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苯并恶嗪类

中文名称 英文名称 CAS号 化学式 结构式图片
—— (2R)-4-acetyl-N-[(1R)-1-[3-(trifluoromethyl)phenyl]ethyl]-2,3-dihydro-1,4-benzoxazine-2-carboxamide —— C20H19F3N2O3
(2R)-4-acetyl-N-[(1R)-1-[3-(trifluoromethyl)phenyl]ethyl]-2,3-dihydro-1,4-benzoxazine-2-carboxamide
—— (2S)-4-acetyl-N-[(1R)-1-[3-(trifluoromethyl)phenyl]ethyl]-2,3-dihydro-1,4-benzoxazine-2-carboxamide —— C20H19F3N2O3
(2S)-4-acetyl-N-[(1R)-1-[3-(trifluoromethyl)phenyl]ethyl]-2,3-dihydro-1,4-benzoxazine-2-carboxamide
—— [(2R)-4-[2-[(4-methylphenoxy)methyl]-1,3-thiazole-4-carbonyl]-2,3-dihydro-1,4-benzoxazin-2-yl]-morpholin-4-ylmethanone —— C25H25N3O5S
[(2R)-4-[2-[(4-methylphenoxy)methyl]-1,3-thiazole-4-carbonyl]-2,3-dihydro-1,4-benzoxazin-2-yl]-morpholin-4-ylmethanone
—— (2R)-4-acetyl-N-[(1R)-1-[4-(2-methylpropyl)phenyl]ethyl]-2,3-dihydro-1,4-benzoxazine-2-carboxamide —— C23H28N2O3
(2R)-4-acetyl-N-[(1R)-1-[4-(2-methylpropyl)phenyl]ethyl]-2,3-dihydro-1,4-benzoxazine-2-carboxamide
—— (2R)-4-acetyl-N-[4-[4-[methyl(methylsulfonyl)amino]phenyl]-1,3-thiazol-2-yl]-2,3-dihydro-1,4-benzoxazine-2-carboxamide —— C22H22N4O5S2
(2R)-4-acetyl-N-[4-[4-[methyl(methylsulfonyl)amino]phenyl]-1,3-thiazol-2-yl]-2,3-dihydro-1,4-benzoxazine-2-carboxamide
—— (2S)-4-acetyl-N-[(1R)-1-[4-(2-methylpropyl)phenyl]ethyl]-2,3-dihydro-1,4-benzoxazine-2-carboxamide —— C23H28N2O3
(2S)-4-acetyl-N-[(1R)-1-[4-(2-methylpropyl)phenyl]ethyl]-2,3-dihydro-1,4-benzoxazine-2-carboxamide
—— (2S)-4-acetyl-N-[(1S)-1-[4-(2-methylpropyl)phenyl]ethyl]-2,3-dihydro-1,4-benzoxazine-2-carboxamide —— C23H28N2O3
(2S)-4-acetyl-N-[(1S)-1-[4-(2-methylpropyl)phenyl]ethyl]-2,3-dihydro-1,4-benzoxazine-2-carboxamide
—— (2S)-4-acetyl-N-[(1S)-1-[3-(trifluoromethyl)phenyl]ethyl]-2,3-dihydro-1,4-benzoxazine-2-carboxamide —— C20H19F3N2O3
(2S)-4-acetyl-N-[(1S)-1-[3-(trifluoromethyl)phenyl]ethyl]-2,3-dihydro-1,4-benzoxazine-2-carboxamide
—— (2R)-4-acetyl-N-[(1S)-1-[4-(2-methylpropyl)phenyl]ethyl]-2,3-dihydro-1,4-benzoxazine-2-carboxamide —— C23H28N2O3
(2R)-4-acetyl-N-[(1S)-1-[4-(2-methylpropyl)phenyl]ethyl]-2,3-dihydro-1,4-benzoxazine-2-carboxamide
—— (2R)-4-acetyl-N-[5-[(4-methylphenyl)methyl]-1,3-thiazol-2-yl]-2,3-dihydro-1,4-benzoxazine-2-carboxamide —— C22H21N3O3S
