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苯并恶嗪类

中文名称 英文名称 CAS号 化学式 结构式图片
—— 4-methyl-5-oxo-N-[(2S)-2-(1,2,4-triazol-1-yl)propyl]spiro[3H-1,4-benzoxazepine-2,4'-cyclohexane]-1'-carboxamide —— C21H27N5O3
4-methyl-5-oxo-N-[(2S)-2-(1,2,4-triazol-1-yl)propyl]spiro[3H-1,4-benzoxazepine-2,4'-cyclohexane]-1'-carboxamide
—— 4-[(2S)-1-(4-hydroxypiperidin-1-yl)-1-oxopropan-2-yl]spiro[3H-1,4-benzoxazepine-2,4'-oxane]-5-one —— C21H28N2O5
4-[(2S)-1-(4-hydroxypiperidin-1-yl)-1-oxopropan-2-yl]spiro[3H-1,4-benzoxazepine-2,4'-oxane]-5-one
—— (2S)-1'-[3-(3-chloro-1,2-oxazol-5-yl)propanoyl]spiro[3,4-dihydro-1,4-benzoxazepine-2,3'-piperidine]-5-one —— C19H20ClN3O4
(2S)-1'-[3-(3-chloro-1,2-oxazol-5-yl)propanoyl]spiro[3,4-dihydro-1,4-benzoxazepine-2,3'-piperidine]-5-one
—— 2-(5-oxospiro[3H-1,4-benzoxazepine-2,4'-oxane]-4-yl)-N-[(2R)-2-(1,2,4-triazol-1-yl)propyl]acetamide —— C20H25N5O4
2-(5-oxospiro[3H-1,4-benzoxazepine-2,4'-oxane]-4-yl)-N-[(2R)-2-(1,2,4-triazol-1-yl)propyl]acetamide
—— (2R)-N-[5-(2-methoxyethyl)-1,3,4-thiadiazol-2-yl]-2-(5-oxospiro[3H-1,4-benzoxazepine-2,4'-oxane]-4-yl)propanamide —— C21H26N4O5S
(2R)-N-[5-(2-methoxyethyl)-1,3,4-thiadiazol-2-yl]-2-(5-oxospiro[3H-1,4-benzoxazepine-2,4'-oxane]-4-yl)propanamide
—— N-(2-methylpropyl)-2-(5-oxospiro[3H-1,4-benzoxazepine-2,4'-oxane]-4-yl)acetamide —— C19H26N2O4
N-(2-methylpropyl)-2-(5-oxospiro[3H-1,4-benzoxazepine-2,4'-oxane]-4-yl)acetamide
—— N-[(3R)-oxan-3-yl]-2-(5-oxospiro[3H-1,4-benzoxazepine-2,4'-oxane]-4-yl)acetamide —— C20H26N2O5
N-[(3R)-oxan-3-yl]-2-(5-oxospiro[3H-1,4-benzoxazepine-2,4'-oxane]-4-yl)acetamide
—— (2R)-1'-[3-(2-fluorophenyl)propanoyl]spiro[3,4-dihydro-1,4-benzoxazepine-2,3'-piperidine]-5-one —— C22H23FN2O3
(2R)-1'-[3-(2-fluorophenyl)propanoyl]spiro[3,4-dihydro-1,4-benzoxazepine-2,3'-piperidine]-5-one
—— 4-[(2R)-1-(4-hydroxypiperidin-1-yl)-1-oxopropan-2-yl]spiro[3H-1,4-benzoxazepine-2,4'-oxane]-5-one —— C21H28N2O5
4-[(2R)-1-(4-hydroxypiperidin-1-yl)-1-oxopropan-2-yl]spiro[3H-1,4-benzoxazepine-2,4'-oxane]-5-one
—— (2S)-1'-[(2R)-2-phenylpropanoyl]spiro[3,4-dihydro-1,4-benzoxazepine-2,3'-piperidine]-5-one —— C22H24N2O3
(2S)-1'-[(2R)-2-phenylpropanoyl]spiro[3,4-dihydro-1,4-benzoxazepine-2,3'-piperidine]-5-one
