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中文名称 英文名称 CAS号 化学式 结构式图片
—— N-[2-(3-{1-ethyl-4-formyl-5-[4-(trifluoromethyl)phenoxy]-1H-pyrazol-3-yl}phenyl)propan-2-yl]-2,2,2-trifluoroethanesulfonamide 1289202-93-2 C24H23F6N3O4S
N-[2-(3-{1-ethyl-4-formyl-5-[4-(trifluoromethyl)phenoxy]-1H-pyrazol-3-yl}phenyl)propan-2-yl]-2,2,2-trifluoroethanesulfonamide
—— N-[2-(3-{4-bromo-1-ethyl-3-[4-(trifluoromethyl)phenoxy]-1H-pyrazol-5-yl}phenyl)propan-2-yl]-2,2,2-trifluoroethanesulfonamide 1289202-89-6 C23H22BrF6N3O3S
N-[2-(3-{4-bromo-1-ethyl-3-[4-(trifluoromethyl)phenoxy]-1H-pyrazol-5-yl}phenyl)propan-2-yl]-2,2,2-trifluoroethanesulfonamide
—— (4R)-4-(2-chloro-2,2-difluoroethyl)-1-{[2-(hydroxymethyl)-6-(trifluoromethyl)imidazo[2,1-b][1,3,4]thiadiazol-5-yl]methyl}pyrrolidin-2-one 1294000-63-7 C13H12ClF5N4O2S
(4R)-4-(2-chloro-2,2-difluoroethyl)-1-{[2-(hydroxymethyl)-6-(trifluoromethyl)imidazo[2,1-b][1,3,4]thiadiazol-5-yl]methyl}pyrrolidin-2-one
—— (4R)-4-(2-chloro-2,2-difluoroethyl)-1-{[2-{[((2)H3)methyloxy]methyl}-6-(trifluoromethyl)imidazo[2,1-b][1,3,4]thiadiazol-5-yl]methyl}pyrrolidin-2-one 1294000-80-8 C14H14ClF5N4O2S
(4R)-4-(2-chloro-2,2-difluoroethyl)-1-{[2-{[((2)H3)methyloxy]methyl}-6-(trifluoromethyl)imidazo[2,1-b][1,3,4]thiadiazol-5-yl]methyl}pyrrolidin-2-one
—— N-[2-(3-{1-ethyl-4-(phenylethynyl)-5-[4-(trifluoromethyl)phenoxy]-1H-pyrazol-3-yl}phenyl)propan-2-yl]-2,2,2-trifluoroethanesulfonamide 1289202-94-3 C31H27F6N3O3S
N-[2-(3-{1-ethyl-4-(phenylethynyl)-5-[4-(trifluoromethyl)phenoxy]-1H-pyrazol-3-yl}phenyl)propan-2-yl]-2,2,2-trifluoroethanesulfonamide
—— N-[1-(3-{1-ethyl-5-[4-(trifluoromethyl)phenoxy]-1H-pyrazol-3-yl}phenyl)-1-methylethyl]-2,2,2-trifluoroethanesulfonamide 1289201-64-4 C23H23F6N3O3S
N-[1-(3-{1-ethyl-5-[4-(trifluoromethyl)phenoxy]-1H-pyrazol-3-yl}phenyl)-1-methylethyl]-2,2,2-trifluoroethanesulfonamide
—— (Z)-5-(diethylamino)-3-ethyl-N'-hydroxy-1-(4-hydroxyphenyl)-1H-pyrazole-4-carboximidamide 1290137-84-6 C16H23N5O2
(Z)-5-(diethylamino)-3-ethyl-N'-hydroxy-1-(4-hydroxyphenyl)-1H-pyrazole-4-carboximidamide
—— 1,3-bis-(2'-diisopropylphosphinoethyl)triazolium bromide 1315562-47-0 Br*C18H38N3P2
1,3-bis-(2'-diisopropylphosphinoethyl)triazolium bromide
—— 2-(2-amino-4-(2,4-dibromophenyl)thiazol-5-ylthio)-N-(2-chloropyridin-3-yl)acetamide 1260403-04-0 C16H11Br2ClN4OS2
2-(2-amino-4-(2,4-dibromophenyl)thiazol-5-ylthio)-N-(2-chloropyridin-3-yl)acetamide
—— N-[2-(3-{4-cyano-1-ethyl-5-[4-(trifluoromethyl)phenoxy]-1H-pyrazol-3-yl}phenyl)propan-2-yl]-2,2,2-trifluoroethanesulfonamide 1289202-92-1 C24H22F6N4O3S
