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苯并恶嗪类

中文名称 英文名称 CAS号 化学式 结构式图片
—— 1',7-dimethyl-4-(2-oxo-2-piperidin-1-ylethyl)spiro[3H-1,4-benzoxazepine-2,4'-piperidine]-5-one —— C22H31N3O3
1',7-dimethyl-4-(2-oxo-2-piperidin-1-ylethyl)spiro[3H-1,4-benzoxazepine-2,4'-piperidine]-5-one
—— 2-(1',7-dimethyl-5-oxospiro[3H-1,4-benzoxazepine-2,4'-piperidine]-4-yl)-N-(2-phenylethyl)acetamide —— C25H31N3O3
2-(1',7-dimethyl-5-oxospiro[3H-1,4-benzoxazepine-2,4'-piperidine]-4-yl)-N-(2-phenylethyl)acetamide
—— 2-(1',7-dimethyl-5-oxospiro[3H-1,4-benzoxazepine-2,4'-piperidine]-4-yl)-N-[2-[(S)-methylsulfinyl]ethyl]acetamide —— C20H29N3O4S
2-(1',7-dimethyl-5-oxospiro[3H-1,4-benzoxazepine-2,4'-piperidine]-4-yl)-N-[2-[(S)-methylsulfinyl]ethyl]acetamide
—— 7-methyl-4-[(2S)-1-[(2R)-2-methylpiperidin-1-yl]-1-oxopropan-2-yl]spiro[3H-1,4-benzoxazepine-2,4'-oxane]-5-one —— C23H32N2O4
7-methyl-4-[(2S)-1-[(2R)-2-methylpiperidin-1-yl]-1-oxopropan-2-yl]spiro[3H-1,4-benzoxazepine-2,4'-oxane]-5-one
—— (2S)-2-(7-methyl-5-oxospiro[3H-1,4-benzoxazepine-2,4'-oxane]-4-yl)-N-(4-methyl-1,3-thiazol-2-yl)propanamide —— C21H25N3O4S
(2S)-2-(7-methyl-5-oxospiro[3H-1,4-benzoxazepine-2,4'-oxane]-4-yl)-N-(4-methyl-1,3-thiazol-2-yl)propanamide
—— N-[(3S)-3-methyl-1,1-dioxothiolan-3-yl]-2-(7-methyl-5-oxospiro[3H-1,4-benzoxazepine-2,4'-oxane]-4-yl)acetamide —— C21H28N2O6S
N-[(3S)-3-methyl-1,1-dioxothiolan-3-yl]-2-(7-methyl-5-oxospiro[3H-1,4-benzoxazepine-2,4'-oxane]-4-yl)acetamide
—— N-[(3-methoxyphenyl)methyl]-7-methyl-5-oxospiro[3,4-dihydro-1,4-benzoxazepine-2,4'-cyclohexane]-1'-carboxamide —— C24H28N2O4
N-[(3-methoxyphenyl)methyl]-7-methyl-5-oxospiro[3,4-dihydro-1,4-benzoxazepine-2,4'-cyclohexane]-1'-carboxamide
—— N-[4-[(2R)-4,7-dimethylspiro[3,5-dihydro-1,4-benzoxazepine-2,3'-piperidine]-1'-yl]sulfonylphenyl]acetamide —— C23H29N3O4S
N-[4-[(2R)-4,7-dimethylspiro[3,5-dihydro-1,4-benzoxazepine-2,3'-piperidine]-1'-yl]sulfonylphenyl]acetamide
—— 4-[2-[(3R,5S)-3,5-dimethylpiperidin-1-yl]-2-oxoethyl]-1',7-dimethylspiro[3H-1,4-benzoxazepine-2,4'-piperidine]-5-one —— C24H35N3O3
4-[2-[(3R,5S)-3,5-dimethylpiperidin-1-yl]-2-oxoethyl]-1',7-dimethylspiro[3H-1,4-benzoxazepine-2,4'-piperidine]-5-one
—— N-(7-methyl-5-oxospiro[3,4-dihydro-1,4-benzoxazepine-2,4'-cyclohexane]-1'-yl)-3-pyridin-3-ylpropanamide —— C23H27N3O3
N-(7-methyl-5-oxospiro[3,4-dihydro-1,4-benzoxazepine-2,4'-cyclohexane]-1'-yl)-3-pyridin-3-ylpropanamide
