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苯并恶嗪类

中文名称 英文名称 CAS号 化学式 结构式图片
—— 1-[(3S)-3-(imidazol-1-ylmethyl)-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-2-(3-methylphenyl)ethanone —— C22H23N3O2
1-[(3S)-3-(imidazol-1-ylmethyl)-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-2-(3-methylphenyl)ethanone
—— 2-(4-ethoxyphenyl)-1-[(3R)-3-(imidazol-1-ylmethyl)-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]ethanone —— C23H25N3O3
2-(4-ethoxyphenyl)-1-[(3R)-3-(imidazol-1-ylmethyl)-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]ethanone
—— (3S)-4-[(2-fluorophenyl)methyl]-3-(imidazol-1-ylmethyl)-3,5-dihydro-2H-1,4-benzoxazepine —— C20H20FN3O
(3S)-4-[(2-fluorophenyl)methyl]-3-(imidazol-1-ylmethyl)-3,5-dihydro-2H-1,4-benzoxazepine
—— 1-[(3R)-3-(imidazol-1-ylmethyl)-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-2-(3-methylphenyl)ethanone —— C22H23N3O2
1-[(3R)-3-(imidazol-1-ylmethyl)-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-2-(3-methylphenyl)ethanone
—— [(3S)-3-(imidazol-1-ylmethyl)-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-pyrimidin-5-ylmethanone —— C18H17N5O2
[(3S)-3-(imidazol-1-ylmethyl)-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-pyrimidin-5-ylmethanone
—— [(3R)-3-(imidazol-1-ylmethyl)-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-(4-methyl-1,3-thiazol-5-yl)methanone —— C18H18N4O2S
[(3R)-3-(imidazol-1-ylmethyl)-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-(4-methyl-1,3-thiazol-5-yl)methanone
—— (2,4-dimethyl-1,3-thiazol-5-yl)-[(3S)-3-(imidazol-1-ylmethyl)-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]methanone —— C19H20N4O2S
(2,4-dimethyl-1,3-thiazol-5-yl)-[(3S)-3-(imidazol-1-ylmethyl)-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]methanone
—— 2-(3-fluorophenyl)-1-[(3S)-3-(imidazol-1-ylmethyl)-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]ethanone —— C21H20FN3O2
2-(3-fluorophenyl)-1-[(3S)-3-(imidazol-1-ylmethyl)-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]ethanone
—— (2,4-dimethyl-1,3-oxazol-5-yl)-[(3S)-3-(imidazol-1-ylmethyl)-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]methanone —— C19H20N4O3
(2,4-dimethyl-1,3-oxazol-5-yl)-[(3S)-3-(imidazol-1-ylmethyl)-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]methanone
—— (3R)-4-[(2-fluorophenyl)methyl]-3-(imidazol-1-ylmethyl)-3,5-dihydro-2H-1,4-benzoxazepine —— C20H20FN3O
(3R)-4-[(2-fluorophenyl)methyl]-3-(imidazol-1-ylmethyl)-3,5-dihydro-2H-1,4-benzoxazepine
—— N-[4-[[4'-(hydroxymethyl)spiro[3,5-dihydro-1,4-benzoxazepine-2,1'-cyclohexane]-4-yl]methyl]phenyl]acetamide —— C24H30N2O3
N-[4-[[4'-(hydroxymethyl)spiro[3,5-dihydro-1,4-benzoxazepine-2,1'-cyclohexane]-4-yl]methyl]phenyl]acetamide
—— 2-Imidazol-1-yl-1-(4-methylsulfonylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-piperidine]-1'-yl)ethanone —— C19H24N4O4S
2-Imidazol-1-yl-1-(4-methylsulfonylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-piperidine]-1'-yl)ethanone
—— 2-(4-fluorophenyl)-1-[(3R)-3-(imidazol-1-ylmethyl)-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]ethanone —— C21H20FN3O2
