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苯并恶嗪类

中文名称 英文名称 CAS号 化学式 结构式图片
—— 1-[4'-(Dimethylamino)spiro[3,5-dihydro-1,4-benzoxazepine-2,1'-cyclohexane]-4-yl]-2-(3-methylphenyl)ethanone —— C25H32N2O2
1-[4'-(Dimethylamino)spiro[3,5-dihydro-1,4-benzoxazepine-2,1'-cyclohexane]-4-yl]-2-(3-methylphenyl)ethanone
—— 3-[(2S)-2-(2-fluorophenyl)-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-1-[4-[(1-methylimidazol-2-yl)methyl]piperazin-1-yl]propan-1-one —— C27H32FN5O2
3-[(2S)-2-(2-fluorophenyl)-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-1-[4-[(1-methylimidazol-2-yl)methyl]piperazin-1-yl]propan-1-one
—— 3-[(2R)-2-(2-fluorophenyl)-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-1-[4-[(1-methylimidazol-2-yl)methyl]piperazin-1-yl]propan-1-one —— C27H32FN5O2
3-[(2R)-2-(2-fluorophenyl)-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-1-[4-[(1-methylimidazol-2-yl)methyl]piperazin-1-yl]propan-1-one
—— 6-Bromo-3',5'-DI-tert-butyl-2-(4-nitrophenyl)-2,4-dihydrospiro[1,4-benzoxazine-3,1'-cyclohexane]-2',5'-dien-4'-one —— C27H29BrN2O4
6-Bromo-3',5'-DI-tert-butyl-2-(4-nitrophenyl)-2,4-dihydrospiro[1,4-benzoxazine-3,1'-cyclohexane]-2',5'-dien-4'-one
—— N-methyl-N-[4-(5-methyl-1-benzofuran-2-carbonyl)spiro[3,5-dihydro-1,4-benzoxazepine-2,4'-cyclohexane]-1'-yl]acetamide —— C27H30N2O4
N-methyl-N-[4-(5-methyl-1-benzofuran-2-carbonyl)spiro[3,5-dihydro-1,4-benzoxazepine-2,4'-cyclohexane]-1'-yl]acetamide
—— N-(4-acetylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-cyclohexane]-1'-yl)-N,5-dimethyl-1-benzofuran-2-carboxamide —— C27H30N2O4
N-(4-acetylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-cyclohexane]-1'-yl)-N,5-dimethyl-1-benzofuran-2-carboxamide
—— N,N-dimethyl-1-[(3S)-7-methyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-3-yl]methanamine —— C13H20N2O
N,N-dimethyl-1-[(3S)-7-methyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-3-yl]methanamine
—— 7-methyl-4-[(2R)-1-(4-methylpiperazin-1-yl)-1-oxopropan-2-yl]spiro[3H-1,4-benzoxazepine-2,4'-oxane]-5-one —— C22H31N3O4
7-methyl-4-[(2R)-1-(4-methylpiperazin-1-yl)-1-oxopropan-2-yl]spiro[3H-1,4-benzoxazepine-2,4'-oxane]-5-one
—— 7-Methyl-4-methylsulfonyl-1'-(2-pyrrolidin-1-ylethyl)spiro[3,5-dihydro-1,4-benzoxazepine-2,4'-piperidine] —— C21H33N3O3S
7-Methyl-4-methylsulfonyl-1'-(2-pyrrolidin-1-ylethyl)spiro[3,5-dihydro-1,4-benzoxazepine-2,4'-piperidine]
