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苯并恶嗪类

中文名称 英文名称 CAS号 化学式 结构式图片
—— 2-[[(2R)-2,6-dimethyl-3-oxo-4H-1,4-benzoxazin-7-yl]sulfonyl-methylamino]-N-(5-methylpyridin-2-yl)acetamide —— C19H22N4O5S
2-[[(2R)-2,6-dimethyl-3-oxo-4H-1,4-benzoxazin-7-yl]sulfonyl-methylamino]-N-(5-methylpyridin-2-yl)acetamide
—— N-cyclopentyl-2-[[(2R)-2,6-dimethyl-3-oxo-4H-1,4-benzoxazin-7-yl]sulfonyl-methylamino]acetamide —— C18H25N3O5S
N-cyclopentyl-2-[[(2R)-2,6-dimethyl-3-oxo-4H-1,4-benzoxazin-7-yl]sulfonyl-methylamino]acetamide
—— (2S)-2-([1,2,4]triazolo[4,3-a]pyrazin-3-yl)-3,4-dihydro-2H-1,4-benzoxazine —— C13H11N5O
(2S)-2-([1,2,4]triazolo[4,3-a]pyrazin-3-yl)-3,4-dihydro-2H-1,4-benzoxazine
—— 2-[[(2S)-2,6-dimethyl-3-oxo-4H-1,4-benzoxazin-7-yl]sulfonyl-methylamino]-N-(3-methoxyphenyl)acetamide —— C20H23N3O6S
2-[[(2S)-2,6-dimethyl-3-oxo-4H-1,4-benzoxazin-7-yl]sulfonyl-methylamino]-N-(3-methoxyphenyl)acetamide
—— N,6-dimethyl-N-[2-[(2R)-2-methylpiperidin-1-yl]-2-oxoethyl]-3-oxo-4H-1,4-benzoxazine-7-sulfonamide —— C18H25N3O5S
N,6-dimethyl-N-[2-[(2R)-2-methylpiperidin-1-yl]-2-oxoethyl]-3-oxo-4H-1,4-benzoxazine-7-sulfonamide
—— 2-[[(2R)-2,6-dimethyl-3-oxo-4H-1,4-benzoxazin-7-yl]sulfonyl-methylamino]-N-(2-methoxy-5-methylphenyl)acetamide —— C21H25N3O6S
2-[[(2R)-2,6-dimethyl-3-oxo-4H-1,4-benzoxazin-7-yl]sulfonyl-methylamino]-N-(2-methoxy-5-methylphenyl)acetamide
—— (2S)-N-[2-(3,4-dihydro-1H-isoquinolin-2-yl)-2-oxoethyl]-N,2,6-trimethyl-3-oxo-4H-1,4-benzoxazine-7-sulfonamide —— C22H25N3O5S
(2S)-N-[2-(3,4-dihydro-1H-isoquinolin-2-yl)-2-oxoethyl]-N,2,6-trimethyl-3-oxo-4H-1,4-benzoxazine-7-sulfonamide
—— N,6-dimethyl-N-[2-[(2S)-2-methylpiperidin-1-yl]-2-oxoethyl]-3-oxo-4H-1,4-benzoxazine-7-sulfonamide —— C18H25N3O5S
N,6-dimethyl-N-[2-[(2S)-2-methylpiperidin-1-yl]-2-oxoethyl]-3-oxo-4H-1,4-benzoxazine-7-sulfonamide
—— (2R)-N-[2-(1,4-dioxa-8-azaspiro[4.5]decan-8-yl)-2-oxoethyl]-N,2,6-trimethyl-3-oxo-4H-1,4-benzoxazine-7-sulfonamide —— C20H27N3O7S
(2R)-N-[2-(1,4-dioxa-8-azaspiro[4.5]decan-8-yl)-2-oxoethyl]-N,2,6-trimethyl-3-oxo-4H-1,4-benzoxazine-7-sulfonamide
—— 2-[[(2R)-2,6-dimethyl-3-oxo-4H-1,4-benzoxazin-7-yl]sulfonyl-methylamino]-N-(2-ethyl-6-methylphenyl)acetamide —— C22H27N3O5S
