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苯并恶嗪类

中文名称 英文名称 CAS号 化学式 结构式图片
—— (2R)-1-[4'-(dimethylamino)spiro[3,5-dihydro-1,4-benzoxazepine-2,1'-cyclohexane]-4-yl]-2-piperidin-1-ylpropan-1-one —— C24H37N3O2
(2R)-1-[4'-(dimethylamino)spiro[3,5-dihydro-1,4-benzoxazepine-2,1'-cyclohexane]-4-yl]-2-piperidin-1-ylpropan-1-one
—— (2S)-1'-[(2S)-2-(4-chloropyrazol-1-yl)propanoyl]spiro[3,4-dihydro-1,4-benzoxazepine-2,3'-piperidine]-5-one —— C19H21ClN4O3
(2S)-1'-[(2S)-2-(4-chloropyrazol-1-yl)propanoyl]spiro[3,4-dihydro-1,4-benzoxazepine-2,3'-piperidine]-5-one
—— (2R)-2-(5-oxospiro[3H-1,4-benzoxazepine-2,4'-oxane]-4-yl)propanoic acid —— C16H19NO5
(2R)-2-(5-oxospiro[3H-1,4-benzoxazepine-2,4'-oxane]-4-yl)propanoic acid
—— (2R)-N-methyl-2-(2-oxopyrrolidin-1-yl)-N-spiro[4,5-dihydro-3H-1,4-benzoxazepine-2,4'-cyclohexane]-1'-ylpropanamide —— C22H31N3O3
(2R)-N-methyl-2-(2-oxopyrrolidin-1-yl)-N-spiro[4,5-dihydro-3H-1,4-benzoxazepine-2,4'-cyclohexane]-1'-ylpropanamide
—— 6-chloro-3-(3,4-dimethylphenyl)-2H-1,3-benzoxazine-2,4(3H)-dione —— C16H12ClNO3
6-chloro-3-(3,4-dimethylphenyl)-2H-1,3-benzoxazine-2,4(3H)-dione
—— (2S)-N-methyl-2-(2-oxopyrrolidin-1-yl)-N-spiro[4,5-dihydro-3H-1,4-benzoxazepine-2,4'-cyclohexane]-1'-ylpropanamide —— C22H31N3O3
(2S)-N-methyl-2-(2-oxopyrrolidin-1-yl)-N-spiro[4,5-dihydro-3H-1,4-benzoxazepine-2,4'-cyclohexane]-1'-ylpropanamide
—— N-[4-(8-methoxy-5-oxospiro[3,4-dihydro-1,4-benzoxazepine-2,4'-piperidine]-1'-carbonyl)-1,3-thiazol-2-yl]acetamide —— C20H22N4O5S
N-[4-(8-methoxy-5-oxospiro[3,4-dihydro-1,4-benzoxazepine-2,4'-piperidine]-1'-carbonyl)-1,3-thiazol-2-yl]acetamide
—— 6-chloro-3-(5-chloro-2-methylphenyl)-2H-1,3-benzoxazine-2,4(3H)-dione —— C15H9Cl2NO3
6-chloro-3-(5-chloro-2-methylphenyl)-2H-1,3-benzoxazine-2,4(3H)-dione
—— N-[4-[(2S)-4-acetylspiro[3,5-dihydro-1,4-benzoxazepine-2,3'-piperidine]-1'-carbonyl]-1,3-thiazol-2-yl]acetamide —— C21H24N4O4S
N-[4-[(2S)-4-acetylspiro[3,5-dihydro-1,4-benzoxazepine-2,3'-piperidine]-1'-carbonyl]-1,3-thiazol-2-yl]acetamide
—— 6-[2-(2,6-dimethylphenyl)imino-3-(1-methoxypropan-2-yl)-1,3-thiazol-4-yl]-4H-1,4-benzoxazin-3-one —— C23H25N3O3S
6-[2-(2,6-dimethylphenyl)imino-3-(1-methoxypropan-2-yl)-1,3-thiazol-4-yl]-4H-1,4-benzoxazin-3-one
—— N-[4-[[4'-[acetyl(methyl)amino]spiro[3,5-dihydro-1,4-benzoxazepine-2,1'-cyclohexane]-4-yl]methyl]phenyl]acetamide —— C26H33N3O3
N-[4-[[4'-[acetyl(methyl)amino]spiro[3,5-dihydro-1,4-benzoxazepine-2,1'-cyclohexane]-4-yl]methyl]phenyl]acetamide
—— N-(5-oxospiro[3,4-dihydro-1,4-benzoxazepine-2,4'-cyclohexane]-1'-yl)acetamide —— C16H20N2O3
N-(5-oxospiro[3,4-dihydro-1,4-benzoxazepine-2,4'-cyclohexane]-1'-yl)acetamide
—— 5-(4-Chloro-3-fluorophenyl)-2-(3,4-dimethoxyphenyl)-1,10b-dihydropyrazolo[1,5-c][1,3]benzoxazine —— C24H20ClFN2O3
5-(4-Chloro-3-fluorophenyl)-2-(3,4-dimethoxyphenyl)-1,10b-dihydropyrazolo[1,5-c][1,3]benzoxazine
—— [2-oxo-2-(3-oxo-4H-1,4-benzoxazin-6-yl)ethyl] 2,4-dichloro-5-morpholin-4-ylsulfonylbenzoate —— C21H18Cl2N2O8S
[2-oxo-2-(3-oxo-4H-1,4-benzoxazin-6-yl)ethyl] 2,4-dichloro-5-morpholin-4-ylsulfonylbenzoate
