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中文名称 英文名称 CAS号 化学式 结构式图片
—— 2,2-dichloro-N-[[(5S)-2-oxo-3-[4-([1,2,4]triazolo[4,3-a]pyrimidin-3-yl)phenyl]-1,3-oxazolidin-5-yl]methyl]acetamide 1309929-37-0 C17H14Cl2N6O3
2,2-dichloro-N-[[(5S)-2-oxo-3-[4-([1,2,4]triazolo[4,3-a]pyrimidin-3-yl)phenyl]-1,3-oxazolidin-5-yl]methyl]acetamide
—— (R)-cyclopropyl(2-(3-m-tolyl-1,2,4-oxadiazol-5-yl)piperidin-1-yl)methanone 1310486-28-2 C18H21N3O2
(R)-cyclopropyl(2-(3-m-tolyl-1,2,4-oxadiazol-5-yl)piperidin-1-yl)methanone
—— (R)-1-(3,4-difluorobenzyl)-5-ethyl-7-isopropyl-2-(4-(trifluoromethoxy)phenyl)-7,8-dihydro-1H-imidazo[2,1-b]purin-4(5H)-one 1314080-27-7 C26H24F5N5O2
(R)-1-(3,4-difluorobenzyl)-5-ethyl-7-isopropyl-2-(4-(trifluoromethoxy)phenyl)-7,8-dihydro-1H-imidazo[2,1-b]purin-4(5H)-one
—— 2-(4-(5-(1-(4-chlorophenyl)cyclobutyl)-4-methyl-4H-1,2,4-triazol-3-yl)-3-fluorophenyl)pyrazine 1296644-85-3 C23H19ClFN5
2-(4-(5-(1-(4-chlorophenyl)cyclobutyl)-4-methyl-4H-1,2,4-triazol-3-yl)-3-fluorophenyl)pyrazine
—— N-[[(5S)-2-oxo-3-[4-([1,2,4]triazolo[4,3-a]pyrimidin-3-yl)phenyl]-1,3-oxazolidin-5-yl]methyl]benzamide 1309929-40-5 C22H18N6O3
N-[[(5S)-2-oxo-3-[4-([1,2,4]triazolo[4,3-a]pyrimidin-3-yl)phenyl]-1,3-oxazolidin-5-yl]methyl]benzamide
—— rac-(2R,3R)-N-((R)-1-(4-(1H-pyrazol-1-yl)phenyl)ethyl)-4-((3S)-2-(3-chlorophenyl)-3-hydroxypyrrolidin-1-yl)-2,3-dihydroxy-4-oxobutanamide 1310416-70-6 C25H27ClN4O5
rac-(2R,3R)-N-((R)-1-(4-(1H-pyrazol-1-yl)phenyl)ethyl)-4-((3S)-2-(3-chlorophenyl)-3-hydroxypyrrolidin-1-yl)-2,3-dihydroxy-4-oxobutanamide
—— sodium;(3R,5R)-7-[5-cyclopropyl-2-(4-fluorophenyl)-4-[(2-methoxyphenyl)methylcarbamoyl]imidazol-1-yl]-3,5-dihydroxyheptanoate 1309777-87-4 C28H31FN3O6*Na
sodium;(3R,5R)-7-[5-cyclopropyl-2-(4-fluorophenyl)-4-[(2-methoxyphenyl)methylcarbamoyl]imidazol-1-yl]-3,5-dihydroxyheptanoate
—— 7-Amino-4-benzyl-10-[2-(dimethylamino)ethyl]-3,4,6,8,10,11-hexazatricyclo[7.3.0.02,6]dodeca-1(9),2,7,11-tetraen-5-one 1303471-19-3 C17H20N8O
7-Amino-4-benzyl-10-[2-(dimethylamino)ethyl]-3,4,6,8,10,11-hexazatricyclo[7.3.0.02,6]dodeca-1(9),2,7,11-tetraen-5-one
—— 3-(2-thienylmethoxycarbonyl)-8-(N-Boc-pyrrol-2-yl)-pyrazolo[5,1-c][1,2,4]benzotriazine 5-oxide 1310053-62-3 C24H21N5O5S
3-(2-thienylmethoxycarbonyl)-8-(N-Boc-pyrrol-2-yl)-pyrazolo[5,1-c][1,2,4]benzotriazine 5-oxide
