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苯并恶嗪类

中文名称 英文名称 CAS号 化学式 结构式图片
—— (2S)-N-[(2S)-1-(4-methoxyphenoxy)propan-2-yl]-2-[(2R)-2-methyl-3-oxo-1,4-benzoxazin-4-yl]propanamide —— C22H26N2O5
(2S)-N-[(2S)-1-(4-methoxyphenoxy)propan-2-yl]-2-[(2R)-2-methyl-3-oxo-1,4-benzoxazin-4-yl]propanamide
—— (2S)-2-imidazol-1-yl-N-[(2S)-2-methyl-3-oxo-4H-1,4-benzoxazin-6-yl]propanamide —— C15H16N4O3
(2S)-2-imidazol-1-yl-N-[(2S)-2-methyl-3-oxo-4H-1,4-benzoxazin-6-yl]propanamide
—— 4-methyl-5-oxo-N-[(1R)-1-pyridin-4-ylethyl]spiro[3H-1,4-benzoxazepine-2,4'-cyclohexane]-1'-carboxamide —— C23H27N3O3
4-methyl-5-oxo-N-[(1R)-1-pyridin-4-ylethyl]spiro[3H-1,4-benzoxazepine-2,4'-cyclohexane]-1'-carboxamide
—— 2,2-dimethyl-6-[(3S)-3-(5-pyridin-3-yl-1,3,4-oxadiazol-2-yl)pyrrolidine-1-carbonyl]-4H-1,4-benzoxazin-3-one —— C22H21N5O4
2,2-dimethyl-6-[(3S)-3-(5-pyridin-3-yl-1,3,4-oxadiazol-2-yl)pyrrolidine-1-carbonyl]-4H-1,4-benzoxazin-3-one
—— N-[2-(3-cyclopropyl-4-pyridin-4-ylpyrazol-1-yl)ethyl]-2,2-dimethyl-3-oxo-4H-1,4-benzoxazine-6-carboxamide —— C24H25N5O3
N-[2-(3-cyclopropyl-4-pyridin-4-ylpyrazol-1-yl)ethyl]-2,2-dimethyl-3-oxo-4H-1,4-benzoxazine-6-carboxamide
—— N-(3-methoxypropyl)-3-oxo-N-[(1S)-1-pyridin-2-ylethyl]-4H-1,4-benzoxazine-6-sulfonamide —— C19H23N3O5S
N-(3-methoxypropyl)-3-oxo-N-[(1S)-1-pyridin-2-ylethyl]-4H-1,4-benzoxazine-6-sulfonamide
—— 2-(7-chloro-5-oxospiro[3H-1,4-benzoxazepine-2,4'-oxane]-4-yl)-N-[(1R)-1-pyridin-4-ylethyl]acetamide —— C22H24ClN3O4
2-(7-chloro-5-oxospiro[3H-1,4-benzoxazepine-2,4'-oxane]-4-yl)-N-[(1R)-1-pyridin-4-ylethyl]acetamide
—— 7-chloro-5-oxo-N-[(1S)-1-thiophen-2-ylethyl]spiro[3,4-dihydro-1,4-benzoxazepine-2,4'-cyclohexane]-1'-carboxamide —— C21H23ClN2O3S
7-chloro-5-oxo-N-[(1S)-1-thiophen-2-ylethyl]spiro[3,4-dihydro-1,4-benzoxazepine-2,4'-cyclohexane]-1'-carboxamide
—— 7-chloro-N-[(1R)-1-(furan-2-yl)ethyl]-5-oxospiro[3,4-dihydro-1,4-benzoxazepine-2,4'-cyclohexane]-1'-carboxamide —— C21H23ClN2O4
7-chloro-N-[(1R)-1-(furan-2-yl)ethyl]-5-oxospiro[3,4-dihydro-1,4-benzoxazepine-2,4'-cyclohexane]-1'-carboxamide
—— (2S)-1-[4'-(dimethylamino)spiro[3,5-dihydro-1,4-benzoxazepine-2,1'-cyclohexane]-4-yl]-2-phenylpropan-1-one —— C25H32N2O2
(2S)-1-[4'-(dimethylamino)spiro[3,5-dihydro-1,4-benzoxazepine-2,1'-cyclohexane]-4-yl]-2-phenylpropan-1-one