2-(4-fluorophenyl)-1-[(3R)-3-(imidazol-1-ylmethyl)-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]ethanone
—— 1-[(3R)-3-(imidazol-1-ylmethyl)-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-3-(2-methoxyphenyl)propan-1-one —— C23H25N3O3
1-[(3R)-3-(imidazol-1-ylmethyl)-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-3-(2-methoxyphenyl)propan-1-one
—— 7-Methyl-1'-[(3-methylimidazol-4-yl)methyl]-4-methylsulfonylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-piperidine] —— C20H28N4O3S
7-Methyl-1'-[(3-methylimidazol-4-yl)methyl]-4-methylsulfonylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-piperidine]
—— 1-[(3R)-3-(imidazol-1-ylmethyl)-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-2-(4-methylphenyl)ethanone —— C22H23N3O2
1-[(3R)-3-(imidazol-1-ylmethyl)-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-2-(4-methylphenyl)ethanone
—— 2-(3,4-dimethoxyphenyl)-1-[(3R)-3-(imidazol-1-ylmethyl)-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]ethanone —— C23H25N3O4
2-(3,4-dimethoxyphenyl)-1-[(3R)-3-(imidazol-1-ylmethyl)-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]ethanone
—— 1-[(3S)-3-(imidazol-1-ylmethyl)-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-2-(4-methylphenyl)ethanone —— C22H23N3O2
1-[(3S)-3-(imidazol-1-ylmethyl)-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-2-(4-methylphenyl)ethanone
—— 1-[4'-[(Dimethylamino)methyl]spiro[3,5-dihydro-1,4-benzoxazepine-2,1'-cyclohexane]-4-yl]-4-imidazol-1-ylbutan-1-one —— C24H34N4O2
1-[4'-[(Dimethylamino)methyl]spiro[3,5-dihydro-1,4-benzoxazepine-2,1'-cyclohexane]-4-yl]-4-imidazol-1-ylbutan-1-one
—— [(3S)-3-(imidazol-1-ylmethyl)-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-pyridin-3-ylmethanone —— C19H18N4O2
[(3S)-3-(imidazol-1-ylmethyl)-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-pyridin-3-ylmethanone
—— 2-(4-ethoxyphenyl)-1-[(3S)-3-(imidazol-1-ylmethyl)-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]ethanone —— C23H25N3O3
2-(4-ethoxyphenyl)-1-[(3S)-3-(imidazol-1-ylmethyl)-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]ethanone
—— 1-[(3S)-3-(imidazol-1-ylmethyl)-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-2-(3-methoxyphenyl)ethanone —— C22H23N3O3
1-[(3S)-3-(imidazol-1-ylmethyl)-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-2-(3-methoxyphenyl)ethanone
—— [4-(Quinoxalin-6-ylmethyl)spiro[3,5-dihydro-1,4-benzoxazepine-2,4'-cyclohexane]-1'-yl]methanol —— C24H27N3O2
[4-(Quinoxalin-6-ylmethyl)spiro[3,5-dihydro-1,4-benzoxazepine-2,4'-cyclohexane]-1'-yl]methanol
—— 1-[(2R)-4-acetylspiro[3,5-dihydro-1,4-benzoxazepine-2,3'-piperidine]-1'-yl]-4-imidazol-1-ylbutan-1-one —— C22H28N4O3
1-[(2R)-4-acetylspiro[3,5-dihydro-1,4-benzoxazepine-2,3'-piperidine]-1'-yl]-4-imidazol-1-ylbutan-1-one
—— 2-(3,4-dimethoxyphenyl)-1-[(3S)-3-(imidazol-1-ylmethyl)-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]ethanone —— C23H25N3O4
2-(3,4-dimethoxyphenyl)-1-[(3S)-3-(imidazol-1-ylmethyl)-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]ethanone