N-[2-(3-{4-cyano-1-ethyl-5-[4-(trifluoromethyl)phenoxy]-1H-pyrazol-3-yl}phenyl)propan-2-yl]-2,2,2-trifluoroethanesulfonamide
—— 2-(2-chloro-4-(2,4-dibromophenyl)thiazol-5-ylthio)-N-(2-chloropyridin-3-yl)acetamide 1260403-14-2 C16H9Br2Cl2N3OS2
2-(2-chloro-4-(2,4-dibromophenyl)thiazol-5-ylthio)-N-(2-chloropyridin-3-yl)acetamide
—— 4-[5-{[4-fluoro-2-(2H-1,2,3-triazol-2-yl)phenyl]carbonyl}hexahydropyrrolo[3,4-c]pyrrol-2(1H)-yl]-6-methoxy-N,N-dimethylpyrimidin-2-amine 1293280-50-8 C22H25FN8O2
4-[5-{[4-fluoro-2-(2H-1,2,3-triazol-2-yl)phenyl]carbonyl}hexahydropyrrolo[3,4-c]pyrrol-2(1H)-yl]-6-methoxy-N,N-dimethylpyrimidin-2-amine
—— 4-[5-{[5-fluoro-2-(2H-1,2,3-triazol-2-yl)phenyl]carbonyl}hexahydropyrrolo[3,4-c]pyrrol-2(1H)-yl]-6-methoxy-N ,N-dimethylpyrimidin-2-amine 1293304-79-6 C22H25FN8O2
4-[5-{[5-fluoro-2-(2H-1,2,3-triazol-2-yl)phenyl]carbonyl}hexahydropyrrolo[3,4-c]pyrrol-2(1H)-yl]-6-methoxy-N ,N-dimethylpyrimidin-2-amine
—— 6-[5-{[5-fluoro-2-(2H-1 ,2,3-triazol-2-yl)phenyl]carbonyl}hexahydropyrrolo[3,4-c]pyrrol-2(1H)-yl]-N,N-dimethyl-2-(trifluoromethyl)pyrimidin-4-amine 1293280-47-3 C22H22F4N8O
6-[5-{[5-fluoro-2-(2H-1 ,2,3-triazol-2-yl)phenyl]carbonyl}hexahydropyrrolo[3,4-c]pyrrol-2(1H)-yl]-N,N-dimethyl-2-(trifluoromethyl)pyrimidin-4-amine
—— 6-[5-{[4-fluoro-2-(2H-1,2,3-triazol-2-yl)phenyl]carbonyl}hexahydropyrrolo[3,4-c]pyrrol-2(1H)-yl]-N,N-dimethyl-2-(trifluoromethyl)pyrimidin-4-amine 1293280-49-5 C22H22F4N8O
6-[5-{[4-fluoro-2-(2H-1,2,3-triazol-2-yl)phenyl]carbonyl}hexahydropyrrolo[3,4-c]pyrrol-2(1H)-yl]-N,N-dimethyl-2-(trifluoromethyl)pyrimidin-4-amine
—— 1-(2-fluoro-4-methyl-5-(2,2,2-trifluoroethylthio)phenyl)-5-(2-nitrophenyl)-3-(trifluoromethyl)-1H-1,2,4-triazole 1293293-79-4 C18H11F7N4O2S
1-(2-fluoro-4-methyl-5-(2,2,2-trifluoroethylthio)phenyl)-5-(2-nitrophenyl)-3-(trifluoromethyl)-1H-1,2,4-triazole
—— methyl 2-(4-chlorophenyl)-9-(2-methoxyethyl)-9H-imidazo[1,2-a]benzoimidazole-6-carboxylate 1266162-66-6 C20H18ClN3O3
methyl 2-(4-chlorophenyl)-9-(2-methoxyethyl)-9H-imidazo[1,2-a]benzoimidazole-6-carboxylate
—— 2-(1-(2-fluoro-4-methyl-5-(2,2,2-trifluoroethylthio)phenyl)-3-(trifluoromethyl)-1H-1,2,4-triazol-5-yl)aniline 1293293-80-7 C18H13F7N4S
2-(1-(2-fluoro-4-methyl-5-(2,2,2-trifluoroethylthio)phenyl)-3-(trifluoromethyl)-1H-1,2,4-triazol-5-yl)aniline
—— (R)-2-(N-(5-(5-(3-cyano-4-isopropoxyphenyl)-1,2,4-oxadiazol-3-yl)-1,2,3,4-tetrahydronaphthalen-1-yl)sulfamoyl)-N,N-dimethylacetamide 1307230-27-8 C26H29N5O5S
