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中文名称 英文名称 CAS号 化学式 结构式图片
—— 4-{8-amino-3-[(6R,8aS)-3-oxooctahydroindolizin-6-yl]imidazo[1,5-a]pyrazin-1-yl}-3-cyano-N-[4-(trifluoromethyl)pyridin-2-yl]benzamide 1620674-42-1 C28H23F3N8O2
4-{8-amino-3-[(6R,8aS)-3-oxooctahydroindolizin-6-yl]imidazo[1,5-a]pyrazin-1-yl}-3-cyano-N-[4-(trifluoromethyl)pyridin-2-yl]benzamide
—— 1-(8-amino-1-(4-(4-(trifluoromethyl)pyridin-2-ylcarbamoyl)phenyl)imidazo[1,5-a]pyrazin-3-yl)-N-isopropylpiperidine-3-carboxamide 1419216-30-0 C28H29F3N8O2
1-(8-amino-1-(4-(4-(trifluoromethyl)pyridin-2-ylcarbamoyl)phenyl)imidazo[1,5-a]pyrazin-3-yl)-N-isopropylpiperidine-3-carboxamide
—— di-(1(2)<i>H</i>-pyrazol-3-yl)-methane 101861-32-9 C7H8N4
di-(1(2)<i>H</i>-pyrazol-3-yl)-methane
—— 4-{8-amino-3-[(7R,9aS)-4-oxooctahydropyrido[2,1-c][1,4]oxazin-7-yl]imidazo[1,5-a]pyrazin-1-yl}-3-fluoro-N-[4-(trifluoromethyl)pyridin-2-yl]benzamide 1620673-47-3 C27H23F4N7O3
4-{8-amino-3-[(7R,9aS)-4-oxooctahydropyrido[2,1-c][1,4]oxazin-7-yl]imidazo[1,5-a]pyrazin-1-yl}-3-fluoro-N-[4-(trifluoromethyl)pyridin-2-yl]benzamide
—— (R)-1-bromo-3-(4-(difluoromethoxy)-3-methylphenyl)-6-methyl-5,6,8,9-tetrahydroimidazo[1,5-d][1,4]oxazepine 1623767-13-4 C16H17BrF2N2O2
(R)-1-bromo-3-(4-(difluoromethoxy)-3-methylphenyl)-6-methyl-5,6,8,9-tetrahydroimidazo[1,5-d][1,4]oxazepine
—— 4-{8-amino-3-[(6R,8aS)-3-oxooctahydroindolizin-6-yl]imidazo[1,5-a]pyrazin-1-yl}-3-(cyclopropyloxy)-N-[4-(trifluoromethyl)pyridin-2-yl]benzamide 1620674-40-9 C30H28F3N7O3
4-{8-amino-3-[(6R,8aS)-3-oxooctahydroindolizin-6-yl]imidazo[1,5-a]pyrazin-1-yl}-3-(cyclopropyloxy)-N-[4-(trifluoromethyl)pyridin-2-yl]benzamide
—— ethyl 1-(3-fluorophenyl)-1H-pyrazole-4-carboxylate 138907-75-2 C12H11FN2O2
ethyl 1-(3-fluorophenyl)-1H-pyrazole-4-carboxylate
—— 4-{8-amino-3-[(6R,8aS)-3-oxooctahydroindolizin-6-yl]imidazo[1,5-a]pyrazin-1-yl}-3-(1,1-difluoroethyl)-N-[4-(trifluoromethyl)pyridin-2-yl]benzamide 1620674-33-0 C29H26F5N7O2
4-{8-amino-3-[(6R,8aS)-3-oxooctahydroindolizin-6-yl]imidazo[1,5-a]pyrazin-1-yl}-3-(1,1-difluoroethyl)-N-[4-(trifluoromethyl)pyridin-2-yl]benzamide
—— (R)-1-bromo-3-(3-methoxy-4-(trifluoromethyl)phenyl)-6-methyl-5,6,8,9-tetrahydroimidazo[1,5-d][1,4]oxazepine 1623767-01-0 C16H16BrF3N2O2
(R)-1-bromo-3-(3-methoxy-4-(trifluoromethyl)phenyl)-6-methyl-5,6,8,9-tetrahydroimidazo[1,5-d][1,4]oxazepine
—— (R)-1-(2,6-dimethylpyridin-4-yl)-3-(3-methoxy-4-(trifluoromethyl)phenyl)-6-methyl-5,6,8,9-tetrahydroimidazo[1,5-d][1,4]oxazepine 1623763-89-2 C23H24F3N3O2
