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中文名称 英文名称 CAS号 化学式 结构式图片
—— 6-(4-(1H-pyrazol-1-yl)phenyl)-1-((tetrahydro-2H-pyran-4-yl)methyl)-1H-imidazo[4,5-b]pyrazin-2(3H)-one 1021917-16-7 C20H20N6O2
6-(4-(1H-pyrazol-1-yl)phenyl)-1-((tetrahydro-2H-pyran-4-yl)methyl)-1H-imidazo[4,5-b]pyrazin-2(3H)-one
—— N-cyclopropyl-4-(8-((tetrahydro-2H-pyran-4-yl)methylamino)imidazo[1,2-a]pyrazin-3-yl)benzamide 1263420-63-8 C22H25N5O2
N-cyclopropyl-4-(8-((tetrahydro-2H-pyran-4-yl)methylamino)imidazo[1,2-a]pyrazin-3-yl)benzamide
—— 4-(3-bromophenyl)-1,3-dihydro-2H-imidazol-2-one 690258-14-1 C9H7BrN2O
4-(3-bromophenyl)-1,3-dihydro-2H-imidazol-2-one
—— 3-(2,4-dichloro-phenyl)-imidazo[1,2-a]pyridine-7-carboxylic acid (tetrahydro-pyran-4-ylmethyl)-amide 1009379-06-9 C20H19Cl2N3O2
3-(2,4-dichloro-phenyl)-imidazo[1,2-a]pyridine-7-carboxylic acid (tetrahydro-pyran-4-ylmethyl)-amide
—— 4-(4-(prop-2-yn-1-yloxy)phenyl)-1,2,4-triazolidine-3,5-dione 1313211-51-6 C11H9N3O3
4-(4-(prop-2-yn-1-yloxy)phenyl)-1,2,4-triazolidine-3,5-dione
—— 4-(6-(sec-butylamino)-8-((tetrahydro-2H-pyran-4-yl)methylamino)imidazo[1,2-b]pyridazin-3-yl)-N-cyclopropylbenzamide 1263423-93-3 C26H34N6O2
4-(6-(sec-butylamino)-8-((tetrahydro-2H-pyran-4-yl)methylamino)imidazo[1,2-b]pyridazin-3-yl)-N-cyclopropylbenzamide
—— tert-butyl 6-(sec-butylamino)-3-(4-(cyclopropylcarbamoyl)phenyl)imidazo[1,2-b]pyridazin-8-yl((tetrahydro-2H-pyran-4-yl)methyl)carbamate 1263425-65-5 C31H42N6O4
tert-butyl 6-(sec-butylamino)-3-(4-(cyclopropylcarbamoyl)phenyl)imidazo[1,2-b]pyridazin-8-yl((tetrahydro-2H-pyran-4-yl)methyl)carbamate
—— 5-chloro-1,2-diphenyl-1<i>H</i>-imidazole 861339-06-2 C15H11ClN2
5-chloro-1,2-diphenyl-1<i>H</i>-imidazole
—— 3-(3-Chloro-phenyl)-imidazo[1,2-a]pyridine-7-carboxylic acid (tetrahydro-pyran-4-ylmethyl)-amide 1009379-04-7 C20H20ClN3O2
3-(3-Chloro-phenyl)-imidazo[1,2-a]pyridine-7-carboxylic acid (tetrahydro-pyran-4-ylmethyl)-amide
—— tert-butyl 2-(4-(oxazol-5-yl)phenylamino)-4-((tetrahydro-2H-pyran-4-yl)methylamino)-7,8-dihydropyrido[4,3-d]pyrimidine-6(5H)-carboxylate 1226889-32-2 C27H34N6O4
tert-butyl 2-(4-(oxazol-5-yl)phenylamino)-4-((tetrahydro-2H-pyran-4-yl)methylamino)-7,8-dihydropyrido[4,3-d]pyrimidine-6(5H)-carboxylate
—— N-cyclopropyl-4-(8-(methylsulfonyl)imidazo[1,2-a]pyrazin-3-yl)benzamide 1263420-64-9 C17H16N4O3S
N-cyclopropyl-4-(8-(methylsulfonyl)imidazo[1,2-a]pyrazin-3-yl)benzamide