(R)-2-(N-(5-(5-(3-cyano-4-isopropoxyphenyl)-1,2,4-oxadiazol-3-yl)-1,2,3,4-tetrahydronaphthalen-1-yl)sulfamoyl)-N,N-dimethylacetamide
—— N-(5-(tert-butyl-D9)isoxazol-3-yl)-N'-{4-[7-(2-morpholin-4-yl-ethoxy)imidazo[2,1-b][1,3]benzothiazol-2-yl]phenyl}urea 1300734-21-7 C29H32N6O4S
N-(5-(tert-butyl-D9)isoxazol-3-yl)-N'-{4-[7-(2-morpholin-4-yl-ethoxy)imidazo[2,1-b][1,3]benzothiazol-2-yl]phenyl}urea
—— 5-chloro-3-(1H-imidazol-5-yl)benzene-1,2-diol 1300729-48-9 C9H7ClN2O2
5-chloro-3-(1H-imidazol-5-yl)benzene-1,2-diol
—— N-(3-(2-fluoropropan-2-yl)isoxazol-5-yl)-N'-{4-[7-(2-morpholin-4-yl-ethoxy)imidazo[2,1-b][1,3]benzothiazol-2-yl]phenyl}urea 1300733-71-4 C28H29FN6O4S
N-(3-(2-fluoropropan-2-yl)isoxazol-5-yl)-N'-{4-[7-(2-morpholin-4-yl-ethoxy)imidazo[2,1-b][1,3]benzothiazol-2-yl]phenyl}urea
—— 7-(5-fluoro-2-methyl-4-(1H-1,2,4-triazol-3-yl)phenyl)-1-isopropyl-3,4-dihydropyrazino[2,3-b]pyrazin-2(1H)-one 1228012-60-9 C18H18FN7O
7-(5-fluoro-2-methyl-4-(1H-1,2,4-triazol-3-yl)phenyl)-1-isopropyl-3,4-dihydropyrazino[2,3-b]pyrazin-2(1H)-one
—— 2-methyl-5-trifluoromethyloxazole-4-carboxylic acid {6-[(2-methoxyethyl)(methyl)amino]pyridin-3-yl}amide 1279083-86-1 C15H17F3N4O3
2-methyl-5-trifluoromethyloxazole-4-carboxylic acid {6-[(2-methoxyethyl)(methyl)amino]pyridin-3-yl}amide
—— (2-{4-[5-(3,8-dihydroindeno[1,2-d] [1,2,3]triazol-6-yl)-4-(pyridin-4-yl)-1H-imidazol-2-yl]-phenoxy}-ethyl)-dimethylamine 1251931-66-4 C27H25N7O
(2-{4-[5-(3,8-dihydroindeno[1,2-d] [1,2,3]triazol-6-yl)-4-(pyridin-4-yl)-1H-imidazol-2-yl]-phenoxy}-ethyl)-dimethylamine
—— [4-[(2-chloro-4,4-difluoro-spiro[5H-thieno[2,3-c]pyran-7,4'-piperidine]-1'-yl)methyl]-1-(2-fluorophenyl)pyrazol-3-yl]methanol 1307313-98-9 C22H21ClF3N3O2S
[4-[(2-chloro-4,4-difluoro-spiro[5H-thieno[2,3-c]pyran-7,4'-piperidine]-1'-yl)methyl]-1-(2-fluorophenyl)pyrazol-3-yl]methanol
—— 2-phenyl-5-trifluoromethyloxazole-4-carboxylic acid {6-[(2-methoxyethyl)(methyl)amino]pyridin-3-yl}methylamide 1279083-87-2 C21H21F3N4O3
2-phenyl-5-trifluoromethyloxazole-4-carboxylic acid {6-[(2-methoxyethyl)(methyl)amino]pyridin-3-yl}methylamide
—— (R)-2-(N-(5-(5-(3-cyano-4-isopropoxyphenyl)-1,2,4-oxadiazol-3-yl)-1,2,3,4-tetrahydronaphthalen-1-yl)sulfamoyl)acetic acid 1307230-23-4 C24H24N4O6S
(R)-2-(N-(5-(5-(3-cyano-4-isopropoxyphenyl)-1,2,4-oxadiazol-3-yl)-1,2,3,4-tetrahydronaphthalen-1-yl)sulfamoyl)acetic acid
—— 4-[(4-chlorophenyl)sulfanyl]-1-(E)-2-[(4-chlorophenyl)sulfanyl]-1-phenyl-1-ethenyl-3-phenyl-1H-pyrazole 1191903-84-0 C29H20Cl2N2S2
