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中文名称 英文名称 CAS号 化学式 结构式图片
—— 2,2,2-Trifluoro-1-[4-[(4-imidazol-1-ylphenyl)methyl]piperazin-1-yl]ethanone 1043508-29-7 C16H17F3N4O
2,2,2-Trifluoro-1-[4-[(4-imidazol-1-ylphenyl)methyl]piperazin-1-yl]ethanone
—— N-{3-[1-ethyl-4-(1H-pyrrolo[2,3-b]pyridin-4-yl)-1H-pyrazol-3-yl]phenyl}-N'-{4-[(phenylmethyl)oxy]phenyl}urea 945865-02-1 C32H28N6O2
N-{3-[1-ethyl-4-(1H-pyrrolo[2,3-b]pyridin-4-yl)-1H-pyrazol-3-yl]phenyl}-N'-{4-[(phenylmethyl)oxy]phenyl}urea
—— 3-ethoxycarbonylpyrazolo[5,1-c]pyrido[4,3-e][1,2,4]triazine 5-oxide 1092790-46-9 C11H9N5O3
3-ethoxycarbonylpyrazolo[5,1-c]pyrido[4,3-e][1,2,4]triazine 5-oxide
—— N-{3-[4-(3-bromo-1H-pyrrolo[2,3-b]pyridin-4-yl)-1-ethyl-1H-pyrazol-3-yl]phenyl}-N'-phenylurea 945865-09-8 C25H21BrN6O
N-{3-[4-(3-bromo-1H-pyrrolo[2,3-b]pyridin-4-yl)-1-ethyl-1H-pyrazol-3-yl]phenyl}-N'-phenylurea
—— N-cyclohexyl-N'-{3-[1-ethyl-4-(1H-pyrrolo[2,3-b]pyridin-4-yl)-1H-pyrazol-3-yl]phenyl}urea 945865-03-2 C25H28N6O
N-cyclohexyl-N'-{3-[1-ethyl-4-(1H-pyrrolo[2,3-b]pyridin-4-yl)-1H-pyrazol-3-yl]phenyl}urea
—— N-(2,6-difluorophenyl)-N'-{3-[1-ethyl-4-(1H-pyrrolo[2,3-b]pyridin-4-yl)-1H-pyrazol-3-yl]phenyl}urea 945865-01-0 C25H20F2N6O
N-(2,6-difluorophenyl)-N'-{3-[1-ethyl-4-(1H-pyrrolo[2,3-b]pyridin-4-yl)-1H-pyrazol-3-yl]phenyl}urea
—— 3-(3-Benzyloxyphenyl)isothiazole-4-carboxylic acid 1062548-11-1 C17H13NO3S
3-(3-Benzyloxyphenyl)isothiazole-4-carboxylic acid
—— 2-(4-chlorophenyl)-5-isopropyl-6,7-dihydropyrazolo[1,5-a]pyrazin-4(5H)-one 1101861-29-3 C15H16ClN3O
2-(4-chlorophenyl)-5-isopropyl-6,7-dihydropyrazolo[1,5-a]pyrazin-4(5H)-one
—— (S)-N-(1-(5-(4-fluorophenyl)-1H-imidazol-2-yl)-7-oxooctyl)-1-methylpiperidine-4-carboxamide 1089661-04-0 C24H33FN4O2
(S)-N-(1-(5-(4-fluorophenyl)-1H-imidazol-2-yl)-7-oxooctyl)-1-methylpiperidine-4-carboxamide
—— 2-(4-chlorophenyl)-5-(3,4-dimethoxyphenethyl)-6,7-dihydropyrazolo[1,5-a]pyrazin-4(5H)-one 1101861-34-0 C22H22ClN3O3
2-(4-chlorophenyl)-5-(3,4-dimethoxyphenethyl)-6,7-dihydropyrazolo[1,5-a]pyrazin-4(5H)-one
—— (2Z)-2-{1-[2-chloro-4-(3-ethyl-1H-pyrazol-1-yl)benzoyl]-4,4-difluoro-1,2,3,4-tetrahydro-5H-1-benzazepin-5-ylidene}-N-(pyridin-2-ylmethyl)acetamide hydrochloride 530090-86-9 C30H26ClF2N5O2*ClH
(2Z)-2-{1-[2-chloro-4-(3-ethyl-1H-pyrazol-1-yl)benzoyl]-4,4-difluoro-1,2,3,4-tetrahydro-5H-1-benzazepin-5-ylidene}-N-(pyridin-2-ylmethyl)acetamide hydrochloride