—— N,N-dimethyl-1-[(3S)-7-methyl-4-[(2-methylpyrimidin-5-yl)methyl]-3,5-dihydro-2H-1,4-benzoxazepin-3-yl]methanamine —— C19H26N4O
N,N-dimethyl-1-[(3S)-7-methyl-4-[(2-methylpyrimidin-5-yl)methyl]-3,5-dihydro-2H-1,4-benzoxazepin-3-yl]methanamine
—— 9'-Bromo-2'-(4-bromophenyl)-4-phenyl-1',10b'-dihydrospiro[cyclohexane-1,5'-pyrazolo[1,5-c][1,3]benzoxazine] —— C27H24Br2N2O
9'-Bromo-2'-(4-bromophenyl)-4-phenyl-1',10b'-dihydrospiro[cyclohexane-1,5'-pyrazolo[1,5-c][1,3]benzoxazine]
—— 1-[(2S)-1'-[2-[2-(3,5-dimethylpyrazol-1-yl)ethoxy]ethyl]-7-methylspiro[3,5-dihydro-1,4-benzoxazepine-2,3'-piperidine]-4-yl]ethanone —— C25H36N4O3
1-[(2S)-1'-[2-[2-(3,5-dimethylpyrazol-1-yl)ethoxy]ethyl]-7-methylspiro[3,5-dihydro-1,4-benzoxazepine-2,3'-piperidine]-4-yl]ethanone
—— 1-[(2S)-4-acetyl-7-methylspiro[3,5-dihydro-1,4-benzoxazepine-2,3'-piperidine]-1'-yl]-3-(1,2,4-triazol-1-yl)propan-1-one —— C21H27N5O3
1-[(2S)-4-acetyl-7-methylspiro[3,5-dihydro-1,4-benzoxazepine-2,3'-piperidine]-1'-yl]-3-(1,2,4-triazol-1-yl)propan-1-one
—— 1',7-dimethylspiro[4,5-dihydro-3H-1,4-benzoxazepine-2,4'-piperidine] —— C15H22N2O
1',7-dimethylspiro[4,5-dihydro-3H-1,4-benzoxazepine-2,4'-piperidine]
—— 1-[(2R)-1'-[2-[2-(3,5-dimethylpyrazol-1-yl)ethoxy]ethyl]-7-methylspiro[3,5-dihydro-1,4-benzoxazepine-2,3'-piperidine]-4-yl]ethanone —— C25H36N4O3
1-[(2R)-1'-[2-[2-(3,5-dimethylpyrazol-1-yl)ethoxy]ethyl]-7-methylspiro[3,5-dihydro-1,4-benzoxazepine-2,3'-piperidine]-4-yl]ethanone
—— 2-(1',7-dimethyl-5-oxospiro[3H-1,4-benzoxazepine-2,4'-piperidine]-4-yl)-N-(3-methoxypropyl)acetamide —— C21H31N3O4
2-(1',7-dimethyl-5-oxospiro[3H-1,4-benzoxazepine-2,4'-piperidine]-4-yl)-N-(3-methoxypropyl)acetamide
—— (2R)-2-(1',7-dimethyl-5-oxospiro[3H-1,4-benzoxazepine-2,4'-piperidine]-4-yl)-N-[[(2R)-oxolan-2-yl]methyl]propanamide —— C23H33N3O4
(2R)-2-(1',7-dimethyl-5-oxospiro[3H-1,4-benzoxazepine-2,4'-piperidine]-4-yl)-N-[[(2R)-oxolan-2-yl]methyl]propanamide
—— N,N-dimethyl-1-[(3R)-7-methyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-3-yl]methanamine —— C13H20N2O
N,N-dimethyl-1-[(3R)-7-methyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-3-yl]methanamine
—— (2R)-2-(1',7-dimethyl-5-oxospiro[3H-1,4-benzoxazepine-2,4'-piperidine]-4-yl)-N-propan-2-ylpropanamide —— C21H31N3O3
(2R)-2-(1',7-dimethyl-5-oxospiro[3H-1,4-benzoxazepine-2,4'-piperidine]-4-yl)-N-propan-2-ylpropanamide
—— 2-(1',7-dimethyl-5-oxospiro[3H-1,4-benzoxazepine-2,4'-piperidine]-4-yl)-N-methylacetamide —— C18H25N3O3