4-[(4-chlorophenyl)sulfanyl]-1-(E)-2-[(4-chlorophenyl)sulfanyl]-1-phenyl-1-ethenyl-3-phenyl-1H-pyrazole
—— N-(phenymethyl)-N'-[3-(1-phenyl-1H-tetrazol-5-yl-thio)propyl]imidodicarbonic diamide 1254556-26-7 C19H21N7O2S
N-(phenymethyl)-N'-[3-(1-phenyl-1H-tetrazol-5-yl-thio)propyl]imidodicarbonic diamide
—— (2R,3R,4S)-3-acetamido-2-((1R,2R)-1,2-dihydroxy-3-(4-(2-hydroxypropan-2-yl)-1H-1,2,3-triazol-1-yl)propyl)-4-hydroxy-3,4-dihydro-2H-pyran-6-carboxylate 1261081-28-0 C16H24N4O8
(2R,3R,4S)-3-acetamido-2-((1R,2R)-1,2-dihydroxy-3-(4-(2-hydroxypropan-2-yl)-1H-1,2,3-triazol-1-yl)propyl)-4-hydroxy-3,4-dihydro-2H-pyran-6-carboxylate
—— 2-(4-(3-(2-amino-1H-imidazol-4-yl)propyl)-1H-1,2,3-triazol-1-yl)-N-(3-phenylpropyl)acetamide hydrochloride 1192357-98-4 C19H25N7O*ClH
2-(4-(3-(2-amino-1H-imidazol-4-yl)propyl)-1H-1,2,3-triazol-1-yl)-N-(3-phenylpropyl)acetamide hydrochloride
—— (R)-N-(5-(5-(3-cyano-4-isopropoxyphenyl)-1,2,4-oxadiazol-3-yl )-1,2, 3, 4-tetrahydronaphthalen-1-yl)-2-hydroxyethanesulfonamide 1307230-25-6 C24H26N4O5S
(R)-N-(5-(5-(3-cyano-4-isopropoxyphenyl)-1,2,4-oxadiazol-3-yl )-1,2, 3, 4-tetrahydronaphthalen-1-yl)-2-hydroxyethanesulfonamide
—— 2-(4-(3-(2-amino-1H-imidazol-4-yl)propyl)-1H-1,2,3-triazol-1-yl)-N-cyclopentylacetamide 1192370-47-0 C15H23N7O
2-(4-(3-(2-amino-1H-imidazol-4-yl)propyl)-1H-1,2,3-triazol-1-yl)-N-cyclopentylacetamide
—— (S)-N-(4-(5-(3-cyano-4-isopropoxyphenyl)-1,2,4-oxadiazol-3-yl)-2,3-dihydro-1H-inden-1-yl)acetamide 1306761-08-9 C23H22N4O3
(S)-N-(4-(5-(3-cyano-4-isopropoxyphenyl)-1,2,4-oxadiazol-3-yl)-2,3-dihydro-1H-inden-1-yl)acetamide
—— (2R,3R,4S)-3-acetamido-2-((1R,2R)-1,2-dihydroxy-3-(4-phenyl-1H-1,2,3-triazol-1-yl)propyl)-4-hydroxy-3,4-dihydro-2H-pyran-6-carboxylate 1261081-20-2 C19H22N4O7
(2R,3R,4S)-3-acetamido-2-((1R,2R)-1,2-dihydroxy-3-(4-phenyl-1H-1,2,3-triazol-1-yl)propyl)-4-hydroxy-3,4-dihydro-2H-pyran-6-carboxylate
—— 5-[[4-(3-Imidazol-1-ylpropyl)-5-methylsulfanyl-1,2,4-triazol-3-yl]methyl]-3-phenyl-1,2,4-oxadiazole 1257330-63-4 C18H19N7OS
5-[[4-(3-Imidazol-1-ylpropyl)-5-methylsulfanyl-1,2,4-triazol-3-yl]methyl]-3-phenyl-1,2,4-oxadiazole
—— 2-(4-(3-(2-amino-1H-imidazol-4-yl)propyl)-1H-1,2,3-triazol-1-yl)-N-(3-phenylpropyl)acetamide 1192370-54-9 C19H25N7O
2-(4-(3-(2-amino-1H-imidazol-4-yl)propyl)-1H-1,2,3-triazol-1-yl)-N-(3-phenylpropyl)acetamide
—— 1-(4-Methyl-2-(3-(piperidin-1-yl)propylthio)thiazol-5-yl)ethanone 1254304-60-3 C14H22N2OS2
