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苯并恶嗪类

中文名称 英文名称 CAS号 化学式 结构式图片
—— (3R,3'S)-1'-(5-ethyl-2,4-dimethylpyrazole-3-carbonyl)-N,N-dimethyl-5-oxospiro[2,4-dihydro-1,4-benzoxazepine-3,4'-pyrrolidine]-3'-carboxamide —— C23H29N5O4
(3R,3'S)-1'-(5-ethyl-2,4-dimethylpyrazole-3-carbonyl)-N,N-dimethyl-5-oxospiro[2,4-dihydro-1,4-benzoxazepine-3,4'-pyrrolidine]-3'-carboxamide
—— (3R,3'S)-1'-(2-methoxypyridine-4-carbonyl)-N,N-dimethyl-5-oxospiro[2,4-dihydro-1,4-benzoxazepine-3,4'-pyrrolidine]-3'-carboxamide —— C22H24N4O5
(3R,3'S)-1'-(2-methoxypyridine-4-carbonyl)-N,N-dimethyl-5-oxospiro[2,4-dihydro-1,4-benzoxazepine-3,4'-pyrrolidine]-3'-carboxamide
—— (3R,3'S)-1'-[(3R)-1,1-dioxothiolane-3-carbonyl]-N,N-dimethyl-5-oxospiro[2,4-dihydro-1,4-benzoxazepine-3,4'-pyrrolidine]-3'-carboxamide —— C20H25N3O6S
(3R,3'S)-1'-[(3R)-1,1-dioxothiolane-3-carbonyl]-N,N-dimethyl-5-oxospiro[2,4-dihydro-1,4-benzoxazepine-3,4'-pyrrolidine]-3'-carboxamide
—— (3R,3'S)-1'-(5-ethyl-1,2-oxazole-3-carbonyl)-N,N-dimethyl-5-oxospiro[2,4-dihydro-1,4-benzoxazepine-3,4'-pyrrolidine]-3'-carboxamide —— C21H24N4O5
(3R,3'S)-1'-(5-ethyl-1,2-oxazole-3-carbonyl)-N,N-dimethyl-5-oxospiro[2,4-dihydro-1,4-benzoxazepine-3,4'-pyrrolidine]-3'-carboxamide
—— (2R)-7-methoxy-1'-[(3R)-piperidine-3-carbonyl]spiro[3,4-dihydro-1,4-benzoxazepine-2,3'-piperidine]-5-one —— C20H27N3O4
(2R)-7-methoxy-1'-[(3R)-piperidine-3-carbonyl]spiro[3,4-dihydro-1,4-benzoxazepine-2,3'-piperidine]-5-one
—— (3R,3'S)-N,N-dimethyl-5-oxo-1'-(1-propan-2-ylpyrazole-4-carbonyl)spiro[2,4-dihydro-1,4-benzoxazepine-3,4'-pyrrolidine]-3'-carboxamide —— C22H27N5O4
(3R,3'S)-N,N-dimethyl-5-oxo-1'-(1-propan-2-ylpyrazole-4-carbonyl)spiro[2,4-dihydro-1,4-benzoxazepine-3,4'-pyrrolidine]-3'-carboxamide
—— (3R,3'S)-N,N-dimethyl-1'-[3-(4-methylphenoxy)propyl]-5-oxospiro[2,4-dihydro-1,4-benzoxazepine-3,4'-pyrrolidine]-3'-carboxamide —— C25H31N3O4
(3R,3'S)-N,N-dimethyl-1'-[3-(4-methylphenoxy)propyl]-5-oxospiro[2,4-dihydro-1,4-benzoxazepine-3,4'-pyrrolidine]-3'-carboxamide
—— (3R,3'S)-1'-(2-fluorobenzoyl)-N,N-dimethyl-5-oxospiro[2,4-dihydro-1,4-benzoxazepine-3,4'-pyrrolidine]-3'-carboxamide —— C22H22FN3O4
(3R,3'S)-1'-(2-fluorobenzoyl)-N,N-dimethyl-5-oxospiro[2,4-dihydro-1,4-benzoxazepine-3,4'-pyrrolidine]-3'-carboxamide
