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苯并恶嗪类

中文名称 英文名称 CAS号 化学式 结构式图片
—— 4-[2-[(3S,4S)-4-hydroxy-3-methylpiperidin-1-yl]-2-oxoethyl]spiro[3H-1,4-benzoxazepine-2,4'-oxane]-5-one —— C21H28N2O5
4-[2-[(3S,4S)-4-hydroxy-3-methylpiperidin-1-yl]-2-oxoethyl]spiro[3H-1,4-benzoxazepine-2,4'-oxane]-5-one
—— N-methyl-4-[[(2R)-2-methyl-2,3-dihydro-1-benzofuran-5-yl]methyl]spiro[3,5-dihydro-1,4-benzoxazepine-2,4'-cyclohexane]-1'-amine —— C25H32N2O2
N-methyl-4-[[(2R)-2-methyl-2,3-dihydro-1-benzofuran-5-yl]methyl]spiro[3,5-dihydro-1,4-benzoxazepine-2,4'-cyclohexane]-1'-amine
—— N-methyl-N-[[(2S)-2-methyl-2,3-dihydro-1-benzofuran-5-yl]methyl]spiro[4,5-dihydro-3H-1,4-benzoxazepine-2,4'-cyclohexane]-1'-amine —— C25H32N2O2
N-methyl-N-[[(2S)-2-methyl-2,3-dihydro-1-benzofuran-5-yl]methyl]spiro[4,5-dihydro-3H-1,4-benzoxazepine-2,4'-cyclohexane]-1'-amine
—— N-methyl-N-[4-[[(2R)-2-methyl-2,3-dihydro-1-benzofuran-5-yl]methyl]spiro[3,5-dihydro-1,4-benzoxazepine-2,4'-cyclohexane]-1'-yl]acetamide —— C27H34N2O3
N-methyl-N-[4-[[(2R)-2-methyl-2,3-dihydro-1-benzofuran-5-yl]methyl]spiro[3,5-dihydro-1,4-benzoxazepine-2,4'-cyclohexane]-1'-yl]acetamide
—— 4-[2-[(2S)-2-methyl-2,3-dihydroindol-1-yl]-2-oxoethyl]-6-(thiophene-2-carbonyl)-1,4-benzoxazin-3-one —— C24H20N2O4S
4-[2-[(2S)-2-methyl-2,3-dihydroindol-1-yl]-2-oxoethyl]-6-(thiophene-2-carbonyl)-1,4-benzoxazin-3-one
—— (2R)-N-(4-acetylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-cyclohexane]-1'-yl)-N,2-dimethyl-2,3-dihydro-1-benzofuran-5-carboxamide —— C27H32N2O4
(2R)-N-(4-acetylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-cyclohexane]-1'-yl)-N,2-dimethyl-2,3-dihydro-1-benzofuran-5-carboxamide
—— (2S)-N-(4-acetylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-cyclohexane]-1'-yl)-N,2-dimethyl-2,3-dihydro-1-benzofuran-5-carboxamide —— C27H32N2O4
(2S)-N-(4-acetylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-cyclohexane]-1'-yl)-N,2-dimethyl-2,3-dihydro-1-benzofuran-5-carboxamide
—— [7-methyl-3-oxo-2-(trifluoromethyl)-4H-1,4-benzoxazin-2-yl] 2-methylprop-2-enoate —— C14H12F3NO4
[7-methyl-3-oxo-2-(trifluoromethyl)-4H-1,4-benzoxazin-2-yl] 2-methylprop-2-enoate
—— 4'-[(3R,4R)-4-hydroxy-3-methylpiperidine-1-carbonyl]spiro[3,4-dihydro-1,4-benzoxazepine-2,1'-cyclohexane]-5-one —— C21H28N2O4
4'-[(3R,4R)-4-hydroxy-3-methylpiperidine-1-carbonyl]spiro[3,4-dihydro-1,4-benzoxazepine-2,1'-cyclohexane]-5-one