—— N-(4-acetylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-cyclohexane]-1'-yl)-5-(furan-2-yl)-N-methyl-1,2-oxazole-3-carboxamide —— C25H27N3O5
N-(4-acetylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-cyclohexane]-1'-yl)-5-(furan-2-yl)-N-methyl-1,2-oxazole-3-carboxamide
—— N-(4-acetylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-cyclohexane]-1'-yl)-N-methyl-1,2-oxazole-5-carboxamide —— C21H25N3O4
N-(4-acetylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-cyclohexane]-1'-yl)-N-methyl-1,2-oxazole-5-carboxamide
—— 1-[4'-[(4-Hydroxyphenyl)methyl-methylamino]spiro[3,5-dihydro-1,4-benzoxazepine-2,1'-cyclohexane]-4-yl]ethanone —— C24H30N2O3
1-[4'-[(4-Hydroxyphenyl)methyl-methylamino]spiro[3,5-dihydro-1,4-benzoxazepine-2,1'-cyclohexane]-4-yl]ethanone
—— N-(4-acetylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-cyclohexane]-1'-yl)-N-methyl-2-phenylacetamide —— C25H30N2O3
N-(4-acetylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-cyclohexane]-1'-yl)-N-methyl-2-phenylacetamide
—— 1-[4'-[Dimethylsulfamoyl(methyl)amino]spiro[3,5-dihydro-1,4-benzoxazepine-2,1'-cyclohexane]-4-yl]ethanone —— C19H29N3O4S
1-[4'-[Dimethylsulfamoyl(methyl)amino]spiro[3,5-dihydro-1,4-benzoxazepine-2,1'-cyclohexane]-4-yl]ethanone
—— N-(4-acetylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-cyclohexane]-1'-yl)-2-methoxy-N-methylacetamide —— C20H28N2O4
N-(4-acetylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-cyclohexane]-1'-yl)-2-methoxy-N-methylacetamide
—— 1-[4'-[Cyclohexen-1-ylmethyl(methyl)amino]spiro[3,5-dihydro-1,4-benzoxazepine-2,1'-cyclohexane]-4-yl]ethanone —— C24H34N2O2
1-[4'-[Cyclohexen-1-ylmethyl(methyl)amino]spiro[3,5-dihydro-1,4-benzoxazepine-2,1'-cyclohexane]-4-yl]ethanone
—— N-(4-acetylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-cyclohexane]-1'-yl)-4-methoxy-N-methylbenzamide —— C25H30N2O4
N-(4-acetylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-cyclohexane]-1'-yl)-4-methoxy-N-methylbenzamide
—— 1-[4'-[Methyl(pyridin-4-ylmethyl)amino]spiro[3,5-dihydro-1,4-benzoxazepine-2,1'-cyclohexane]-4-yl]ethanone —— C23H29N3O2
1-[4'-[Methyl(pyridin-4-ylmethyl)amino]spiro[3,5-dihydro-1,4-benzoxazepine-2,1'-cyclohexane]-4-yl]ethanone
—— N-(4-acetylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-cyclohexane]-1'-yl)-N-methyl-1-benzofuran-2-carboxamide —— C26H28N2O4
N-(4-acetylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-cyclohexane]-1'-yl)-N-methyl-1-benzofuran-2-carboxamide
—— 1-[4'-[Methyl(thiophen-2-ylmethyl)amino]spiro[3,5-dihydro-1,4-benzoxazepine-2,1'-cyclohexane]-4-yl]ethanone —— C22H28N2O2S
1-[4'-[Methyl(thiophen-2-ylmethyl)amino]spiro[3,5-dihydro-1,4-benzoxazepine-2,1'-cyclohexane]-4-yl]ethanone
—— N-(4-acetylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-cyclohexane]-1'-yl)-N,1-dimethylpyrazole-4-carboxamide —— C22H28N4O3
N-(4-acetylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-cyclohexane]-1'-yl)-N,1-dimethylpyrazole-4-carboxamide
