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苯并恶嗪类

中文名称 英文名称 CAS号 化学式 结构式图片
—— 1-[(3S)-3-[(dimethylamino)methyl]-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-2-[(3S)-1,1-dioxothiolan-3-yl]ethanone —— C18H26N2O4S
1-[(3S)-3-[(dimethylamino)methyl]-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-2-[(3S)-1,1-dioxothiolan-3-yl]ethanone
—— [(3S)-3-[(dimethylamino)methyl]-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-[(3S)-1,1-dioxothiolan-3-yl]methanone —— C17H24N2O4S
[(3S)-3-[(dimethylamino)methyl]-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-[(3S)-1,1-dioxothiolan-3-yl]methanone
—— [4-[(2-Ethylpyrimidin-5-yl)methyl]spiro[3,5-dihydro-1,4-benzoxazepine-2,4'-cyclohexane]-1'-yl]methanol —— C22H29N3O2
[4-[(2-Ethylpyrimidin-5-yl)methyl]spiro[3,5-dihydro-1,4-benzoxazepine-2,4'-cyclohexane]-1'-yl]methanol
—— [(3S)-3-[(dimethylamino)methyl]-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-(5-methylpyrazin-2-yl)methanone —— C18H22N4O2
[(3S)-3-[(dimethylamino)methyl]-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-(5-methylpyrazin-2-yl)methanone
—— (2R)-7-methoxy-1'-methyl-4-[[(3S)-oxolan-3-yl]methyl]spiro[3,5-dihydro-1,4-benzoxazepine-2,4'-azepane] —— C21H32N2O3
(2R)-7-methoxy-1'-methyl-4-[[(3S)-oxolan-3-yl]methyl]spiro[3,5-dihydro-1,4-benzoxazepine-2,4'-azepane]
—— [(3S)-3-[(dimethylamino)methyl]-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-[1-(3-fluorophenyl)cyclopropyl]methanone —— C22H25FN2O2
[(3S)-3-[(dimethylamino)methyl]-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-[1-(3-fluorophenyl)cyclopropyl]methanone
—— [(3S)-3-[(dimethylamino)methyl]-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-pyrazolo[1,5-a]pyrimidin-3-ylmethanone —— C19H21N5O2
[(3S)-3-[(dimethylamino)methyl]-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-pyrazolo[1,5-a]pyrimidin-3-ylmethanone
—— 2-(4-acetyl-7-methylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-piperidine]-1'-yl)-1-[(2R)-2-methylpiperidin-1-yl]ethanone —— C24H35N3O3
2-(4-acetyl-7-methylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-piperidine]-1'-yl)-1-[(2R)-2-methylpiperidin-1-yl]ethanone
—— 1-[(3S)-3-[(dimethylamino)methyl]-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-2-(4-methylsulfonylphenyl)ethanone —— C21H26N2O4S
1-[(3S)-3-[(dimethylamino)methyl]-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-2-(4-methylsulfonylphenyl)ethanone
—— 1-[(3S)-3-[(dimethylamino)methyl]-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-2-(4-methoxy-3-methylphenyl)ethanone —— C22H28N2O3
1-[(3S)-3-[(dimethylamino)methyl]-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-2-(4-methoxy-3-methylphenyl)ethanone
—— 1-[(3R)-3-[(dimethylamino)methyl]-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-2-[(3R)-1,1-dioxothiolan-3-yl]ethanone —— C18H26N2O4S
1-[(3R)-3-[(dimethylamino)methyl]-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-2-[(3R)-1,1-dioxothiolan-3-yl]ethanone
—— [(3R)-3-[(dimethylamino)methyl]-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-pyrazolo[1,5-a]pyrimidin-3-ylmethanone —— C19H21N5O2
[(3R)-3-[(dimethylamino)methyl]-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-pyrazolo[1,5-a]pyrimidin-3-ylmethanone
