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中文名称 英文名称 CAS号 化学式 结构式图片
—— 2-[2-(3-chlorobenzylidene)hydrazinyl]-4-phenyl-1,3-thiazole 464200-09-7 C16H12ClN3S
2-[2-(3-chlorobenzylidene)hydrazinyl]-4-phenyl-1,3-thiazole
—— N-(2,4-dichlorophenyl)-2-(2-(2,4-dichlorophenyl)-2H-1,2,4-triazol-3-ylthio)acetamide 1259007-21-0 C16H10Cl4N4OS
N-(2,4-dichlorophenyl)-2-(2-(2,4-dichlorophenyl)-2H-1,2,4-triazol-3-ylthio)acetamide
—— 1-(5-tert-butyl-2-{3-[2-(tetrahydro-pyran-2-yloxy)-ethoxy]-phenyl}-2H-pyrazol-3-yl)-3-[(1S,4R)-4-(3-piperidin-1-yl-[1,2,4] triazolo[4,3-a]pyridin-6-yloxy)-1,2,3,4-tetrahydro-naphthalen-1-yl]-urea 1443243-62-6 C42H52N8O5
1-(5-tert-butyl-2-{3-[2-(tetrahydro-pyran-2-yloxy)-ethoxy]-phenyl}-2H-pyrazol-3-yl)-3-[(1S,4R)-4-(3-piperidin-1-yl-[1,2,4] triazolo[4,3-a]pyridin-6-yloxy)-1,2,3,4-tetrahydro-naphthalen-1-yl]-urea
—— 1-{5-tert-butyl-2-[3-(2-hydroxy-ethoxy)-phenyl]-2H-pyrazol-3-yl}-3-[(1S,4R)-4-(3-piperidin-1-yl-[1,2,4]triazolo[4,3-a]pyridin-6-yloxy)-1,2,3,4-tetrahydro-naphthalen-1-yl]-urea 1443240-07-0 C37H44N8O4
1-{5-tert-butyl-2-[3-(2-hydroxy-ethoxy)-phenyl]-2H-pyrazol-3-yl}-3-[(1S,4R)-4-(3-piperidin-1-yl-[1,2,4]triazolo[4,3-a]pyridin-6-yloxy)-1,2,3,4-tetrahydro-naphthalen-1-yl]-urea
—— methane sulfonic acid 3-(3-tert-butyl-5-{3-[(1S,4R)-4-(3-piperidin-1-yl-[1,2,4]triazolo[4,3-a]pyridin-6-yloxy)-1,2,3,4-tetrahydro-naphthalen-1-yl]-ureido}-pyrazol-1-yl)-benzyl ester 1443243-76-2 C37H44N8O5S
methane sulfonic acid 3-(3-tert-butyl-5-{3-[(1S,4R)-4-(3-piperidin-1-yl-[1,2,4]triazolo[4,3-a]pyridin-6-yloxy)-1,2,3,4-tetrahydro-naphthalen-1-yl]-ureido}-pyrazol-1-yl)-benzyl ester
—— 3-methyl-1-phenyl-1H-pyrazole-4-carboxylic acid ethylester 113502-46-8 C13H14N2O2
3-methyl-1-phenyl-1H-pyrazole-4-carboxylic acid ethylester
—— 3-(4-chloro-3-methoxyphenyl)-N-(2-(4-methylpiperazin-1-yl)ethyl)-4-(pyridin-4-yl)-1H-pyrazole-1-carboxamide 1352810-93-5 C23H27ClN6O2
3-(4-chloro-3-methoxyphenyl)-N-(2-(4-methylpiperazin-1-yl)ethyl)-4-(pyridin-4-yl)-1H-pyrazole-1-carboxamide
—— 7-(4-Chloro-phenyl)-2-[3-methoxy-4-(4-methyl-imidazol-1-yl)-phenylamino]-6,7-dihydro-4H-[1,2,4]triazolo[1,5-a]pyrimidin-5-one 1319065-72-9 C22H20ClN7O2
7-(4-Chloro-phenyl)-2-[3-methoxy-4-(4-methyl-imidazol-1-yl)-phenylamino]-6,7-dihydro-4H-[1,2,4]triazolo[1,5-a]pyrimidin-5-one