—— 2-(2-(5-bromo-1-tert-butyl-1H-pyrazol-4-yl)thiazol-4-yl)-N-((tetrahydro-2H-pyran-4-yl)methyl)acetamide 1421849-22-0 C18H25BrN4O2S
2-(2-(5-bromo-1-tert-butyl-1H-pyrazol-4-yl)thiazol-4-yl)-N-((tetrahydro-2H-pyran-4-yl)methyl)acetamide
—— 6-{4-[2-(2-trimethylsilanylethoxymethyl)-2H-pyrazol-3-yl]phenoxy}-2,3-dihydrobenzofuran-2-carbaldehyde 1541188-64-0 C24H28N2O4Si
6-{4-[2-(2-trimethylsilanylethoxymethyl)-2H-pyrazol-3-yl]phenoxy}-2,3-dihydrobenzofuran-2-carbaldehyde
—— 4-Methyl-2-ethyl-5-propylthiazole 104256-96-4 C9H15NS
4-Methyl-2-ethyl-5-propylthiazole
—— 3-(4-(cyclopropylcarbamoyl)phenyl)-8-((tetrahydro-2H-pyran-4-yl)methylamino)imidazo[1,2-a]pyrazine-6-carboxamide 1263422-97-4 C23H26N6O3
3-(4-(cyclopropylcarbamoyl)phenyl)-8-((tetrahydro-2H-pyran-4-yl)methylamino)imidazo[1,2-a]pyrazine-6-carboxamide
—— 2-{2-[1-tert-butyl-5-(4-fluorophenyl)-1H-pyrazol-4-yl]-1,3-thiazol-4-yl}-3-phenyl-N-(tetrahydro-2H-pyran-4-ylmethyl)propanamide 1421848-19-2 C31H35FN4O2S
2-{2-[1-tert-butyl-5-(4-fluorophenyl)-1H-pyrazol-4-yl]-1,3-thiazol-4-yl}-3-phenyl-N-(tetrahydro-2H-pyran-4-ylmethyl)propanamide
—— (1aS,5aS)-2-(2,4-difluorophenyl)-1a,2,5,5a-tetrahydro-1H-2,3-diazacyclopropa[a]pentalene-4-carboxylic acid (tetrahydro-pyran-4-ylmethyl)amide 1268878-32-5 C20H21F2N3O2
(1aS,5aS)-2-(2,4-difluorophenyl)-1a,2,5,5a-tetrahydro-1H-2,3-diazacyclopropa[a]pentalene-4-carboxylic acid (tetrahydro-pyran-4-ylmethyl)amide
—— 2-{2-[1-tert-butyl-5-(4-fluorophenyl)-1H-pyrazol-4-yl]-1,3-thiazol-4-yl}-N-(tetrahydro-2H-pyran-4-ylmethyl)acetamide 1421847-06-4 C24H29FN4O2S
2-{2-[1-tert-butyl-5-(4-fluorophenyl)-1H-pyrazol-4-yl]-1,3-thiazol-4-yl}-N-(tetrahydro-2H-pyran-4-ylmethyl)acetamide
—— (2E)-3-{2-[1-tert-butyl-5-(4-methoxyphenyl)-1H-pyrazol-4-yl]-1,3-thiazol-4-yl}-N-(tetrahydro-2H-pyran-4-ylmethyl)prop-2-enamide 1421848-24-9 C26H32N4O3S
(2E)-3-{2-[1-tert-butyl-5-(4-methoxyphenyl)-1H-pyrazol-4-yl]-1,3-thiazol-4-yl}-N-(tetrahydro-2H-pyran-4-ylmethyl)prop-2-enamide
—— (E)-3-(2-(1-(tert-butyl)-5-(4-methoxyphenyl)-1H-pyrazol-4-yl)thiazol-4-yl)acrylic acid 1421850-07-8 C20H21N3O3S
(E)-3-(2-(1-(tert-butyl)-5-(4-methoxyphenyl)-1H-pyrazol-4-yl)thiazol-4-yl)acrylic acid
—— N-cyclopropyl-4-(6-(piperidine-1-carbonyl)-8-((tetrahydro-2H-pyran-4-yl)methylamino)imidazo[1,2-a]pyrazin-3-yl)benzamide 1263423-06-8 C28H34N6O3