2-[[(2R)-2,6-dimethyl-3-oxo-4H-1,4-benzoxazin-7-yl]sulfonyl-methylamino]-N-(2-ethyl-6-methylphenyl)acetamide
—— (2S)-N,2,6-trimethyl-3-oxo-N-[2-oxo-2-(4-phenyl-3,6-dihydro-2H-pyridin-1-yl)ethyl]-4H-1,4-benzoxazine-7-sulfonamide —— C24H27N3O5S
(2S)-N,2,6-trimethyl-3-oxo-N-[2-oxo-2-(4-phenyl-3,6-dihydro-2H-pyridin-1-yl)ethyl]-4H-1,4-benzoxazine-7-sulfonamide
—— 2-[[(2R)-2,6-dimethyl-3-oxo-4H-1,4-benzoxazin-7-yl]sulfonyl-methylamino]-N-(3-methylbutyl)acetamide —— C18H27N3O5S
2-[[(2R)-2,6-dimethyl-3-oxo-4H-1,4-benzoxazin-7-yl]sulfonyl-methylamino]-N-(3-methylbutyl)acetamide
—— 7-amino-6-[(2S)-2-methylmorpholin-4-yl]-4H-1,4-benzoxazin-3-one —— C13H17N3O3
7-amino-6-[(2S)-2-methylmorpholin-4-yl]-4H-1,4-benzoxazin-3-one
—— 2-[[(2S)-2,6-dimethyl-3-oxo-4H-1,4-benzoxazin-7-yl]sulfonyl-methylamino]-N-[(3-methoxyphenyl)methyl]acetamide —— C21H25N3O6S
2-[[(2S)-2,6-dimethyl-3-oxo-4H-1,4-benzoxazin-7-yl]sulfonyl-methylamino]-N-[(3-methoxyphenyl)methyl]acetamide
—— 2-[[(2R)-2,6-dimethyl-3-oxo-4H-1,4-benzoxazin-7-yl]sulfonyl-methylamino]-N-(pyridin-2-ylmethyl)acetamide —— C19H22N4O5S
2-[[(2R)-2,6-dimethyl-3-oxo-4H-1,4-benzoxazin-7-yl]sulfonyl-methylamino]-N-(pyridin-2-ylmethyl)acetamide
—— 2-[[(2R)-2,6-dimethyl-3-oxo-4H-1,4-benzoxazin-7-yl]sulfonyl-methylamino]-N-propylacetamide —— C16H23N3O5S
2-[[(2R)-2,6-dimethyl-3-oxo-4H-1,4-benzoxazin-7-yl]sulfonyl-methylamino]-N-propylacetamide
—— N-(2,4-dimethoxyphenyl)-2-[[(2S)-2,6-dimethyl-3-oxo-4H-1,4-benzoxazin-7-yl]sulfonyl-methylamino]acetamide —— C21H25N3O7S
N-(2,4-dimethoxyphenyl)-2-[[(2S)-2,6-dimethyl-3-oxo-4H-1,4-benzoxazin-7-yl]sulfonyl-methylamino]acetamide
—— 2-[[(2R)-2,6-dimethyl-3-oxo-4H-1,4-benzoxazin-7-yl]sulfonyl-methylamino]-N-(4-methylpyridin-2-yl)acetamide —— C19H22N4O5S
2-[[(2R)-2,6-dimethyl-3-oxo-4H-1,4-benzoxazin-7-yl]sulfonyl-methylamino]-N-(4-methylpyridin-2-yl)acetamide
—— 2-[[(2S)-2,6-dimethyl-3-oxo-4H-1,4-benzoxazin-7-yl]sulfonyl-methylamino]-N-(3,5-dimethylphenyl)acetamide —— C21H25N3O5S
2-[[(2S)-2,6-dimethyl-3-oxo-4H-1,4-benzoxazin-7-yl]sulfonyl-methylamino]-N-(3,5-dimethylphenyl)acetamide
—— N-[2-(cyclohexen-1-yl)ethyl]-2-[[(2S)-2,6-dimethyl-3-oxo-4H-1,4-benzoxazin-7-yl]sulfonyl-methylamino]acetamide —— C21H29N3O5S