2-(1',7-dimethyl-5-oxospiro[3H-1,4-benzoxazepine-2,4'-piperidine]-4-yl)-N-methylacetamide
—— 1',7-dimethyl-4-(2-oxo-2-thiomorpholin-4-ylethyl)spiro[3H-1,4-benzoxazepine-2,4'-piperidine]-5-one —— C21H29N3O3S
1',7-dimethyl-4-(2-oxo-2-thiomorpholin-4-ylethyl)spiro[3H-1,4-benzoxazepine-2,4'-piperidine]-5-one
—— 7-methyl-4-[2-(4-methylpiperazin-1-yl)-2-oxoethyl]spiro[3H-1,4-benzoxazepine-2,4'-oxane]-5-one —— C21H29N3O4
7-methyl-4-[2-(4-methylpiperazin-1-yl)-2-oxoethyl]spiro[3H-1,4-benzoxazepine-2,4'-oxane]-5-one
—— 1-[(3S)-4-[(3-methoxyphenyl)methyl]-7-methyl-3,5-dihydro-2H-1,4-benzoxazepin-3-yl]-N,N-dimethylmethanamine —— C21H28N2O2
1-[(3S)-4-[(3-methoxyphenyl)methyl]-7-methyl-3,5-dihydro-2H-1,4-benzoxazepin-3-yl]-N,N-dimethylmethanamine
—— 2-(1',7-dimethyl-5-oxospiro[3H-1,4-benzoxazepine-2,4'-piperidine]-4-yl)-N-[(1S,2R)-2-methylcyclohexyl]acetamide —— C24H35N3O3
2-(1',7-dimethyl-5-oxospiro[3H-1,4-benzoxazepine-2,4'-piperidine]-4-yl)-N-[(1S,2R)-2-methylcyclohexyl]acetamide
—— 2-(1',7-dimethyl-5-oxospiro[3H-1,4-benzoxazepine-2,4'-piperidine]-4-yl)-N-(pyridin-4-ylmethyl)acetamide —— C23H28N4O3
2-(1',7-dimethyl-5-oxospiro[3H-1,4-benzoxazepine-2,4'-piperidine]-4-yl)-N-(pyridin-4-ylmethyl)acetamide
—— (2S)-2-(7-methyl-5-oxospiro[3H-1,4-benzoxazepine-2,4'-oxane]-4-yl)-N-(1-propan-2-ylpiperidin-4-yl)propanamide —— C25H37N3O4
(2S)-2-(7-methyl-5-oxospiro[3H-1,4-benzoxazepine-2,4'-oxane]-4-yl)-N-(1-propan-2-ylpiperidin-4-yl)propanamide
—— 2-imidazol-1-yl-1-[(2S)-7-methyl-4-methylsulfonylspiro[3,5-dihydro-1,4-benzoxazepine-2,3'-piperidine]-1'-yl]ethanone —— C20H26N4O4S
2-imidazol-1-yl-1-[(2S)-7-methyl-4-methylsulfonylspiro[3,5-dihydro-1,4-benzoxazepine-2,3'-piperidine]-1'-yl]ethanone
—— 2-(1',7-dimethyl-5-oxospiro[3H-1,4-benzoxazepine-2,4'-piperidine]-4-yl)-N-[(3R)-oxan-3-yl]acetamide —— C22H31N3O4
2-(1',7-dimethyl-5-oxospiro[3H-1,4-benzoxazepine-2,4'-piperidine]-4-yl)-N-[(3R)-oxan-3-yl]acetamide
—— 4-[(2R)-1-[2,2-bis(prop-2-enyl)azetidin-1-yl]-1-oxopropan-2-yl]-7-methylspiro[3H-1,4-benzoxazepine-2,4'-oxane]-5-one —— C26H34N2O4
4-[(2R)-1-[2,2-bis(prop-2-enyl)azetidin-1-yl]-1-oxopropan-2-yl]-7-methylspiro[3H-1,4-benzoxazepine-2,4'-oxane]-5-one
—— 4-[2-(azepan-1-yl)-2-oxoethyl]-1',7-dimethylspiro[3H-1,4-benzoxazepine-2,4'-piperidine]-5-one —— C23H33N3O3
4-[2-(azepan-1-yl)-2-oxoethyl]-1',7-dimethylspiro[3H-1,4-benzoxazepine-2,4'-piperidine]-5-one