—— (+)-2-{(E)-2-[3-methoxy-4-(4-methyl-1H-imidazol-1-yl)phenyl]vinyl}-8-(3,4,5-trifluorophenyl)-5,6,7,8-tetrahydro[1,2,4]triazolo[1,5-a]pyridine 949170-25-6 C25H22F3N5O
(+)-2-{(E)-2-[3-methoxy-4-(4-methyl-1H-imidazol-1-yl)phenyl]vinyl}-8-(3,4,5-trifluorophenyl)-5,6,7,8-tetrahydro[1,2,4]triazolo[1,5-a]pyridine
—— 7-(4-chlorophenyl)-2-(3-methoxy-4-(4-methyl-1H-imidazol-1-yl)phenylamino)-4-propyl-6,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidin-5(4H)-one 1319066-03-9 C25H26ClN7O2
7-(4-chlorophenyl)-2-(3-methoxy-4-(4-methyl-1H-imidazol-1-yl)phenylamino)-4-propyl-6,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidin-5(4H)-one
—— 1-{5-tert-butyl-2-[3-(2-hydroxy-ethoxymethyl)-phenyl]-2H-pyrazol-3-yl}-3-[(1S,4R)-4-(3-piperidin-1-yl-[1,2,4]triazolo[4,3-a]pyridin-6-yloxy)-1,2,3,4-tetrahydro-naphthalen-1-yl]-urea 1443240-18-3 C38H46N8O4
1-{5-tert-butyl-2-[3-(2-hydroxy-ethoxymethyl)-phenyl]-2H-pyrazol-3-yl}-3-[(1S,4R)-4-(3-piperidin-1-yl-[1,2,4]triazolo[4,3-a]pyridin-6-yloxy)-1,2,3,4-tetrahydro-naphthalen-1-yl]-urea
—— methanesulfonic acid 2-[3-(3-tert-butyl-5-{3-[(1S,4R)-4-(3-piperidin-1-yl-[1,2,4]triazolo[4,3-a]pyridin-6-yloxy)-1,2,3,4-tetrahydro-naphthalen-1-yl]-ureido}-pyrazol-1-yl)-phenoxy]-ethyl ester 1443243-63-7 C38H46N8O6S
methanesulfonic acid 2-[3-(3-tert-butyl-5-{3-[(1S,4R)-4-(3-piperidin-1-yl-[1,2,4]triazolo[4,3-a]pyridin-6-yloxy)-1,2,3,4-tetrahydro-naphthalen-1-yl]-ureido}-pyrazol-1-yl)-phenoxy]-ethyl ester
—— 1-(2-tert-butyl-5-p-tolyl-3H-imidazol-4-yl)-3-[(1S,4R)-4-(3-piperidin-1-yl-[1,2,4]triazolo[4,3-a]pyridin-6-yloxy)-1,2,3,4-tetrahydro-naphthalen-1-yl]-urea 1443240-21-8 C36H42N8O2
1-(2-tert-butyl-5-p-tolyl-3H-imidazol-4-yl)-3-[(1S,4R)-4-(3-piperidin-1-yl-[1,2,4]triazolo[4,3-a]pyridin-6-yloxy)-1,2,3,4-tetrahydro-naphthalen-1-yl]-urea
—— methyl 5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-1H-1,2,4-triazole-3-carboxylate 676457-40-2 C16H10Cl3N3O2
methyl 5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-1H-1,2,4-triazole-3-carboxylate
—— 1-{4-[3-(4-chloro-3-methoxyphenyl)-4-(pyridin-4-yl)-1H-pyrazol-1-yl]phenyl}-3-(2,3-dichlorophenyl)urea 1350473-77-6 C28H20Cl3N5O2
1-{4-[3-(4-chloro-3-methoxyphenyl)-4-(pyridin-4-yl)-1H-pyrazol-1-yl]phenyl}-3-(2,3-dichlorophenyl)urea