—— (3R,3'S)-1'-(1,5-dimethylpyrazole-4-carbonyl)-N,N-dimethyl-5-oxospiro[2,4-dihydro-1,4-benzoxazepine-3,4'-pyrrolidine]-3'-carboxamide —— C21H25N5O4
(3R,3'S)-1'-(1,5-dimethylpyrazole-4-carbonyl)-N,N-dimethyl-5-oxospiro[2,4-dihydro-1,4-benzoxazepine-3,4'-pyrrolidine]-3'-carboxamide
—— [4'-[(dimethylamino)methyl]spiro[3,5-dihydro-1,4-benzoxazepine-2,1'-cyclohexane]-4-yl]-(1H-pyrazol-5-yl)methanone —— C21H28N4O2
[4'-[(dimethylamino)methyl]spiro[3,5-dihydro-1,4-benzoxazepine-2,1'-cyclohexane]-4-yl]-(1H-pyrazol-5-yl)methanone
—— [4-[(2,4,5-Trimethoxyphenyl)methyl]spiro[3,5-dihydro-1,4-benzoxazepine-2,4'-cyclohexane]-1'-yl]methanol —— C25H33NO5
[4-[(2,4,5-Trimethoxyphenyl)methyl]spiro[3,5-dihydro-1,4-benzoxazepine-2,4'-cyclohexane]-1'-yl]methanol
—— (7-methyl-4-methylsulfonylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-piperidine]-1'-yl)-(1H-pyrazol-5-yl)methanone —— C19H24N4O4S
(7-methyl-4-methylsulfonylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-piperidine]-1'-yl)-(1H-pyrazol-5-yl)methanone
—— 2-(4-fluorophenyl)-1-[(3S)-3-(imidazol-1-ylmethyl)-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]ethanone —— C21H20FN3O2
2-(4-fluorophenyl)-1-[(3S)-3-(imidazol-1-ylmethyl)-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]ethanone
—— 1-[(2S)-4-acetylspiro[3,5-dihydro-1,4-benzoxazepine-2,3'-piperidine]-1'-yl]-4-imidazol-1-ylbutan-1-one —— C22H28N4O3
1-[(2S)-4-acetylspiro[3,5-dihydro-1,4-benzoxazepine-2,3'-piperidine]-1'-yl]-4-imidazol-1-ylbutan-1-one
—— (3R,3'S)-N,N-dimethyl-1'-(1-methylpyrazole-3-carbonyl)-5-oxospiro[2,4-dihydro-1,4-benzoxazepine-3,4'-pyrrolidine]-3'-carboxamide —— C20H23N5O4
(3R,3'S)-N,N-dimethyl-1'-(1-methylpyrazole-3-carbonyl)-5-oxospiro[2,4-dihydro-1,4-benzoxazepine-3,4'-pyrrolidine]-3'-carboxamide
—— 4-[[2-(2-Methoxyethyl)pyrimidin-5-yl]methyl]spiro[3,5-dihydro-1,4-benzoxazepine-2,4'-oxane] —— C21H27N3O3
4-[[2-(2-Methoxyethyl)pyrimidin-5-yl]methyl]spiro[3,5-dihydro-1,4-benzoxazepine-2,4'-oxane]
—— [4-[(2-Fluoro-3-methoxyphenyl)methyl]spiro[3,5-dihydro-1,4-benzoxazepine-2,4'-cyclohexane]-1'-yl]methanol —— C23H28FNO3
[4-[(2-Fluoro-3-methoxyphenyl)methyl]spiro[3,5-dihydro-1,4-benzoxazepine-2,4'-cyclohexane]-1'-yl]methanol
—— [4-[(2,3,4-Trimethoxyphenyl)methyl]spiro[3,5-dihydro-1,4-benzoxazepine-2,4'-cyclohexane]-1'-yl]methanol —— C25H33NO5
[4-[(2,3,4-Trimethoxyphenyl)methyl]spiro[3,5-dihydro-1,4-benzoxazepine-2,4'-cyclohexane]-1'-yl]methanol
—— [(3R)-3-(imidazol-1-ylmethyl)-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-pyridin-3-ylmethanone —— C19H18N4O2
[(3R)-3-(imidazol-1-ylmethyl)-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-pyridin-3-ylmethanone
—— [4-[(5-Methylfuran-2-yl)methyl]spiro[3,5-dihydro-1,4-benzoxazepine-2,4'-cyclohexane]-1'-yl]methanol —— C21H27NO3
[4-[(5-Methylfuran-2-yl)methyl]spiro[3,5-dihydro-1,4-benzoxazepine-2,4'-cyclohexane]-1'-yl]methanol
—— [4-[(5-Chloro-1,3-dimethylpyrazol-4-yl)methyl]spiro[3,5-dihydro-1,4-benzoxazepine-2,4'-cyclohexane]-1'-yl]methanol —— C21H28ClN3O2
[4-[(5-Chloro-1,3-dimethylpyrazol-4-yl)methyl]spiro[3,5-dihydro-1,4-benzoxazepine-2,4'-cyclohexane]-1'-yl]methanol
