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中文名称 英文名称 CAS号 化学式 结构式图片
—— 3-(3,5-difluoro-4-((1-phenyl-1H-1,2,3-triazol-5-yl)methoxy)phenyl)propanoic acid 1224102-19-5 C18H15F2N3O3
3-(3,5-difluoro-4-((1-phenyl-1H-1,2,3-triazol-5-yl)methoxy)phenyl)propanoic acid
—— 2-(2-(4-((1-(4-chlorophenyl)-3-methyl-1H-pyrazol-5-yl)methoxy)-3,5-difluoro-phenyl)cyclopropyl)acetic acid 1224102-18-4 C22H19ClF2N2O3
2-(2-(4-((1-(4-chlorophenyl)-3-methyl-1H-pyrazol-5-yl)methoxy)-3,5-difluoro-phenyl)cyclopropyl)acetic acid
—— 2,4,5,6-Tetrahydrocyclopenta[c]pyrazol-3-ylmethanol 1215295-82-1 C7H10N2O
2,4,5,6-Tetrahydrocyclopenta[c]pyrazol-3-ylmethanol
—— 1-(4-(4-amino-1-(3-hydroxypropyl)-1H-pyrazolo[3,4-d]pyrimidin-3-yl)phenyl)-3-(3-(trifluoromethyl)phenyl)urea 1221743-66-3 C22H20F3N7O2
1-(4-(4-amino-1-(3-hydroxypropyl)-1H-pyrazolo[3,4-d]pyrimidin-3-yl)phenyl)-3-(3-(trifluoromethyl)phenyl)urea
—— Carbamic acid, N-[(1R)-1-[1-(2,2,2-trifluoroethyl)-1H-imidazol-5-yl]ethyl]-, 1,1-dimethylethyl ester 1893470-00-2 C12H18F3N3O2
Carbamic acid, N-[(1R)-1-[1-(2,2,2-trifluoroethyl)-1H-imidazol-5-yl]ethyl]-, 1,1-dimethylethyl ester
—— 2-(Pyridin-4-YL)thiazole-5-carbaldehyde 21346-36-1 C9H6N2OS
2-(Pyridin-4-YL)thiazole-5-carbaldehyde
—— 1-(ethylsulfonyl)-N-[1-(4-methoxyphenyl)-1H-imidazol-4-yl]-1,2-dihydro-1'H-spiro[indole-3,4'-piperidine]-1'-carboxamide 1185761-99-2 C25H29N5O4S
1-(ethylsulfonyl)-N-[1-(4-methoxyphenyl)-1H-imidazol-4-yl]-1,2-dihydro-1'H-spiro[indole-3,4'-piperidine]-1'-carboxamide
—— 3-(4-Chlorophenyl)imidazo[1,2-a]pyridine-2-carboxylic acid 1244949-49-2 C14H9ClN2O2
3-(4-Chlorophenyl)imidazo[1,2-a]pyridine-2-carboxylic acid
—— N-cycloheptyl 1-(2,4-difluorophenyl)-4-methyl-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamide 1185915-70-1 C22H24F2N4O
N-cycloheptyl 1-(2,4-difluorophenyl)-4-methyl-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamide
—— 4-(4-Methyl-1H-imidazol-1-yl)benzenemethanamine 1244949-44-7 C11H13N3
4-(4-Methyl-1H-imidazol-1-yl)benzenemethanamine
—— 1-{3-[4-Chloro-3-(4-chloro-phenylethynyl)-phenyl]-5-methanesulfonyl-4,5,6,7-tetrahydro-pyrazolo[4,3-c]pyridin-1-yl}-3-piperidin-1-yl-propan-2-ol 1049809-31-5 C29H32Cl2N4O3S
1-{3-[4-Chloro-3-(4-chloro-phenylethynyl)-phenyl]-5-methanesulfonyl-4,5,6,7-tetrahydro-pyrazolo[4,3-c]pyridin-1-yl}-3-piperidin-1-yl-propan-2-ol
—— 3-cyano-4-(thiophen-2-yl)-1,2,5-oxadiazole 2-oxide 1147335-85-0 C7H3N3O2S
3-cyano-4-(thiophen-2-yl)-1,2,5-oxadiazole 2-oxide