—— (2-((E)-2-[3-methoxy-4-(4-methyl-1H-imidazol-1-yl)phenyl]vinyl)-8-(3,4,5-trifluorophenyl)-5,6,7,8-tetrahydro[1,2,4]triazolo[1,5-a]pyridin-8-yl)methanol 1123191-35-4 C26H24F3N5O2
(2-((E)-2-[3-methoxy-4-(4-methyl-1H-imidazol-1-yl)phenyl]vinyl)-8-(3,4,5-trifluorophenyl)-5,6,7,8-tetrahydro[1,2,4]triazolo[1,5-a]pyridin-8-yl)methanol
—— 1-{4-[3-(4-chloro-3-methoxyphenyl)-4-(pyridin-4-yl)-1H-pyrazol-1-yl]phenyl}-3-(4-chloro-3-(trifluoromethyl)phenyl)urea 1350473-79-8 C29H20Cl2F3N5O2
1-{4-[3-(4-chloro-3-methoxyphenyl)-4-(pyridin-4-yl)-1H-pyrazol-1-yl]phenyl}-3-(4-chloro-3-(trifluoromethyl)phenyl)urea
—— 3-(4-fluoro-3-methyl-phenyl)-5-phenyl-pyrazole 1439306-15-6 C16H13FN2
3-(4-fluoro-3-methyl-phenyl)-5-phenyl-pyrazole
—— 3-(4-chloro-3-methoxyphenyl)-N-(2-(2,6-dimethylmorpholino)ethyl)-4-(pyridin-4-yl)-1H-pyrazole-1-carboxamide 1352810-92-4 C24H28ClN5O3
3-(4-chloro-3-methoxyphenyl)-N-(2-(2,6-dimethylmorpholino)ethyl)-4-(pyridin-4-yl)-1H-pyrazole-1-carboxamide
—— 1-(5-tert-butyl-2-p-tolyl-2H-pyrazol-3-yl)-3-[(1S,4S)-4-(3-piperidin-1-yl-[1,2,4]triazolo[4,3-a]pyridin-6-yloxy)-1,2,3,4-tetrahydro-naphthalen-1-yl]-urea 1443240-25-2 C36H42N8O2
1-(5-tert-butyl-2-p-tolyl-2H-pyrazol-3-yl)-3-[(1S,4S)-4-(3-piperidin-1-yl-[1,2,4]triazolo[4,3-a]pyridin-6-yloxy)-1,2,3,4-tetrahydro-naphthalen-1-yl]-urea
—— 1-{5-tert-butyl-2-[3-(4-methyl-piperazin-1-ylmethyl)-phenyl]-2H-pyrazol-3-yl}-3-[(1S,4R)-4-(3-piperidin-1-yl-[1,2,4]triazolo[4,3-a]pyridin-6-yloxy)-1,2,3,4-tetrahydro-naphthalen-1-yl]-urea 1443240-10-5 C41H52N10O2
1-{5-tert-butyl-2-[3-(4-methyl-piperazin-1-ylmethyl)-phenyl]-2H-pyrazol-3-yl}-3-[(1S,4R)-4-(3-piperidin-1-yl-[1,2,4]triazolo[4,3-a]pyridin-6-yloxy)-1,2,3,4-tetrahydro-naphthalen-1-yl]-urea
—— 1-(5-tert-butyl-2-{3-[4-(2-hydroxy-ethyl)-piperazin-1-ylmethyl]-phenyl}-2H-pyrazol-3-yl)-3-[(1S,4R)-4-(3-piperidin-1-yl-[1,2,4]triazolo[4,3-a]pyridin-6-yloxy)-1,2,3,4-tetrahydro-naphthalen-1-yl]-urea 1443240-20-7 C42H54N10O3
1-(5-tert-butyl-2-{3-[4-(2-hydroxy-ethyl)-piperazin-1-ylmethyl]-phenyl}-2H-pyrazol-3-yl)-3-[(1S,4R)-4-(3-piperidin-1-yl-[1,2,4]triazolo[4,3-a]pyridin-6-yloxy)-1,2,3,4-tetrahydro-naphthalen-1-yl]-urea
—— 2-(1-Phenyl-1H-pyrazol-5-yl)-propanoic acid 130216-56-7 C12H12N2O2
2-(1-Phenyl-1H-pyrazol-5-yl)-propanoic acid