—— N-[[(2S)-oxolan-2-yl]methyl]-2-(5-oxospiro[3H-1,4-benzoxazepine-2,4'-oxane]-4-yl)acetamide —— C20H26N2O5
N-[[(2S)-oxolan-2-yl]methyl]-2-(5-oxospiro[3H-1,4-benzoxazepine-2,4'-oxane]-4-yl)acetamide
—— (2S)-8-methoxy-1'-(pyridin-2-ylmethyl)spiro[3,4-dihydro-1,4-benzoxazepine-2,3'-piperidine]-5-one —— C20H23N3O3
(2S)-8-methoxy-1'-(pyridin-2-ylmethyl)spiro[3,4-dihydro-1,4-benzoxazepine-2,3'-piperidine]-5-one
—— N-methyl-5-oxo-N-(pyridin-4-ylmethyl)spiro[3,4-dihydro-1,4-benzoxazepine-2,4'-cyclohexane]-1'-carboxamide —— C22H25N3O3
N-methyl-5-oxo-N-(pyridin-4-ylmethyl)spiro[3,4-dihydro-1,4-benzoxazepine-2,4'-cyclohexane]-1'-carboxamide
—— (2R)-1'-[(3R)-3-(3,5-dimethylpyrazol-1-yl)butanoyl]spiro[3,4-dihydro-1,4-benzoxazepine-2,3'-piperidine]-5-one —— C22H28N4O3
(2R)-1'-[(3R)-3-(3,5-dimethylpyrazol-1-yl)butanoyl]spiro[3,4-dihydro-1,4-benzoxazepine-2,3'-piperidine]-5-one
—— 4-methyl-N-[2-(5-methylpyrazol-1-yl)ethyl]-5-oxospiro[3H-1,4-benzoxazepine-2,4'-cyclohexane]-1'-carboxamide —— C22H28N4O3
4-methyl-N-[2-(5-methylpyrazol-1-yl)ethyl]-5-oxospiro[3H-1,4-benzoxazepine-2,4'-cyclohexane]-1'-carboxamide
—— (2R)-4-[2-(azepan-1-yl)-2-oxoethyl]-1'-methylspiro[3H-1,4-benzoxazepine-2,5'-azepane]-2',5-dione —— C23H31N3O4
(2R)-4-[2-(azepan-1-yl)-2-oxoethyl]-1'-methylspiro[3H-1,4-benzoxazepine-2,5'-azepane]-2',5-dione
—— (2R)-1'-[3-(tetrazol-1-yl)propanoyl]spiro[3,4-dihydro-1,4-benzoxazepine-2,3'-piperidine]-5-one —— C17H20N6O3
(2R)-1'-[3-(tetrazol-1-yl)propanoyl]spiro[3,4-dihydro-1,4-benzoxazepine-2,3'-piperidine]-5-one
—— (2R)-N-[[(2S)-1,4-dioxan-2-yl]methyl]-2-(5-oxospiro[3H-1,4-benzoxazepine-2,4'-oxane]-4-yl)propanamide —— C21H28N2O6
(2R)-N-[[(2S)-1,4-dioxan-2-yl]methyl]-2-(5-oxospiro[3H-1,4-benzoxazepine-2,4'-oxane]-4-yl)propanamide
—— 2-[(2R)-1'-methyl-2',5-dioxospiro[3H-1,4-benzoxazepine-2,5'-azepane]-4-yl]-N-[[(2R)-oxolan-2-yl]methyl]acetamide —— C22H29N3O5
2-[(2R)-1'-methyl-2',5-dioxospiro[3H-1,4-benzoxazepine-2,5'-azepane]-4-yl]-N-[[(2R)-oxolan-2-yl]methyl]acetamide
—— (2S)-1'-[3-(5-methyltetrazol-1-yl)propanoyl]spiro[3,4-dihydro-1,4-benzoxazepine-2,3'-piperidine]-5-one —— C18H22N6O3
(2S)-1'-[3-(5-methyltetrazol-1-yl)propanoyl]spiro[3,4-dihydro-1,4-benzoxazepine-2,3'-piperidine]-5-one