—— N,N-dimethyl-1-[(3R)-7-methyl-4-[(5-methylthiophen-2-yl)methyl]-3,5-dihydro-2H-1,4-benzoxazepin-3-yl]methanamine —— C19H26N2OS
N,N-dimethyl-1-[(3R)-7-methyl-4-[(5-methylthiophen-2-yl)methyl]-3,5-dihydro-2H-1,4-benzoxazepin-3-yl]methanamine
—— 2-(1',7-dimethyl-5-oxospiro[3H-1,4-benzoxazepine-2,4'-piperidine]-4-yl)-N-[(2R)-3-methylbutan-2-yl]acetamide —— C22H33N3O3
2-(1',7-dimethyl-5-oxospiro[3H-1,4-benzoxazepine-2,4'-piperidine]-4-yl)-N-[(2R)-3-methylbutan-2-yl]acetamide
—— N,N-dimethyl-1-[(3R)-7-methyl-4-[(2-methylpyrimidin-5-yl)methyl]-3,5-dihydro-2H-1,4-benzoxazepin-3-yl]methanamine —— C19H26N4O
N,N-dimethyl-1-[(3R)-7-methyl-4-[(2-methylpyrimidin-5-yl)methyl]-3,5-dihydro-2H-1,4-benzoxazepin-3-yl]methanamine
—— N-[2-(4-fluorophenyl)ethyl]-7-methyl-5-oxospiro[3,4-dihydro-1,4-benzoxazepine-2,4'-cyclohexane]-1'-carboxamide —— C24H27FN2O3
N-[2-(4-fluorophenyl)ethyl]-7-methyl-5-oxospiro[3,4-dihydro-1,4-benzoxazepine-2,4'-cyclohexane]-1'-carboxamide
—— 7-methyl-4-[(2S)-1-(4-methylpiperazin-1-yl)-1-oxopropan-2-yl]spiro[3H-1,4-benzoxazepine-2,4'-oxane]-5-one —— C22H31N3O4
7-methyl-4-[(2S)-1-(4-methylpiperazin-1-yl)-1-oxopropan-2-yl]spiro[3H-1,4-benzoxazepine-2,4'-oxane]-5-one
—— 7-methyl-5-oxo-N-[[4-(trifluoromethyl)phenyl]methyl]spiro[3,4-dihydro-1,4-benzoxazepine-2,4'-cyclohexane]-1'-carboxamide —— C24H25F3N2O3
7-methyl-5-oxo-N-[[4-(trifluoromethyl)phenyl]methyl]spiro[3,4-dihydro-1,4-benzoxazepine-2,4'-cyclohexane]-1'-carboxamide
—— 1',7-dimethyl-4-[2-[(3R)-3-methylpiperidin-1-yl]-2-oxoethyl]spiro[3H-1,4-benzoxazepine-2,4'-piperidine]-5-one —— C23H33N3O3
1',7-dimethyl-4-[2-[(3R)-3-methylpiperidin-1-yl]-2-oxoethyl]spiro[3H-1,4-benzoxazepine-2,4'-piperidine]-5-one
—— N-[2-(2,4-dioxo-1,3-thiazolidin-3-yl)ethyl]-7-methyl-5-oxospiro[3,4-dihydro-1,4-benzoxazepine-2,4'-cyclohexane]-1'-carboxamide —— C21H25N3O5S
N-[2-(2,4-dioxo-1,3-thiazolidin-3-yl)ethyl]-7-methyl-5-oxospiro[3,4-dihydro-1,4-benzoxazepine-2,4'-cyclohexane]-1'-carboxamide
—— (2S)-N-(3,5-dimethyl-1H-pyrazol-4-yl)-2-(7-methyl-5-oxospiro[3H-1,4-benzoxazepine-2,4'-oxane]-4-yl)propanamide —— C22H28N4O4
(2S)-N-(3,5-dimethyl-1H-pyrazol-4-yl)-2-(7-methyl-5-oxospiro[3H-1,4-benzoxazepine-2,4'-oxane]-4-yl)propanamide
—— (2R)-N-(3,5-dimethyl-1H-pyrazol-4-yl)-2-(7-methyl-5-oxospiro[3H-1,4-benzoxazepine-2,4'-oxane]-4-yl)propanamide —— C22H28N4O4