(2R)-4-acetyl-N-[5-[(4-methylphenyl)methyl]-1,3-thiazol-2-yl]-2,3-dihydro-1,4-benzoxazine-2-carboxamide
—— (2R)-4-acetyl-N-[(1S)-1-[3-(trifluoromethyl)phenyl]ethyl]-2,3-dihydro-1,4-benzoxazine-2-carboxamide —— C20H19F3N2O3
(2R)-4-acetyl-N-[(1S)-1-[3-(trifluoromethyl)phenyl]ethyl]-2,3-dihydro-1,4-benzoxazine-2-carboxamide
—— N,N-diethyl-4-[(6-methyl-3-oxo-1,4-benzoxazin-4-yl)methyl]benzamide —— C21H24N2O3
N,N-diethyl-4-[(6-methyl-3-oxo-1,4-benzoxazin-4-yl)methyl]benzamide
—— (2S)-4-[2-[2-[(4-chlorophenoxy)methyl]-1,3-thiazol-4-yl]acetyl]-N-methyl-2,3-dihydro-1,4-benzoxazine-2-carboxamide —— C22H20ClN3O4S
(2S)-4-[2-[2-[(4-chlorophenoxy)methyl]-1,3-thiazol-4-yl]acetyl]-N-methyl-2,3-dihydro-1,4-benzoxazine-2-carboxamide
—— 1-[3-[(2R)-2-(morpholine-4-carbonyl)-2,3-dihydro-1,4-benzoxazin-4-yl]-3-oxopropyl]-3-propylbenzimidazol-2-one —— C26H30N4O5
1-[3-[(2R)-2-(morpholine-4-carbonyl)-2,3-dihydro-1,4-benzoxazin-4-yl]-3-oxopropyl]-3-propylbenzimidazol-2-one
—— (2S)-4-[3-[5-(4-methoxyphenyl)furan-2-yl]propanoyl]-N-methyl-2,3-dihydro-1,4-benzoxazine-2-carboxamide —— C24H24N2O5
(2S)-4-[3-[5-(4-methoxyphenyl)furan-2-yl]propanoyl]-N-methyl-2,3-dihydro-1,4-benzoxazine-2-carboxamide
—— 1-[2-[(2S)-2-(morpholine-4-carbonyl)-2,3-dihydro-1,4-benzoxazin-4-yl]-2-oxoethyl]-3-propylbenzimidazol-2-one —— C25H28N4O5
1-[2-[(2S)-2-(morpholine-4-carbonyl)-2,3-dihydro-1,4-benzoxazin-4-yl]-2-oxoethyl]-3-propylbenzimidazol-2-one
—— (2R)-4-[3-[5-(4-methoxyphenyl)furan-2-yl]propanoyl]-N-methyl-2,3-dihydro-1,4-benzoxazine-2-carboxamide —— C24H24N2O5
(2R)-4-[3-[5-(4-methoxyphenyl)furan-2-yl]propanoyl]-N-methyl-2,3-dihydro-1,4-benzoxazine-2-carboxamide
—— (2R)-4-[2-[2-[(4-chlorophenoxy)methyl]-1,3-thiazol-4-yl]acetyl]-N-methyl-2,3-dihydro-1,4-benzoxazine-2-carboxamide —— C22H20ClN3O4S
(2R)-4-[2-[2-[(4-chlorophenoxy)methyl]-1,3-thiazol-4-yl]acetyl]-N-methyl-2,3-dihydro-1,4-benzoxazine-2-carboxamide
—— 1-[2-[(2R)-2-(morpholine-4-carbonyl)-2,3-dihydro-1,4-benzoxazin-4-yl]-2-oxoethyl]-3-propylbenzimidazol-2-one —— C25H28N4O5
1-[2-[(2R)-2-(morpholine-4-carbonyl)-2,3-dihydro-1,4-benzoxazin-4-yl]-2-oxoethyl]-3-propylbenzimidazol-2-one
—— 1-[3-[(2S)-2-(morpholine-4-carbonyl)-2,3-dihydro-1,4-benzoxazin-4-yl]-3-oxopropyl]-3-propylbenzimidazol-2-one —— C26H30N4O5