—— 4'-[(3S,4R)-4-hydroxy-3-methylpiperidine-1-carbonyl]spiro[3,4-dihydro-1,4-benzoxazepine-2,1'-cyclohexane]-5-one —— C21H28N2O4
4'-[(3S,4R)-4-hydroxy-3-methylpiperidine-1-carbonyl]spiro[3,4-dihydro-1,4-benzoxazepine-2,1'-cyclohexane]-5-one
—— 7-chloro-4'-[(3S,4R)-4-hydroxy-3-methylpiperidine-1-carbonyl]spiro[3,4-dihydro-1,4-benzoxazepine-2,1'-cyclohexane]-5-one —— C21H27ClN2O4
7-chloro-4'-[(3S,4R)-4-hydroxy-3-methylpiperidine-1-carbonyl]spiro[3,4-dihydro-1,4-benzoxazepine-2,1'-cyclohexane]-5-one
—— 4-[2-[(2R,6R)-2,6-dimethylmorpholin-4-yl]-2-oxoethyl]-1'-methylspiro[3H-1,4-benzoxazepine-2,4'-piperidine]-5-one —— C22H31N3O4
4-[2-[(2R,6R)-2,6-dimethylmorpholin-4-yl]-2-oxoethyl]-1'-methylspiro[3H-1,4-benzoxazepine-2,4'-piperidine]-5-one
—— 4-[2-[(2S,6S)-2,6-dimethylmorpholin-4-yl]-2-oxoethyl]-1'-methylspiro[3H-1,4-benzoxazepine-2,4'-piperidine]-5-one —— C22H31N3O4
4-[2-[(2S,6S)-2,6-dimethylmorpholin-4-yl]-2-oxoethyl]-1'-methylspiro[3H-1,4-benzoxazepine-2,4'-piperidine]-5-one
—— 4-[2-[(2S,6R)-2,6-dimethylmorpholin-4-yl]-2-oxoethyl]-1'-methylspiro[3H-1,4-benzoxazepine-2,4'-piperidine]-5-one —— C22H31N3O4
4-[2-[(2S,6R)-2,6-dimethylmorpholin-4-yl]-2-oxoethyl]-1'-methylspiro[3H-1,4-benzoxazepine-2,4'-piperidine]-5-one
—— 1'-methyl-4-[2-(4-methylpiperidin-1-yl)-2-oxoethyl]spiro[3H-1,4-benzoxazepine-2,4'-piperidine]-5-one —— C22H31N3O3
1'-methyl-4-[2-(4-methylpiperidin-1-yl)-2-oxoethyl]spiro[3H-1,4-benzoxazepine-2,4'-piperidine]-5-one
—— 1-[4'-(Dimethylamino)spiro[3,5-dihydro-1,4-benzoxazepine-2,1'-cyclohexane]-4-yl]-2-(4-methylpiperidin-1-yl)ethanone —— C24H37N3O2
1-[4'-(Dimethylamino)spiro[3,5-dihydro-1,4-benzoxazepine-2,1'-cyclohexane]-4-yl]-2-(4-methylpiperidin-1-yl)ethanone
—— N-[5-(diethylamino)pentan-2-yl]-2-(7-methyl-3-oxo-1,4-benzoxazin-4-yl)acetamide —— C20H31N3O3
N-[5-(diethylamino)pentan-2-yl]-2-(7-methyl-3-oxo-1,4-benzoxazin-4-yl)acetamide
—— 7-chloro-4'-[(2S,3S)-2,3-dimethylpiperidine-1-carbonyl]spiro[3,4-dihydro-1,4-benzoxazepine-2,1'-cyclohexane]-5-one —— C22H29ClN2O3
7-chloro-4'-[(2S,3S)-2,3-dimethylpiperidine-1-carbonyl]spiro[3,4-dihydro-1,4-benzoxazepine-2,1'-cyclohexane]-5-one
—— (2R)-2-[(2R)-2-methyl-3-oxo-1,4-benzoxazin-4-yl]-N-[(2R)-2-(4-methylpiperidin-1-yl)propyl]propanamide —— C21H31N3O3
(2R)-2-[(2R)-2-methyl-3-oxo-1,4-benzoxazin-4-yl]-N-[(2R)-2-(4-methylpiperidin-1-yl)propyl]propanamide
—— (2R)-2-[(2R)-2-methyl-3-oxo-1,4-benzoxazin-4-yl]-N-[(2S)-2-(4-methylpiperidin-1-yl)propyl]propanamide —— C21H31N3O3