—— N-(4-acetylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-cyclohexane]-1'-yl)-2-cyclopentyl-N-methylacetamide —— C24H34N2O3
N-(4-acetylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-cyclohexane]-1'-yl)-2-cyclopentyl-N-methylacetamide
—— N-(4-acetylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-cyclohexane]-1'-yl)-5-tert-butyl-N-methyl-1H-pyrazole-3-carboxamide —— C25H34N4O3
N-(4-acetylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-cyclohexane]-1'-yl)-5-tert-butyl-N-methyl-1H-pyrazole-3-carboxamide
—— N-(4-acetylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-cyclohexane]-1'-yl)-N-methylpyridine-4-carboxamide —— C23H27N3O3
N-(4-acetylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-cyclohexane]-1'-yl)-N-methylpyridine-4-carboxamide
—— 1-[(2R)-2-[(3R)-1-[[(1R)-cyclohex-3-en-1-yl]methyl]piperidin-3-yl]-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]ethanone —— C23H32N2O2
1-[(2R)-2-[(3R)-1-[[(1R)-cyclohex-3-en-1-yl]methyl]piperidin-3-yl]-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]ethanone
—— N-(4-acetylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-cyclohexane]-1'-yl)-2-(4-amino-1,2,5-oxadiazol-3-yl)-N-methylacetamide —— C21H27N5O4
N-(4-acetylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-cyclohexane]-1'-yl)-2-(4-amino-1,2,5-oxadiazol-3-yl)-N-methylacetamide
—— (2R)-N-(4-acetylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-cyclohexane]-1'-yl)-N-methyloxolane-2-carboxamide —— C22H30N2O4
(2R)-N-(4-acetylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-cyclohexane]-1'-yl)-N-methyloxolane-2-carboxamide
—— 1-{4,5-dihydro-3H-spiro[1,4-benzoxazepine-2,4'-piperidin]-4-yl}ethan-1-one —— C15H20N2O2
1-{4,5-dihydro-3H-spiro[1,4-benzoxazepine-2,4'-piperidin]-4-yl}ethan-1-one
—— 1-[(2S)-2-[(3R)-1-[[(1R)-cyclohex-3-en-1-yl]methyl]piperidin-3-yl]-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]ethanone —— C23H32N2O2
1-[(2S)-2-[(3R)-1-[[(1R)-cyclohex-3-en-1-yl]methyl]piperidin-3-yl]-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]ethanone
—— 1-[4'-[(2-Chlorophenyl)methyl-methylamino]spiro[3,5-dihydro-1,4-benzoxazepine-2,1'-cyclohexane]-4-yl]ethanone —— C24H29ClN2O2
1-[4'-[(2-Chlorophenyl)methyl-methylamino]spiro[3,5-dihydro-1,4-benzoxazepine-2,1'-cyclohexane]-4-yl]ethanone
—— 1-[4'-[2,3-Dihydro-1,4-benzodioxin-6-ylmethyl(methyl)amino]spiro[3,5-dihydro-1,4-benzoxazepine-2,1'-cyclohexane]-4-yl]ethanone —— C26H32N2O4
1-[4'-[2,3-Dihydro-1,4-benzodioxin-6-ylmethyl(methyl)amino]spiro[3,5-dihydro-1,4-benzoxazepine-2,1'-cyclohexane]-4-yl]ethanone
—— N-(4-acetylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-cyclohexane]-1'-yl)-N-methylacetamide —— C19H26N2O3
N-(4-acetylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-cyclohexane]-1'-yl)-N-methylacetamide
—— 1-[(2R)-2-[(3S)-1-[[2-(dimethylamino)pyrimidin-5-yl]methyl]piperidin-3-yl]-7-methoxy-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]ethanone —— C24H33N5O3
1-[(2R)-2-[(3S)-1-[[2-(dimethylamino)pyrimidin-5-yl]methyl]piperidin-3-yl]-7-methoxy-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]ethanone
