pyrrolidin-1-yl]propyl]isoindole-1,3-dione —— C22H24BrN5O3
5-bromo-2-[3-oxo-3-[(2R)-2-(6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-a]azepin-3-yl)pyrrolidin-1-yl]propyl]isoindole-1,3-dione
—— [5-cyclopropyl-1-(2,4-dichlorophenyl)pyrazol-4-yl]-[(3S)-3-(6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-a]azepin-3-yl)piperidin-1-yl]methanone —— C25H28Cl2N6O
[5-cyclopropyl-1-(2,4-dichlorophenyl)pyrazol-4-yl]-[(3S)-3-(6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-a]azepin-3-yl)piperidin-1-yl]methanone
—— 5-{2-[2-(3-chloro-phenyl)-2-hydroxy-ethylamino]-propyl}-benzo[1,3]dioxole-2,2-dicarboxylic acid dihexyl ester —— C32H44ClNO7
5-{2-[2-(3-chloro-phenyl)-2-hydroxy-ethylamino]-propyl}-benzo[1,3]dioxole-2,2-dicarboxylic acid dihexyl ester
—— 5-(4-aminophenyl)-7-[3-[4-(2-fluorophenyl)piperazin-1-yl]propanoyl]-8-methyl-9H-[1,3]dioxolo[4,5-h][2,3]benzodiazepine-8-carbonitrile —— C31H31FN6O3
5-(4-aminophenyl)-7-[3-[4-(2-fluorophenyl)piperazin-1-yl]propanoyl]-8-methyl-9H-[1,3]dioxolo[4,5-h][2,3]benzodiazepine-8-carbonitrile
—— 5-chloro-N-[(1R)-1-[1-methyl-5-(4-morpholin-4-ylphenyl)imidazol-2-yl]-2-pyridin-2-ylethyl]-1-benzofuran-2-carboxamide —— C30H28ClN5O3
5-chloro-N-[(1R)-1-[1-methyl-5-(4-morpholin-4-ylphenyl)imidazol-2-yl]-2-pyridin-2-ylethyl]-1-benzofuran-2-carboxamide
—— 5-(diaminomethylideneamino)-2-[[4-(5,7-difluoro-2-phenyl-1H-indol-3-yl)-1-oxobutyl]amino]pentanoic acid methyl ester —— C25H29F2N5O3
5-(diaminomethylideneamino)-2-[[4-(5,7-difluoro-2-phenyl-1H-indol-3-yl)-1-oxobutyl]amino]pentanoic acid methyl ester
—— 5-(2-Methoxyphenyl)-3-[[8-(4-methylpiperazin-1-yl)naphthalen-2-yl]oxymethyl]-1,2,4-oxadiazole;hydrate;dihydrochloride —— C25H30Cl2N4O4
5-(2-Methoxyphenyl)-3-[[8-(4-methylpiperazin-1-yl)naphthalen-2-yl]oxymethyl]-1,2,4-oxadiazole;hydrate;dihydrochloride
—— 5-[4-(Trifluoromethyl)pyridin-3-yl]-3-[2-[2-[5-[4-(trifluoromethyl)pyridin-3-yl]-1,2,4-oxadiazol-3-yl]ethylsulfanyl]ethyl]-1,2,4-oxadiazole —— C20H14F6N6O2S
5-[4-(Trifluoromethyl)pyridin-3-yl]-3-[2-[2-[5-[4-(trifluoromethyl)pyridin-3-yl]-1,2,4-oxadiazol-3-yl]ethylsulfanyl]ethyl]-1,2,4-oxadiazole
—— [5-[(1-methylimidazol-2-yl)sulfanylmethyl]furan-2-yl]-[(4S)-4-phenyl-6,7-dihydro-4H-thieno[3,2-c]pyridin-5-yl]methanone —— C23H21N3O2S2
[5-[(1-methylimidazol-2-yl)sulfanylmethyl]furan-2-yl]-[(4S)-4-phenyl-6,7-dihydro-4H-thieno[3,2-c]pyridin-5-yl]methanone
—— (5-methoxy-2,3-dihydro-1,4-benzodioxin-7-yl)-[(2S)-2-(6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-a]azepin-3-yl)pyrrolidin-1-yl]methanone —— C21H26N4O4