(2R)-2-[(2R)-2-methyl-3-oxo-1,4-benzoxazin-4-yl]-N-[(2S)-2-(4-methylpiperidin-1-yl)propyl]propanamide
—— (2R)-N-[2-methyl-1-[(3R)-3-methylpiperidin-1-yl]propan-2-yl]-2-[(2R)-2-methyl-3-oxo-1,4-benzoxazin-4-yl]propanamide —— C22H33N3O3
(2R)-N-[2-methyl-1-[(3R)-3-methylpiperidin-1-yl]propan-2-yl]-2-[(2R)-2-methyl-3-oxo-1,4-benzoxazin-4-yl]propanamide
—— N-methyl-2-(4-methylpiperidin-1-yl)-N-spiro[4,5-dihydro-3H-1,4-benzoxazepine-2,4'-cyclohexane]-1'-ylacetamide —— C23H35N3O2
N-methyl-2-(4-methylpiperidin-1-yl)-N-spiro[4,5-dihydro-3H-1,4-benzoxazepine-2,4'-cyclohexane]-1'-ylacetamide
—— N-methyl-2-(4-methylpiperidin-1-yl)-N-(4-methylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-cyclohexane]-1'-yl)acetamide —— C24H37N3O2
N-methyl-2-(4-methylpiperidin-1-yl)-N-(4-methylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-cyclohexane]-1'-yl)acetamide
—— (2S)-2-[(2R)-2-methyl-3-oxo-1,4-benzoxazin-4-yl]-N-[(2S)-2-(4-methylpiperidin-1-yl)propyl]propanamide —— C21H31N3O3
(2S)-2-[(2R)-2-methyl-3-oxo-1,4-benzoxazin-4-yl]-N-[(2S)-2-(4-methylpiperidin-1-yl)propyl]propanamide
—— 2,2-dimethyl-N-[(1R)-1-[2-(4-methylpiperidin-1-yl)-6-oxo-1H-pyrimidin-4-yl]ethyl]-3-oxo-4H-1,4-benzoxazine-6-carboxamide —— C23H29N5O4
2,2-dimethyl-N-[(1R)-1-[2-(4-methylpiperidin-1-yl)-6-oxo-1H-pyrimidin-4-yl]ethyl]-3-oxo-4H-1,4-benzoxazine-6-carboxamide
—— 7-chloro-4'-[(2R,3R)-2,3-dimethylpiperidine-1-carbonyl]spiro[3,4-dihydro-1,4-benzoxazepine-2,1'-cyclohexane]-5-one —— C22H29ClN2O3
7-chloro-4'-[(2R,3R)-2,3-dimethylpiperidine-1-carbonyl]spiro[3,4-dihydro-1,4-benzoxazepine-2,1'-cyclohexane]-5-one
—— N-methyl-2-[(3S)-3-methylpiperidin-1-yl]-N-spiro[4,5-dihydro-3H-1,4-benzoxazepine-2,4'-cyclohexane]-1'-ylacetamide —— C23H35N3O2
N-methyl-2-[(3S)-3-methylpiperidin-1-yl]-N-spiro[4,5-dihydro-3H-1,4-benzoxazepine-2,4'-cyclohexane]-1'-ylacetamide
—— 7-chloro-4-[2-[(3R)-3-methylpiperidin-1-yl]-2-oxoethyl]spiro[3H-1,4-benzoxazepine-2,4'-oxane]-5-one —— C21H27ClN2O4
7-chloro-4-[2-[(3R)-3-methylpiperidin-1-yl]-2-oxoethyl]spiro[3H-1,4-benzoxazepine-2,4'-oxane]-5-one
—— 2,2-dimethyl-N-[(1S)-1-[2-(4-methylpiperidin-1-yl)-6-oxo-1H-pyrimidin-4-yl]ethyl]-3-oxo-4H-1,4-benzoxazine-6-carboxamide —— C23H29N5O4
2,2-dimethyl-N-[(1S)-1-[2-(4-methylpiperidin-1-yl)-6-oxo-1H-pyrimidin-4-yl]ethyl]-3-oxo-4H-1,4-benzoxazine-6-carboxamide
—— 7-Chloro-4'-(4-methylpiperidine-1-carbonyl)spiro[3,4-dihydro-1,4-benzoxazepine-2,1'-cyclohexane]-5-one —— C21H27ClN2O3