—— 2-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-1-[(3R)-3-[(dimethylamino)methyl]-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]ethanone —— C23H28N2O4
2-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-1-[(3R)-3-[(dimethylamino)methyl]-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]ethanone
—— [(3S)-3-[(dimethylamino)methyl]-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-[(3R)-1,1-dioxothiolan-3-yl]methanone —— C17H24N2O4S
[(3S)-3-[(dimethylamino)methyl]-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-[(3R)-1,1-dioxothiolan-3-yl]methanone
—— [(3S)-3-[(dimethylamino)methyl]-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-(1,3-dimethylpyrazol-4-yl)methanone —— C18H24N4O2
[(3S)-3-[(dimethylamino)methyl]-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-(1,3-dimethylpyrazol-4-yl)methanone
—— 1-[(3R)-3-[(dimethylamino)methyl]-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-2-(4-methylphenyl)ethanone —— C21H26N2O2
1-[(3R)-3-[(dimethylamino)methyl]-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-2-(4-methylphenyl)ethanone
—— 1-[(2S)-7-methoxy-1'-[[(3S)-oxolan-3-yl]methyl]spiro[3,5-dihydro-1,4-benzoxazepine-2,4'-azepane]-4-yl]ethanone —— C22H32N2O4
1-[(2S)-7-methoxy-1'-[[(3S)-oxolan-3-yl]methyl]spiro[3,5-dihydro-1,4-benzoxazepine-2,4'-azepane]-4-yl]ethanone
—— [4'-[(dimethylamino)methyl]spiro[3,5-dihydro-1,4-benzoxazepine-2,1'-cyclohexane]-4-yl]-[(3R)-oxolan-3-yl]methanone —— C22H32N2O3
[4'-[(dimethylamino)methyl]spiro[3,5-dihydro-1,4-benzoxazepine-2,1'-cyclohexane]-4-yl]-[(3R)-oxolan-3-yl]methanone
—— 1-[(3R)-3-[(dimethylamino)methyl]-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-2-(4-ethoxyphenyl)ethanone —— C22H28N2O3
1-[(3R)-3-[(dimethylamino)methyl]-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-2-(4-ethoxyphenyl)ethanone
—— 1-[(2S)-1'-(2-methylpyridine-3-carbonyl)spiro[3,5-dihydro-1,4-benzoxazepine-2,4'-azepane]-4-yl]ethanone —— C23H27N3O3
1-[(2S)-1'-(2-methylpyridine-3-carbonyl)spiro[3,5-dihydro-1,4-benzoxazepine-2,4'-azepane]-4-yl]ethanone
—— 7-[(2-bromoethyl)amino]-8H-naphtho[2,3-a]phenoxazine-8,13(14H)-dione —— C22H15BrN2O3
7-[(2-bromoethyl)amino]-8H-naphtho[2,3-a]phenoxazine-8,13(14H)-dione
—— 4-[2-[(3S)-3-[(dimethylamino)methyl]-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-2-oxoethyl]benzenesulfonamide —— C20H25N3O4S
4-[2-[(3S)-3-[(dimethylamino)methyl]-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-2-oxoethyl]benzenesulfonamide
—— 1-[(3S)-3-[(dimethylamino)methyl]-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-3-(1,2,4-triazol-1-yl)propan-1-one —— C17H23N5O2
1-[(3S)-3-[(dimethylamino)methyl]-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-3-(1,2,4-triazol-1-yl)propan-1-one
—— [(3R)-3-[(dimethylamino)methyl]-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-[1-(4-methylphenyl)cyclopropyl]methanone —— C23H28N2O2
[(3R)-3-[(dimethylamino)methyl]-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-[1-(4-methylphenyl)cyclopropyl]methanone
—— 1-[(3R)-3-[(dimethylamino)methyl]-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-3-(1,2,4-triazol-1-yl)propan-1-one —— C17H23N5O2