—— 4-methyl-5-oxo-N-[(1S)-1-pyridin-4-ylethyl]spiro[3H-1,4-benzoxazepine-2,4'-cyclohexane]-1'-carboxamide —— C23H27N3O3
4-methyl-5-oxo-N-[(1S)-1-pyridin-4-ylethyl]spiro[3H-1,4-benzoxazepine-2,4'-cyclohexane]-1'-carboxamide
—— 7-chloro-N-[(1S)-1-(furan-2-yl)ethyl]-5-oxospiro[3,4-dihydro-1,4-benzoxazepine-2,4'-cyclohexane]-1'-carboxamide —— C21H23ClN2O4
7-chloro-N-[(1S)-1-(furan-2-yl)ethyl]-5-oxospiro[3,4-dihydro-1,4-benzoxazepine-2,4'-cyclohexane]-1'-carboxamide
—— 7-chloro-5-oxo-N-[(1R)-1-thiophen-2-ylethyl]spiro[3,4-dihydro-1,4-benzoxazepine-2,4'-cyclohexane]-1'-carboxamide —— C21H23ClN2O3S
7-chloro-5-oxo-N-[(1R)-1-thiophen-2-ylethyl]spiro[3,4-dihydro-1,4-benzoxazepine-2,4'-cyclohexane]-1'-carboxamide
—— N-(3-methoxypropyl)-3-oxo-N-[(1R)-1-pyridin-2-ylethyl]-4H-1,4-benzoxazine-6-sulfonamide —— C19H23N3O5S
N-(3-methoxypropyl)-3-oxo-N-[(1R)-1-pyridin-2-ylethyl]-4H-1,4-benzoxazine-6-sulfonamide
—— (2R)-1-[4'-(dimethylamino)spiro[3,5-dihydro-1,4-benzoxazepine-2,1'-cyclohexane]-4-yl]-2-phenylpropan-1-one —— C25H32N2O2
(2R)-1-[4'-(dimethylamino)spiro[3,5-dihydro-1,4-benzoxazepine-2,1'-cyclohexane]-4-yl]-2-phenylpropan-1-one
—— 2-(7-chloro-5-oxospiro[3H-1,4-benzoxazepine-2,4'-oxane]-4-yl)-N-[(1S)-1-pyridin-4-ylethyl]acetamide —— C22H24ClN3O4
2-(7-chloro-5-oxospiro[3H-1,4-benzoxazepine-2,4'-oxane]-4-yl)-N-[(1S)-1-pyridin-4-ylethyl]acetamide
—— 2,2-dimethyl-6-[(3R)-3-(5-pyridin-3-yl-1,3,4-oxadiazol-2-yl)pyrrolidine-1-carbonyl]-4H-1,4-benzoxazin-3-one —— C22H21N5O4
2,2-dimethyl-6-[(3R)-3-(5-pyridin-3-yl-1,3,4-oxadiazol-2-yl)pyrrolidine-1-carbonyl]-4H-1,4-benzoxazin-3-one
—— (2S)-2-methyl-1-[4'-(methylamino)spiro[3,5-dihydro-1,4-benzoxazepine-2,1'-cyclohexane]-4-yl]-3-pyrazol-1-ylpropan-1-one —— C22H30N4O2
(2S)-2-methyl-1-[4'-(methylamino)spiro[3,5-dihydro-1,4-benzoxazepine-2,1'-cyclohexane]-4-yl]-3-pyrazol-1-ylpropan-1-one
—— 1-(3-Phenoxypropyl)-3,1-benzoxazine-2,4-dione —— C17H15NO4
1-(3-Phenoxypropyl)-3,1-benzoxazine-2,4-dione
—— (2R)-2-methyl-1-[4'-(methylamino)spiro[3,5-dihydro-1,4-benzoxazepine-2,1'-cyclohexane]-4-yl]-3-pyrazol-1-ylpropan-1-one —— C22H30N4O2
(2R)-2-methyl-1-[4'-(methylamino)spiro[3,5-dihydro-1,4-benzoxazepine-2,1'-cyclohexane]-4-yl]-3-pyrazol-1-ylpropan-1-one
—— 2-(7-chloro-5-oxospiro[3H-1,4-benzoxazepine-2,4'-oxane]-4-yl)-N-[(2S)-2-phenylpropyl]acetamide —— C24H27ClN2O4
2-(7-chloro-5-oxospiro[3H-1,4-benzoxazepine-2,4'-oxane]-4-yl)-N-[(2S)-2-phenylpropyl]acetamide