(5-methoxy-2,3-dihydro-1,4-benzodioxin-7-yl)-[(2S)-2-(6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-a]azepin-3-yl)pyrrolidin-1-yl]methanone
—— 5-[(1-methylimidazol-2-yl)sulfanylmethyl]-N-[(1R,2R,4S)-1,7,7-trimethyl-2-bicyclo[2.2.1]heptanyl]furan-2-carboxamide —— C20H27N3O2S
5-[(1-methylimidazol-2-yl)sulfanylmethyl]-N-[(1R,2R,4S)-1,7,7-trimethyl-2-bicyclo[2.2.1]heptanyl]furan-2-carboxamide
—— 5-[2-Ethoxy-5-(4-methylpiperazin-1-ylsulphonyl)pyridin-3-yl]-3-ethyl-2-[2-methoxyethyl]-2,6-dihydro-7h-pyrazolo[4,3-d]pyrimidin-7-one —— C22H31N7O5S
5-[2-Ethoxy-5-(4-methylpiperazin-1-ylsulphonyl)pyridin-3-yl]-3-ethyl-2-[2-methoxyethyl]-2,6-dihydro-7h-pyrazolo[4,3-d]pyrimidin-7-one
—— [5-[(1-methylimidazol-2-yl)sulfanylmethyl]furan-2-yl]-[(3S)-3-(6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-a]azepin-3-yl)piperidin-1-yl]methanone —— C22H28N6O2S
[5-[(1-methylimidazol-2-yl)sulfanylmethyl]furan-2-yl]-[(3S)-3-(6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-a]azepin-3-yl)piperidin-1-yl]methanone
—— 5-[(1-methylimidazol-2-yl)sulfanylmethyl]-N-[(1S,2R,4R)-1,7,7-trimethyl-2-bicyclo[2.2.1]heptanyl]furan-2-carboxamide —— C20H27N3O2S
5-[(1-methylimidazol-2-yl)sulfanylmethyl]-N-[(1S,2R,4R)-1,7,7-trimethyl-2-bicyclo[2.2.1]heptanyl]furan-2-carboxamide
—— [5-[(1-methylimidazol-2-yl)sulfanylmethyl]furan-2-yl]-[(2R)-2-(4-methylphenyl)pyrrolidin-1-yl]methanone —— C21H23N3O2S
[5-[(1-methylimidazol-2-yl)sulfanylmethyl]furan-2-yl]-[(2R)-2-(4-methylphenyl)pyrrolidin-1-yl]methanone
—— 5-bromo-2-[3-oxo-3-[(2S)-2-(6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-a]azepin-3-yl)pyrrolidin-1-yl]propyl]isoindole-1,3-dione —— C22H24BrN5O3
5-bromo-2-[3-oxo-3-[(2S)-2-(6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-a]azepin-3-yl)pyrrolidin-1-yl]propyl]isoindole-1,3-dione
—— 5-(4-carbamimidoylphenyl)-N-[(3S)-5-oxo-2-phenyloxolan-3-yl]pentanamide —— C22H25N3O3
5-(4-carbamimidoylphenyl)-N-[(3S)-5-oxo-2-phenyloxolan-3-yl]pentanamide
—— [5-[(1-methylimidazol-2-yl)sulfanylmethyl]furan-2-yl]-[(2S)-2-(4-methylphenyl)pyrrolidin-1-yl]methanone —— C21H23N3O2S
[5-[(1-methylimidazol-2-yl)sulfanylmethyl]furan-2-yl]-[(2S)-2-(4-methylphenyl)pyrrolidin-1-yl]methanone
—— 5,6-dimethyl-3-[3-oxo-3-[(2S)-2-(6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-a]azepin-3-yl)pyrrolidin-1-yl]propyl]thieno[2,3-d]pyrimidin-4-one —— C22H28N6O2S
5,6-dimethyl-3-[3-oxo-3-[(2S)-2-(6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-a]azepin-3-yl)pyrrolidin-1-yl]propyl]thieno[2,3-d]pyrimidin-4-one