1-[(3R)-3-[(dimethylamino)methyl]-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-3-(1,2,4-triazol-1-yl)propan-1-one
—— 1-[(2S)-1'-(pyridine-3-carbonyl)spiro[3,5-dihydro-1,4-benzoxazepine-2,4'-azepane]-4-yl]ethanone —— C22H25N3O3
1-[(2S)-1'-(pyridine-3-carbonyl)spiro[3,5-dihydro-1,4-benzoxazepine-2,4'-azepane]-4-yl]ethanone
—— (3,4-dimethoxyphenyl)-[(3R)-3-[(dimethylamino)methyl]-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]methanone —— C21H26N2O4
(3,4-dimethoxyphenyl)-[(3R)-3-[(dimethylamino)methyl]-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]methanone
—— [(3R)-3-[(dimethylamino)methyl]-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-[(3S)-1,1-dioxothiolan-3-yl]methanone —— C17H24N2O4S
[(3R)-3-[(dimethylamino)methyl]-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-[(3S)-1,1-dioxothiolan-3-yl]methanone
—— 2-(3,4-dimethoxyphenyl)-1-[(3S)-3-[(dimethylamino)methyl]-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]ethanone —— C22H28N2O4
2-(3,4-dimethoxyphenyl)-1-[(3S)-3-[(dimethylamino)methyl]-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]ethanone
—— 1-[(3S)-3-[(dimethylamino)methyl]-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-2-(4-methyl-1,2,5-oxadiazol-3-yl)ethanone —— C17H22N4O3
1-[(3S)-3-[(dimethylamino)methyl]-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-2-(4-methyl-1,2,5-oxadiazol-3-yl)ethanone
—— 1-[(2R)-4,7-dimethylspiro[3,5-dihydro-1,4-benzoxazepine-2,3'-piperidine]-1'-yl]-2-phenylethanone —— C23H28N2O2
1-[(2R)-4,7-dimethylspiro[3,5-dihydro-1,4-benzoxazepine-2,3'-piperidine]-1'-yl]-2-phenylethanone
—— 1-[(3S)-3-[(dimethylamino)methyl]-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-2-[(3R)-1,1-dioxothiolan-3-yl]ethanone —— C18H26N2O4S
1-[(3S)-3-[(dimethylamino)methyl]-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-2-[(3R)-1,1-dioxothiolan-3-yl]ethanone
—— [(3R)-3-[(dimethylamino)methyl]-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-[1-(2-fluorophenyl)cyclopropyl]methanone —— C22H25FN2O2
[(3R)-3-[(dimethylamino)methyl]-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-[1-(2-fluorophenyl)cyclopropyl]methanone
—— 1-[(3S)-3-[(dimethylamino)methyl]-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-2-(3,5-dimethyl-1,2,4-triazol-1-yl)ethanone —— C18H25N5O2
1-[(3S)-3-[(dimethylamino)methyl]-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-2-(3,5-dimethyl-1,2,4-triazol-1-yl)ethanone
—— 1-[(3R)-3-[(dimethylamino)methyl]-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-2-(3,5-dimethyl-1,2,4-triazol-1-yl)ethanone —— C18H25N5O2
1-[(3R)-3-[(dimethylamino)methyl]-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-2-(3,5-dimethyl-1,2,4-triazol-1-yl)ethanone
—— 2-(1,3-benzodioxol-5-yl)-1-[(3S)-3-[(dimethylamino)methyl]-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]ethanone —— C21H24N2O4
2-(1,3-benzodioxol-5-yl)-1-[(3S)-3-[(dimethylamino)methyl]-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]ethanone
—— 1-[(2S)-1'-(3-phenoxypropyl)spiro[3,5-dihydro-1,4-benzoxazepine-2,4'-azepane]-4-yl]ethanone —— C25H32N2O3
1-[(2S)-1'-(3-phenoxypropyl)spiro[3,5-dihydro-1,4-benzoxazepine-2,4'-azepane]-4-yl]ethanone