7-Chloro-4'-(4-methylpiperidine-1-carbonyl)spiro[3,4-dihydro-1,4-benzoxazepine-2,1'-cyclohexane]-5-one
—— 7-chloro-4'-[(2S,3R)-2,3-dimethylpiperidine-1-carbonyl]spiro[3,4-dihydro-1,4-benzoxazepine-2,1'-cyclohexane]-5-one —— C22H29ClN2O3
7-chloro-4'-[(2S,3R)-2,3-dimethylpiperidine-1-carbonyl]spiro[3,4-dihydro-1,4-benzoxazepine-2,1'-cyclohexane]-5-one
—— N-methyl-2-[(3R)-3-methylpiperidin-1-yl]-N-spiro[4,5-dihydro-3H-1,4-benzoxazepine-2,4'-cyclohexane]-1'-ylacetamide —— C23H35N3O2
N-methyl-2-[(3R)-3-methylpiperidin-1-yl]-N-spiro[4,5-dihydro-3H-1,4-benzoxazepine-2,4'-cyclohexane]-1'-ylacetamide
—— 7-chloro-4-[2-[(3S)-3-methylpiperidin-1-yl]-2-oxoethyl]spiro[3H-1,4-benzoxazepine-2,4'-oxane]-5-one —— C21H27ClN2O4
7-chloro-4-[2-[(3S)-3-methylpiperidin-1-yl]-2-oxoethyl]spiro[3H-1,4-benzoxazepine-2,4'-oxane]-5-one
—— 7-chloro-N-[(1R,2R)-2-methylcyclohexyl]-5-oxospiro[3,4-dihydro-1,4-benzoxazepine-2,4'-cyclohexane]-1'-carboxamide —— C22H29ClN2O3
7-chloro-N-[(1R,2R)-2-methylcyclohexyl]-5-oxospiro[3,4-dihydro-1,4-benzoxazepine-2,4'-cyclohexane]-1'-carboxamide
—— 7-chloro-4'-[(2R,3S)-2,3-dimethylpiperidine-1-carbonyl]spiro[3,4-dihydro-1,4-benzoxazepine-2,1'-cyclohexane]-5-one —— C22H29ClN2O3
7-chloro-4'-[(2R,3S)-2,3-dimethylpiperidine-1-carbonyl]spiro[3,4-dihydro-1,4-benzoxazepine-2,1'-cyclohexane]-5-one
—— N-[(1R,2S)-2-methylcyclohexyl]-2-(1'-methyl-5-oxospiro[3H-1,4-benzoxazepine-2,4'-piperidine]-4-yl)acetamide —— C23H33N3O3
N-[(1R,2S)-2-methylcyclohexyl]-2-(1'-methyl-5-oxospiro[3H-1,4-benzoxazepine-2,4'-piperidine]-4-yl)acetamide
—— 1'-methyl-4-[2-[(3S)-3-methylpiperidin-1-yl]-2-oxoethyl]spiro[3H-1,4-benzoxazepine-2,4'-piperidine]-5-one —— C22H31N3O3
1'-methyl-4-[2-[(3S)-3-methylpiperidin-1-yl]-2-oxoethyl]spiro[3H-1,4-benzoxazepine-2,4'-piperidine]-5-one
—— (2S)-1'-methyl-4-[2-[(2S)-2-methylpiperidin-1-yl]-2-oxoethyl]spiro[3H-1,4-benzoxazepine-2,5'-azepane]-2',5-dione —— C23H31N3O4
(2S)-1'-methyl-4-[2-[(2S)-2-methylpiperidin-1-yl]-2-oxoethyl]spiro[3H-1,4-benzoxazepine-2,5'-azepane]-2',5-dione
—— 1'-methyl-4-[2-[(3R)-3-methylpiperidin-1-yl]-2-oxoethyl]spiro[3H-1,4-benzoxazepine-2,4'-piperidine]-5-one —— C22H31N3O3
1'-methyl-4-[2-[(3R)-3-methylpiperidin-1-yl]-2-oxoethyl]spiro[3H-1,4-benzoxazepine-2,4'-piperidine]-5-one
—— N-methyl-2-[(2S)-2-methylpiperidin-1-yl]-N-spiro[4,5-dihydro-3H-1,4-benzoxazepine-2,4'-cyclohexane]-1'-ylacetamide —— C23H35N3O2
N-methyl-2-[(2S)-2-methylpiperidin-1-yl]-N-spiro[4,5-dihydro-3H-1,4-benzoxazepine-2,4'-cyclohexane]-1'-ylacetamide