N-cyclopropyl-4-(6-(piperidine-1-carbonyl)-8-((tetrahydro-2H-pyran-4-yl)methylamino)imidazo[1,2-a]pyrazin-3-yl)benzamide
—— 3-(4-(cyclopropylcarbamoyl)phenyl)-8-(methylsulfonyl)imidazo[1,2-a]pyrazine-6-carboxamide 1263425-55-3 C18H17N5O4S
3-(4-(cyclopropylcarbamoyl)phenyl)-8-(methylsulfonyl)imidazo[1,2-a]pyrazine-6-carboxamide
—— 2-{4-[1-tert-butyl-5-(4-methoxyphenyl)-1H-pyrazol-4-yl]-1,3-thiazol-2-yl}-N-(tetrahydro-2H-pyran-4-ylmethyl)acetamide 1421847-26-8 C25H32N4O3S
2-{4-[1-tert-butyl-5-(4-methoxyphenyl)-1H-pyrazol-4-yl]-1,3-thiazol-2-yl}-N-(tetrahydro-2H-pyran-4-ylmethyl)acetamide
—— {2-[5-(4-fluorophenyl)-1-phenyl-1H-pyrazol-4-yl]-1,3-thiazol-4-yl}acetic acid 1421848-91-0 C20H14FN3O2S
{2-[5-(4-fluorophenyl)-1-phenyl-1H-pyrazol-4-yl]-1,3-thiazol-4-yl}acetic acid
—— 2-(4-(1-tert-butyl-5-(4-methoxyphenyl)-1H-pyrazol-4-yl)thiazol-2-yl)acetic acid 1421848-86-3 C19H21N3O3S
2-(4-(1-tert-butyl-5-(4-methoxyphenyl)-1H-pyrazol-4-yl)thiazol-2-yl)acetic acid
—— 2-(2-(1-(tert-butyl)-5-(4-fluorophenyl)-1H-pyrazol-4-yl)thiazol-4-yl)-3-phenylpropanoic acid 1421849-98-0 C25H24FN3O2S
2-(2-(1-(tert-butyl)-5-(4-fluorophenyl)-1H-pyrazol-4-yl)thiazol-4-yl)-3-phenylpropanoic acid
—— 2-[1-tert-butyl-5-(4-fluorophenyl)-1H-pyrazol-4-yl]-N-(tetrahydro-2H-pyran-4-ylmethyl)-4,5-dihydro-1,3-thiazole-4-carboxamide 1421850-80-7 C23H29FN4O2S
2-[1-tert-butyl-5-(4-fluorophenyl)-1H-pyrazol-4-yl]-N-(tetrahydro-2H-pyran-4-ylmethyl)-4,5-dihydro-1,3-thiazole-4-carboxamide
—— 2-(2-(1-tert-butyl-5-(4-fluorophenyl)-1H-pyrazol-4-yl)thiazol-4-yl)acetic acid 1421848-76-1 C18H18FN3O2S
2-(2-(1-tert-butyl-5-(4-fluorophenyl)-1H-pyrazol-4-yl)thiazol-4-yl)acetic acid
—— N-((tetrahydro-2H-pyran-4-yl)methyl)-3-(3-(trifluoromethoxy)phenyl)imidazo[1,2-b]pyridazin-6-amine 1361951-04-3 C19H19F3N4O2
N-((tetrahydro-2H-pyran-4-yl)methyl)-3-(3-(trifluoromethoxy)phenyl)imidazo[1,2-b]pyridazin-6-amine
—— N-cyclopropyl-4-(8-(methylsulfonyl)-6-(piperidine-1-carbonyl)imidazo[1,2-a]pyrazin-3-yl)benzamide 1263425-58-6 C23H25N5O4S
N-cyclopropyl-4-(8-(methylsulfonyl)-6-(piperidine-1-carbonyl)imidazo[1,2-a]pyrazin-3-yl)benzamide
—— 2-[5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-4-methyl-1H-pyrazol-3-yl]-5,5-dimethyl-3,5-dihydroimidazol-4-one 1170700-89-6 C21H17Cl3N4O
2-[5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-4-methyl-1H-pyrazol-3-yl]-5,5-dimethyl-3,5-dihydroimidazol-4-one