1-(4-Methyl-2-(3-(piperidin-1-yl)propylthio)thiazol-5-yl)ethanone
—— 2-(4-(3-(2-amino-1H-imidazol-4-yl)propyl)-1H-1,2,3-triazol-1-yl)-N-benzylacetamide hydrochloride 1192357-96-2 C17H21N7O*ClH
2-(4-(3-(2-amino-1H-imidazol-4-yl)propyl)-1H-1,2,3-triazol-1-yl)-N-benzylacetamide hydrochloride
—— 5-methyl-2-(3-methylphenyl)-1H-imidazole-4-carboxylic acid 1225511-16-9 C12H12N2O2
5-methyl-2-(3-methylphenyl)-1H-imidazole-4-carboxylic acid
—— 2-(4-(3-(2-amino-1H-imidazol-4-yl)propyl)-1H-1,2,3-triazol-1-yl)-N-benzylacetamide 1192370-52-7 C17H21N7O
2-(4-(3-(2-amino-1H-imidazol-4-yl)propyl)-1H-1,2,3-triazol-1-yl)-N-benzylacetamide
—— (2R,3R,4S)-3-acetamido-2-((1R,2R)-1,2-dihydroxy-3-(4-(2-hydroxyethyl)-1H-1,2,3-triazol-1-yl)propyl)-4-hydroxy-3,4-dihydro-2H-pyran-6-carboxylate 1261081-26-8 C15H22N4O8
(2R,3R,4S)-3-acetamido-2-((1R,2R)-1,2-dihydroxy-3-(4-(2-hydroxyethyl)-1H-1,2,3-triazol-1-yl)propyl)-4-hydroxy-3,4-dihydro-2H-pyran-6-carboxylate
—— N-[4-[4-amino-1-[1-(1-methylpiperidin-4-yl)piperidin-4-yl]pyrazolo[3,4-d]pyrimidin-3-yl]phenyl]-7-chloro-1,3-benzoxazol-2-amine 1253107-58-2 C29H32ClN9O
N-[4-[4-amino-1-[1-(1-methylpiperidin-4-yl)piperidin-4-yl]pyrazolo[3,4-d]pyrimidin-3-yl]phenyl]-7-chloro-1,3-benzoxazol-2-amine
—— 2-(4-(3-(2-amino-1H-imidazol-4-yl)propyl)-1H-1,2,3-triazol-1-yl)-N-tert-butylacetamide 1192370-45-8 C14H23N7O
2-(4-(3-(2-amino-1H-imidazol-4-yl)propyl)-1H-1,2,3-triazol-1-yl)-N-tert-butylacetamide
—— 2-(4-(3-(2-amino-1H-imidazol-4-yl)propyl)-1H-1,2,3-triazol-1-yl)-N-tert-butylacetamide hydrochloride 1192357-89-3 C14H23N7O*ClH
2-(4-(3-(2-amino-1H-imidazol-4-yl)propyl)-1H-1,2,3-triazol-1-yl)-N-tert-butylacetamide hydrochloride
—— 2-(4-(3-(2-amino-1H-imidazol-4-yl)propyl)-1H-1,2,3-triazol-1-yl)-N-cyclopentylacetamide hydrochloride 1192357-91-7 C15H23N7O*ClH
2-(4-(3-(2-amino-1H-imidazol-4-yl)propyl)-1H-1,2,3-triazol-1-yl)-N-cyclopentylacetamide hydrochloride
—— 2-(4-(5-(2-amino-1H-imidazol-4-yl)pentyl)-1H-1,2,3-triazol-1-yl)-N-octylacetamide 1257692-57-1 C20H35N7O
2-(4-(5-(2-amino-1H-imidazol-4-yl)pentyl)-1H-1,2,3-triazol-1-yl)-N-octylacetamide
—— 2-(4-(5-(2-amino-1H-imidazol-4-yl)pentyl)-1H-1,2,3-triazol-1-yl)-N-octylacetamide hydrochloride 1257629-50-7 C20H35N7O*ClH
2-(4-(5-(2-amino-1H-imidazol-4-yl)pentyl)-1H-1,2,3-triazol-1-yl)-N-octylacetamide hydrochloride
—— 2-(4-(3-(2-amino-1H-imidazol-4-yl)propyl)-1H-1,2,3-triazol-1-yl)-N-hexylacetamide 1192370-53-8 C16H27N7O
2-(4-(3-(2-amino-1H-imidazol-4-yl)propyl)-1H-1,2,3-triazol-1-yl)-N-hexylacetamide