—— 1-[(2S)-4-acetyl-7-methylspiro[3,5-dihydro-1,4-benzoxazepine-2,3'-piperidine]-1'-yl]-3-(3,5-dimethyl-1,2,4-triazol-1-yl)propan-1-one —— C23H31N5O3
1-[(2S)-4-acetyl-7-methylspiro[3,5-dihydro-1,4-benzoxazepine-2,3'-piperidine]-1'-yl]-3-(3,5-dimethyl-1,2,4-triazol-1-yl)propan-1-one
—— (1,5-dimethylpyrazol-4-yl)-[(2R)-7-methyl-4-methylsulfonylspiro[3,5-dihydro-1,4-benzoxazepine-2,3'-piperidine]-1'-yl]methanone —— C21H28N4O4S
(1,5-dimethylpyrazol-4-yl)-[(2R)-7-methyl-4-methylsulfonylspiro[3,5-dihydro-1,4-benzoxazepine-2,3'-piperidine]-1'-yl]methanone
—— 7-methyl-4-[(2S)-1-[(2S)-2-methylpiperidin-1-yl]-1-oxopropan-2-yl]spiro[3H-1,4-benzoxazepine-2,4'-oxane]-5-one —— C23H32N2O4
7-methyl-4-[(2S)-1-[(2S)-2-methylpiperidin-1-yl]-1-oxopropan-2-yl]spiro[3H-1,4-benzoxazepine-2,4'-oxane]-5-one
—— (2R)-2-(7-methyl-5-oxospiro[3H-1,4-benzoxazepine-2,4'-oxane]-4-yl)-N-[[(2S)-oxolan-2-yl]methyl]propanamide —— C22H30N2O5
(2R)-2-(7-methyl-5-oxospiro[3H-1,4-benzoxazepine-2,4'-oxane]-4-yl)-N-[[(2S)-oxolan-2-yl]methyl]propanamide
—— (2R)-2-(7-methyl-5-oxospiro[3H-1,4-benzoxazepine-2,4'-oxane]-4-yl)-N-(4-methyl-1,3-thiazol-2-yl)propanamide —— C21H25N3O4S
(2R)-2-(7-methyl-5-oxospiro[3H-1,4-benzoxazepine-2,4'-oxane]-4-yl)-N-(4-methyl-1,3-thiazol-2-yl)propanamide
—— N-(3,5-dimethyl-1H-pyrazol-4-yl)-2-(7-methyl-5-oxospiro[3H-1,4-benzoxazepine-2,4'-oxane]-4-yl)acetamide —— C21H26N4O4
N-(3,5-dimethyl-1H-pyrazol-4-yl)-2-(7-methyl-5-oxospiro[3H-1,4-benzoxazepine-2,4'-oxane]-4-yl)acetamide
—— 1-[(3S)-4-[(3,4-dimethoxyphenyl)methyl]-7-methyl-3,5-dihydro-2H-1,4-benzoxazepin-3-yl]-N,N-dimethylmethanamine —— C22H30N2O3
1-[(3S)-4-[(3,4-dimethoxyphenyl)methyl]-7-methyl-3,5-dihydro-2H-1,4-benzoxazepin-3-yl]-N,N-dimethylmethanamine
—— 1',7-dimethyl-4-(2-oxo-2-pyrrolidin-1-ylethyl)spiro[3H-1,4-benzoxazepine-2,4'-piperidine]-5-one —— C21H29N3O3
1',7-dimethyl-4-(2-oxo-2-pyrrolidin-1-ylethyl)spiro[3H-1,4-benzoxazepine-2,4'-piperidine]-5-one
—— 2-(1',7-dimethyl-5-oxospiro[3H-1,4-benzoxazepine-2,4'-piperidine]-4-yl)-N-(3,5-dimethyl-1H-pyrazol-4-yl)acetamide —— C22H29N5O3
2-(1',7-dimethyl-5-oxospiro[3H-1,4-benzoxazepine-2,4'-piperidine]-4-yl)-N-(3,5-dimethyl-1H-pyrazol-4-yl)acetamide
—— (2R)-2-(1',7-dimethyl-5-oxospiro[3H-1,4-benzoxazepine-2,4'-piperidine]-4-yl)-N-[(2R)-3-methylbutan-2-yl]propanamide —— C23H35N3O3