—— N-cyclopropyl-4-[6-(2,3-difluoro-4-methoxyphenoxy)-8-(methylsulfonyl)imidazo[1,2-b]pyridazin-3-yl]-2-methylbenzamide 1554460-88-6 C25H22F2N4O5S
N-cyclopropyl-4-[6-(2,3-difluoro-4-methoxyphenoxy)-8-(methylsulfonyl)imidazo[1,2-b]pyridazin-3-yl]-2-methylbenzamide
—— 2-(2-(1-cyclohexyl-5-(4-fluorophenyl)-1H-pyrazol-4-yl)thiazol-4-yl)acetic acid 1421849-62-8 C20H20FN3O2S
2-(2-(1-cyclohexyl-5-(4-fluorophenyl)-1H-pyrazol-4-yl)thiazol-4-yl)acetic acid
—— 2-{2-[5-(4-fluorophenyl)-1-phenyl-1H-pyrazol-4-yl]-1,3-thiazol-4-yl}-N-(tetrahydro-2H-pyran-4-ylmethyl)acetamide 1421847-27-9 C26H25FN4O2S
2-{2-[5-(4-fluorophenyl)-1-phenyl-1H-pyrazol-4-yl]-1,3-thiazol-4-yl}-N-(tetrahydro-2H-pyran-4-ylmethyl)acetamide
—— (2-[1-(difluoromethyl)-5-(4-fluorophenyl)-1H-pyrazol-4-yl]-1,3-thiazol-4-yl)acetic acid 1421849-12-8 C15H10F3N3O2S
(2-[1-(difluoromethyl)-5-(4-fluorophenyl)-1H-pyrazol-4-yl]-1,3-thiazol-4-yl)acetic acid
—— 2-(1-tert-butyl-5-(4-fluorophenyl)-1H-pyrazol-4-yl)thiazole-4-carboxylic acid 1421848-78-3 C17H16FN3O2S
2-(1-tert-butyl-5-(4-fluorophenyl)-1H-pyrazol-4-yl)thiazole-4-carboxylic acid
—— 2-[1-tert-butyl-5-(4-fluorophenyl)-1H-pyrazol-4-yl]-N-(tetrahydro-2H-pyran-4-ylmethyl)-1,3-thiazole-4-carboxamide 1421847-12-2 C23H27FN4O2S
2-[1-tert-butyl-5-(4-fluorophenyl)-1H-pyrazol-4-yl]-N-(tetrahydro-2H-pyran-4-ylmethyl)-1,3-thiazole-4-carboxamide
—— N-cyclopropyl-4-{6-(2,3-difluoro-4-methoxyphenoxy)-8-[(tetrahydro-2H-pyran-4-ylmethyl)amino]imidazo[ 1,2-b]pyridazin-3-yl}-2-methylbenzamide 1554458-55-7 C30H31F2N5O4
N-cyclopropyl-4-{6-(2,3-difluoro-4-methoxyphenoxy)-8-[(tetrahydro-2H-pyran-4-ylmethyl)amino]imidazo[ 1,2-b]pyridazin-3-yl}-2-methylbenzamide
—— methyl-[6-methyl-3-(3-trifluoromethoxy-phenyl)-7,8-dihydro-6H-9-oxa-1,2,3a,4,6-pentaaza-cyclopenta[a]naphthalen-5-yl]-piperidin-4-ylmethyl-amine 1313732-78-3 C22H26F3N7O2
methyl-[6-methyl-3-(3-trifluoromethoxy-phenyl)-7,8-dihydro-6H-9-oxa-1,2,3a,4,6-pentaaza-cyclopenta[a]naphthalen-5-yl]-piperidin-4-ylmethyl-amine
—— 2-(2-(5-bromo-1-tert-butyl-1H-pyrazol-4-yl)thiazol-4-yl)acetic acid 1421849-21-9 C12H14BrN3O2S
2-(2-(5-bromo-1-tert-butyl-1H-pyrazol-4-yl)thiazol-4-yl)acetic acid
—— 2-{2-[1-cyclohexyl-5-(4-fluorophenyl)-1H-pyrazol-4-yl]-1,3-thiazol-4-yl}-N-(tetrahydro-2H-pyran-4-ylmethyl)acetamide 1421847-45-1 C26H31FN4O2S
2-{2-[1-cyclohexyl-5-(4-fluorophenyl)-1H-pyrazol-4-yl]-1,3-thiazol-4-yl}-N-(tetrahydro-2H-pyran-4-ylmethyl)acetamide