—— 1-[(2R)-1'-(3-phenoxypropyl)spiro[3,5-dihydro-1,4-benzoxazepine-2,4'-azepane]-4-yl]ethanone —— C25H32N2O3
1-[(2R)-1'-(3-phenoxypropyl)spiro[3,5-dihydro-1,4-benzoxazepine-2,4'-azepane]-4-yl]ethanone
—— [(3R)-3-[(dimethylamino)methyl]-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-[(3R)-1,1-dioxothiolan-3-yl]methanone —— C17H24N2O4S
[(3R)-3-[(dimethylamino)methyl]-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-[(3R)-1,1-dioxothiolan-3-yl]methanone
—— 1-[(3R)-3-[(dimethylamino)methyl]-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-4-(1,2,4-triazol-1-yl)butan-1-one —— C18H25N5O2
1-[(3R)-3-[(dimethylamino)methyl]-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-4-(1,2,4-triazol-1-yl)butan-1-one
—— 4-[(3S)-3-[(dimethylamino)methyl]-3,5-dihydro-2H-1,4-benzoxazepine-4-carbonyl]benzenesulfonamide —— C19H23N3O4S
4-[(3S)-3-[(dimethylamino)methyl]-3,5-dihydro-2H-1,4-benzoxazepine-4-carbonyl]benzenesulfonamide
—— [(3R)-3-[(dimethylamino)methyl]-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-(1,5-dimethylpyrazol-4-yl)methanone —— C18H24N4O2
[(3R)-3-[(dimethylamino)methyl]-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-(1,5-dimethylpyrazol-4-yl)methanone
—— 1-[(3S)-3-[(dimethylamino)methyl]-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-4-(1,2,4-triazol-1-yl)butan-1-one —— C18H25N5O2
1-[(3S)-3-[(dimethylamino)methyl]-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-4-(1,2,4-triazol-1-yl)butan-1-one
—— 2-(2-methoxyphenyl)-1-[(2S)-4-methylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-azepane]-1'-yl]ethanone —— C24H30N2O3
2-(2-methoxyphenyl)-1-[(2S)-4-methylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-azepane]-1'-yl]ethanone
—— [(3R)-3-[(dimethylamino)methyl]-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-(1,3-dimethylpyrazol-4-yl)methanone —— C18H24N4O2
[(3R)-3-[(dimethylamino)methyl]-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-(1,3-dimethylpyrazol-4-yl)methanone
—— 1-[(3S)-3-[(dimethylamino)methyl]-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-2-(4-methylphenyl)ethanone —— C21H26N2O2
1-[(3S)-3-[(dimethylamino)methyl]-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-2-(4-methylphenyl)ethanone
—— 1-[7-methyl-1'-[[(3S)-oxolan-3-yl]methyl]spiro[3,5-dihydro-1,4-benzoxazepine-2,4'-piperidine]-4-yl]ethanone —— C21H30N2O3
1-[7-methyl-1'-[[(3S)-oxolan-3-yl]methyl]spiro[3,5-dihydro-1,4-benzoxazepine-2,4'-piperidine]-4-yl]ethanone
—— [(3R)-3-[(dimethylamino)methyl]-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-(1-phenylcyclopropyl)methanone —— C22H26N2O2
[(3R)-3-[(dimethylamino)methyl]-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-(1-phenylcyclopropyl)methanone
—— 1-[(3S)-3-[(dimethylamino)methyl]-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-2-(2-fluorophenyl)ethanone —— C20H23FN2O2
1-[(3S)-3-[(dimethylamino)methyl]-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-2-(2-fluorophenyl)ethanone
—— 1-[(2S)-1'-(2-phenylethyl)spiro[3,5-dihydro-1,4-benzoxazepine-2,4'-azepane]-4-yl]ethanone —— C24H30N2O2
1-[(2S)-1'-(2-phenylethyl)spiro[3,5-dihydro-1,4-benzoxazepine-2,4'-azepane]-4-yl]ethanone