1-[3-[(2S)-2-(morpholine-4-carbonyl)-2,3-dihydro-1,4-benzoxazin-4-yl]-3-oxopropyl]-3-propylbenzimidazol-2-one
—— 3-ethoxy-4-[2-[(2S)-2-(morpholine-4-carbonyl)-2,3-dihydro-1,4-benzoxazin-4-yl]-2-oxoethoxy]benzonitrile —— C24H25N3O6
3-ethoxy-4-[2-[(2S)-2-(morpholine-4-carbonyl)-2,3-dihydro-1,4-benzoxazin-4-yl]-2-oxoethoxy]benzonitrile
—— [(2R)-4-(6-chloro-2H-chromene-3-carbonyl)-2,3-dihydro-1,4-benzoxazin-2-yl]-morpholin-4-ylmethanone —— C23H21ClN2O5
[(2R)-4-(6-chloro-2H-chromene-3-carbonyl)-2,3-dihydro-1,4-benzoxazin-2-yl]-morpholin-4-ylmethanone
—— (2S)-4-acetyl-N'-[4-[(4-chlorophenyl)sulfanylmethyl]benzoyl]-2,3-dihydro-1,4-benzoxazine-2-carbohydrazide —— C25H22ClN3O4S
(2S)-4-acetyl-N'-[4-[(4-chlorophenyl)sulfanylmethyl]benzoyl]-2,3-dihydro-1,4-benzoxazine-2-carbohydrazide
—— 2-(4-BR-Phenyl)-5-(2-chlorophenyl)-1,10B-dihydropyrazolo(1,5-C)(1,3)benzoxazine —— C22H16BrClN2O
2-(4-BR-Phenyl)-5-(2-chlorophenyl)-1,10B-dihydropyrazolo(1,5-C)(1,3)benzoxazine
—— (2R)-4-(6-chloro-2H-chromene-3-carbonyl)-N-methyl-2,3-dihydro-1,4-benzoxazine-2-carboxamide —— C20H17ClN2O4
(2R)-4-(6-chloro-2H-chromene-3-carbonyl)-N-methyl-2,3-dihydro-1,4-benzoxazine-2-carboxamide
—— [(2S)-4-(6-chloro-2H-chromene-3-carbonyl)-2,3-dihydro-1,4-benzoxazin-2-yl]-morpholin-4-ylmethanone —— C23H21ClN2O5
[(2S)-4-(6-chloro-2H-chromene-3-carbonyl)-2,3-dihydro-1,4-benzoxazin-2-yl]-morpholin-4-ylmethanone
—— (2R)-4-acetyl-N'-[4-[(4-chlorophenyl)sulfanylmethyl]benzoyl]-2,3-dihydro-1,4-benzoxazine-2-carbohydrazide —— C25H22ClN3O4S
(2R)-4-acetyl-N'-[4-[(4-chlorophenyl)sulfanylmethyl]benzoyl]-2,3-dihydro-1,4-benzoxazine-2-carbohydrazide
—— 6-(2-Methylbutan-2-yl)-4-(4-oxo-4-pyrrolidin-1-ylbutyl)-1,4-benzoxazin-3-one —— C21H30N2O3
6-(2-Methylbutan-2-yl)-4-(4-oxo-4-pyrrolidin-1-ylbutyl)-1,4-benzoxazin-3-one
—— 5-[(6-tert-butyl-3-oxo-1,4-benzoxazin-4-yl)methyl]-N,N-dipropylfuran-2-carboxamide —— C24H32N2O4
5-[(6-tert-butyl-3-oxo-1,4-benzoxazin-4-yl)methyl]-N,N-dipropylfuran-2-carboxamide
—— 3-[5,7-dimethyl-2-(trifluoromethyl)-[1,2,4]triazolo[1,5-a]pyrimidin-6-yl]-N-[[(2R)-4-ethyl-2,3-dihydro-1,4-benzoxazin-2-yl]methyl]-N-methylpropanamide —— C23H27F3N6O2
3-[5,7-dimethyl-2-(trifluoromethyl)-[1,2,4]triazolo[1,5-a]pyrimidin-6-yl]-N-[[(2R)-4-ethyl-2,3-dihydro-1,4-benzoxazin-2-yl]methyl]-N-methylpropanamide