—— (3R,3'S)-1'-(2,4-dimethylpyrimidine-5-carbonyl)-N,N-dimethyl-5-oxospiro[2,4-dihydro-1,4-benzoxazepine-3,4'-pyrrolidine]-3'-carboxamide —— C22H25N5O4
(3R,3'S)-1'-(2,4-dimethylpyrimidine-5-carbonyl)-N,N-dimethyl-5-oxospiro[2,4-dihydro-1,4-benzoxazepine-3,4'-pyrrolidine]-3'-carboxamide
—— (3R,3'S)-N,N-dimethyl-1'-(2-methyl-5-propan-2-ylpyrazole-3-carbonyl)-5-oxospiro[2,4-dihydro-1,4-benzoxazepine-3,4'-pyrrolidine]-3'-carboxamide —— C23H29N5O4
(3R,3'S)-N,N-dimethyl-1'-(2-methyl-5-propan-2-ylpyrazole-3-carbonyl)-5-oxospiro[2,4-dihydro-1,4-benzoxazepine-3,4'-pyrrolidine]-3'-carboxamide
—— (3R,3'S)-1'-[2-(2,4-dimethyl-1,3-thiazol-5-yl)acetyl]-N,N-dimethyl-5-oxospiro[2,4-dihydro-1,4-benzoxazepine-3,4'-pyrrolidine]-3'-carboxamide —— C22H26N4O4S
(3R,3'S)-1'-[2-(2,4-dimethyl-1,3-thiazol-5-yl)acetyl]-N,N-dimethyl-5-oxospiro[2,4-dihydro-1,4-benzoxazepine-3,4'-pyrrolidine]-3'-carboxamide
—— (3R,3'S)-1'-(3-ethyl-1,2-oxazole-5-carbonyl)-N,N-dimethyl-5-oxospiro[2,4-dihydro-1,4-benzoxazepine-3,4'-pyrrolidine]-3'-carboxamide —— C21H24N4O5
(3R,3'S)-1'-(3-ethyl-1,2-oxazole-5-carbonyl)-N,N-dimethyl-5-oxospiro[2,4-dihydro-1,4-benzoxazepine-3,4'-pyrrolidine]-3'-carboxamide
—— [4-(4-Methoxyphenyl)sulfonylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-cyclohexane]-1'-yl]methanol —— C22H27NO5S
[4-(4-Methoxyphenyl)sulfonylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-cyclohexane]-1'-yl]methanol
—— 1-[(2R)-1'-[(3R)-piperidine-3-carbonyl]spiro[3,5-dihydro-1,4-benzoxazepine-2,3'-piperidine]-4-yl]ethanone —— C21H29N3O3
1-[(2R)-1'-[(3R)-piperidine-3-carbonyl]spiro[3,5-dihydro-1,4-benzoxazepine-2,3'-piperidine]-4-yl]ethanone
—— 2-(7-chloro-5-oxospiro[3H-1,4-benzoxazepine-2,4'-oxane]-4-yl)-N-(2-thiophen-2-ylethyl)acetamide —— C21H23ClN2O4S
2-(7-chloro-5-oxospiro[3H-1,4-benzoxazepine-2,4'-oxane]-4-yl)-N-(2-thiophen-2-ylethyl)acetamide
—— 1-[(2S)-7-methyl-1'-(3-phenoxypropyl)spiro[3,5-dihydro-1,4-benzoxazepine-2,3'-piperidine]-4-yl]ethanone —— C25H32N2O3
1-[(2S)-7-methyl-1'-(3-phenoxypropyl)spiro[3,5-dihydro-1,4-benzoxazepine-2,3'-piperidine]-4-yl]ethanone
—— 1-[4-[(3,4-dimethoxyphenyl)methyl]spiro[3,5-dihydro-1,4-benzoxazepine-2,4'-cyclohexane]-1'-yl]-N,N-dimethylmethanamine —— C26H36N2O3
1-[4-[(3,4-dimethoxyphenyl)methyl]spiro[3,5-dihydro-1,4-benzoxazepine-2,4'-cyclohexane]-1'-yl]-N,N-dimethylmethanamine