—— 2-{2-[1-(difluoromethyl)-5-(4-fluorophenyl)-1H-pyrazol-4-yl]-1,3-thiazol-4-yl}-N-(tetrahydro-2H-pyran-4-ylmethyl)acetamide 1421847-30-4 C21H21F3N4O2S
2-{2-[1-(difluoromethyl)-5-(4-fluorophenyl)-1H-pyrazol-4-yl]-1,3-thiazol-4-yl}-N-(tetrahydro-2H-pyran-4-ylmethyl)acetamide
—— 2-(2-(1-tert-butyl-5-(4-methoxyphenyl)-1H-pyrazol-4-yl)thiazol-4-yl)acetic acid 1421849-26-4 C19H21N3O3S
2-(2-(1-tert-butyl-5-(4-methoxyphenyl)-1H-pyrazol-4-yl)thiazol-4-yl)acetic acid
—— {2-[5-(4-fluorophenyl)-1H-pyrazol-4-yl]-1,3-thiazol-4-yl}acetic acid 1421849-75-3 C14H10FN3O2S
{2-[5-(4-fluorophenyl)-1H-pyrazol-4-yl]-1,3-thiazol-4-yl}acetic acid
—— methyl-{1-[6-methyl-3-(3-trifluoromethoxy-phenyl)-7,8-dihydro-6H-9-oxa-1,2,3a,4,6-pentaaza-cyclopenta[a]naphthalen-5-yl]-piperidin-4-ylmethyl}-amine 1313732-77-2 C22H26F3N7O2
methyl-{1-[6-methyl-3-(3-trifluoromethoxy-phenyl)-7,8-dihydro-6H-9-oxa-1,2,3a,4,6-pentaaza-cyclopenta[a]naphthalen-5-yl]-piperidin-4-ylmethyl}-amine
—— 2-{2-[5-(4-fluorophenyl)-1-methyl-1H-pyrazol-4-yl]-1,3-thiazol-4-yl}-N-(tetrahydro-2H-pyran-4-ylmethyl)acetamide 1421847-28-0 C21H23FN4O2S
2-{2-[5-(4-fluorophenyl)-1-methyl-1H-pyrazol-4-yl]-1,3-thiazol-4-yl}-N-(tetrahydro-2H-pyran-4-ylmethyl)acetamide
—— N-(5-allyl-2-(2,4-dichlorophenyl)-7,7-difluoro-6-(4-methoxyphenyl)-4,5,6,7-tetrahydro-2H-pyrazolo[4,3-c]pyridin-3-yl)-4-fluorobenzenesulfonamide 1562996-86-4 C28H23Cl2F3N4O3S
N-(5-allyl-2-(2,4-dichlorophenyl)-7,7-difluoro-6-(4-methoxyphenyl)-4,5,6,7-tetrahydro-2H-pyrazolo[4,3-c]pyridin-3-yl)-4-fluorobenzenesulfonamide
—— {2-[5-(4-fluorophenyl)-1-methyl-1H-pyrazol-4-yl]-1,3-thiazol-4-yl}acetic acid 1421848-97-6 C15H12FN3O2S
{2-[5-(4-fluorophenyl)-1-methyl-1H-pyrazol-4-yl]-1,3-thiazol-4-yl}acetic acid
—— 2-{2-[1-tert-butyl-5-(4-methoxyphenyl)-1H-pyrazol-4-yl]-1,3-thiazol-4-yl}-N-(tetrahydro-2H-pyran-4-ylmethyl)acetamide 1421847-33-7 C25H32N4O3S
2-{2-[1-tert-butyl-5-(4-methoxyphenyl)-1H-pyrazol-4-yl]-1,3-thiazol-4-yl}-N-(tetrahydro-2H-pyran-4-ylmethyl)acetamide
—— 1-(5-allyl-2-(2,4-dichlorophenyl)-7,7-difluoro-4,5,6,7-tetrahydro-6-(4-methoxyphenyl)-2H-pyrazolo[4,3-c]pyridin-3-yl)-3-(4-(trifluoromethyl)phenyl)thiourea 1562996-92-2 C30H24Cl2F5N5OS
1-(5-allyl-2-(2,4-dichlorophenyl)-7,7-difluoro-4,5,6,7-tetrahydro-6-(4-methoxyphenyl)-2H-pyrazolo[4,3-c]pyridin-3-yl)-3-(4-(trifluoromethyl)phenyl)thiourea