N-[2-(cyclohexen-1-yl)ethyl]-2-[[(2S)-2,6-dimethyl-3-oxo-4H-1,4-benzoxazin-7-yl]sulfonyl-methylamino]acetamide
—— (2R)-N-[2-(2,3-dihydroindol-1-yl)-2-oxoethyl]-N,2,6-trimethyl-3-oxo-4H-1,4-benzoxazine-7-sulfonamide —— C21H23N3O5S
(2R)-N-[2-(2,3-dihydroindol-1-yl)-2-oxoethyl]-N,2,6-trimethyl-3-oxo-4H-1,4-benzoxazine-7-sulfonamide
—— 2-[[(2R)-2,6-dimethyl-3-oxo-4H-1,4-benzoxazin-7-yl]sulfonyl-methylamino]-N-(4-fluoro-2-methylphenyl)acetamide —— C20H22FN3O5S
2-[[(2R)-2,6-dimethyl-3-oxo-4H-1,4-benzoxazin-7-yl]sulfonyl-methylamino]-N-(4-fluoro-2-methylphenyl)acetamide
—— 2-[[(2S)-2,6-dimethyl-3-oxo-4H-1,4-benzoxazin-7-yl]sulfonyl-methylamino]-N-(2,3-dimethylphenyl)acetamide —— C21H25N3O5S
2-[[(2S)-2,6-dimethyl-3-oxo-4H-1,4-benzoxazin-7-yl]sulfonyl-methylamino]-N-(2,3-dimethylphenyl)acetamide
—— N-(2,4-difluorophenyl)-2-[[(2R)-2,6-dimethyl-3-oxo-4H-1,4-benzoxazin-7-yl]sulfonyl-methylamino]acetamide —— C19H19F2N3O5S
N-(2,4-difluorophenyl)-2-[[(2R)-2,6-dimethyl-3-oxo-4H-1,4-benzoxazin-7-yl]sulfonyl-methylamino]acetamide
—— N-(2-bromo-4-methylphenyl)-2-[[(2R)-2,6-dimethyl-3-oxo-4H-1,4-benzoxazin-7-yl]sulfonyl-methylamino]acetamide —— C20H22BrN3O5S
N-(2-bromo-4-methylphenyl)-2-[[(2R)-2,6-dimethyl-3-oxo-4H-1,4-benzoxazin-7-yl]sulfonyl-methylamino]acetamide
—— 7-amino-6-[[(2S)-pentan-2-yl]amino]-4H-1,4-benzoxazin-3-one —— C13H19N3O2
7-amino-6-[[(2S)-pentan-2-yl]amino]-4H-1,4-benzoxazin-3-one
—— N-(4-bromo-3-methylphenyl)-2-[[(2R)-2,6-dimethyl-3-oxo-4H-1,4-benzoxazin-7-yl]sulfonyl-methylamino]acetamide —— C20H22BrN3O5S
N-(4-bromo-3-methylphenyl)-2-[[(2R)-2,6-dimethyl-3-oxo-4H-1,4-benzoxazin-7-yl]sulfonyl-methylamino]acetamide
—— 2-[[(2R)-2,6-dimethyl-3-oxo-4H-1,4-benzoxazin-7-yl]sulfonyl-methylamino]-N-[(5-methylfuran-2-yl)methyl]acetamide —— C19H23N3O6S
2-[[(2R)-2,6-dimethyl-3-oxo-4H-1,4-benzoxazin-7-yl]sulfonyl-methylamino]-N-[(5-methylfuran-2-yl)methyl]acetamide
—— N-[(2R)-butan-2-yl]-2-[(6-chloro-3-oxo-4H-1,4-benzoxazin-7-yl)sulfonyl-methylamino]acetamide —— C15H20ClN3O5S
N-[(2R)-butan-2-yl]-2-[(6-chloro-3-oxo-4H-1,4-benzoxazin-7-yl)sulfonyl-methylamino]acetamide
—— N-(2-chloro-4-methylphenyl)-2-[[(2S)-2,6-dimethyl-3-oxo-4H-1,4-benzoxazin-7-yl]sulfonyl-methylamino]acetamide —— C20H22ClN3O5S