—— 1-[5-tert-butyl-2-(4-cyano-phenyl)-2H-pyrazol-3-yl]-3-[(1S,4R)-4-(3-piperidin-1-yl-[1,2,4]triazolo[4,3-a]pyridin-6-yloxy)-1,2,3,4-tetrahydro-naphthalen-1-yl]-urea 1443240-48-9 C36H39N9O2
1-[5-tert-butyl-2-(4-cyano-phenyl)-2H-pyrazol-3-yl]-3-[(1S,4R)-4-(3-piperidin-1-yl-[1,2,4]triazolo[4,3-a]pyridin-6-yloxy)-1,2,3,4-tetrahydro-naphthalen-1-yl]-urea
—— 3-(4-chloro-3-hydroxyphenyl)-N-(2-(piperidin-1-yl)ethyl)-4-(pyridin-4-yl)-1H-pyrazole-1-carboxamide 1352811-04-1 C22H24ClN5O2
3-(4-chloro-3-hydroxyphenyl)-N-(2-(piperidin-1-yl)ethyl)-4-(pyridin-4-yl)-1H-pyrazole-1-carboxamide
—— 1-[5-tert-butyl-2-(4-hydroxymethyl-phenyl)-2H-pyrazol-3-yl]-3-[(1S,4R)-4-(3-piperidin-1-yl-[1,2,4]triazolo[4,3-a]pyridin-6-yloxy)-1,2,3,4-tetrahydro-naphthalen-1-yl]-urea 1443240-02-5 C36H42N8O3
1-[5-tert-butyl-2-(4-hydroxymethyl-phenyl)-2H-pyrazol-3-yl]-3-[(1S,4R)-4-(3-piperidin-1-yl-[1,2,4]triazolo[4,3-a]pyridin-6-yloxy)-1,2,3,4-tetrahydro-naphthalen-1-yl]-urea
—— 1-{5-tert-butyl-2-[3-(2-hydroxy-ethylsulfanyl)-phenyl]-2H-pyrazol-3-yl}-3-[(1S,4R)-4-(3-piperidin-1-yl-[1,2,4]triazolo[4,3-a]pyridin-6-yloxy)-1,2,3,4-tetrahydro-naphthalen-1-yl]-urea 1443240-23-0 C37H44N8O3S
1-{5-tert-butyl-2-[3-(2-hydroxy-ethylsulfanyl)-phenyl]-2H-pyrazol-3-yl}-3-[(1S,4R)-4-(3-piperidin-1-yl-[1,2,4]triazolo[4,3-a]pyridin-6-yloxy)-1,2,3,4-tetrahydro-naphthalen-1-yl]-urea
—— 3-(4-methoxyphenyl)-4-piperidin-1-yl-1H-1,2,4-triazole-5-thione 1254359-28-8 C14H18N4OS
3-(4-methoxyphenyl)-4-piperidin-1-yl-1H-1,2,4-triazole-5-thione
—— 1-[5-tert-butyl-2-(4-chloromethyl-phenyl)-2H-pyrazol-3-yl]-3-[(1S,4R)-4-(3-piperidin-1-yl-[1,2,4]triazolo[4,3-a]pyridin-6-yloxy)-1,2,3,4-tetrahydro-naphthalen-1-yl]-urea 1443245-55-3 C36H41ClN8O2
1-[5-tert-butyl-2-(4-chloromethyl-phenyl)-2H-pyrazol-3-yl]-3-[(1S,4R)-4-(3-piperidin-1-yl-[1,2,4]triazolo[4,3-a]pyridin-6-yloxy)-1,2,3,4-tetrahydro-naphthalen-1-yl]-urea
—— 3-(4-chloro-3-hydroxyphenyl)-N-(2-(2,6-dimethylmorpholino)ethyl)-4-(pyridin-4-yl)-1H-pyrazole-1-carboxamide 1352811-01-8 C23H26ClN5O3
3-(4-chloro-3-hydroxyphenyl)-N-(2-(2,6-dimethylmorpholino)ethyl)-4-(pyridin-4-yl)-1H-pyrazole-1-carboxamide
—— 1-{5-tert-butyl-2-[4-(4-methyl-piperazin-1-ylmethyl)-phenyl]-2H-pyrazol-3-yl}-3-[(1S,4R)-4-(3-piperidin-1-yl-[1,2,4]triazolo[4,3-a]pyridin-6-yloxy)-1,2,3,4-tetrahydro-naphthalen-1-yl]-urea 1443240-99-0 C41H52N10O2