(R)-1-(2,6-dimethylpyridin-4-yl)-3-(3-methoxy-4-(trifluoromethyl)phenyl)-6-methyl-5,6,8,9-tetrahydroimidazo[1,5-d][1,4]oxazepine
—— methyl 1-(8-amino-1-(4-(4-(trifluoromethyl)pyridin-2-ylcarbamoyl)phenyl)imidazo[1,5-a]pyrazin-3-yl)piperidine-3-carboxylate 1419222-77-7 C26H24F3N7O3
methyl 1-(8-amino-1-(4-(4-(trifluoromethyl)pyridin-2-ylcarbamoyl)phenyl)imidazo[1,5-a]pyrazin-3-yl)piperidine-3-carboxylate
—— 4-{8-amino-3-[(6R,8aS)-3-oxooctahydroindolizin-6-yl]imidazo[1,5-a]pyrazin-1-yl}-N-1-[4-(trifluoromethyl)pyridin-2-yl]benzene-1,3-dicarboxamide 1620674-43-2 C28H25F3N8O3
4-{8-amino-3-[(6R,8aS)-3-oxooctahydroindolizin-6-yl]imidazo[1,5-a]pyrazin-1-yl}-N-1-[4-(trifluoromethyl)pyridin-2-yl]benzene-1,3-dicarboxamide
—— 4-{8-amino-3-[(6R,8aS)-3-oxooctahydroindolizin-6-yl]imidazo[1,5-a]pyrazin-1-yl}-3-(difluoromethoxy)-N-[4-(trifluoromethyl)pyridin-2-yl]benzamide 1620673-91-7 C28H24F5N7O3
4-{8-amino-3-[(6R,8aS)-3-oxooctahydroindolizin-6-yl]imidazo[1,5-a]pyrazin-1-yl}-3-(difluoromethoxy)-N-[4-(trifluoromethyl)pyridin-2-yl]benzamide
—— 4-{8-amino-3-[(6R,8aS)-3-oxooctahydroindolizin-6-yl]imidazo[1,5-a]pyrazin-1-yl}-3-(1-methylethoxy)-N-[4-(trifluoromethyl)pyridin-2-yl]benzamide 1620674-58-9 C30H30F3N7O3
4-{8-amino-3-[(6R,8aS)-3-oxooctahydroindolizin-6-yl]imidazo[1,5-a]pyrazin-1-yl}-3-(1-methylethoxy)-N-[4-(trifluoromethyl)pyridin-2-yl]benzamide
—— 4-{8-amino-3-[(6R,8aS)-3-oxooctahydroindolizin-6-yl]imidazo[1,5-a]pyrazin-1-yl}-3-fluoro-N-[4-(trifluoromethyl)pyridin-2-yl]benzamide 1620673-30-4 C27H23F4N7O2
4-{8-amino-3-[(6R,8aS)-3-oxooctahydroindolizin-6-yl]imidazo[1,5-a]pyrazin-1-yl}-3-fluoro-N-[4-(trifluoromethyl)pyridin-2-yl]benzamide
—— 2-{8-amino-3-[(6R,8aS)-3-oxooctahydroindolizin-6-yl]imidazo[1,5-a]pyrazin-1-yl}-5-{[4-(trifluoromethyl)pyridin-2-yl]carbamoyl}benzoic acid 1620674-46-5 C28H24F3N7O4
2-{8-amino-3-[(6R,8aS)-3-oxooctahydroindolizin-6-yl]imidazo[1,5-a]pyrazin-1-yl}-5-{[4-(trifluoromethyl)pyridin-2-yl]carbamoyl}benzoic acid
—— 4-{8-amino-3-[(3R,8aR)-6-oxohexahydro-1H-pyrrolo[2,1-c][1,4]oxazin-3-yl]imidazo[1,5-a]pyrazin-1-yl}-N-[4-(trifluoromethyl)pyridin-2-yl]benzamide 1620674-26-1 C26H22F3N7O3
4-{8-amino-3-[(3R,8aR)-6-oxohexahydro-1H-pyrrolo[2,1-c][1,4]oxazin-3-yl]imidazo[1,5-a]pyrazin-1-yl}-N-[4-(trifluoromethyl)pyridin-2-yl]benzamide