—— 4-[[5-(Pyrrolidine-1-carbonyl)furan-2-yl]methyl]-1,4-benzoxazin-3-one —— C18H18N2O4
4-[[5-(Pyrrolidine-1-carbonyl)furan-2-yl]methyl]-1,4-benzoxazin-3-one
—— 9-bromo-5'-methyl-2-(4-methylphenyl)spiro[1,10b-dihydropyrazolo[1,5-c][1,3]benzoxazine-5,3'-1H-indole]-2'-one —— C25H20BrN3O2
9-bromo-5'-methyl-2-(4-methylphenyl)spiro[1,10b-dihydropyrazolo[1,5-c][1,3]benzoxazine-5,3'-1H-indole]-2'-one
—— 1-[(2R)-7-methoxy-2-[(3S)-1-[(1-propan-2-ylpyrrol-2-yl)methyl]piperidin-3-yl]-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]ethanone —— C25H35N3O3
1-[(2R)-7-methoxy-2-[(3S)-1-[(1-propan-2-ylpyrrol-2-yl)methyl]piperidin-3-yl]-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]ethanone
—— (2S)-1'-[(3S)-3-imidazol-1-ylbutanoyl]spiro[3,4-dihydro-1,4-benzoxazepine-2,3'-piperidine]-5-one —— C20H24N4O3
(2S)-1'-[(3S)-3-imidazol-1-ylbutanoyl]spiro[3,4-dihydro-1,4-benzoxazepine-2,3'-piperidine]-5-one
—— (2R)-1'-[(3S)-3-imidazol-1-ylbutanoyl]spiro[3,4-dihydro-1,4-benzoxazepine-2,3'-piperidine]-5-one —— C20H24N4O3
(2R)-1'-[(3S)-3-imidazol-1-ylbutanoyl]spiro[3,4-dihydro-1,4-benzoxazepine-2,3'-piperidine]-5-one
—— (2R)-1'-[(3R)-3-imidazol-1-ylbutanoyl]spiro[3,4-dihydro-1,4-benzoxazepine-2,3'-piperidine]-5-one —— C20H24N4O3
(2R)-1'-[(3R)-3-imidazol-1-ylbutanoyl]spiro[3,4-dihydro-1,4-benzoxazepine-2,3'-piperidine]-5-one
—— 2-(5-oxospiro[3H-1,4-benzoxazepine-2,4'-oxane]-4-yl)-N-(2-propan-2-ylpyrazol-3-yl)acetamide —— C21H26N4O4
2-(5-oxospiro[3H-1,4-benzoxazepine-2,4'-oxane]-4-yl)-N-(2-propan-2-ylpyrazol-3-yl)acetamide
—— 2-(1'-methyl-5-oxospiro[3H-1,4-benzoxazepine-2,4'-piperidine]-4-yl)-N-(2-propan-2-ylpyrazol-3-yl)acetamide —— C22H29N5O3
2-(1'-methyl-5-oxospiro[3H-1,4-benzoxazepine-2,4'-piperidine]-4-yl)-N-(2-propan-2-ylpyrazol-3-yl)acetamide
—— (2S)-1'-[3-(2-propan-2-ylimidazol-1-yl)propanoyl]spiro[3,4-dihydro-1,4-benzoxazepine-2,3'-piperidine]-5-one —— C22H28N4O3
(2S)-1'-[3-(2-propan-2-ylimidazol-1-yl)propanoyl]spiro[3,4-dihydro-1,4-benzoxazepine-2,3'-piperidine]-5-one
—— 1-[(2R)-7-methoxy-2-[(3R)-1-[(1-propan-2-ylpyrrol-2-yl)methyl]piperidin-3-yl]-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]ethanone —— C25H35N3O3
1-[(2R)-7-methoxy-2-[(3R)-1-[(1-propan-2-ylpyrrol-2-yl)methyl]piperidin-3-yl]-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]ethanone