—— 1-(7-Chlorospiro[3,5-dihydro-1,4-benzoxazepine-2,4'-oxane]-4-yl)-3-(1,2,4-triazol-1-yl)propan-1-one —— C18H21ClN4O3
1-(7-Chlorospiro[3,5-dihydro-1,4-benzoxazepine-2,4'-oxane]-4-yl)-3-(1,2,4-triazol-1-yl)propan-1-one
—— [5-[[4'-[(Dimethylamino)methyl]spiro[3,5-dihydro-1,4-benzoxazepine-2,1'-cyclohexane]-4-yl]methyl]-2-methoxyphenyl]methanol —— C26H36N2O3
[5-[[4'-[(Dimethylamino)methyl]spiro[3,5-dihydro-1,4-benzoxazepine-2,1'-cyclohexane]-4-yl]methyl]-2-methoxyphenyl]methanol
—— 4-(3,6-dihydro-2H-pyran-5-ylmethyl)spiro[3,5-dihydro-1,4-benzoxazepine-2,4'-oxane] —— C19H25NO3
4-(3,6-dihydro-2H-pyran-5-ylmethyl)spiro[3,5-dihydro-1,4-benzoxazepine-2,4'-oxane]
—— 1-[(2S)-1'-[2-(benzenesulfonyl)ethyl]-7-methylspiro[3,5-dihydro-1,4-benzoxazepine-2,3'-piperidine]-4-yl]ethanone —— C24H30N2O4S
1-[(2S)-1'-[2-(benzenesulfonyl)ethyl]-7-methylspiro[3,5-dihydro-1,4-benzoxazepine-2,3'-piperidine]-4-yl]ethanone
—— 2-(4-Amino-1,2,5-oxadiazol-3-yl)-1-spiro[3,5-dihydro-1,4-benzoxazepine-2,4'-oxane]-4-ylethanone —— C17H20N4O4
2-(4-Amino-1,2,5-oxadiazol-3-yl)-1-spiro[3,5-dihydro-1,4-benzoxazepine-2,4'-oxane]-4-ylethanone
—— (5-Methylpyrazin-2-yl)-spiro[3,5-dihydro-1,4-benzoxazepine-2,4'-oxane]-4-ylmethanone —— C19H21N3O3
(5-Methylpyrazin-2-yl)-spiro[3,5-dihydro-1,4-benzoxazepine-2,4'-oxane]-4-ylmethanone
—— ethyl (3S,3'R)-5-oxo-1'-(piperidine-4-carbonyl)spiro[2,4-dihydro-1,4-benzoxazepine-3,4'-pyrrolidine]-3'-carboxylate —— C21H27N3O5
ethyl (3S,3'R)-5-oxo-1'-(piperidine-4-carbonyl)spiro[2,4-dihydro-1,4-benzoxazepine-3,4'-pyrrolidine]-3'-carboxylate
—— Spiro[3,5-dihydro-1,4-benzoxazepine-2,4'-oxane]-4-yl-(3,4,5-trimethoxyphenyl)methanone —— C23H27NO6
Spiro[3,5-dihydro-1,4-benzoxazepine-2,4'-oxane]-4-yl-(3,4,5-trimethoxyphenyl)methanone
—— Oxan-4-yl(spiro[3,5-dihydro-1,4-benzoxazepine-2,4'-oxane]-4-yl)methanone —— C19H25NO4
Oxan-4-yl(spiro[3,5-dihydro-1,4-benzoxazepine-2,4'-oxane]-4-yl)methanone
—— (2S)-7-methoxy-1'-[(3R)-piperidine-3-carbonyl]spiro[3,4-dihydro-1,4-benzoxazepine-2,3'-piperidine]-5-one —— C20H27N3O4
(2S)-7-methoxy-1'-[(3R)-piperidine-3-carbonyl]spiro[3,4-dihydro-1,4-benzoxazepine-2,3'-piperidine]-5-one
—— 4-[[(3R)-oxolan-3-yl]methyl]spiro[3,5-dihydro-1,4-benzoxazepine-2,4'-oxane] —— C18H25NO3
4-[[(3R)-oxolan-3-yl]methyl]spiro[3,5-dihydro-1,4-benzoxazepine-2,4'-oxane]