—— [4-[(4-Methoxy-3-methylphenyl)methyl]spiro[3,5-dihydro-1,4-benzoxazepine-2,4'-cyclohexane]-1'-yl]methanol —— C24H31NO3
[4-[(4-Methoxy-3-methylphenyl)methyl]spiro[3,5-dihydro-1,4-benzoxazepine-2,4'-cyclohexane]-1'-yl]methanol
—— (3R,3'S)-1'-[3-(2-fluorophenoxy)propyl]-N,N-dimethyl-5-oxospiro[2,4-dihydro-1,4-benzoxazepine-3,4'-pyrrolidine]-3'-carboxamide —— C24H28FN3O4
(3R,3'S)-1'-[3-(2-fluorophenoxy)propyl]-N,N-dimethyl-5-oxospiro[2,4-dihydro-1,4-benzoxazepine-3,4'-pyrrolidine]-3'-carboxamide
—— 1-[(2R)-7-methyl-1'-(3-phenoxypropyl)spiro[3,5-dihydro-1,4-benzoxazepine-2,3'-piperidine]-4-yl]ethanone —— C25H32N2O3
1-[(2R)-7-methyl-1'-(3-phenoxypropyl)spiro[3,5-dihydro-1,4-benzoxazepine-2,3'-piperidine]-4-yl]ethanone
—— (3R,3'S)-N,N-dimethyl-1'-(5-methyl-3-propan-2-yl-1,2-oxazole-4-carbonyl)-5-oxospiro[2,4-dihydro-1,4-benzoxazepine-3,4'-pyrrolidine]-3'-carboxamide —— C23H28N4O5
(3R,3'S)-N,N-dimethyl-1'-(5-methyl-3-propan-2-yl-1,2-oxazole-4-carbonyl)-5-oxospiro[2,4-dihydro-1,4-benzoxazepine-3,4'-pyrrolidine]-3'-carboxamide
—— (3R,3'S)-N,N-dimethyl-5-oxo-1'-(3-phenoxypropyl)spiro[2,4-dihydro-1,4-benzoxazepine-3,4'-pyrrolidine]-3'-carboxamide —— C24H29N3O4
(3R,3'S)-N,N-dimethyl-5-oxo-1'-(3-phenoxypropyl)spiro[2,4-dihydro-1,4-benzoxazepine-3,4'-pyrrolidine]-3'-carboxamide
—— (2S)-7-methoxy-1'-(piperidine-4-carbonyl)spiro[3,4-dihydro-1,4-benzoxazepine-2,3'-piperidine]-5-one —— C20H27N3O4
(2S)-7-methoxy-1'-(piperidine-4-carbonyl)spiro[3,4-dihydro-1,4-benzoxazepine-2,3'-piperidine]-5-one
—— (3R,3'S)-1'-(2,4-dimethyl-1,3-oxazole-5-carbonyl)-N,N-dimethyl-5-oxospiro[2,4-dihydro-1,4-benzoxazepine-3,4'-pyrrolidine]-3'-carboxamide —— C21H24N4O5
(3R,3'S)-1'-(2,4-dimethyl-1,3-oxazole-5-carbonyl)-N,N-dimethyl-5-oxospiro[2,4-dihydro-1,4-benzoxazepine-3,4'-pyrrolidine]-3'-carboxamide
—— 1-[(2S)-1'-[(3S)-piperidine-3-carbonyl]spiro[3,5-dihydro-1,4-benzoxazepine-2,3'-piperidine]-4-yl]ethanone —— C21H29N3O3
1-[(2S)-1'-[(3S)-piperidine-3-carbonyl]spiro[3,5-dihydro-1,4-benzoxazepine-2,3'-piperidine]-4-yl]ethanone
—— (3R,3'S)-N,N-dimethyl-1'-(5-methylthiophene-3-carbonyl)-5-oxospiro[2,4-dihydro-1,4-benzoxazepine-3,4'-pyrrolidine]-3'-carboxamide —— C21H23N3O4S
(3R,3'S)-N,N-dimethyl-1'-(5-methylthiophene-3-carbonyl)-5-oxospiro[2,4-dihydro-1,4-benzoxazepine-3,4'-pyrrolidine]-3'-carboxamide
—— (3R,3'S)-N,N-dimethyl-5-oxo-1'-(pyridine-4-carbonyl)spiro[2,4-dihydro-1,4-benzoxazepine-3,4'-pyrrolidine]-3'-carboxamide —— C21H22N4O4
(3R,3'S)-N,N-dimethyl-5-oxo-1'-(pyridine-4-carbonyl)spiro[2,4-dihydro-1,4-benzoxazepine-3,4'-pyrrolidine]-3'-carboxamide
—— (3R,3'S)-1'-(5-ethyl-3-methyl-1,2-oxazole-4-carbonyl)-N,N-dimethyl-5-oxospiro[2,4-dihydro-1,4-benzoxazepine-3,4'-pyrrolidine]-3'-carboxamide —— C22H26N4O5
(3R,3'S)-1'-(5-ethyl-3-methyl-1,2-oxazole-4-carbonyl)-N,N-dimethyl-5-oxospiro[2,4-dihydro-1,4-benzoxazepine-3,4'-pyrrolidine]-3'-carboxamide
—— (3R,3'S)-N,N-dimethyl-5-oxo-1'-(5-propan-2-yl-1,2-oxazole-3-carbonyl)spiro[2,4-dihydro-1,4-benzoxazepine-3,4'-pyrrolidine]-3'-carboxamide —— C22H26N4O5
(3R,3'S)-N,N-dimethyl-5-oxo-1'-(5-propan-2-yl-1,2-oxazole-3-carbonyl)spiro[2,4-dihydro-1,4-benzoxazepine-3,4'-pyrrolidine]-3'-carboxamide