—— Ethyl 2-(3-bromobenzyl)thiazole-4-carboxylate 954241-25-9 C13H12BrNO2S
Ethyl 2-(3-bromobenzyl)thiazole-4-carboxylate
—— 4-bromothiazole-5-carboxylic acid 1244949-48-1 C4H2BrNO2S
4-bromothiazole-5-carboxylic acid
—— 1-(ethylsulfonyl)-N-[1-(2-methoxyphenyl)-1H-imidazol-4-yl]-1,2-dihydro-1'H-spiro[indole-3,4'-piperidine]-1'-carboxamide 1185773-49-2 C25H29N5O4S
1-(ethylsulfonyl)-N-[1-(2-methoxyphenyl)-1H-imidazol-4-yl]-1,2-dihydro-1'H-spiro[indole-3,4'-piperidine]-1'-carboxamide
—— 5-(4-carboxymethylphenyl)-1-(4-methanesulfonylphenyl)-3-trifluoromethyl-1H-pyrazole 1186423-56-2 C19H15F3N2O4S
5-(4-carboxymethylphenyl)-1-(4-methanesulfonylphenyl)-3-trifluoromethyl-1H-pyrazole
—— 2-((1-(4-methoxy-2-methylphenyl)-3,6-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl)(propyl)amino)-N,N-dimethylacetamide 1197371-66-6 C22H30N6O2
2-((1-(4-methoxy-2-methylphenyl)-3,6-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl)(propyl)amino)-N,N-dimethylacetamide
—— 1-(ethylsulfonyl)-N-[1-(4-fluorophenyl)-1H-imidazol-4-yl]-1,2-dihydro-1'H-spiro[indole-3,4'-piperidine]-1'-carboxamide 1185761-97-0 C24H26FN5O3S
1-(ethylsulfonyl)-N-[1-(4-fluorophenyl)-1H-imidazol-4-yl]-1,2-dihydro-1'H-spiro[indole-3,4'-piperidine]-1'-carboxamide
—— 1-(3-{3-[4-Chloro-3-(4-chloro-phenylethynyl)-phenyl]-5-methanesulfonyl-4,5,6,7-tetrahydro-pyrazolo[4,3-c]pyridin-1-yl}-2-hydroxy-propyl)-piperidine-4-carboxylic acid methyl ester 1049809-33-7 C31H34Cl2N4O5S
1-(3-{3-[4-Chloro-3-(4-chloro-phenylethynyl)-phenyl]-5-methanesulfonyl-4,5,6,7-tetrahydro-pyrazolo[4,3-c]pyridin-1-yl}-2-hydroxy-propyl)-piperidine-4-carboxylic acid methyl ester
—— 5-chloro-N-{(1S)-1-[1-(4-hydroxyphenyl)-1H-pyrazol-5-yl]-2-methylpropyl}thiophene-2-sulfonamide 1178876-51-1 C17H18ClN3O3S2
5-chloro-N-{(1S)-1-[1-(4-hydroxyphenyl)-1H-pyrazol-5-yl]-2-methylpropyl}thiophene-2-sulfonamide
—— 1-{3-[4-Chloro-3-(4-chloro-phenylethynyl)-phenyl]-5-methanesulfonyl-4,5,6,7-tetrahydro-pyrazolo[4,3-c]pyridin-1-yl}-3-morpholin-4-yl-propan-2-ol 1049809-30-4 C28H30Cl2N4O4S
1-{3-[4-Chloro-3-(4-chloro-phenylethynyl)-phenyl]-5-methanesulfonyl-4,5,6,7-tetrahydro-pyrazolo[4,3-c]pyridin-1-yl}-3-morpholin-4-yl-propan-2-ol
—— 5-[2,3-dimethyl-4-(2-methylene-1-oxopropyl)phenoxymethyl]-3-(4-nitrobenzyl)-1,2,4-oxadiazol 1258065-03-0 C21H19N3O5
5-[2,3-dimethyl-4-(2-methylene-1-oxopropyl)phenoxymethyl]-3-(4-nitrobenzyl)-1,2,4-oxadiazol