—— [4'-[(Dimethylamino)methyl]spiro[3,5-dihydro-1,4-benzoxazepine-2,1'-cyclohexane]-4-yl]-(oxan-4-yl)methanone —— C23H34N2O3
[4'-[(Dimethylamino)methyl]spiro[3,5-dihydro-1,4-benzoxazepine-2,1'-cyclohexane]-4-yl]-(oxan-4-yl)methanone
—— 2-(3,5-Dimethylpyrazol-1-yl)-1-spiro[3,5-dihydro-1,4-benzoxazepine-2,4'-oxane]-4-ylethanone —— C20H25N3O3
2-(3,5-Dimethylpyrazol-1-yl)-1-spiro[3,5-dihydro-1,4-benzoxazepine-2,4'-oxane]-4-ylethanone
—— 2-(4-Methylsulfonylphenyl)-1-spiro[3,5-dihydro-1,4-benzoxazepine-2,4'-oxane]-4-ylethanone —— C22H25NO5S
2-(4-Methylsulfonylphenyl)-1-spiro[3,5-dihydro-1,4-benzoxazepine-2,4'-oxane]-4-ylethanone
—— 2-(4-Methoxyphenyl)-5-(3,4,5-trimethoxyphenyl)-1,10b-dihydropyrazolo[1,5-c][1,3]benzoxazine —— C26H26N2O5
2-(4-Methoxyphenyl)-5-(3,4,5-trimethoxyphenyl)-1,10b-dihydropyrazolo[1,5-c][1,3]benzoxazine
—— (2S)-2-methyl-1-spiro[3,5-dihydro-1,4-benzoxazepine-2,4'-oxane]-4-yl-3-(1,2,4-triazol-1-yl)propan-1-one —— C19H24N4O3
(2S)-2-methyl-1-spiro[3,5-dihydro-1,4-benzoxazepine-2,4'-oxane]-4-yl-3-(1,2,4-triazol-1-yl)propan-1-one
—— [4-[(2-Fluoro-4-methoxyphenyl)methyl]spiro[3,5-dihydro-1,4-benzoxazepine-2,4'-cyclohexane]-1'-yl]methanol —— C23H28FNO3
[4-[(2-Fluoro-4-methoxyphenyl)methyl]spiro[3,5-dihydro-1,4-benzoxazepine-2,4'-cyclohexane]-1'-yl]methanol
—— [4'-[(Dimethylamino)methyl]spiro[3,5-dihydro-1,4-benzoxazepine-2,1'-cyclohexane]-4-yl]-pyridin-3-ylmethanone —— C23H29N3O2
[4'-[(Dimethylamino)methyl]spiro[3,5-dihydro-1,4-benzoxazepine-2,1'-cyclohexane]-4-yl]-pyridin-3-ylmethanone
—— 4-[(3-Methoxyphenyl)methyl]spiro[3,5-dihydro-1,4-benzoxazepine-2,4'-oxane] —— C21H25NO3
4-[(3-Methoxyphenyl)methyl]spiro[3,5-dihydro-1,4-benzoxazepine-2,4'-oxane]
—— 4-(Spiro[3,5-dihydro-1,4-benzoxazepine-2,4'-oxane]-4-carbonyl)benzenesulfonamide —— C20H22N2O5S
4-(Spiro[3,5-dihydro-1,4-benzoxazepine-2,4'-oxane]-4-carbonyl)benzenesulfonamide
—— 1-Spiro[3,5-dihydro-1,4-benzoxazepine-2,4'-oxane]-4-yl-2-(3,4,5-trimethoxyphenyl)ethanone —— C24H29NO6
1-Spiro[3,5-dihydro-1,4-benzoxazepine-2,4'-oxane]-4-yl-2-(3,4,5-trimethoxyphenyl)ethanone
—— 4-[(2-Ethylpyrimidin-5-yl)methyl]spiro[3,5-dihydro-1,4-benzoxazepine-2,4'-oxane] —— C20H25N3O2
4-[(2-Ethylpyrimidin-5-yl)methyl]spiro[3,5-dihydro-1,4-benzoxazepine-2,4'-oxane]
—— 4-[(2,3-Dimethoxyphenyl)methyl]spiro[3,5-dihydro-1,4-benzoxazepine-2,4'-oxane] —— C22H27NO4