—— [5-cyclopropyl-1-(2,4-dichlorophenyl)pyrazol-4-yl]-[(2S)-2-(4-fluorophenyl)morpholin-4-yl]methanone —— C23H20Cl2FN3O2
[5-cyclopropyl-1-(2,4-dichlorophenyl)pyrazol-4-yl]-[(2S)-2-(4-fluorophenyl)morpholin-4-yl]methanone
—— [5-cyclopropyl-1-(2,4-dichlorophenyl)pyrazol-4-yl]-[(2R)-2-(4-fluorophenyl)morpholin-4-yl]methanone —— C23H20Cl2FN3O2
[5-cyclopropyl-1-(2,4-dichlorophenyl)pyrazol-4-yl]-[(2R)-2-(4-fluorophenyl)morpholin-4-yl]methanone
—— 5,6-dimethyl-3-[3-oxo-3-[(2R)-2-(6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-a]azepin-3-yl)pyrrolidin-1-yl]propyl]thieno[2,3-d]pyrimidin-4-one —— C22H28N6O2S
5,6-dimethyl-3-[3-oxo-3-[(2R)-2-(6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-a]azepin-3-yl)pyrrolidin-1-yl]propyl]thieno[2,3-d]pyrimidin-4-one
—— 5-[(2R)-2-[(1R,3aS,4E,7aR)-4-[(2Z)-2-[(3S,5R)-3,5-dihydroxy-2-methylidenecyclohexylidene]ethylidene]-7a-methyl-2,3,3a,5,6,7-hexahydro-1H-inden-1-yl]propyl]-4-methyl-3-methylideneoxolan-2-one —— C28H40O4
5-[(2R)-2-[(1R,3aS,4E,7aR)-4-[(2Z)-2-[(3S,5R)-3,5-dihydroxy-2-methylidenecyclohexylidene]ethylidene]-7a-methyl-2,3,3a,5,6,7-hexahydro-1H-inden-1-yl]propyl]-4-methyl-3-methylideneoxolan-2-one
—— 5-[2-(3,4-Diethoxyphenyl)-1,3-thiazol-4-yl]-3-(2-ethoxyethyl)-2-methoxybenzoic acid —— C25H29NO6S
5-[2-(3,4-Diethoxyphenyl)-1,3-thiazol-4-yl]-3-(2-ethoxyethyl)-2-methoxybenzoic acid
—— 5-[(3S)-dithiolan-3-yl]-1-[4-[[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]methyl]piperazin-1-yl]pentan-1-one —— C22H30N4O2S2
5-[(3S)-dithiolan-3-yl]-1-[4-[[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]methyl]piperazin-1-yl]pentan-1-one
—— 5-(80Br)bromanyl-1-[(2R,4R,5R)-4-hydroxy-5-[[(2R,3R,4S,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]oxymethyl]oxolan-2-yl]pyridine-2,4-dione —— C16H22BrNO10
5-(80Br)bromanyl-1-[(2R,4R,5R)-4-hydroxy-5-[[(2R,3R,4S,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]oxymethyl]oxolan-2-yl]pyridine-2,4-dione
—— 5-(ethylsulfamoyl)-N-[(1S)-1-[1-(4-fluorophenyl)-5-methylpyrazol-4-yl]ethyl]-2-methylbenzamide —— C22H25FN4O3S
5-(ethylsulfamoyl)-N-[(1S)-1-[1-(4-fluorophenyl)-5-methylpyrazol-4-yl]ethyl]-2-methylbenzamide
—— 5-[[3-[3-[4-(Trifluoromethyl)phenyl]propanoyl]-4-methoxyphenyl]methyl]thiazolidine-2,4-dione —— C21H18F3NO4S
5-[[3-[3-[4-(Trifluoromethyl)phenyl]propanoyl]-4-methoxyphenyl]methyl]thiazolidine-2,4-dione
—— 5-[(3R)-dithiolan-3-yl]-1-[4-[[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]methyl]piperazin-1-yl]pentan-1-one —— C22H30N4O2S2