—— (S)-N-(1-(5-(4-chlorophenyl)-1H-imidazol-2-yl)-7-oxooctyl)-1-methylpiperidine-4-carboxamide 1089661-02-8 C24H33ClN4O2
(S)-N-(1-(5-(4-chlorophenyl)-1H-imidazol-2-yl)-7-oxooctyl)-1-methylpiperidine-4-carboxamide
—— Spiro[1,2-benzisoxazole-5(4H),1a(2)-cyclopropane]-4-carboxylic acid, 6,7-dihydro-3-methyl- 1550937-09-1 C11H13NO3
Spiro[1,2-benzisoxazole-5(4H),1a(2)-cyclopropane]-4-carboxylic acid, 6,7-dihydro-3-methyl-
—— (S)-N-(1-(5-(3-chlorophenyl)-1H-imidazol-2-yl)-7-oxooctyl)-1-methylpiperidine-4-carboxamide 891259-78-2 C24H33ClN4O2
(S)-N-(1-(5-(3-chlorophenyl)-1H-imidazol-2-yl)-7-oxooctyl)-1-methylpiperidine-4-carboxamide
—— (2Z)-2-{1-[2-chloro-4-(5-methyl-1H-pyrazol-1-yl)benzoyl]-4,4-difluoro-1,2,3,4-tetrahydro-5H-1-benzazepin-5-ylidene}-N-(pyridin-2-ylmethyl)acetamide hydrochloride 530090-85-8 C29H24ClF2N5O2*ClH
(2Z)-2-{1-[2-chloro-4-(5-methyl-1H-pyrazol-1-yl)benzoyl]-4,4-difluoro-1,2,3,4-tetrahydro-5H-1-benzazepin-5-ylidene}-N-(pyridin-2-ylmethyl)acetamide hydrochloride
—— 5-butyl-2-(4-chlorophenyl)-6,7-dihydropyrazolo[1,5-a]pyrazin-4(5H)-one 1101861-30-6 C16H18ClN3O
5-butyl-2-(4-chlorophenyl)-6,7-dihydropyrazolo[1,5-a]pyrazin-4(5H)-one
—— Ethyl 5-(3,4-dihydroxyphenyl)-1,3-oxazole-4-carboxylate 1141892-73-0 C12H11NO5
Ethyl 5-(3,4-dihydroxyphenyl)-1,3-oxazole-4-carboxylate
—— 2-(4-chlorophenyl)-5-((6-chloropyridin-3-yl)methyl)-6,7-dihydropyrazolo[1,5-a]pyrazin-4(5H)-one 1101861-33-9 C18H14Cl2N4O
2-(4-chlorophenyl)-5-((6-chloropyridin-3-yl)methyl)-6,7-dihydropyrazolo[1,5-a]pyrazin-4(5H)-one
—— N-cyclopentyl-5-(3,4-dihydroxyphenyl)-1,3-oxazole-4-carboxamide 1141892-74-1 C15H16N2O4
N-cyclopentyl-5-(3,4-dihydroxyphenyl)-1,3-oxazole-4-carboxamide
—— (S)-1-methyl-N-(1-(4-methyl-5-phenyl-1H-imidazol-2-yl)-7-oxooctyl)piperidine-4-carboxamide 891259-72-6 C25H36N4O2
(S)-1-methyl-N-(1-(4-methyl-5-phenyl-1H-imidazol-2-yl)-7-oxooctyl)piperidine-4-carboxamide
—— ethyl (E)-3-[5-(3-fluorophenyl)-1H-tetrazol-1-yl]propenoate 1077626-99-3 C12H11FN4O2
ethyl (E)-3-[5-(3-fluorophenyl)-1H-tetrazol-1-yl]propenoate
—— (S)-N-(1-(5-(2-chlorophenyl)-1H-imidazol-2-yl)-7-oxooctyl)-1-methylpiperidine-4-carboxamide 1089661-03-9 C24H33ClN4O2
(S)-N-(1-(5-(2-chlorophenyl)-1H-imidazol-2-yl)-7-oxooctyl)-1-methylpiperidine-4-carboxamide
—— KMI-1293 1160850-87-2 C33H29IN8O5
KMI-1293
—— (S)-1-methyl-N-(7-oxo-1-(5-phenyl-1H-imidazol-2-yl)octyl)piperidine-4-carboxamide 891259-10-2 C24H34N4O2