4-[(2,3-Dimethoxyphenyl)methyl]spiro[3,5-dihydro-1,4-benzoxazepine-2,4'-oxane]
—— (1-Propan-2-ylpyrazol-4-yl)-spiro[3,5-dihydro-1,4-benzoxazepine-2,4'-oxane]-4-ylmethanone —— C20H25N3O3
(1-Propan-2-ylpyrazol-4-yl)-spiro[3,5-dihydro-1,4-benzoxazepine-2,4'-oxane]-4-ylmethanone
—— (3S)-3-(3,5-dimethyl-1,2,4-triazol-1-yl)-1-spiro[3,5-dihydro-1,4-benzoxazepine-2,4'-oxane]-4-ylbutan-1-one —— C21H28N4O3
(3S)-3-(3,5-dimethyl-1,2,4-triazol-1-yl)-1-spiro[3,5-dihydro-1,4-benzoxazepine-2,4'-oxane]-4-ylbutan-1-one
—— [2-(Dimethylamino)-4-methylpyrimidin-5-yl]-spiro[3,5-dihydro-1,4-benzoxazepine-2,4'-oxane]-4-ylmethanone —— C21H26N4O3
[2-(Dimethylamino)-4-methylpyrimidin-5-yl]-spiro[3,5-dihydro-1,4-benzoxazepine-2,4'-oxane]-4-ylmethanone
—— 1-(7-Chlorospiro[3,5-dihydro-1,4-benzoxazepine-2,4'-oxane]-4-yl)-2-(3,5-dimethyl-1,2,4-triazol-1-yl)ethanone —— C19H23ClN4O3
1-(7-Chlorospiro[3,5-dihydro-1,4-benzoxazepine-2,4'-oxane]-4-yl)-2-(3,5-dimethyl-1,2,4-triazol-1-yl)ethanone
—— [4-[(2-Methylpyrimidin-5-yl)methyl]spiro[3,5-dihydro-1,4-benzoxazepine-2,4'-cyclohexane]-1'-yl]methanol —— C21H27N3O2
[4-[(2-Methylpyrimidin-5-yl)methyl]spiro[3,5-dihydro-1,4-benzoxazepine-2,4'-cyclohexane]-1'-yl]methanol
—— 1-[4-[(2,3-dimethoxyphenyl)methyl]spiro[3,5-dihydro-1,4-benzoxazepine-2,4'-cyclohexane]-1'-yl]-N,N-dimethylmethanamine —— C26H36N2O3
1-[4-[(2,3-dimethoxyphenyl)methyl]spiro[3,5-dihydro-1,4-benzoxazepine-2,4'-cyclohexane]-1'-yl]-N,N-dimethylmethanamine
—— 2-(3,5-Dimethyl-1,2,4-triazol-1-yl)-1-spiro[3,5-dihydro-1,4-benzoxazepine-2,4'-oxane]-4-ylethanone —— C19H24N4O3
2-(3,5-Dimethyl-1,2,4-triazol-1-yl)-1-spiro[3,5-dihydro-1,4-benzoxazepine-2,4'-oxane]-4-ylethanone
—— (4S)-1-methyl-4-(spiro[3,5-dihydro-1,4-benzoxazepine-2,4'-oxane]-4-carbonyl)pyrrolidin-2-one —— C19H24N2O4
(4S)-1-methyl-4-(spiro[3,5-dihydro-1,4-benzoxazepine-2,4'-oxane]-4-carbonyl)pyrrolidin-2-one
—— (2-Methylpyrazol-3-yl)-spiro[3,5-dihydro-1,4-benzoxazepine-2,4'-oxane]-4-ylmethanone —— C18H21N3O3
(2-Methylpyrazol-3-yl)-spiro[3,5-dihydro-1,4-benzoxazepine-2,4'-oxane]-4-ylmethanone
—— 2-(4-Acetyl-3,5-dimethylpyrazol-1-yl)-1-spiro[3,5-dihydro-1,4-benzoxazepine-2,4'-oxane]-4-ylethanone —— C22H27N3O4
2-(4-Acetyl-3,5-dimethylpyrazol-1-yl)-1-spiro[3,5-dihydro-1,4-benzoxazepine-2,4'-oxane]-4-ylethanone