(2R)-N-(3,5-dimethyl-1H-pyrazol-4-yl)-2-(7-methyl-5-oxospiro[3H-1,4-benzoxazepine-2,4'-oxane]-4-yl)propanamide
—— 1',7-dimethyl-4-[(2S)-1-[(3R)-3-methylpiperidin-1-yl]-1-oxopropan-2-yl]spiro[3H-1,4-benzoxazepine-2,4'-piperidine]-5-one —— C24H35N3O3
1',7-dimethyl-4-[(2S)-1-[(3R)-3-methylpiperidin-1-yl]-1-oxopropan-2-yl]spiro[3H-1,4-benzoxazepine-2,4'-piperidine]-5-one
—— 2-(1',7-dimethyl-5-oxospiro[3H-1,4-benzoxazepine-2,4'-piperidine]-4-yl)-N-[(4-fluorophenyl)methyl]acetamide —— C24H28FN3O3
2-(1',7-dimethyl-5-oxospiro[3H-1,4-benzoxazepine-2,4'-piperidine]-4-yl)-N-[(4-fluorophenyl)methyl]acetamide
—— 4-[2-(3,3-dimethylpiperidin-1-yl)-2-oxoethyl]-1',7-dimethylspiro[3H-1,4-benzoxazepine-2,4'-piperidine]-5-one —— C24H35N3O3
4-[2-(3,3-dimethylpiperidin-1-yl)-2-oxoethyl]-1',7-dimethylspiro[3H-1,4-benzoxazepine-2,4'-piperidine]-5-one
—— 1-[2-(1',7-dimethyl-5-oxospiro[3H-1,4-benzoxazepine-2,4'-piperidine]-4-yl)acetyl]piperidine-4-carboxamide —— C23H32N4O4
1-[2-(1',7-dimethyl-5-oxospiro[3H-1,4-benzoxazepine-2,4'-piperidine]-4-yl)acetyl]piperidine-4-carboxamide
—— N-(4,5-dimethyl-1,3-thiazol-2-yl)-2-(7-methyl-5-oxospiro[3H-1,4-benzoxazepine-2,4'-oxane]-4-yl)acetamide —— C21H25N3O4S
N-(4,5-dimethyl-1,3-thiazol-2-yl)-2-(7-methyl-5-oxospiro[3H-1,4-benzoxazepine-2,4'-oxane]-4-yl)acetamide
—— 2-(1',7-dimethyl-5-oxospiro[3H-1,4-benzoxazepine-2,4'-piperidine]-4-yl)-N-[[(2R)-1,4-dioxan-2-yl]methyl]acetamide —— C22H31N3O5
2-(1',7-dimethyl-5-oxospiro[3H-1,4-benzoxazepine-2,4'-piperidine]-4-yl)-N-[[(2R)-1,4-dioxan-2-yl]methyl]acetamide
—— 2-(1',7-dimethyl-5-oxospiro[3H-1,4-benzoxazepine-2,4'-piperidine]-4-yl)acetic acid —— C17H22N2O4
2-(1',7-dimethyl-5-oxospiro[3H-1,4-benzoxazepine-2,4'-piperidine]-4-yl)acetic acid
—— N,N-dimethyl-1-[(3S)-7-methyl-4-[(5-methylthiophen-2-yl)methyl]-3,5-dihydro-2H-1,4-benzoxazepin-3-yl]methanamine —— C19H26N2OS
N,N-dimethyl-1-[(3S)-7-methyl-4-[(5-methylthiophen-2-yl)methyl]-3,5-dihydro-2H-1,4-benzoxazepin-3-yl]methanamine
—— 1-[(3R)-4-[(3-fluorophenyl)methyl]-7-methyl-3,5-dihydro-2H-1,4-benzoxazepin-3-yl]-N,N-dimethylmethanamine —— C20H25FN2O
1-[(3R)-4-[(3-fluorophenyl)methyl]-7-methyl-3,5-dihydro-2H-1,4-benzoxazepin-3-yl]-N,N-dimethylmethanamine
—— 4-[2-[(2S,3R)-2,3-dimethylpiperidin-1-yl]-2-oxoethyl]-1',7-dimethylspiro[3H-1,4-benzoxazepine-2,4'-piperidine]-5-one —— C24H35N3O3
4-[2-[(2S,3R)-2,3-dimethylpiperidin-1-yl]-2-oxoethyl]-1',7-dimethylspiro[3H-1,4-benzoxazepine-2,4'-piperidine]-5-one