(2R)-2-(1',7-dimethyl-5-oxospiro[3H-1,4-benzoxazepine-2,4'-piperidine]-4-yl)-N-[(2R)-3-methylbutan-2-yl]propanamide
—— 2-(1',7-dimethyl-5-oxospiro[3H-1,4-benzoxazepine-2,4'-piperidine]-4-yl)-N-(2-methoxyethyl)acetamide —— C20H29N3O4
2-(1',7-dimethyl-5-oxospiro[3H-1,4-benzoxazepine-2,4'-piperidine]-4-yl)-N-(2-methoxyethyl)acetamide
—— N-cyclohexyl-2-(1',7-dimethyl-5-oxospiro[3H-1,4-benzoxazepine-2,4'-piperidine]-4-yl)-N-methylacetamide —— C24H35N3O3
N-cyclohexyl-2-(1',7-dimethyl-5-oxospiro[3H-1,4-benzoxazepine-2,4'-piperidine]-4-yl)-N-methylacetamide
—— (3R)-3-[(dimethylamino)methyl]-7-methyl-3,4-dihydro-2H-1,4-benzoxazepin-5-one —— C13H18N2O2
(3R)-3-[(dimethylamino)methyl]-7-methyl-3,4-dihydro-2H-1,4-benzoxazepin-5-one
—— 2-(1',7-dimethyl-5-oxospiro[3H-1,4-benzoxazepine-2,4'-piperidine]-4-yl)-N-[(1R,2S)-2-methylcyclohexyl]acetamide —— C24H35N3O3
2-(1',7-dimethyl-5-oxospiro[3H-1,4-benzoxazepine-2,4'-piperidine]-4-yl)-N-[(1R,2S)-2-methylcyclohexyl]acetamide
—— 7-methyl-5-oxo-N-[[3-(trifluoromethyl)phenyl]methyl]spiro[3,4-dihydro-1,4-benzoxazepine-2,4'-cyclohexane]-1'-carboxamide —— C24H25F3N2O3
7-methyl-5-oxo-N-[[3-(trifluoromethyl)phenyl]methyl]spiro[3,4-dihydro-1,4-benzoxazepine-2,4'-cyclohexane]-1'-carboxamide
—— 1',7-dimethyl-4-[(2R)-1-[(3R)-3-methylpiperidin-1-yl]-1-oxopropan-2-yl]spiro[3H-1,4-benzoxazepine-2,4'-piperidine]-5-one —— C24H35N3O3
1',7-dimethyl-4-[(2R)-1-[(3R)-3-methylpiperidin-1-yl]-1-oxopropan-2-yl]spiro[3H-1,4-benzoxazepine-2,4'-piperidine]-5-one
—— 2-(1',7-dimethyl-5-oxospiro[3H-1,4-benzoxazepine-2,4'-piperidine]-4-yl)-N-(1,5-dimethylpyrazol-3-yl)acetamide —— C22H29N5O3
2-(1',7-dimethyl-5-oxospiro[3H-1,4-benzoxazepine-2,4'-piperidine]-4-yl)-N-(1,5-dimethylpyrazol-3-yl)acetamide
—— (2R)-2-(1',7-dimethyl-5-oxospiro[3H-1,4-benzoxazepine-2,4'-piperidine]-4-yl)propanoic acid —— C18H24N2O4
(2R)-2-(1',7-dimethyl-5-oxospiro[3H-1,4-benzoxazepine-2,4'-piperidine]-4-yl)propanoic acid
—— 2-(1',7-dimethyl-5-oxospiro[3H-1,4-benzoxazepine-2,4'-piperidine]-4-yl)-N-[(2S)-3-methylbutan-2-yl]acetamide —— C22H33N3O3
2-(1',7-dimethyl-5-oxospiro[3H-1,4-benzoxazepine-2,4'-piperidine]-4-yl)-N-[(2S)-3-methylbutan-2-yl]acetamide
—— (1,5-dimethylpyrazol-4-yl)-[(2S)-7-methyl-4-methylsulfonylspiro[3,5-dihydro-1,4-benzoxazepine-2,3'-piperidine]-1'-yl]methanone —— C21H28N4O4S
(1,5-dimethylpyrazol-4-yl)-[(2S)-7-methyl-4-methylsulfonylspiro[3,5-dihydro-1,4-benzoxazepine-2,3'-piperidine]-1'-yl]methanone