—— N-{[4-cyano-2-(trifluoromethyl)phenyl]methyl}-2-(4-{4-methyl-5-[2-(trifluoromethyl)phenyl]-4H-1,2,4-triazol-3-yl}bicyclo[2.2.2]oct-1-yl)acetamide 1206686-99-8 C28H28F6N4O
N-{[4-cyano-2-(trifluoromethyl)phenyl]methyl}-2-(4-{4-methyl-5-[2-(trifluoromethyl)phenyl]-4H-1,2,4-triazol-3-yl}bicyclo[2.2.2]oct-1-yl)acetamide
—— (1Z)-2-[3-(5-chlorothiophen-2-yl)-4-(2-fluorobenzyl)-5-oxo-4,5-dihydro-1H-1,2,4-triazol-1-yl]-N'-hydroxyethaneimidamide 1332647-58-1 C15H13ClFN5O2S
(1Z)-2-[3-(5-chlorothiophen-2-yl)-4-(2-fluorobenzyl)-5-oxo-4,5-dihydro-1H-1,2,4-triazol-1-yl]-N'-hydroxyethaneimidamide
—— N-(4-fluorophenyl)-2-phenyl-5,6,7,8-tetrahydroimidazo[1,2-a]pyrazin-3-amine 1261117-43-4 C18H17FN4
N-(4-fluorophenyl)-2-phenyl-5,6,7,8-tetrahydroimidazo[1,2-a]pyrazin-3-amine
—— N-(4-(4-chloro-1H-imidazol-1-yl)-3-methoxyphenyl)-2-(3-(trifluoromethyl)phenyl)acetamide 1555543-61-7 C19H15ClF3N3O2
N-(4-(4-chloro-1H-imidazol-1-yl)-3-methoxyphenyl)-2-(3-(trifluoromethyl)phenyl)acetamide
—— 3-Methyl-4-[3-(trifluoromethyl)phenyl]-1H-pyrazol-5-amine 851975-08-1 C11H10F3N3
3-Methyl-4-[3-(trifluoromethyl)phenyl]-1H-pyrazol-5-amine
—— (R)-1-bromo-3-(3-methoxy-4-(trifluoromethoxy)phenyl)-6-methyl-5,6,8,9-tetrahydroimidazo[1,5-d][1,4]oxazepine 1623767-29-2 C16H16BrF3N2O3
(R)-1-bromo-3-(3-methoxy-4-(trifluoromethoxy)phenyl)-6-methyl-5,6,8,9-tetrahydroimidazo[1,5-d][1,4]oxazepine
—— (R)-3-(3-chloro-4-isopropoxyphenyl)-1-(2,6-dimethylpyridin-4-yl)-6-methyl-5,6,8,9-tetrahydroimidazo[1,5-d][1,4]oxazepine 1623764-17-9 C24H28ClN3O2
(R)-3-(3-chloro-4-isopropoxyphenyl)-1-(2,6-dimethylpyridin-4-yl)-6-methyl-5,6,8,9-tetrahydroimidazo[1,5-d][1,4]oxazepine
—— N-(tetrahydro-2H-pyran-4-yl)-3-(3-(trifluoromethyl)phenyl)pyrazolo[1,5-a]pyrimidin-5-amine 1361951-40-7 C18H17F3N4O
N-(tetrahydro-2H-pyran-4-yl)-3-(3-(trifluoromethyl)phenyl)pyrazolo[1,5-a]pyrimidin-5-amine
—— (R)-3-(3-chloro-4-methoxyphenyl)-1-(2,6-dimethylpyridin-4-yl)-6-methyl-5,6,8,9-tetrahydroimidazo[1,5-d][1,4]oxazepine 1623764-15-7 C22H24ClN3O2
(R)-3-(3-chloro-4-methoxyphenyl)-1-(2,6-dimethylpyridin-4-yl)-6-methyl-5,6,8,9-tetrahydroimidazo[1,5-d][1,4]oxazepine
—— (R)-(4-(3-(4-chloro-3-methoxyphenyl)-6-methyl-5,6,8,9-tetrahydroimidazo[1,5-d][1,4]oxazepin-1-yl)-6-methylpyridin-2-yl)methanol 1623767-10-1 C22H24ClN3O3
(R)-(4-(3-(4-chloro-3-methoxyphenyl)-6-methyl-5,6,8,9-tetrahydroimidazo[1,5-d][1,4]oxazepin-1-yl)-6-methylpyridin-2-yl)methanol
—— (R)-3-(4-chloro-3-methoxyphenyl)-1-(2-(fluoromethyl)-6-methylpyridin-4-yl)-6-methyl-5,6,8,9-tetrahydroimidazo[1,5-d][1,4]oxazepine 1623763-95-0 C22H23ClFN3O2