—— N-(4-acetylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-cyclohexane]-1'-yl)-N-methyl-1-propan-2-ylpyrazole-4-carboxamide —— C24H32N4O3
N-(4-acetylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-cyclohexane]-1'-yl)-N-methyl-1-propan-2-ylpyrazole-4-carboxamide
—— N-methyl-1-propan-2-yl-N-spiro[4,5-dihydro-3H-1,4-benzoxazepine-2,4'-cyclohexane]-1'-ylpyrazole-4-carboxamide —— C22H30N4O2
N-methyl-1-propan-2-yl-N-spiro[4,5-dihydro-3H-1,4-benzoxazepine-2,4'-cyclohexane]-1'-ylpyrazole-4-carboxamide
—— (2R)-1'-[3-(2-propan-2-ylimidazol-1-yl)propanoyl]spiro[3,4-dihydro-1,4-benzoxazepine-2,3'-piperidine]-5-one —— C22H28N4O3
(2R)-1'-[3-(2-propan-2-ylimidazol-1-yl)propanoyl]spiro[3,4-dihydro-1,4-benzoxazepine-2,3'-piperidine]-5-one
—— N-methyl-N-[(2-propan-2-ylpyrimidin-5-yl)methyl]spiro[4,5-dihydro-3H-1,4-benzoxazepine-2,4'-cyclohexane]-1'-amine —— C23H32N4O
N-methyl-N-[(2-propan-2-ylpyrimidin-5-yl)methyl]spiro[4,5-dihydro-3H-1,4-benzoxazepine-2,4'-cyclohexane]-1'-amine
—— N-methyl-4-[(2-propan-2-ylpyrimidin-5-yl)methyl]spiro[3,5-dihydro-1,4-benzoxazepine-2,4'-cyclohexane]-1'-amine —— C23H32N4O
N-methyl-4-[(2-propan-2-ylpyrimidin-5-yl)methyl]spiro[3,5-dihydro-1,4-benzoxazepine-2,4'-cyclohexane]-1'-amine
—— N,4-dimethyl-N-[(2-propan-2-ylpyrimidin-5-yl)methyl]spiro[3,5-dihydro-1,4-benzoxazepine-2,4'-cyclohexane]-1'-amine —— C24H34N4O
N,4-dimethyl-N-[(2-propan-2-ylpyrimidin-5-yl)methyl]spiro[3,5-dihydro-1,4-benzoxazepine-2,4'-cyclohexane]-1'-amine
—— N,N-dimethyl-4-[(2-propan-2-ylpyrimidin-5-yl)methyl]spiro[3,5-dihydro-1,4-benzoxazepine-2,4'-cyclohexane]-1'-amine —— C24H34N4O
N,N-dimethyl-4-[(2-propan-2-ylpyrimidin-5-yl)methyl]spiro[3,5-dihydro-1,4-benzoxazepine-2,4'-cyclohexane]-1'-amine
—— 5-(4-fluorophenyl)-7-methoxy-2-(4-methylsulfanylphenyl)-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine —— C24H21FN2O2S
5-(4-fluorophenyl)-7-methoxy-2-(4-methylsulfanylphenyl)-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine
—— N-methyl-N-[4-[(2-propan-2-ylpyrimidin-5-yl)methyl]spiro[3,5-dihydro-1,4-benzoxazepine-2,4'-cyclohexane]-1'-yl]acetamide —— C25H34N4O2
N-methyl-N-[4-[(2-propan-2-ylpyrimidin-5-yl)methyl]spiro[3,5-dihydro-1,4-benzoxazepine-2,4'-cyclohexane]-1'-yl]acetamide
—— N-methyl-3-propan-2-yl-N-spiro[4,5-dihydro-3H-1,4-benzoxazepine-2,4'-cyclohexane]-1'-yl-1,2-oxazole-5-carboxamide —— C22H29N3O3
N-methyl-3-propan-2-yl-N-spiro[4,5-dihydro-3H-1,4-benzoxazepine-2,4'-cyclohexane]-1'-yl-1,2-oxazole-5-carboxamide