—— N-cycloheptyl 1-(2,4-dichlorophenyl)-4-methyl-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamide 1185915-36-9 C22H24Cl2N4O
N-cycloheptyl 1-(2,4-dichlorophenyl)-4-methyl-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamide
—— N-(2-bromo-3,4,5-trimethoxybenzyl) 1-(2,4-difluorophenyl)-4-methyl-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamide 1185915-64-3 C25H23BrF2N4O4
N-(2-bromo-3,4,5-trimethoxybenzyl) 1-(2,4-difluorophenyl)-4-methyl-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamide
—— (1R,2S,5S,10S,14R,15R,23R)-1,2,8,8,15,22,22-heptamethyl-20-phenyl-19,20-diazahexacyclo[12.11.0.02,11.05,10.015,23.017,21]pentacosa-11,17(21),18-triene-5-carboxylic acid 1202006-27-6 C37H50N2O2
(1R,2S,5S,10S,14R,15R,23R)-1,2,8,8,15,22,22-heptamethyl-20-phenyl-19,20-diazahexacyclo[12.11.0.02,11.05,10.015,23.017,21]pentacosa-11,17(21),18-triene-5-carboxylic acid
—— (Z)-acetyloxymethoxyimino-[methyl-[2-[2-[4-[2-(4-sulfamoylphenyl)-5-(trifluoromethyl)pyrazol-3-yl]phenyl]acetyl]oxyethyl]amino]-oxidoazanium 1186423-59-5 C24H25F3N6O8S
(Z)-acetyloxymethoxyimino-[methyl-[2-[2-[4-[2-(4-sulfamoylphenyl)-5-(trifluoromethyl)pyrazol-3-yl]phenyl]acetyl]oxyethyl]amino]-oxidoazanium
—— (2R)-2-({[4-({2-Chloro-5-[5-(methylsulfonyl)-1-(3-morpholin-4-ylpropyl)-4,5,6,7-tetrahydro-1H-pyrazolo[4,3-c]pyridin-3-yl]phenyl}ethynyl)phenyl]methyl}amino)-2-phenylethanol 1049810-65-2 C37H42ClN5O4S
(2R)-2-({[4-({2-Chloro-5-[5-(methylsulfonyl)-1-(3-morpholin-4-ylpropyl)-4,5,6,7-tetrahydro-1H-pyrazolo[4,3-c]pyridin-3-yl]phenyl}ethynyl)phenyl]methyl}amino)-2-phenylethanol
—— (Z)-acetyloxymethoxyimino-[methyl-[2-[2-[4-[2-(4-methylsulfonylphenyl)-5-(trifluoromethyl)pyrazol-3-yl]phenyl]acetyl]oxyethyl]amino]-oxidoazanium 1186423-58-4 C25H26F3N5O8S
(Z)-acetyloxymethoxyimino-[methyl-[2-[2-[4-[2-(4-methylsulfonylphenyl)-5-(trifluoromethyl)pyrazol-3-yl]phenyl]acetyl]oxyethyl]amino]-oxidoazanium
—— 1-(4-methoxy-2-methylphenyl)-N-((S)-1-methoxybutan-2-yl)-3,6-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine 1197371-72-4 C20H27N5O2
1-(4-methoxy-2-methylphenyl)-N-((S)-1-methoxybutan-2-yl)-3,6-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
—— 1,12-bis[(4-ethyl-1,2,4-oxadiazol-5-(4H)-one)-3-yl]dodecane 1190625-07-0 C20H34N4O4
1,12-bis[(4-ethyl-1,2,4-oxadiazol-5-(4H)-one)-3-yl]dodecane
—— 1-(4-methoxy-2-methylphenyl)-N,N-bis(2-methoxyethyl)-3,6-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine 1197371-64-4 C21H29N5O3