—— 1-(4-methyl-5-oxospiro[3H-1,4-benzoxazepine-2,4'-cyclohexane]-1'-carbonyl)piperidine-4-carboxamide —— C22H29N3O4
1-(4-methyl-5-oxospiro[3H-1,4-benzoxazepine-2,4'-cyclohexane]-1'-carbonyl)piperidine-4-carboxamide
—— (2S)-4-[2-(azepan-1-yl)-2-oxoethyl]-1'-methylspiro[3H-1,4-benzoxazepine-2,5'-azepane]-2',5-dione —— C23H31N3O4
(2S)-4-[2-(azepan-1-yl)-2-oxoethyl]-1'-methylspiro[3H-1,4-benzoxazepine-2,5'-azepane]-2',5-dione
—— (2R)-1'-[(2S)-2-phenylpropanoyl]spiro[3,4-dihydro-1,4-benzoxazepine-2,3'-piperidine]-5-one —— C22H24N2O3
(2R)-1'-[(2S)-2-phenylpropanoyl]spiro[3,4-dihydro-1,4-benzoxazepine-2,3'-piperidine]-5-one
—— (2R)-8-methoxy-1'-(6-oxo-4,5-dihydro-1H-pyridazine-3-carbonyl)spiro[3,4-dihydro-1,4-benzoxazepine-2,3'-piperidine]-5-one —— C19H22N4O5
(2R)-8-methoxy-1'-(6-oxo-4,5-dihydro-1H-pyridazine-3-carbonyl)spiro[3,4-dihydro-1,4-benzoxazepine-2,3'-piperidine]-5-one
—— (2R)-1'-[(3S)-3-(3,5-dimethylpyrazol-1-yl)butanoyl]spiro[3,4-dihydro-1,4-benzoxazepine-2,3'-piperidine]-5-one —— C22H28N4O3
(2R)-1'-[(3S)-3-(3,5-dimethylpyrazol-1-yl)butanoyl]spiro[3,4-dihydro-1,4-benzoxazepine-2,3'-piperidine]-5-one
—— (2R)-1'-[3-(3-chloro-1,2-oxazol-5-yl)propanoyl]spiro[3,4-dihydro-1,4-benzoxazepine-2,3'-piperidine]-5-one —— C19H20ClN3O4
(2R)-1'-[3-(3-chloro-1,2-oxazol-5-yl)propanoyl]spiro[3,4-dihydro-1,4-benzoxazepine-2,3'-piperidine]-5-one
—— (2S)-1'-[3-(tetrazol-1-yl)propanoyl]spiro[3,4-dihydro-1,4-benzoxazepine-2,3'-piperidine]-5-one —— C17H20N6O3
(2S)-1'-[3-(tetrazol-1-yl)propanoyl]spiro[3,4-dihydro-1,4-benzoxazepine-2,3'-piperidine]-5-one
—— N-methyl-2-(5-oxospiro[3H-1,4-benzoxazepine-2,4'-oxane]-4-yl)-N-[2-(1H-pyrazol-4-yl)ethyl]acetamide —— C21H26N4O4
N-methyl-2-(5-oxospiro[3H-1,4-benzoxazepine-2,4'-oxane]-4-yl)-N-[2-(1H-pyrazol-4-yl)ethyl]acetamide
—— (2S)-8-methoxy-1'-(pyridine-3-carbonyl)spiro[3,4-dihydro-1,4-benzoxazepine-2,3'-piperidine]-5-one —— C20H21N3O4
(2S)-8-methoxy-1'-(pyridine-3-carbonyl)spiro[3,4-dihydro-1,4-benzoxazepine-2,3'-piperidine]-5-one
—— (2R)-8-methoxy-1'-(pyridine-3-carbonyl)spiro[3,4-dihydro-1,4-benzoxazepine-2,3'-piperidine]-5-one —— C20H21N3O4
(2R)-8-methoxy-1'-(pyridine-3-carbonyl)spiro[3,4-dihydro-1,4-benzoxazepine-2,3'-piperidine]-5-one