—— (2R)-1'-(5-propan-2-yl-1H-pyrazole-3-carbonyl)spiro[3,4-dihydro-1,4-benzoxazepine-2,3'-piperidine]-5-one —— C20H24N4O3
(2R)-1'-(5-propan-2-yl-1H-pyrazole-3-carbonyl)spiro[3,4-dihydro-1,4-benzoxazepine-2,3'-piperidine]-5-one
—— [4'-(methylamino)spiro[3,5-dihydro-1,4-benzoxazepine-2,1'-cyclohexane]-4-yl]-(5-propan-2-yl-1H-pyrazol-3-yl)methanone —— C22H30N4O2
[4'-(methylamino)spiro[3,5-dihydro-1,4-benzoxazepine-2,1'-cyclohexane]-4-yl]-(5-propan-2-yl-1H-pyrazol-3-yl)methanone
—— [4'-(Methylamino)spiro[3,5-dihydro-1,4-benzoxazepine-2,1'-cyclohexane]-4-yl]-(5-propan-2-ylthiophen-3-yl)methanone —— C23H30N2O2S
[4'-(Methylamino)spiro[3,5-dihydro-1,4-benzoxazepine-2,1'-cyclohexane]-4-yl]-(5-propan-2-ylthiophen-3-yl)methanone
—— N-methyl-5-propan-2-yl-N-spiro[4,5-dihydro-3H-1,4-benzoxazepine-2,4'-cyclohexane]-1'-ylthiophene-3-carboxamide —— C23H30N2O2S
N-methyl-5-propan-2-yl-N-spiro[4,5-dihydro-3H-1,4-benzoxazepine-2,4'-cyclohexane]-1'-ylthiophene-3-carboxamide
—— N-methyl-N-[4-(5-propan-2-ylthiophene-3-carbonyl)spiro[3,5-dihydro-1,4-benzoxazepine-2,4'-cyclohexane]-1'-yl]acetamide —— C25H32N2O3S
N-methyl-N-[4-(5-propan-2-ylthiophene-3-carbonyl)spiro[3,5-dihydro-1,4-benzoxazepine-2,4'-cyclohexane]-1'-yl]acetamide
—— N-methyl-N-[4-(5-propan-2-yl-1H-pyrazole-3-carbonyl)spiro[3,5-dihydro-1,4-benzoxazepine-2,4'-cyclohexane]-1'-yl]acetamide —— C24H32N4O3
N-methyl-N-[4-(5-propan-2-yl-1H-pyrazole-3-carbonyl)spiro[3,5-dihydro-1,4-benzoxazepine-2,4'-cyclohexane]-1'-yl]acetamide
—— N-(4-acetylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-cyclohexane]-1'-yl)-N-methyl-5-propan-2-yl-1H-pyrazole-3-carboxamide —— C24H32N4O3
N-(4-acetylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-cyclohexane]-1'-yl)-N-methyl-5-propan-2-yl-1H-pyrazole-3-carboxamide
—— N-methyl-N-(4-methylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-cyclohexane]-1'-yl)-5-propan-2-yl-1H-pyrazole-3-carboxamide —— C23H32N4O2
N-methyl-N-(4-methylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-cyclohexane]-1'-yl)-5-propan-2-yl-1H-pyrazole-3-carboxamide
—— N-methyl-5-propan-2-yl-N-spiro[4,5-dihydro-3H-1,4-benzoxazepine-2,4'-cyclohexane]-1'-yl-1H-pyrazole-3-carboxamide —— C22H30N4O2
N-methyl-5-propan-2-yl-N-spiro[4,5-dihydro-3H-1,4-benzoxazepine-2,4'-cyclohexane]-1'-yl-1H-pyrazole-3-carboxamide