1-(4-methoxy-2-methylphenyl)-N,N-bis(2-methoxyethyl)-3,6-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
—— (R)-N-(1-(3-(4-cyanophenyl)-8-methylimidazo[1,2-a]pyrazin-2-yl)ethyl)-N-(2-(ethylsulfonyl)ethyl)-2-(3-fluoro-4-(trifluoromethyl)phenyl)acetamide 1190969-56-2 C29H27F4N5O3S
(R)-N-(1-(3-(4-cyanophenyl)-8-methylimidazo[1,2-a]pyrazin-2-yl)ethyl)-N-(2-(ethylsulfonyl)ethyl)-2-(3-fluoro-4-(trifluoromethyl)phenyl)acetamide
—— 1,12-bis[(4-methyl-1,2,4-oxadiazol-5-(4H)-one)-3-yl]dodecane 1190625-05-8 C18H30N4O4
1,12-bis[(4-methyl-1,2,4-oxadiazol-5-(4H)-one)-3-yl]dodecane
—— 2-tert-butyl-5-(5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-4-(5-methyl-1,3,4-oxadiazol-2-yl)-1H-pyrazol-3-yl)-1,3,4-oxadiazole 1202256-92-5 C24H19Cl3N6O2
2-tert-butyl-5-(5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-4-(5-methyl-1,3,4-oxadiazol-2-yl)-1H-pyrazol-3-yl)-1,3,4-oxadiazole
—— 2-((1-(4-methoxy-2-methylphenyl)-3,6-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl)(propyl)amino)ethanol 1197371-65-5 C20H27N5O2
2-((1-(4-methoxy-2-methylphenyl)-3,6-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl)(propyl)amino)ethanol
—— (R)-N-(1-(3-(4-cyanophenyl)-8-methoxyimidazo[1,2-a]pyrazin-2-yl)ethyl)-N-(2-(ethylsulfonyl)ethyl)-2-(3-fluoro-4-(trifluoromethyl)phenyl)acetamide 1190969-55-1 C29H27F4N5O4S
(R)-N-(1-(3-(4-cyanophenyl)-8-methoxyimidazo[1,2-a]pyrazin-2-yl)ethyl)-N-(2-(ethylsulfonyl)ethyl)-2-(3-fluoro-4-(trifluoromethyl)phenyl)acetamide
—— 1-(4-(2-(diethylamino)ethoxy)-3-(1-methyl-1H-pyrazol-5-yl)phenyl)-3-(4-fluorophenyl)urea 1190953-85-5 C23H28FN5O2
1-(4-(2-(diethylamino)ethoxy)-3-(1-methyl-1H-pyrazol-5-yl)phenyl)-3-(4-fluorophenyl)urea
—— Ethyl 3-(3-(4-(1,3,4-oxadiazol-2-yl)phenyl)-2-(pyridin-4-yl)-1,2-dihydropyrazolo[1,5-a]pyrimidin-7-yl)-8-azabicyclo[3.2.1]octane-8-carboxylate 1202183-89-8 C29H27N7O3
Ethyl 3-(3-(4-(1,3,4-oxadiazol-2-yl)phenyl)-2-(pyridin-4-yl)-1,2-dihydropyrazolo[1,5-a]pyrimidin-7-yl)-8-azabicyclo[3.2.1]octane-8-carboxylate
—— 2-tert-butyl-5-(5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-4-(5-methyl-1,3,4-thiadiazol-2-yl)-1H-pyrazol-3-yl)-1,3,4-oxadiazole 1202256-96-9 C24H19Cl3N6OS
2-tert-butyl-5-(5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-4-(5-methyl-1,3,4-thiadiazol-2-yl)-1H-pyrazol-3-yl)-1,3,4-oxadiazole
—— (S)-1,1,1-trifluoro-2-[(5aR,6S)-1-(4-fluorophenyl)-5a-methyl-5,5a,6,7,8,9-hexahydroimidazo[1,5-b]isoquinolin-6-yl]propan-2-ol 1150845-42-3 C21H22F4N2O