—— N-(4-acetylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-cyclohexane]-1'-yl)-N-methylfuran-3-carboxamide —— C22H26N2O4
N-(4-acetylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-cyclohexane]-1'-yl)-N-methylfuran-3-carboxamide
—— N-(4-acetylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-cyclohexane]-1'-yl)-3,4-dimethoxy-N-methylfuran-2-carboxamide —— C24H30N2O6
N-(4-acetylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-cyclohexane]-1'-yl)-3,4-dimethoxy-N-methylfuran-2-carboxamide
—— N-(4-acetylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-cyclohexane]-1'-yl)-1-(difluoromethyl)-N-methylpyrazole-3-carboxamide —— C22H26F2N4O3
N-(4-acetylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-cyclohexane]-1'-yl)-1-(difluoromethyl)-N-methylpyrazole-3-carboxamide
—— 1-[4'-[(3-Fluorophenyl)methyl-methylamino]spiro[3,5-dihydro-1,4-benzoxazepine-2,1'-cyclohexane]-4-yl]ethanone —— C24H29FN2O2
1-[4'-[(3-Fluorophenyl)methyl-methylamino]spiro[3,5-dihydro-1,4-benzoxazepine-2,1'-cyclohexane]-4-yl]ethanone
—— N-(4-acetylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-cyclohexane]-1'-yl)-N-methylpyridine-3-carboxamide —— C23H27N3O3
N-(4-acetylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-cyclohexane]-1'-yl)-N-methylpyridine-3-carboxamide
—— (2S)-N-(4-acetylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-cyclohexane]-1'-yl)-N-methyloxolane-2-carboxamide —— C22H30N2O4
(2S)-N-(4-acetylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-cyclohexane]-1'-yl)-N-methyloxolane-2-carboxamide
—— 1-[(2R)-2-[(3S)-1-(pyridin-2-ylmethyl)piperidin-3-yl]-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]ethanone —— C22H27N3O2
1-[(2R)-2-[(3S)-1-(pyridin-2-ylmethyl)piperidin-3-yl]-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]ethanone
—— 1-(4'-Morpholin-4-ylspiro[3,5-dihydro-1,4-benzoxazepine-2,1'-cyclohexane]-4-yl)ethanone —— C20H28N2O3
1-(4'-Morpholin-4-ylspiro[3,5-dihydro-1,4-benzoxazepine-2,1'-cyclohexane]-4-yl)ethanone
—— 1-[4'-[Cyclohexylmethyl(methyl)amino]spiro[3,5-dihydro-1,4-benzoxazepine-2,1'-cyclohexane]-4-yl]ethanone —— C24H36N2O2
1-[4'-[Cyclohexylmethyl(methyl)amino]spiro[3,5-dihydro-1,4-benzoxazepine-2,1'-cyclohexane]-4-yl]ethanone
—— N-(4-acetylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-cyclohexane]-1'-yl)-2-(difluoromethyl)-N-methylpyrazole-3-carboxamide —— C22H26F2N4O3
N-(4-acetylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-cyclohexane]-1'-yl)-2-(difluoromethyl)-N-methylpyrazole-3-carboxamide
—— 1-[4'-[(2-Fluorophenyl)methyl-methylamino]spiro[3,5-dihydro-1,4-benzoxazepine-2,1'-cyclohexane]-4-yl]ethanone —— C24H29FN2O2
1-[4'-[(2-Fluorophenyl)methyl-methylamino]spiro[3,5-dihydro-1,4-benzoxazepine-2,1'-cyclohexane]-4-yl]ethanone
—— N-(4-acetylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-cyclohexane]-1'-yl)-2-[(1R)-cyclopent-2-en-1-yl]-N-methylacetamide —— C24H32N2O3
N-(4-acetylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-cyclohexane]-1'-yl)-2-[(1R)-cyclopent-2-en-1-yl]-N-methylacetamide