(R)-3-(4-chloro-3-methoxyphenyl)-1-(2-(fluoromethyl)-6-methylpyridin-4-yl)-6-methyl-5,6,8,9-tetrahydroimidazo[1,5-d][1,4]oxazepine
—— (R)-3-(4-chloro-3-methoxyphenyl)-1-(2,6-dimethylpyridin-4-yl)-6-methyl-5,6,8,9-tetrahydroimidazo[1,5-d][1,4]oxazepine 1623763-83-6 C22H24ClN3O2
(R)-3-(4-chloro-3-methoxyphenyl)-1-(2,6-dimethylpyridin-4-yl)-6-methyl-5,6,8,9-tetrahydroimidazo[1,5-d][1,4]oxazepine
—— (R)-4-(3-(4-chloro-3-methoxyphenyl)-6-methyl-5,6,8,9-tetrahydroimidazo[1,5-d][1,4]oxazepin-1-yl)-2,6-dimethylpyridine 1-oxide 1623767-11-2 C22H24ClN3O3
(R)-4-(3-(4-chloro-3-methoxyphenyl)-6-methyl-5,6,8,9-tetrahydroimidazo[1,5-d][1,4]oxazepin-1-yl)-2,6-dimethylpyridine 1-oxide
—— (R)-1-bromo-3-(3-chloro-4-(methoxymethoxy)phenyl)-6-methyl-5,6,8,9-tetrahydroimidazo[1,5-d][1,4]oxazepine 1623767-38-3 C16H18BrClN2O3
(R)-1-bromo-3-(3-chloro-4-(methoxymethoxy)phenyl)-6-methyl-5,6,8,9-tetrahydroimidazo[1,5-d][1,4]oxazepine
—— (R)-3-(4-(difluoromethoxy)-3-methylphenyl)-1-(2,6-dimethylpyridin-4-yl)-6-methyl-5,6,8,9-tetrahydroimidazo[1,5-d][1,4]oxazepine 1623763-96-1 C23H25F2N3O2
(R)-3-(4-(difluoromethoxy)-3-methylphenyl)-1-(2,6-dimethylpyridin-4-yl)-6-methyl-5,6,8,9-tetrahydroimidazo[1,5-d][1,4]oxazepine
—— (R)-3-(3-methoxy-4-(trifluoromethoxy)phenyl)-6-methyl-1-(2-methylpyridin-4-yl)-5,6,8,9-tetrahydroimidazo[1,5-d][1,4]oxazepine 1623764-06-6 C22H22F3N3O3
(R)-3-(3-methoxy-4-(trifluoromethoxy)phenyl)-6-methyl-1-(2-methylpyridin-4-yl)-5,6,8,9-tetrahydroimidazo[1,5-d][1,4]oxazepine
—— (R)-3-(3-chloro-4-(methoxymethoxy)phenyl)-1-(2,6-dimethylpyridin-4-yl)-6-methyl-5,6,8,9-tetrahydroimidazo[1,5-d][1,4]oxazepine 1623767-39-4 C23H26ClN3O3
(R)-3-(3-chloro-4-(methoxymethoxy)phenyl)-1-(2,6-dimethylpyridin-4-yl)-6-methyl-5,6,8,9-tetrahydroimidazo[1,5-d][1,4]oxazepine
—— 1-isopropyl-1H-pyrazole-3-carbonyl chloride 1435244-63-5 C7H9ClN2O
1-isopropyl-1H-pyrazole-3-carbonyl chloride
—— 2-(1-isopropyl-1H-pyrazol-3-yl)acetic acid 1260658-97-6 C8H12N2O2
2-(1-isopropyl-1H-pyrazol-3-yl)acetic acid
—— 4-chloro-1-isopropyl-1H-pyrazole-3-carboxylic acid 1006493-69-1 C7H9ClN2O2
4-chloro-1-isopropyl-1H-pyrazole-3-carboxylic acid
—— methyl 1-(propan-2-yl)-1H-pyrazole-5-carboxylate 1006319-17-0 C8H12N2O2
methyl 1-(propan-2-yl)-1H-pyrazole-5-carboxylate
—— N-(4-fluorophenyl)-2-(4-methylphenyl)-5,6,7,8-tetrahydroimidazo[1,2-a]pyrazin-3-amine 1261117-56-9 C19H19FN4