—— (2S)-4-acetyl-N-[(1R)-1-(4-bromophenyl)ethyl]-2,3-dihydro-1,4-benzoxazine-2-carboxamide —— C19H19BrN2O3
(2S)-4-acetyl-N-[(1R)-1-(4-bromophenyl)ethyl]-2,3-dihydro-1,4-benzoxazine-2-carboxamide
—— (2R)-4-acetyl-N-[(1R)-1-(4-bromophenyl)ethyl]-2,3-dihydro-1,4-benzoxazine-2-carboxamide —— C19H19BrN2O3
(2R)-4-acetyl-N-[(1R)-1-(4-bromophenyl)ethyl]-2,3-dihydro-1,4-benzoxazine-2-carboxamide
—— (2R)-4-acetyl-N-[(1S)-1-(4-bromophenyl)ethyl]-2,3-dihydro-1,4-benzoxazine-2-carboxamide —— C19H19BrN2O3
(2R)-4-acetyl-N-[(1S)-1-(4-bromophenyl)ethyl]-2,3-dihydro-1,4-benzoxazine-2-carboxamide
—— (2S)-N-methyl-4-(4-morpholin-4-ylsulfonylphenyl)sulfonyl-2,3-dihydro-1,4-benzoxazine-2-carboxamide —— C20H23N3O7S2
(2S)-N-methyl-4-(4-morpholin-4-ylsulfonylphenyl)sulfonyl-2,3-dihydro-1,4-benzoxazine-2-carboxamide
—— (2R)-N-methyl-4-(4-morpholin-4-ylsulfonylphenyl)sulfonyl-2,3-dihydro-1,4-benzoxazine-2-carboxamide —— C20H23N3O7S2
(2R)-N-methyl-4-(4-morpholin-4-ylsulfonylphenyl)sulfonyl-2,3-dihydro-1,4-benzoxazine-2-carboxamide
—— (2R)-4-(3-bromo-4-methoxyphenyl)sulfonyl-N-methyl-2,3-dihydro-1,4-benzoxazine-2-carboxamide —— C17H17BrN2O5S
(2R)-4-(3-bromo-4-methoxyphenyl)sulfonyl-N-methyl-2,3-dihydro-1,4-benzoxazine-2-carboxamide
—— (2S)-4-(3-bromo-4-methoxyphenyl)sulfonyl-N-methyl-2,3-dihydro-1,4-benzoxazine-2-carboxamide —— C17H17BrN2O5S
(2S)-4-(3-bromo-4-methoxyphenyl)sulfonyl-N-methyl-2,3-dihydro-1,4-benzoxazine-2-carboxamide
—— 9-Bromo-2-(4-ethylphenyl)-5-isopropyl-1,10b-dihydropyrazolo[1,5-c][1,3]benzoxazine —— C21H23BrN2O
9-Bromo-2-(4-ethylphenyl)-5-isopropyl-1,10b-dihydropyrazolo[1,5-c][1,3]benzoxazine
—— N-[(4R)-6-fluoro-3,4-dihydro-2H-thiochromen-4-yl]-2-(4-oxo-2,3-dihydro-1,5-benzoxazepin-5-yl)acetamide —— C20H19FN2O3S
N-[(4R)-6-fluoro-3,4-dihydro-2H-thiochromen-4-yl]-2-(4-oxo-2,3-dihydro-1,5-benzoxazepin-5-yl)acetamide
—— N-[(4S)-6-fluoro-3,4-dihydro-2H-thiochromen-4-yl]-2-(4-oxo-2,3-dihydro-1,5-benzoxazepin-5-yl)acetamide —— C20H19FN2O3S
N-[(4S)-6-fluoro-3,4-dihydro-2H-thiochromen-4-yl]-2-(4-oxo-2,3-dihydro-1,5-benzoxazepin-5-yl)acetamide
—— [(2R)-4-(3-fluoro-4-methylbenzoyl)-2,3-dihydro-1,4-benzoxazin-2-yl]-morpholin-4-ylmethanone —— C21H21FN2O4
[(2R)-4-(3-fluoro-4-methylbenzoyl)-2,3-dihydro-1,4-benzoxazin-2-yl]-morpholin-4-ylmethanone