(S)-1-methyl-N-(7-oxo-1-(5-phenyl-1H-imidazol-2-yl)octyl)piperidine-4-carboxamide
—— (2Z)-2-{1-[2-chloro-4-(3-isopropyl-1H-pyrazol-1-yl)benzoyl]-4,4-difluoro-1,2,3,4-tetrahydro-5H-1-benzazepin-5-ylidene}-N-(pyridin-2-ylmethyl)acetamide hydrochloride 530090-87-0 C31H28ClF2N5O2*ClH
(2Z)-2-{1-[2-chloro-4-(3-isopropyl-1H-pyrazol-1-yl)benzoyl]-4,4-difluoro-1,2,3,4-tetrahydro-5H-1-benzazepin-5-ylidene}-N-(pyridin-2-ylmethyl)acetamide hydrochloride
—— ethyl (Z)-3-[5-(3-iodophenyl)-1H-tetrazol-1-yl]propenoate 1077627-09-8 C12H11IN4O2
ethyl (Z)-3-[5-(3-iodophenyl)-1H-tetrazol-1-yl]propenoate
—— (S)-N-(1-(5-(3-cyanophenyl)-1H-imidazol-2-yl)-7-oxooctyl)-1-methylpiperidine-4-carboxamide 1089661-06-2 C25H33N5O2
(S)-N-(1-(5-(3-cyanophenyl)-1H-imidazol-2-yl)-7-oxooctyl)-1-methylpiperidine-4-carboxamide
—— N-but-3-enyl-5-(3,4-dihydroxyphenyl)-1,3-oxazole-4-carboxamide 1141892-75-2 C14H14N2O4
N-but-3-enyl-5-(3,4-dihydroxyphenyl)-1,3-oxazole-4-carboxamide
—— ethyl (Z)-3-[5-(3-fluorophenyl)-1H-tetrazol-1-yl]propenoate 1077627-07-6 C12H11FN4O2
ethyl (Z)-3-[5-(3-fluorophenyl)-1H-tetrazol-1-yl]propenoate
—— (S)-N-(1-(5-(4-cyanophenyl)-1H-imidazol-2-yl)-7-oxooctyl)-1-methylpiperidine-4-carboxamide 1089661-05-1 C25H33N5O2
(S)-N-(1-(5-(4-cyanophenyl)-1H-imidazol-2-yl)-7-oxooctyl)-1-methylpiperidine-4-carboxamide
—— (2Z)-2-{1-[2-chloro-4-(3,5-dimethyl-1H-pyrazol-1-yl)benzoyl]-4,4-difluoro-1,2,3,4-tetrahydro-5H-1-benzazepin-5-ylidene}-N-(pyridin-2-ylmethyl)acetamide hydrochloride 530090-89-2 C30H26ClF2N5O2*ClH
(2Z)-2-{1-[2-chloro-4-(3,5-dimethyl-1H-pyrazol-1-yl)benzoyl]-4,4-difluoro-1,2,3,4-tetrahydro-5H-1-benzazepin-5-ylidene}-N-(pyridin-2-ylmethyl)acetamide hydrochloride
—— ethyl (E)-3-[5-(3-iodophenyl)-1H-tetrazol-1-yl]propenoate 1077627-01-0 C12H11IN4O2
ethyl (E)-3-[5-(3-iodophenyl)-1H-tetrazol-1-yl]propenoate
—— (S)-4-cyano-N-(7-oxo-1-(5-phenyl-1H-imidazol-2-yl)octyl)benzenesulfonamide 891259-22-6 C24H26N4O3S
(S)-4-cyano-N-(7-oxo-1-(5-phenyl-1H-imidazol-2-yl)octyl)benzenesulfonamide
—— 6-Chloro-2-(4-fluorophenyl)-3-(pyridin-4-yl)pyrazolo[1,5-a]pyridine 1085712-27-1 C18H11ClFN3
6-Chloro-2-(4-fluorophenyl)-3-(pyridin-4-yl)pyrazolo[1,5-a]pyridine
—— (S)-N-(7-oxo-1-(5-phenyl-1H-imidazol-2-yl)octyl)thiazole-5-carboxamide 891259-14-6 C21H24N4O2S
(S)-N-(7-oxo-1-(5-phenyl-1H-imidazol-2-yl)octyl)thiazole-5-carboxamide