5-[(3R)-dithiolan-3-yl]-1-[4-[[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]methyl]piperazin-1-yl]pentan-1-one
—— (5R,9S)-2-[[(2R,6R)-4-acetyl-6-methylmorpholin-2-yl]oxymethyl]-9-cyano-5-methyl-13-propan-2-yltetracyclo[7.4.0.02,11.04,8]tridec-12-ene-1-carboxylic acid —— C27H38N2O5
(5R,9S)-2-[[(2R,6R)-4-acetyl-6-methylmorpholin-2-yl]oxymethyl]-9-cyano-5-methyl-13-propan-2-yltetracyclo[7.4.0.02,11.04,8]tridec-12-ene-1-carboxylic acid
—— 5-(ethylsulfamoyl)-N-[(1R)-1-[1-(4-fluorophenyl)-5-methylpyrazol-4-yl]ethyl]-2-methylbenzamide —— C22H25FN4O3S
5-(ethylsulfamoyl)-N-[(1R)-1-[1-(4-fluorophenyl)-5-methylpyrazol-4-yl]ethyl]-2-methylbenzamide
—— [5-[(3-Methoxyphenyl)-(2-phenylethylamino)methyl]-2-(2-phenylethoxy)phenyl]methanol —— C31H33NO3
[5-[(3-Methoxyphenyl)-(2-phenylethylamino)methyl]-2-(2-phenylethoxy)phenyl]methanol
—— 5-[4-[(3-tert-butylphenyl)carbamoylamino]phenoxy]-2-methoxy-N-methylbenzamide —— C26H29N3O4
5-[4-[(3-tert-butylphenyl)carbamoylamino]phenoxy]-2-methoxy-N-methylbenzamide
—— 5-[(3S)-dithiolan-3-yl]-N-[(1S)-1-[1-(4-fluorophenyl)-5-methylpyrazol-4-yl]ethyl]pentanamide —— C20H26FN3OS2
5-[(3S)-dithiolan-3-yl]-N-[(1S)-1-[1-(4-fluorophenyl)-5-methylpyrazol-4-yl]ethyl]pentanamide
—— 5-Chloro-1,1-dioxo-2-(4-spiro[1,2-dihydroindene-3,4'-piperidine]-1'-ylbutyl)-1,2-benzothiazol-3-one —— C24H27ClN2O3S
5-Chloro-1,1-dioxo-2-(4-spiro[1,2-dihydroindene-3,4'-piperidine]-1'-ylbutyl)-1,2-benzothiazol-3-one
—— 5-[Cyclohexyl-[3-[4-(3-hydroxyphenyl)-3,4-dimethylpiperidin-1-yl]propyl]amino]-5-oxopentanoic acid —— C27H42N2O4
5-[Cyclohexyl-[3-[4-(3-hydroxyphenyl)-3,4-dimethylpiperidin-1-yl]propyl]amino]-5-oxopentanoic acid
—— 5-[(3R)-dithiolan-3-yl]-N-[(1S)-1-[1-(4-fluorophenyl)-5-methylpyrazol-4-yl]ethyl]pentanamide —— C20H26FN3OS2
5-[(3R)-dithiolan-3-yl]-N-[(1S)-1-[1-(4-fluorophenyl)-5-methylpyrazol-4-yl]ethyl]pentanamide
—— (5Z)-5-[[4-chloro-3-(3,5,5,8,8-pentamethyl-6,7-dihydronaphthalen-2-yl)phenyl]methylidene]-1,3-thiazolidine-2,4-dione —— C25H26ClNO2S
(5Z)-5-[[4-chloro-3-(3,5,5,8,8-pentamethyl-6,7-dihydronaphthalen-2-yl)phenyl]methylidene]-1,3-thiazolidine-2,4-dione
—— 5,7-dihydroxy-6,8-bis(pyrrolidin-1-ylmethyl)-3-[4-[(2R,3R,4R,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]oxyphenyl]chromen-4-one —— C31H38N2O10
5,7-dihydroxy-6,8-bis(pyrrolidin-1-ylmethyl)-3-[4-[(2R,3R,4R,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]oxyphenyl]chromen-4-one
—— [5-(4-Bromophenyl)-4-methyl-6-morpholin-4-ylpyridin-2-yl]-morpholin-4-ylmethanone —— C21H24BrN3O3
[5-(4-Bromophenyl)-4-methyl-6-morpholin-4-ylpyridin-2-yl]-morpholin-4-ylmethanone