(S)-1,1,1-trifluoro-2-[(5aR,6S)-1-(4-fluorophenyl)-5a-methyl-5,5a,6,7,8,9-hexahydroimidazo[1,5-b]isoquinolin-6-yl]propan-2-ol
—— 1-(4-(6-aminoquinazolin-4-ylamino)phenyl)-3-(3-tert-butyl-1-p-tolyl-1H-pyrazol-5-yl)urea 1163731-06-3 C29H30N8O
1-(4-(6-aminoquinazolin-4-ylamino)phenyl)-3-(3-tert-butyl-1-p-tolyl-1H-pyrazol-5-yl)urea
—— Ethyl 3-(3-(3,4-difluorophenyl)-2-(pyridin-4-yl)-1,2-dihydropyrazolo[1,5-a]pyrimidin-7-yl)-8-azabicyclo[3.2.1]octane-8-carboxylate 1202183-88-7 C27H25F2N5O2
Ethyl 3-(3-(3,4-difluorophenyl)-2-(pyridin-4-yl)-1,2-dihydropyrazolo[1,5-a]pyrimidin-7-yl)-8-azabicyclo[3.2.1]octane-8-carboxylate
—— 1-(4-chlorophenyl)-3-(4-(2-(diethylamino)ethoxy)-3-(1-methyl-1H-pyrazol-5-yl)phenyl)urea 1190953-83-3 C23H28ClN5O2
1-(4-chlorophenyl)-3-(4-(2-(diethylamino)ethoxy)-3-(1-methyl-1H-pyrazol-5-yl)phenyl)urea
—— N-(4-(3-(3-(tert-butyl-1-p-tolyl-1H-pyrazol-5-yl)ureido)phenylamino)quinolin-6-yl)propionamide 1163731-00-7 C33H35N7O2
N-(4-(3-(3-(tert-butyl-1-p-tolyl-1H-pyrazol-5-yl)ureido)phenylamino)quinolin-6-yl)propionamide
—— 1-(4-tert-butylbenzyl)-N-phenethyl-3-phenyl-1H-pyrazole-5-carboxamide 1191284-77-1 C29H31N3O
1-(4-tert-butylbenzyl)-N-phenethyl-3-phenyl-1H-pyrazole-5-carboxamide
—— N-[1-[3-(4-cyanophenyl)-8-methoxyimidazo[1,2-a]pyrazin-2-yl]ethyl]-N-(2-ethylsulfonylethyl)-2-[3-fluoro-4-(trifluoromethyl)phenyl]acetamide 1190969-54-0 C29H27F4N5O4S
N-[1-[3-(4-cyanophenyl)-8-methoxyimidazo[1,2-a]pyrazin-2-yl]ethyl]-N-(2-ethylsulfonylethyl)-2-[3-fluoro-4-(trifluoromethyl)phenyl]acetamide
—— 1-(4-Chloro-phenyl)-3-[4-[2-((2S,6R)-2,6-dimethyl-piperidin-1-yl)-ethoxy]-3-(2-methyl-2H-pyrazol-3-yl)-phenyl]-urea 887932-54-9 C26H32ClN5O2
1-(4-Chloro-phenyl)-3-[4-[2-((2S,6R)-2,6-dimethyl-piperidin-1-yl)-ethoxy]-3-(2-methyl-2H-pyrazol-3-yl)-phenyl]-urea
—— 1-(4-Chloro-phenyl)-3-[4-[2-(2-methyl-piperidin-1-yl)-ethoxy]-3-(2-methyl-2H-pyrazol-3-yl)-phenyl]-urea 887933-96-2 C25H30ClN5O2
1-(4-Chloro-phenyl)-3-[4-[2-(2-methyl-piperidin-1-yl)-ethoxy]-3-(2-methyl-2H-pyrazol-3-yl)-phenyl]-urea
—— 2-(4-fluorophenyl)-3-(4-pyridyl)-5-chloro-(2-hydroxyethyl)imidazo[1,2-a]pyridine 1201526-69-3 C20H15ClFN3O
2-(4-fluorophenyl)-3-(4-pyridyl)-5-chloro-(2-hydroxyethyl)imidazo[1,2-a]pyridine
—— N-((2S,3R)-4-(3-(3-(1H-pyrazol-1-yl)phenyl)tetrahydrofuran-3-ylamino)-1-(3,5-difluorophenyl)-3-hydroxybutan-2-yl)acetamide 1350060-85-3 C25H28F2N4O3
N-((2S,3R)-4-(3-(3-(1H-pyrazol-1-yl)phenyl)tetrahydrofuran-3-ylamino)-1-(3,5-difluorophenyl)-3-hydroxybutan-2-yl)acetamide