—— 2-[(2S)-1'-methyl-2',5-dioxospiro[3H-1,4-benzoxazepine-2,5'-azepane]-4-yl]-N-propan-2-ylacetamide —— C20H27N3O4
2-[(2S)-1'-methyl-2',5-dioxospiro[3H-1,4-benzoxazepine-2,5'-azepane]-4-yl]-N-propan-2-ylacetamide
—— N-cyclopentyl-2-[(2S)-1'-methyl-2',5-dioxospiro[3H-1,4-benzoxazepine-2,5'-azepane]-4-yl]acetamide —— C22H29N3O4
N-cyclopentyl-2-[(2S)-1'-methyl-2',5-dioxospiro[3H-1,4-benzoxazepine-2,5'-azepane]-4-yl]acetamide
—— 2-[(2S)-1'-methyl-2',5-dioxospiro[3H-1,4-benzoxazepine-2,5'-azepane]-4-yl]-N-[[(2R)-oxolan-2-yl]methyl]acetamide —— C22H29N3O5
2-[(2S)-1'-methyl-2',5-dioxospiro[3H-1,4-benzoxazepine-2,5'-azepane]-4-yl]-N-[[(2R)-oxolan-2-yl]methyl]acetamide
—— (2R)-8-methoxy-1'-(2-phenylethyl)spiro[3,4-dihydro-1,4-benzoxazepine-2,3'-piperidine]-5-one —— C22H26N2O3
(2R)-8-methoxy-1'-(2-phenylethyl)spiro[3,4-dihydro-1,4-benzoxazepine-2,3'-piperidine]-5-one
—— Ethyl 1-(5-oxospiro[3,4-dihydro-1,4-benzoxazepine-2,4'-cyclohexane]-1'-carbonyl)piperidine-4-carboxylate —— C23H30N2O5
Ethyl 1-(5-oxospiro[3,4-dihydro-1,4-benzoxazepine-2,4'-cyclohexane]-1'-carbonyl)piperidine-4-carboxylate
—— (2S)-8-methoxy-1'-(6-oxo-4,5-dihydro-1H-pyridazine-3-carbonyl)spiro[3,4-dihydro-1,4-benzoxazepine-2,3'-piperidine]-5-one —— C19H22N4O5
(2S)-8-methoxy-1'-(6-oxo-4,5-dihydro-1H-pyridazine-3-carbonyl)spiro[3,4-dihydro-1,4-benzoxazepine-2,3'-piperidine]-5-one
—— (2S)-1'-(2-phenylethyl)spiro[3,4-dihydro-1,4-benzoxazepine-2,3'-piperidine]-5-one —— C21H24N2O2
(2S)-1'-(2-phenylethyl)spiro[3,4-dihydro-1,4-benzoxazepine-2,3'-piperidine]-5-one
—— (2S)-1'-[3-(2-fluorophenyl)propanoyl]spiro[3,4-dihydro-1,4-benzoxazepine-2,3'-piperidine]-5-one —— C22H23FN2O3
(2S)-1'-[3-(2-fluorophenyl)propanoyl]spiro[3,4-dihydro-1,4-benzoxazepine-2,3'-piperidine]-5-one
—— (2R)-1'-(2-phenylethyl)spiro[3,4-dihydro-1,4-benzoxazepine-2,3'-piperidine]-5-one —— C21H24N2O2
(2R)-1'-(2-phenylethyl)spiro[3,4-dihydro-1,4-benzoxazepine-2,3'-piperidine]-5-one
—— 5-oxo-N-(1,3,5-trimethylpyrazol-4-yl)spiro[3,4-dihydro-1,4-benzoxazepine-2,4'-cyclohexane]-1'-carboxamide —— C21H26N4O3
5-oxo-N-(1,3,5-trimethylpyrazol-4-yl)spiro[3,4-dihydro-1,4-benzoxazepine-2,4'-cyclohexane]-1'-carboxamide