1-{5-tert-butyl-2-[4-(4-methyl-piperazin-1-ylmethyl)-phenyl]-2H-pyrazol-3-yl}-3-[(1S,4R)-4-(3-piperidin-1-yl-[1,2,4]triazolo[4,3-a]pyridin-6-yloxy)-1,2,3,4-tetrahydro-naphthalen-1-yl]-urea
—— 3-(4-chloro-3-methoxyphenyl)-N-(2-(dimethylamino)-ethyl)-4-(pyridin-4-yl)-1H-pyrazole-1-carboxamide 1352810-89-9 C20H22ClN5O2
3-(4-chloro-3-methoxyphenyl)-N-(2-(dimethylamino)-ethyl)-4-(pyridin-4-yl)-1H-pyrazole-1-carboxamide
—— 3-(5-tert-butyl-1,3,4-oxadiazol-2-yl)-5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-N-(piperidin-1-yl)-1H-pyrazoIe-4-carboxamide 1161827-18-4 C27H27Cl3N6O2
3-(5-tert-butyl-1,3,4-oxadiazol-2-yl)-5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-N-(piperidin-1-yl)-1H-pyrazoIe-4-carboxamide
—— 2-amino-5-N-morpholyl-4-phenylthiazole 446065-21-0 C13H15N3OS
2-amino-5-N-morpholyl-4-phenylthiazole
—— 3-(4-chloro-3-hydroxyphenyl)-N-(2-(diethylamino)ethyl)-4-(pyridin-4-yl)-1H-pyrazole-1-carboxamide 1352810-99-1 C21H24ClN5O2
3-(4-chloro-3-hydroxyphenyl)-N-(2-(diethylamino)ethyl)-4-(pyridin-4-yl)-1H-pyrazole-1-carboxamide
—— 1-{4-[3-(4-chloro-3-hydroxyphenyl)-4-(pyridin-4-yl)-1H-pyrazol-1-yl]phenyl}-3-(4-chloro-3-(trifluoromethyl)phenyl)urea 1350473-93-6 C28H18Cl2F3N5O2
1-{4-[3-(4-chloro-3-hydroxyphenyl)-4-(pyridin-4-yl)-1H-pyrazol-1-yl]phenyl}-3-(4-chloro-3-(trifluoromethyl)phenyl)urea
—— N-(4-chloro-3-(oxazolo[4,5-b]pyridin-2-yl)phenyl)piperidine-1-carboxamide 1533398-90-1 C18H17ClN4O2
N-(4-chloro-3-(oxazolo[4,5-b]pyridin-2-yl)phenyl)piperidine-1-carboxamide
—— 1-{4-[3-(4-chloro-3-hydroxyphenyl)-4-(pyridin-4-yl)-1H-pyrazol-1-yl]phenyl}-3-(3,5-bis(trifluoromethyl)phenyl)urea 1350473-95-8 C29H18ClF6N5O2
1-{4-[3-(4-chloro-3-hydroxyphenyl)-4-(pyridin-4-yl)-1H-pyrazol-1-yl]phenyl}-3-(3,5-bis(trifluoromethyl)phenyl)urea
—— 3-(4-chloro-3-hydroxyphenyl)-N-(2-(dimethylamino)ethyl)-4-(pyridin-4-yl)-1H-pyrazole-1-carboxamide 1352810-98-0 C19H20ClN5O2
3-(4-chloro-3-hydroxyphenyl)-N-(2-(dimethylamino)ethyl)-4-(pyridin-4-yl)-1H-pyrazole-1-carboxamide
—— 1-{4-[3-(4-chloro-3-hydroxyphenyl)-4-(pyridin-4-yl)-1H-pyrazol-1-yl]phenyl}-3-(3,4-dichlorophenyl)urea 1350473-90-3 C27H18Cl3N5O2