N-(2-chloro-4-methylphenyl)-2-[[(2S)-2,6-dimethyl-3-oxo-4H-1,4-benzoxazin-7-yl]sulfonyl-methylamino]acetamide
—— 2-[[(2S)-2,6-dimethyl-3-oxo-4H-1,4-benzoxazin-7-yl]sulfonyl-methylamino]-N-[(4-methylphenyl)methyl]acetamide —— C21H25N3O5S
2-[[(2S)-2,6-dimethyl-3-oxo-4H-1,4-benzoxazin-7-yl]sulfonyl-methylamino]-N-[(4-methylphenyl)methyl]acetamide
—— N-tert-butyl-2-[[(2S)-2,6-dimethyl-3-oxo-4H-1,4-benzoxazin-7-yl]sulfonyl-methylamino]acetamide —— C17H25N3O5S
N-tert-butyl-2-[[(2S)-2,6-dimethyl-3-oxo-4H-1,4-benzoxazin-7-yl]sulfonyl-methylamino]acetamide
—— 7-amino-6-[(2R)-2-methylmorpholin-4-yl]-4H-1,4-benzoxazin-3-one —— C13H17N3O3
7-amino-6-[(2R)-2-methylmorpholin-4-yl]-4H-1,4-benzoxazin-3-one
—— N-(2,4-difluorophenyl)-2-[[(2S)-2,6-dimethyl-3-oxo-4H-1,4-benzoxazin-7-yl]sulfonyl-methylamino]acetamide —— C19H19F2N3O5S
N-(2,4-difluorophenyl)-2-[[(2S)-2,6-dimethyl-3-oxo-4H-1,4-benzoxazin-7-yl]sulfonyl-methylamino]acetamide
—— 2-[[(2R)-2,6-dimethyl-3-oxo-4H-1,4-benzoxazin-7-yl]sulfonyl-methylamino]-N-(2-methylbutan-2-yl)acetamide —— C18H27N3O5S
2-[[(2R)-2,6-dimethyl-3-oxo-4H-1,4-benzoxazin-7-yl]sulfonyl-methylamino]-N-(2-methylbutan-2-yl)acetamide
—— N-[2-(cyclohexen-1-yl)ethyl]-2-[[(2R)-2,6-dimethyl-3-oxo-4H-1,4-benzoxazin-7-yl]sulfonyl-methylamino]acetamide —— C21H29N3O5S
N-[2-(cyclohexen-1-yl)ethyl]-2-[[(2R)-2,6-dimethyl-3-oxo-4H-1,4-benzoxazin-7-yl]sulfonyl-methylamino]acetamide
—— 7-amino-6-[[(2R)-butan-2-yl]amino]-4H-1,4-benzoxazin-3-one —— C12H17N3O2
7-amino-6-[[(2R)-butan-2-yl]amino]-4H-1,4-benzoxazin-3-one
—— 2-[[(2R)-2,6-dimethyl-3-oxo-4H-1,4-benzoxazin-7-yl]sulfonyl-methylamino]-N-(2,4-dimethylphenyl)acetamide —— C21H25N3O5S
2-[[(2R)-2,6-dimethyl-3-oxo-4H-1,4-benzoxazin-7-yl]sulfonyl-methylamino]-N-(2,4-dimethylphenyl)acetamide
—— 2-[[(2S)-2,6-dimethyl-3-oxo-4H-1,4-benzoxazin-7-yl]sulfonyl-methylamino]-N-(2-ethyl-6-methylphenyl)acetamide —— C22H27N3O5S
2-[[(2S)-2,6-dimethyl-3-oxo-4H-1,4-benzoxazin-7-yl]sulfonyl-methylamino]-N-(2-ethyl-6-methylphenyl)acetamide
—— (2S)-N-[2-(3,4-dihydro-2H-quinolin-1-yl)-2-oxoethyl]-N,2,6-trimethyl-3-oxo-4H-1,4-benzoxazine-7-sulfonamide —— C22H25N3O5S
(2S)-N-[2-(3,4-dihydro-2H-quinolin-1-yl)-2-oxoethyl]-N,2,6-trimethyl-3-oxo-4H-1,4-benzoxazine-7-sulfonamide