—— (2S)-1'-(3-phenylpropanoyl)spiro[3,4-dihydro-1,4-benzoxazepine-2,3'-piperidine]-5-one —— C22H24N2O3
(2S)-1'-(3-phenylpropanoyl)spiro[3,4-dihydro-1,4-benzoxazepine-2,3'-piperidine]-5-one
—— N-[2-(4-fluorophenyl)ethyl]-5-oxospiro[3,4-dihydro-1,4-benzoxazepine-2,4'-cyclohexane]-1'-carboxamide —— C23H25FN2O3
N-[2-(4-fluorophenyl)ethyl]-5-oxospiro[3,4-dihydro-1,4-benzoxazepine-2,4'-cyclohexane]-1'-carboxamide
—— (2R)-1'-(1-ethyl-5-methylpyrazole-4-carbonyl)spiro[3,4-dihydro-1,4-benzoxazepine-2,3'-piperidine]-5-one —— C20H24N4O3
(2R)-1'-(1-ethyl-5-methylpyrazole-4-carbonyl)spiro[3,4-dihydro-1,4-benzoxazepine-2,3'-piperidine]-5-one
—— (2R)-1'-[(2R)-2-phenylpropanoyl]spiro[3,4-dihydro-1,4-benzoxazepine-2,3'-piperidine]-5-one —— C22H24N2O3
(2R)-1'-[(2R)-2-phenylpropanoyl]spiro[3,4-dihydro-1,4-benzoxazepine-2,3'-piperidine]-5-one
—— (2S)-8-methoxy-1'-(5-propan-2-yl-1H-pyrazole-3-carbonyl)spiro[3,4-dihydro-1,4-benzoxazepine-2,3'-piperidine]-5-one —— C21H26N4O4
(2S)-8-methoxy-1'-(5-propan-2-yl-1H-pyrazole-3-carbonyl)spiro[3,4-dihydro-1,4-benzoxazepine-2,3'-piperidine]-5-one
—— (2R)-1'-[2-(3,4,5-trimethylpyrazol-1-yl)acetyl]spiro[3,4-dihydro-1,4-benzoxazepine-2,3'-piperidine]-5-one —— C21H26N4O3
(2R)-1'-[2-(3,4,5-trimethylpyrazol-1-yl)acetyl]spiro[3,4-dihydro-1,4-benzoxazepine-2,3'-piperidine]-5-one
—— (2S)-4-[2-[(2S,6R)-2,6-dimethylmorpholin-4-yl]-2-oxoethyl]-1'-methylspiro[3H-1,4-benzoxazepine-2,5'-azepane]-2',5-dione —— C23H31N3O5
(2S)-4-[2-[(2S,6R)-2,6-dimethylmorpholin-4-yl]-2-oxoethyl]-1'-methylspiro[3H-1,4-benzoxazepine-2,5'-azepane]-2',5-dione
—— N-cyclohexyl-N-methyl-2-[(2R)-1'-methyl-2',5-dioxospiro[3H-1,4-benzoxazepine-2,5'-azepane]-4-yl]acetamide —— C24H33N3O4
N-cyclohexyl-N-methyl-2-[(2R)-1'-methyl-2',5-dioxospiro[3H-1,4-benzoxazepine-2,5'-azepane]-4-yl]acetamide
—— (2R)-1'-[2-(4-chloropyrazol-1-yl)acetyl]spiro[3,4-dihydro-1,4-benzoxazepine-2,3'-piperidine]-5-one —— C18H19ClN4O3
(2R)-1'-[2-(4-chloropyrazol-1-yl)acetyl]spiro[3,4-dihydro-1,4-benzoxazepine-2,3'-piperidine]-5-one
—— (2S)-1'-[2-(4-chloropyrazol-1-yl)acetyl]spiro[3,4-dihydro-1,4-benzoxazepine-2,3'-piperidine]-5-one —— C18H19ClN4O3
(2S)-1'-[2-(4-chloropyrazol-1-yl)acetyl]spiro[3,4-dihydro-1,4-benzoxazepine-2,3'-piperidine]-5-one