—— 8-methoxy-1'-methyl-4-[2-[(2S)-2-methylpiperidin-1-yl]-2-oxoethyl]spiro[3H-1,4-benzoxazepine-2,4'-piperidine]-5-one —— C23H33N3O4
8-methoxy-1'-methyl-4-[2-[(2S)-2-methylpiperidin-1-yl]-2-oxoethyl]spiro[3H-1,4-benzoxazepine-2,4'-piperidine]-5-one
—— (2R)-7-methoxy-1'-methyl-4-[2-[(2R)-2-methylpiperidin-1-yl]-2-oxoethyl]spiro[3H-1,4-benzoxazepine-2,5'-azepane]-2',5-dione —— C24H33N3O5
(2R)-7-methoxy-1'-methyl-4-[2-[(2R)-2-methylpiperidin-1-yl]-2-oxoethyl]spiro[3H-1,4-benzoxazepine-2,5'-azepane]-2',5-dione
—— 7-chloro-4'-[(2S)-2-methylpiperidine-1-carbonyl]spiro[3,4-dihydro-1,4-benzoxazepine-2,1'-cyclohexane]-5-one —— C21H27ClN2O3
7-chloro-4'-[(2S)-2-methylpiperidine-1-carbonyl]spiro[3,4-dihydro-1,4-benzoxazepine-2,1'-cyclohexane]-5-one
—— (2R)-1'-methyl-4-[2-[(2R)-2-methylpiperidin-1-yl]-2-oxoethyl]spiro[3H-1,4-benzoxazepine-2,5'-azepane]-2',5-dione —— C23H31N3O4
(2R)-1'-methyl-4-[2-[(2R)-2-methylpiperidin-1-yl]-2-oxoethyl]spiro[3H-1,4-benzoxazepine-2,5'-azepane]-2',5-dione
—— 1-[4'-(dimethylamino)spiro[3,5-dihydro-1,4-benzoxazepine-2,1'-cyclohexane]-4-yl]-2-[(2S)-2-methylpiperidin-1-yl]ethanone —— C24H37N3O2
1-[4'-(dimethylamino)spiro[3,5-dihydro-1,4-benzoxazepine-2,1'-cyclohexane]-4-yl]-2-[(2S)-2-methylpiperidin-1-yl]ethanone
—— 2-(7-chloro-5-oxospiro[3H-1,4-benzoxazepine-2,4'-oxane]-4-yl)-N-[(1R,2R)-2-methylcyclohexyl]acetamide —— C22H29ClN2O4
2-(7-chloro-5-oxospiro[3H-1,4-benzoxazepine-2,4'-oxane]-4-yl)-N-[(1R,2R)-2-methylcyclohexyl]acetamide
—— 4-methyl-N-[(1S,2R)-2-methylcyclohexyl]-5-oxospiro[3H-1,4-benzoxazepine-2,4'-cyclohexane]-1'-carboxamide —— C23H32N2O3
4-methyl-N-[(1S,2R)-2-methylcyclohexyl]-5-oxospiro[3H-1,4-benzoxazepine-2,4'-cyclohexane]-1'-carboxamide
—— 1'-methyl-4-[2-[(2R)-2-methylpiperidin-1-yl]-2-oxoethyl]spiro[3H-1,4-benzoxazepine-2,4'-piperidine]-5-one —— C22H31N3O3
1'-methyl-4-[2-[(2R)-2-methylpiperidin-1-yl]-2-oxoethyl]spiro[3H-1,4-benzoxazepine-2,4'-piperidine]-5-one
—— (2R)-7-methoxy-1'-methyl-4-[2-[(2S)-2-methylpiperidin-1-yl]-2-oxoethyl]spiro[3H-1,4-benzoxazepine-2,5'-azepane]-2',5-dione —— C24H33N3O5
(2R)-7-methoxy-1'-methyl-4-[2-[(2S)-2-methylpiperidin-1-yl]-2-oxoethyl]spiro[3H-1,4-benzoxazepine-2,5'-azepane]-2',5-dione
—— 4-methyl-N-[(1R,2R)-2-methylcyclohexyl]-5-oxospiro[3H-1,4-benzoxazepine-2,4'-cyclohexane]-1'-carboxamide —— C23H32N2O3
4-methyl-N-[(1R,2R)-2-methylcyclohexyl]-5-oxospiro[3H-1,4-benzoxazepine-2,4'-cyclohexane]-1'-carboxamide