—— 2-[(6-chloro-3-oxo-4H-1,4-benzoxazin-7-yl)sulfonyl-methylamino]-N-[[(2S)-oxolan-2-yl]methyl]acetamide —— C16H20ClN3O6S
2-[(6-chloro-3-oxo-4H-1,4-benzoxazin-7-yl)sulfonyl-methylamino]-N-[[(2S)-oxolan-2-yl]methyl]acetamide
—— 6-chloro-N-[2-[(2S)-2-ethylpiperidin-1-yl]-2-oxoethyl]-N-methyl-3-oxo-4H-1,4-benzoxazine-7-sulfonamide —— C18H24ClN3O5S
6-chloro-N-[2-[(2S)-2-ethylpiperidin-1-yl]-2-oxoethyl]-N-methyl-3-oxo-4H-1,4-benzoxazine-7-sulfonamide
—— (2R)-2-([1,2,4]triazolo[4,3-a]pyrazin-3-yl)-3,4-dihydro-2H-1,4-benzoxazine —— C13H11N5O
(2R)-2-([1,2,4]triazolo[4,3-a]pyrazin-3-yl)-3,4-dihydro-2H-1,4-benzoxazine
—— ethyl (3R)-1-[2-[methyl-[(6-methyl-3-oxo-4H-1,4-benzoxazin-7-yl)sulfonyl]amino]acetyl]piperidine-3-carboxylate —— C20H27N3O7S
ethyl (3R)-1-[2-[methyl-[(6-methyl-3-oxo-4H-1,4-benzoxazin-7-yl)sulfonyl]amino]acetyl]piperidine-3-carboxylate
—— N-(5-chloropyridin-2-yl)-2-[[(2S)-2,6-dimethyl-3-oxo-4H-1,4-benzoxazin-7-yl]sulfonyl-methylamino]acetamide —— C18H19ClN4O5S
N-(5-chloropyridin-2-yl)-2-[[(2S)-2,6-dimethyl-3-oxo-4H-1,4-benzoxazin-7-yl]sulfonyl-methylamino]acetamide
—— N-(2-chloro-4-methylphenyl)-2-[[(2R)-2,6-dimethyl-3-oxo-4H-1,4-benzoxazin-7-yl]sulfonyl-methylamino]acetamide —— C20H22ClN3O5S
N-(2-chloro-4-methylphenyl)-2-[[(2R)-2,6-dimethyl-3-oxo-4H-1,4-benzoxazin-7-yl]sulfonyl-methylamino]acetamide
—— 2-[[(2R)-2,6-dimethyl-3-oxo-4H-1,4-benzoxazin-7-yl]sulfonyl-methylamino]-N-[(2-methoxyphenyl)methyl]acetamide —— C21H25N3O6S
2-[[(2R)-2,6-dimethyl-3-oxo-4H-1,4-benzoxazin-7-yl]sulfonyl-methylamino]-N-[(2-methoxyphenyl)methyl]acetamide
—— 2-[[(2R)-2,6-dimethyl-3-oxo-4H-1,4-benzoxazin-7-yl]sulfonyl-methylamino]-N-ethyl-N-(3-methylphenyl)acetamide —— C22H27N3O5S
2-[[(2R)-2,6-dimethyl-3-oxo-4H-1,4-benzoxazin-7-yl]sulfonyl-methylamino]-N-ethyl-N-(3-methylphenyl)acetamide
—— 2-[[(2R)-2,6-dimethyl-3-oxo-4H-1,4-benzoxazin-7-yl]sulfonyl-methylamino]-N-[3-(trifluoromethyl)phenyl]acetamide —— C20H20F3N3O5S
2-[[(2R)-2,6-dimethyl-3-oxo-4H-1,4-benzoxazin-7-yl]sulfonyl-methylamino]-N-[3-(trifluoromethyl)phenyl]acetamide
—— 2-[[(2S)-2,6-dimethyl-3-oxo-4H-1,4-benzoxazin-7-yl]sulfonyl-methylamino]-N-(2-methylphenyl)acetamide —— C20H23N3O5S
2-[[(2S)-2,6-dimethyl-3-oxo-4H-1,4-benzoxazin-7-yl]sulfonyl-methylamino]-N-(2-methylphenyl)acetamide