—— (3-(4-chlorophenyl)-1H-pyrazol-5-yl)(4-(2-methoxybenzyl)piperazin-1-yl)methanone 1277167-57-3 C22H23ClN4O2
(3-(4-chlorophenyl)-1H-pyrazol-5-yl)(4-(2-methoxybenzyl)piperazin-1-yl)methanone
—— (7R)-1-(3,4-difluorobenzyl)-5-ethyl-2-(2-fluorophenyl)-7-isopropyl-7,8-dihydro-1H-imidazo[2,1-b]purin-4(5H)-one 1314080-26-6 C25H24F3N5O
(7R)-1-(3,4-difluorobenzyl)-5-ethyl-2-(2-fluorophenyl)-7-isopropyl-7,8-dihydro-1H-imidazo[2,1-b]purin-4(5H)-one
—— 5-chloro-N-(4-(3,5-dimethyl-1H-1,2,4-triazol-1-yl)phenyl)-4-(1-methyl-1H-pyrazol-3-yl)pyridin-2-amine 1309880-11-2 C19H18ClN7
5-chloro-N-(4-(3,5-dimethyl-1H-1,2,4-triazol-1-yl)phenyl)-4-(1-methyl-1H-pyrazol-3-yl)pyridin-2-amine
—— sodium;(3R,5R)-7-[5-cyclopropyl-2-(4-fluorophenyl)-4-[(4-fluorophenyl)methylcarbamoyl]imidazol-1-yl]-3,5-dihydroxyheptanoate 1309777-88-5 C27H28F2N3O5*Na
sodium;(3R,5R)-7-[5-cyclopropyl-2-(4-fluorophenyl)-4-[(4-fluorophenyl)methylcarbamoyl]imidazol-1-yl]-3,5-dihydroxyheptanoate
—— 1-tert-butyl-3-[[(5S)-2-oxo-3-[4-([1,2,4]triazolo[4,3-a]pyrimidin-3-yl)phenyl]-1,3-oxazolidin-5-yl]methyl]urea 1309929-47-2 C20H23N7O3
1-tert-butyl-3-[[(5S)-2-oxo-3-[4-([1,2,4]triazolo[4,3-a]pyrimidin-3-yl)phenyl]-1,3-oxazolidin-5-yl]methyl]urea
—— 5-chloro-4-(1-methyl-1H-pyrazol-3-yl)-N-(4-(3-morpholino-1H-1,2,4-triazol-1-yl)phenyl)pyridin-2-amine 1309880-12-3 C21H21ClN8O
5-chloro-4-(1-methyl-1H-pyrazol-3-yl)-N-(4-(3-morpholino-1H-1,2,4-triazol-1-yl)phenyl)pyridin-2-amine
—— sodium;(3R,5R)-7-[5-cyclopropyl-2-(4-fluorophenyl)-4-[(3-methoxyphenyl)methylcarbamoyl]imidazol-1-yl]-3,5-dihydroxyheptanoate 1309777-86-3 C28H31FN3O6*Na
sodium;(3R,5R)-7-[5-cyclopropyl-2-(4-fluorophenyl)-4-[(3-methoxyphenyl)methylcarbamoyl]imidazol-1-yl]-3,5-dihydroxyheptanoate
—— 1-(2,3-dichlorophenyl)-N-[[2-(difluoromethoxy)phenyl]methyl]tetrazol-5-amine 870066-61-8 C15H11Cl2F2N5O
1-(2,3-dichlorophenyl)-N-[[2-(difluoromethoxy)phenyl]methyl]tetrazol-5-amine
—— (S)-cyclobutyl(3-(3-(3-fluorophenyl)-1,2,4-oxadiazol-5-yl)piperidin-1-yl)methanone 1310486-08-8 C18H20FN3O2
(S)-cyclobutyl(3-(3-(3-fluorophenyl)-1,2,4-oxadiazol-5-yl)piperidin-1-yl)methanone
—— 1-[[(5S)-2-oxo-3-[4-([1,2,4]triazolo[4,3-a]pyrimidin-3-yl)phenyl]-1,3-oxazolidin-5-yl]methyl]-3-propan-2-ylthiourea 1309929-49-4 C19H21N7O2S
1-[[(5S)-2-oxo-3-[4-([1,2,4]triazolo[4,3-a]pyrimidin-3-yl)phenyl]-1,3-oxazolidin-5-yl]methyl]-3-propan-2-ylthiourea