N-(4-fluorophenyl)-2-(4-methylphenyl)-5,6,7,8-tetrahydroimidazo[1,2-a]pyrazin-3-amine
—— 1-(4-cyanophenyl)-5-(3,6-dimethyl-2,4-dioxo-1-(3-(trifluoromethyl)phenyl)-1,2,3,4-tetrahydropyrimidin-5-yl)-1H-pyrazole-4-carboxylic acid methyl ester 1421963-13-4 C25H18F3N5O4
1-(4-cyanophenyl)-5-(3,6-dimethyl-2,4-dioxo-1-(3-(trifluoromethyl)phenyl)-1,2,3,4-tetrahydropyrimidin-5-yl)-1H-pyrazole-4-carboxylic acid methyl ester
—— methyl N-[[5-[3-(2,4-dimethoxyphenyl)-1H-pyrazol-1-yl]-2-methylphenyl]methyl]carbamate 1604808-15-2 C21H23N3O4
methyl N-[[5-[3-(2,4-dimethoxyphenyl)-1H-pyrazol-1-yl]-2-methylphenyl]methyl]carbamate
—— 2-(2-fluorophenyl)-N-(4-fluorophenyl)-5,6,7,8-tetrahydroimidazo[1,2-a]pyrazin-3-amine 1261117-42-3 C18H16F2N4
2-(2-fluorophenyl)-N-(4-fluorophenyl)-5,6,7,8-tetrahydroimidazo[1,2-a]pyrazin-3-amine
—— 2-(4-chlorophenyl)-N-(4-fluorophenyl)imidazo[1,2-a]pyrazin-3-amine 1286677-25-5 C18H12ClFN4
2-(4-chlorophenyl)-N-(4-fluorophenyl)imidazo[1,2-a]pyrazin-3-amine
—— 2-(4-chlorophenyl)-N-(4-fluorophenyl)-5,6,7,8-tetrahydroimidazo[1,2-a]pyrazin-3-amine 1261117-59-2 C18H16ClFN4
2-(4-chlorophenyl)-N-(4-fluorophenyl)-5,6,7,8-tetrahydroimidazo[1,2-a]pyrazin-3-amine
—— 3-amino-1-(2-(4-fluorophenyl)-3-(4-fluorophenylamino)-5,6-dihydroimidazo[1,2-a]pyrazin-7(8H)-yl)propan-1-one 1261110-20-6 C21H21F2N5O
3-amino-1-(2-(4-fluorophenyl)-3-(4-fluorophenylamino)-5,6-dihydroimidazo[1,2-a]pyrazin-7(8H)-yl)propan-1-one
—— 4-(5-phenylpentyl)-1H-imidazol-2-amine hydrochloride —— C14H19N3*(x)ClH
4-(5-phenylpentyl)-1H-imidazol-2-amine hydrochloride
—— 2-(6-bromoquinolin-3-yl)-N-(4-fluorophenyl)-6-(5-p-tolyl-1H-imidazol-2-yl)imidazo[1,2-a]pyridin-3-amine 1297399-20-2 C32H22BrFN6
2-(6-bromoquinolin-3-yl)-N-(4-fluorophenyl)-6-(5-p-tolyl-1H-imidazol-2-yl)imidazo[1,2-a]pyridin-3-amine
—— N-(4-fluorophenyl)-2-(4-methoxyphenyl)-5,6,7,8-tetrahydroimidazo[1,2-a]pyrazin-3-amine 1261117-57-0 C19H19FN4O
N-(4-fluorophenyl)-2-(4-methoxyphenyl)-5,6,7,8-tetrahydroimidazo[1,2-a]pyrazin-3-amine
—— 2-(3-fluorophenyl)-N-(4-fluorophenyl)-5H,6H,7H,8H-imidazo[1,2-a]pyrazin-3-amine 1261111-77-6 C18H16F2N4
2-(3-fluorophenyl)-N-(4-fluorophenyl)-5H,6H,7H,8H-imidazo[1,2-a]pyrazin-3-amine
—— 2-(6-bromoquinolin-3-yl)-N-(4-fluorophenyl)-6-(5-(4-fluorophenyl)-1H-imidazol-2-yl)imidazo[1,2-a]pyridin-3-amine 1297399-19-9 C31H19BrF2N6
2-(6-bromoquinolin-3-yl)-N-(4-fluorophenyl)-6-(5-(4-fluorophenyl)-1H-imidazol-2-yl)imidazo[1,2-a]pyridin-3-amine