—— (2R)-N-methyl-4-[2-[2-[2-(4-methyl-1,3-thiazol-2-yl)acetyl]hydrazinyl]-2-oxoethyl]-2,3-dihydro-1,4-benzoxazine-2-carboxamide —— C18H21N5O4S
(2R)-N-methyl-4-[2-[2-[2-(4-methyl-1,3-thiazol-2-yl)acetyl]hydrazinyl]-2-oxoethyl]-2,3-dihydro-1,4-benzoxazine-2-carboxamide
—— 2-[2-(2-chlorophenyl)-1,3-thiazol-4-yl]-1-[(2R)-2-(morpholine-4-carbonyl)-2,3-dihydro-1,4-benzoxazin-4-yl]ethanone —— C24H22ClN3O4S
2-[2-(2-chlorophenyl)-1,3-thiazol-4-yl]-1-[(2R)-2-(morpholine-4-carbonyl)-2,3-dihydro-1,4-benzoxazin-4-yl]ethanone
—— (2S)-4-[2-[[2-[4-chloro-3-(trifluoromethyl)anilino]-2-oxoethyl]-methylamino]-2-oxoethyl]-N-methyl-2,3-dihydro-1,4-benzoxazine-2-carboxamide —— C22H22ClF3N4O4
(2S)-4-[2-[[2-[4-chloro-3-(trifluoromethyl)anilino]-2-oxoethyl]-methylamino]-2-oxoethyl]-N-methyl-2,3-dihydro-1,4-benzoxazine-2-carboxamide
—— [(2R)-4-(2,5-dichlorothiophene-3-carbonyl)-2,3-dihydro-1,4-benzoxazin-2-yl]-morpholin-4-ylmethanone —— C18H16Cl2N2O4S
[(2R)-4-(2,5-dichlorothiophene-3-carbonyl)-2,3-dihydro-1,4-benzoxazin-2-yl]-morpholin-4-ylmethanone
—— (2R)-N-methyl-4-[[4-(trifluoromethyl)phenyl]methyl]-2,3-dihydro-1,4-benzoxazine-2-carboxamide —— C18H17F3N2O2
(2R)-N-methyl-4-[[4-(trifluoromethyl)phenyl]methyl]-2,3-dihydro-1,4-benzoxazine-2-carboxamide
—— (2R)-4-[2-[[2-[4-chloro-3-(trifluoromethyl)anilino]-2-oxoethyl]-methylamino]-2-oxoethyl]-N-methyl-2,3-dihydro-1,4-benzoxazine-2-carboxamide —— C22H22ClF3N4O4
(2R)-4-[2-[[2-[4-chloro-3-(trifluoromethyl)anilino]-2-oxoethyl]-methylamino]-2-oxoethyl]-N-methyl-2,3-dihydro-1,4-benzoxazine-2-carboxamide
—— (2S)-N-methyl-4-[2-[2-[2-(4-methyl-1,3-thiazol-2-yl)acetyl]hydrazinyl]-2-oxoethyl]-2,3-dihydro-1,4-benzoxazine-2-carboxamide —— C18H21N5O4S
(2S)-N-methyl-4-[2-[2-[2-(4-methyl-1,3-thiazol-2-yl)acetyl]hydrazinyl]-2-oxoethyl]-2,3-dihydro-1,4-benzoxazine-2-carboxamide
—— 1-[(2S)-2-(morpholine-4-carbonyl)-2,3-dihydro-1,4-benzoxazin-4-yl]-3-(5-phenylfuran-2-yl)propan-1-one —— C26H26N2O5
1-[(2S)-2-(morpholine-4-carbonyl)-2,3-dihydro-1,4-benzoxazin-4-yl]-3-(5-phenylfuran-2-yl)propan-1-one
—— (2R)-2-(4-bromophenoxy)-1-[(2S)-2-(morpholine-4-carbonyl)-2,3-dihydro-1,4-benzoxazin-4-yl]propan-1-one —— C22H23BrN2O5
(2R)-2-(4-bromophenoxy)-1-[(2S)-2-(morpholine-4-carbonyl)-2,3-dihydro-1,4-benzoxazin-4-yl]propan-1-one