1-{4-[3-(4-chloro-3-hydroxyphenyl)-4-(pyridin-4-yl)-1H-pyrazol-1-yl]phenyl}-3-(3,4-dichlorophenyl)urea
—— 3-(4-chloro-3-hydroxyphenyl)-N-(2-(4-methylpiperazin-1-yl)ethyl)-4-(pyridin-4-yl)-1H-pyrazole-1-carboxamide 1352811-02-9 C22H25ClN6O2
3-(4-chloro-3-hydroxyphenyl)-N-(2-(4-methylpiperazin-1-yl)ethyl)-4-(pyridin-4-yl)-1H-pyrazole-1-carboxamide
—— 1-{4-[3-(4-chloro-3-methoxyphenyl)-4-(pyridin-4-yl)-1H-pyrazol-1-yl]phenyl}-3-(3,5-bis(trifluoromethyl)phenyl)urea 1350473-80-1 C30H20ClF6N5O2
1-{4-[3-(4-chloro-3-methoxyphenyl)-4-(pyridin-4-yl)-1H-pyrazol-1-yl]phenyl}-3-(3,5-bis(trifluoromethyl)phenyl)urea
—— 1-{4-[3-(4-chloro-3-hydroxyphenyl)-4-(pyridin-4-yl)-1H-pyrazol-1-yl]phenyl}-3-(2,3-dichlorophenyl)urea 1350473-88-9 C27H18Cl3N5O2
1-{4-[3-(4-chloro-3-hydroxyphenyl)-4-(pyridin-4-yl)-1H-pyrazol-1-yl]phenyl}-3-(2,3-dichlorophenyl)urea
—— 9-Benzoyl-2-(3-chlorophenyl)-7,8,9,10-tetrahydro-imidazo[1,2-c]pyrido[3,4-e] pyrimidin-5(6H)-one 141056-87-3 C22H17ClN4O2
9-Benzoyl-2-(3-chlorophenyl)-7,8,9,10-tetrahydro-imidazo[1,2-c]pyrido[3,4-e] pyrimidin-5(6H)-one
—— 3-(4-chloro-3-hydroxyphenyl)-N-(2-morpholinoethyl)-4-(pyridin-4-yl)-1H-pyrazole-1-carboxamide 1352811-00-7 C21H22ClN5O3
3-(4-chloro-3-hydroxyphenyl)-N-(2-morpholinoethyl)-4-(pyridin-4-yl)-1H-pyrazole-1-carboxamide
—— 3-(4-Chloro-3-methoxyphenyl)-N-(2-(2-methylpiperidin-1-yl)ethyl)-4-(pyridin-4-yl)-1H-pyrazole-1-carboxamide 1352810-96-8 C24H28ClN5O2
3-(4-Chloro-3-methoxyphenyl)-N-(2-(2-methylpiperidin-1-yl)ethyl)-4-(pyridin-4-yl)-1H-pyrazole-1-carboxamide
—— 3,5-bis(adamantyl)-1H-pyrazole 125995-71-3 C23H32N2
3,5-bis(adamantyl)-1H-pyrazole
—— 3-(4-chloro-3-methoxyphenyl)-N-(2-morpholinoethyl)-4-(pyridin-4-yl)-1H-pyrazole-1-carboxamide 1352810-91-3 C22H24ClN5O3
3-(4-chloro-3-methoxyphenyl)-N-(2-morpholinoethyl)-4-(pyridin-4-yl)-1H-pyrazole-1-carboxamide
—— N-(2-(4-acetylpiperazin-1-yl)ethyl)-3-(4-chloro-3-methoxyphenyl)-4-(pyridin-4-yl)-1H-pyrazole-1-carboxamide 1352810-94-6 C24H27ClN6O3
N-(2-(4-acetylpiperazin-1-yl)ethyl)-3-(4-chloro-3-methoxyphenyl)-4-(pyridin-4-yl)-1H-pyrazole-1-carboxamide
—— 3-(4-chloro-3-methoxyphenyl)-4-(pyridin-4-yl)-N-(2-(pyrrolidin-1-yl)ethyl)-1H-pyrazole-1-carboxamide 1352810-97-9 C22H24ClN5O2
3-(4-chloro-3-methoxyphenyl)-4-(pyridin-4-yl)-N-(2-(pyrrolidin-1-yl)ethyl)-1H-pyrazole-1-carboxamide