—— 1-(2,3-dichlorophenyl)-N-[(3-methoxyphenyl)methyl]tetrazol-5-amine 870066-57-2 C15H13Cl2N5O
1-(2,3-dichlorophenyl)-N-[(3-methoxyphenyl)methyl]tetrazol-5-amine
—— N-(4-(3,5-dimethyl-1H-1,2,4-triazol-1-yl)phenyl)-4-(1-(3-methoxyphenyl)-1H-pyrazol-3-yl)pyridin-2-amine 1309880-28-1 C25H23N7O
N-(4-(3,5-dimethyl-1H-1,2,4-triazol-1-yl)phenyl)-4-(1-(3-methoxyphenyl)-1H-pyrazol-3-yl)pyridin-2-amine
—— (E)-3-[5-[4-[[2-(5-acetyl-2-thienyl)-5-(morpholine-4-carbonyl)phenyl]methoxy]phenyl]-1-cyclohexyl-pyrazol-3-yl]-2-methyl-prop-2-enoic acid 1310458-92-4 C37H39N3O6S
(E)-3-[5-[4-[[2-(5-acetyl-2-thienyl)-5-(morpholine-4-carbonyl)phenyl]methoxy]phenyl]-1-cyclohexyl-pyrazol-3-yl]-2-methyl-prop-2-enoic acid
—— sodium;(3R,5R)-7-[5-cyclopropyl-4-[[4-(dimethylsulfamoyl)phenyl]methylcarbamoyl]-2-(4-fluorophenyl)imidazol-1-yl]-3,5-dihydroxyheptanoate 1309777-96-5 C29H34FN4O7S*Na
sodium;(3R,5R)-7-[5-cyclopropyl-4-[[4-(dimethylsulfamoyl)phenyl]methylcarbamoyl]-2-(4-fluorophenyl)imidazol-1-yl]-3,5-dihydroxyheptanoate
—— methyl N-[[(5S)-2-oxo-3-[4-([1,2,4]triazolo[4,3-a]pyrimidin-3-yl)phenyl]-1,3-oxazolidin-5-yl]methyl]carbamate 1309929-43-8 C17H16N6O4
methyl N-[[(5S)-2-oxo-3-[4-([1,2,4]triazolo[4,3-a]pyrimidin-3-yl)phenyl]-1,3-oxazolidin-5-yl]methyl]carbamate
—— 5-chloro-4-(1-methyl-1H-pyrazol-3-yl)-N-(4-(3-morpholino-1H-1,2,4-triazol-1-yl)phenyl)pyrimidin-2-amine 1309880-07-6 C20H20ClN9O
5-chloro-4-(1-methyl-1H-pyrazol-3-yl)-N-(4-(3-morpholino-1H-1,2,4-triazol-1-yl)phenyl)pyrimidin-2-amine
—— 4-[4-methyl-2-[(2R)-2-[4-(5-phenylpentylsulfanyl)phenoxy]propanoyl]-1,3-thiazol-5-yl]butanoic acid 1310809-77-8 C28H33NO4S2
4-[4-methyl-2-[(2R)-2-[4-(5-phenylpentylsulfanyl)phenoxy]propanoyl]-1,3-thiazol-5-yl]butanoic acid
—— sodium;(3R,5R)-7-[5-cyclopropyl-2-(4-fluorophenyl)-4-[(4-methylphenyl)methylcarbamoyl]imidazol-1-yl]-3,5-dihydroxyheptanoate 1309777-83-0 C28H31FN3O5*Na
sodium;(3R,5R)-7-[5-cyclopropyl-2-(4-fluorophenyl)-4-[(4-methylphenyl)methylcarbamoyl]imidazol-1-yl]-3,5-dihydroxyheptanoate
—— 4-[4-methyl-2-[(2S)-2-[4-(5-phenylpentylsulfanyl)phenoxy]propanoyl]-1,3-thiazol-5-yl]butanoic acid 1310809-76-7 C28H33NO4S2
4-[4-methyl-2-[(2S)-2-[4-(5-phenylpentylsulfanyl)phenoxy]propanoyl]-1,3-thiazol-5-yl]butanoic acid
—— sodium;(3R,5R)-7-[5-cyclopropyl-2-(4-fluorophenyl)-4-[(2-methylphenyl)methylcarbamoyl]imidazol-1-yl]-3,5-dihydroxyheptanoate 1309777-85-2 C28H31FN3O5*Na