—— (S)-3-cyano-N-(7-oxo-1-(5-phenyl-1H-imidazol-2-yl)octyl)benzamide 891260-86-9 C25H26N4O2
(S)-3-cyano-N-(7-oxo-1-(5-phenyl-1H-imidazol-2-yl)octyl)benzamide
—— 5-methyl-2-p-tolyl-2H-pyrazolo[4,3-d]pyrimidin-7(6H)-one 1190305-79-3 C13H12N4O
5-methyl-2-p-tolyl-2H-pyrazolo[4,3-d]pyrimidin-7(6H)-one
—— (S)-2-Ethoxy-3-{4-[2-(5-methyl-2-phenyl-oxazol-4-yl)-ethoxy]-benzo[b]thiophen-7-yl}-propionic acid 475479-35-7 C25H25NO5S
(S)-2-Ethoxy-3-{4-[2-(5-methyl-2-phenyl-oxazol-4-yl)-ethoxy]-benzo[b]thiophen-7-yl}-propionic acid
—— 4-(5-(5-Tert-butyl-1,2,4-oxadiazol-3-yl)-2-methylphenylsulfonyl)morpholine 1123297-09-5 C17H23N3O4S
4-(5-(5-Tert-butyl-1,2,4-oxadiazol-3-yl)-2-methylphenylsulfonyl)morpholine
—— KMI-1283 1160850-88-3 C33H28ClFN8O5
KMI-1283
—— (S)-3-(4-(2-(5-methyl-2-phenyloxazol-4-yl)ethoxy)benzo[b]thiophen-7-yl)-2-propoxypropanoic acid 1160810-86-5 C26H27NO5S
(S)-3-(4-(2-(5-methyl-2-phenyloxazol-4-yl)ethoxy)benzo[b]thiophen-7-yl)-2-propoxypropanoic acid
—— 4-(5-(5-tert-butyl-1H-pyrazol-3-yl)-2-methylphenylsulfonyl)morpholine 1123297-12-0 C18H25N3O3S
4-(5-(5-tert-butyl-1H-pyrazol-3-yl)-2-methylphenylsulfonyl)morpholine
—— (S)-2-Ethoxy-3-(4-{2-[5-methyl-2-(4-trifluoromethyl-phenyl)-oxazol-4-yl]-ethoxy}-benzo[b]thiophen-7-yl)-propionic acid 475479-47-1 C26H24F3NO5S
(S)-2-Ethoxy-3-(4-{2-[5-methyl-2-(4-trifluoromethyl-phenyl)-oxazol-4-yl]-ethoxy}-benzo[b]thiophen-7-yl)-propionic acid
—— 4-(2-methyl-5-(2H-tetrazol-5-yl)phenylsulfonyl)morpholine 1123296-99-0 C12H15N5O3S
4-(2-methyl-5-(2H-tetrazol-5-yl)phenylsulfonyl)morpholine
—— 4-(3-(4-chlorophenyl)-1H-pyrazol-4-yl)-N-cyclopentylpyrimidin-2-amine 1158908-30-5 C18H18ClN5
4-(3-(4-chlorophenyl)-1H-pyrazol-4-yl)-N-cyclopentylpyrimidin-2-amine
—— 4-(2-Methyl-5-(5-neopentyl-1,2,4-oxadiazol-3-yl)phenylsulfonyl)morpholine 1123297-06-2 C18H25N3O4S
4-(2-Methyl-5-(5-neopentyl-1,2,4-oxadiazol-3-yl)phenylsulfonyl)morpholine
—— 4-(5-(2-(cyclohexylmethyl)-2H-tetrazol-5-yl)-2-methylphenylsulfonyl)morpholine 1123296-98-9 C19H27N5O3S
4-(5-(2-(cyclohexylmethyl)-2H-tetrazol-5-yl)-2-methylphenylsulfonyl)morpholine
—— N-(5-(1-(4-(2-cyanopropan-2-yl)phenyl)-3-methyl-3H-pyrazolo[3,4-c]quinolin-8-yl)pyridin-3-yl)methanesulfonamide 1201646-09-4 C27H24N6O2S
N-(5-(1-(4-(2-cyanopropan-2-yl)phenyl)-3-methyl-3H-pyrazolo[3,4-c]quinolin-8-yl)pyridin-3-yl)methanesulfonamide
—— KMI-1302 1160850-90-7 C33H28FIN8O5
KMI-1302
—— KMI-1256 1160850-86-1 C33H29BrN8O5
KMI-1256