—— 1',7-dimethyl-4-[(2R)-1-[(3S)-3-methylpiperidin-1-yl]-1-oxopropan-2-yl]spiro[3H-1,4-benzoxazepine-2,4'-piperidine]-5-one —— C24H35N3O3
1',7-dimethyl-4-[(2R)-1-[(3S)-3-methylpiperidin-1-yl]-1-oxopropan-2-yl]spiro[3H-1,4-benzoxazepine-2,4'-piperidine]-5-one
—— 1-[(2R)-1'-[3-(4-fluorophenoxy)propyl]-7-methylspiro[3,5-dihydro-1,4-benzoxazepine-2,3'-piperidine]-4-yl]ethanone —— C25H31FN2O3
1-[(2R)-1'-[3-(4-fluorophenoxy)propyl]-7-methylspiro[3,5-dihydro-1,4-benzoxazepine-2,3'-piperidine]-4-yl]ethanone
—— N-cyclohexyl-2-(1',7-dimethyl-5-oxospiro[3H-1,4-benzoxazepine-2,4'-piperidine]-4-yl)acetamide —— C23H33N3O3
N-cyclohexyl-2-(1',7-dimethyl-5-oxospiro[3H-1,4-benzoxazepine-2,4'-piperidine]-4-yl)acetamide
—— N-[4-[[(3S)-3-[(dimethylamino)methyl]-7-methyl-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]methyl]phenyl]acetamide —— C22H29N3O2
N-[4-[[(3S)-3-[(dimethylamino)methyl]-7-methyl-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]methyl]phenyl]acetamide
—— 1-[(2S)-1'-[3-(4-fluorophenoxy)propyl]-7-methylspiro[3,5-dihydro-1,4-benzoxazepine-2,3'-piperidine]-4-yl]ethanone —— C25H31FN2O3
1-[(2S)-1'-[3-(4-fluorophenoxy)propyl]-7-methylspiro[3,5-dihydro-1,4-benzoxazepine-2,3'-piperidine]-4-yl]ethanone
—— (2S)-2-(1',7-dimethyl-5-oxospiro[3H-1,4-benzoxazepine-2,4'-piperidine]-4-yl)-N-[[(2S)-oxolan-2-yl]methyl]propanamide —— C23H33N3O4
(2S)-2-(1',7-dimethyl-5-oxospiro[3H-1,4-benzoxazepine-2,4'-piperidine]-4-yl)-N-[[(2S)-oxolan-2-yl]methyl]propanamide
—— 1-[(3S)-4-[(3-fluorophenyl)methyl]-7-methyl-3,5-dihydro-2H-1,4-benzoxazepin-3-yl]-N,N-dimethylmethanamine —— C20H25FN2O
1-[(3S)-4-[(3-fluorophenyl)methyl]-7-methyl-3,5-dihydro-2H-1,4-benzoxazepin-3-yl]-N,N-dimethylmethanamine
—— 1-[(2R)-4-acetyl-7-methylspiro[3,5-dihydro-1,4-benzoxazepine-2,3'-piperidine]-1'-yl]-3-(3,5-dimethyl-1,2,4-triazol-1-yl)propan-1-one —— C23H31N5O3
1-[(2R)-4-acetyl-7-methylspiro[3,5-dihydro-1,4-benzoxazepine-2,3'-piperidine]-1'-yl]-3-(3,5-dimethyl-1,2,4-triazol-1-yl)propan-1-one
—— 1-[(2R)-4-acetyl-7-methylspiro[3,5-dihydro-1,4-benzoxazepine-2,3'-piperidine]-1'-yl]-3-(1,2,4-triazol-1-yl)propan-1-one —— C21H27N5O3
1-[(2R)-4-acetyl-7-methylspiro[3,5-dihydro-1,4-benzoxazepine-2,3'-piperidine]-1'-yl]-3-(1,2,4-triazol-1-yl)propan-1-one
—— 7-methyl-4-[(2R)-1-[(2R)-2-methylpiperidin-1-yl]-1-oxopropan-2-yl]spiro[3H-1,4-benzoxazepine-2,4'-oxane]-5-one —— C23H32N2O4