sodium;(3R,5R)-7-[5-cyclopropyl-2-(4-fluorophenyl)-4-[(2-methylphenyl)methylcarbamoyl]imidazol-1-yl]-3,5-dihydroxyheptanoate
—— 4-(5-(1-(4-chlorophenyl)cyclobutyl)-4-methyl-4H-1,2,4-triazol-3-yl)benzoic acid 1296644-48-8 C20H18ClN3O2
4-(5-(1-(4-chlorophenyl)cyclobutyl)-4-methyl-4H-1,2,4-triazol-3-yl)benzoic acid
—— N-[(2-chlorophenyl)methyl]-1-(2,3-dichlorophenyl)tetrazol-5-amine 870066-50-5 C14H10Cl3N5
N-[(2-chlorophenyl)methyl]-1-(2,3-dichlorophenyl)tetrazol-5-amine
—— 4-methyl-3-(4-((4-(methylsulfonyl)phenoxy)methyl)bicyclo[2.2.2]octan-1-yl)-5-(2-(trifluoromethyl)phenyl)-4H-1,2,4-triazole 1304515-68-1 C26H28F3N3O3S
4-methyl-3-(4-((4-(methylsulfonyl)phenoxy)methyl)bicyclo[2.2.2]octan-1-yl)-5-(2-(trifluoromethyl)phenyl)-4H-1,2,4-triazole
—— [3-(4-Chlorophenyl)-1-(4-hydroxyphenyl)-1H-pyrazol-4-yl]acetic acid 89435-60-9 C17H13ClN2O3
[3-(4-Chlorophenyl)-1-(4-hydroxyphenyl)-1H-pyrazol-4-yl]acetic acid
—— N-(4-(5-(1-(4-chlorophenyl)cyclobutyl)-4-methyl-4H-1,2,4-triazol-3-yl)phenyl)acetamide 1296644-60-4 C21H21ClN4O
N-(4-(5-(1-(4-chlorophenyl)cyclobutyl)-4-methyl-4H-1,2,4-triazol-3-yl)phenyl)acetamide
—— 1-(2,3-dichlorophenyl)-N-[(4-fluorophenyl)methyl]tetrazol-5-amine 870066-55-0 C14H10Cl2FN5
1-(2,3-dichlorophenyl)-N-[(4-fluorophenyl)methyl]tetrazol-5-amine
—— N-[(4-chlorophenyl)methyl]-1-(2,3-dichlorophenyl)tetrazol-5-amine 870066-52-7 C14H10Cl3N5
N-[(4-chlorophenyl)methyl]-1-(2,3-dichlorophenyl)tetrazol-5-amine
—— N-[3-(diethylamino)propyl]-2,4-diphenyl-thiazole-5-carboxamide 1314802-58-8 C23H27N3OS
N-[3-(diethylamino)propyl]-2,4-diphenyl-thiazole-5-carboxamide
—— 5-chloro-N-(4-(3-methyl-1H-1,2,4-triazol-1-yl)phenyl)-4-(1-methyl-1H-pyrazol-3-yl)pyrimidin-2-amine 1309880-06-5 C17H15ClN8
5-chloro-N-(4-(3-methyl-1H-1,2,4-triazol-1-yl)phenyl)-4-(1-methyl-1H-pyrazol-3-yl)pyrimidin-2-amine
—— (Z)-carbamoylimino-(1,5-dimethyl-3-thiophen-2-ylpyrazol-4-yl)-oxidoazanium 1312672-00-6 C10H11N5O2S
(Z)-carbamoylimino-(1,5-dimethyl-3-thiophen-2-ylpyrazol-4-yl)-oxidoazanium
—— N-[[(5S)-2-oxo-3-[4-([1,2,4]triazolo[4,3-a]pyrimidin-3-yl)phenyl]-1,3-oxazolidin-5-yl]methyl]cyclobutanecarboxamide 1309929-39-2 C20H20N6O3
N-[[(5S)-2-oxo-3-[4-([1,2,4]triazolo[4,3-a]pyrimidin-3-yl)phenyl]-1,3-oxazolidin-5-yl]methyl]cyclobutanecarboxamide
—— (S)-cyclobutyl(2-(3-(3-fluorophenyl)-1,2,4-oxadiazol-5-yl)piperidin-1-yl)methanone 1310486-20-4 C18H20FN3O2
(S)-cyclobutyl(2-(3-(3-fluorophenyl)-1,2,4-oxadiazol-5-yl)piperidin-1-yl)methanone
—— sodium;(3R,5R)-7-[5-cyclopropyl-4-[(2,4-difluorophenyl)methylcarbamoyl]-2-(4-fluorophenyl)imidazol-1-yl]-3,5-dihydroxyheptanoate 1309777-92-1 C27H27F3N3O5*Na
sodium;(3R,5R)-7-[5-cyclopropyl-4-[(2,4-difluorophenyl)methylcarbamoyl]-2-(4-fluorophenyl)imidazol-1-yl]-3,5-dihydroxyheptanoate
—— N-[[(5S)-2-oxo-3-[4-([1,2,4]triazolo[4,3-a]pyrimidin-3-yl)phenyl]-1,3-oxazolidin-5-yl]methyl]cyclopropanecarboxamide 1309929-38-1 C19H18N6O3
N-[[(5S)-2-oxo-3-[4-([1,2,4]triazolo[4,3-a]pyrimidin-3-yl)phenyl]-1,3-oxazolidin-5-yl]methyl]cyclopropanecarboxamide
—— phenyl N-[[(5S)-2-oxo-3-[4-([1,2,4]triazolo[4,3-a]pyrimidin-3-yl)phenyl]-1,3-oxazolidin-5-yl]methyl]carbamate 1309929-45-0 C22H18N6O4
phenyl N-[[(5S)-2-oxo-3-[4-([1,2,4]triazolo[4,3-a]pyrimidin-3-yl)phenyl]-1,3-oxazolidin-5-yl]methyl]carbamate
—— 4,5,6,7-tetrahydro-2H-indazol-7-ol 1306606-66-5 C7H10N2O
4,5,6,7-tetrahydro-2H-indazol-7-ol
—— (R)-5-(1-(3,4-difluorobenzyl)-5-ethyl-7-isopropyl-4-oxo-4,5,7,8-tetrahydro-1H-imidazo[2,1-b]purin-2-yl)-2-fluorobenzonitrile 1314080-31-3 C26H23F3N6O
(R)-5-(1-(3,4-difluorobenzyl)-5-ethyl-7-isopropyl-4-oxo-4,5,7,8-tetrahydro-1H-imidazo[2,1-b]purin-2-yl)-2-fluorobenzonitrile
—— 3-methoxycarbonyl-8-(pyrrol-2-yl)pyrazolo[5,1-c][1,2,4]-benzotriazine 5-oxide 1310053-63-4 C15H11N5O3
3-methoxycarbonyl-8-(pyrrol-2-yl)pyrazolo[5,1-c][1,2,4]-benzotriazine 5-oxide
—— 2-chloro-N-[[(5S)-2-oxo-3-[4-([1,2,4]triazolo[4,3-a]pyrimidin-3-yl)phenyl]-1,3-oxazolidin-5-yl]methyl]acetamide 1309929-36-9 C17H15ClN6O3
2-chloro-N-[[(5S)-2-oxo-3-[4-([1,2,4]triazolo[4,3-a]pyrimidin-3-yl)phenyl]-1,3-oxazolidin-5-yl]methyl]acetamide
—— N-[[(5S)-2-oxo-3-[4-([1,2,4]triazolo[4,3-a]pyrimidin-3-yl)phenyl]-1,3-oxazolidin-5-yl]methyl]propanethioamide 1309929-42-7 C18H18N6O2S
N-[[(5S)-2-oxo-3-[4-([1,2,4]triazolo[4,3-a]pyrimidin-3-yl)phenyl]-1,3-oxazolidin-5-yl]methyl]propanethioamide
—— sodium;(3R,5R)-7-[4-[(4-carbamoylphenyl)methylcarbamoyl]-5-cyclopropyl-2-(4-fluorophenyl)imidazol-1-yl]-3,5-dihydroxyheptanoate 1309777-95-4 C28H30FN4O6*Na
sodium;(3R,5R)-7-[4-[(4-carbamoylphenyl)methylcarbamoyl]-5-cyclopropyl-2-(4-fluorophenyl)imidazol-1-yl]-3,5-dihydroxyheptanoate