7-methyl-4-[(2R)-1-[(2R)-2-methylpiperidin-1-yl]-1-oxopropan-2-yl]spiro[3H-1,4-benzoxazepine-2,4'-oxane]-5-one
—— 1',7-Dimethylspiro[3,4-dihydro-1,4-benzoxazepine-2,4'-piperidine]-5-one —— C15H20N2O2
1',7-Dimethylspiro[3,4-dihydro-1,4-benzoxazepine-2,4'-piperidine]-5-one
—— 1',7-dimethyl-4-[(2S)-1-(4-methylpiperazin-1-yl)-1-oxopropan-2-yl]spiro[3H-1,4-benzoxazepine-2,4'-piperidine]-5-one —— C23H34N4O3
1',7-dimethyl-4-[(2S)-1-(4-methylpiperazin-1-yl)-1-oxopropan-2-yl]spiro[3H-1,4-benzoxazepine-2,4'-piperidine]-5-one
—— (2S)-2-(7-methyl-5-oxospiro[3H-1,4-benzoxazepine-2,4'-oxane]-4-yl)-N-(pyridin-2-ylmethyl)propanamide —— C23H27N3O4
(2S)-2-(7-methyl-5-oxospiro[3H-1,4-benzoxazepine-2,4'-oxane]-4-yl)-N-(pyridin-2-ylmethyl)propanamide
—— N-tert-butyl-2-(1',7-dimethyl-5-oxospiro[3H-1,4-benzoxazepine-2,4'-piperidine]-4-yl)acetamide —— C21H31N3O3
N-tert-butyl-2-(1',7-dimethyl-5-oxospiro[3H-1,4-benzoxazepine-2,4'-piperidine]-4-yl)acetamide
—— N-cycloheptyl-2-(1',7-dimethyl-5-oxospiro[3H-1,4-benzoxazepine-2,4'-piperidine]-4-yl)acetamide —— C24H35N3O3
N-cycloheptyl-2-(1',7-dimethyl-5-oxospiro[3H-1,4-benzoxazepine-2,4'-piperidine]-4-yl)acetamide
—— (2R)-2-(7-methyl-5-oxospiro[3H-1,4-benzoxazepine-2,4'-oxane]-4-yl)-N-(1-propan-2-ylpiperidin-4-yl)propanamide —— C25H37N3O4
(2R)-2-(7-methyl-5-oxospiro[3H-1,4-benzoxazepine-2,4'-oxane]-4-yl)-N-(1-propan-2-ylpiperidin-4-yl)propanamide
—— 1-[(3R)-4-[(3-methoxyphenyl)methyl]-7-methyl-3,5-dihydro-2H-1,4-benzoxazepin-3-yl]-N,N-dimethylmethanamine —— C21H28N2O2
1-[(3R)-4-[(3-methoxyphenyl)methyl]-7-methyl-3,5-dihydro-2H-1,4-benzoxazepin-3-yl]-N,N-dimethylmethanamine
—— 2-(1',7-dimethyl-5-oxospiro[3H-1,4-benzoxazepine-2,4'-piperidine]-4-yl)-N-(4-methyl-1,3-thiazol-2-yl)acetamide —— C21H26N4O3S
2-(1',7-dimethyl-5-oxospiro[3H-1,4-benzoxazepine-2,4'-piperidine]-4-yl)-N-(4-methyl-1,3-thiazol-2-yl)acetamide
—— 1-[(3R)-4-[(3,4-dimethoxyphenyl)methyl]-7-methyl-3,5-dihydro-2H-1,4-benzoxazepin-3-yl]-N,N-dimethylmethanamine —— C22H30N2O3
1-[(3R)-4-[(3,4-dimethoxyphenyl)methyl]-7-methyl-3,5-dihydro-2H-1,4-benzoxazepin-3-yl]-N,N-dimethylmethanamine
—— 1',7-dimethyl-4-[(2S)-1-[(3S)-3-methylpiperidin-1-yl]-1-oxopropan-2-yl]spiro[3H-1,4-benzoxazepine-2,4'-piperidine]-5-one —— C24H35N3O3
1',7-dimethyl-4-[(2S)-1-[(3S)-3-methylpiperidin-1-yl]-1-oxopropan-2-yl]spiro[3H-1,4-benzoxazepine-2,4'-piperidine]-5-one