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二嗪类

中文名称 英文名称 CAS号 化学式 结构式图片
—— N-[[(3R)-1-[(5-chloro-1,3-dimethylpyrazol-4-yl)methyl]pyrrolidin-3-yl]methyl]pyrazine-2-carboxamide —— C16H21ClN6O
N-[[(3R)-1-[(5-chloro-1,3-dimethylpyrazol-4-yl)methyl]pyrrolidin-3-yl]methyl]pyrazine-2-carboxamide
—— 5-[4-[(3R)-3-(pyrrolidine-1-carbonyl)piperidin-1-yl]piperidine-1-carbonyl]-1H-pyrazin-2-one —— C20H29N5O3
5-[4-[(3R)-3-(pyrrolidine-1-carbonyl)piperidin-1-yl]piperidine-1-carbonyl]-1H-pyrazin-2-one
—— 5-[(3S)-1-(2-cyclopropyl-4-methylpyrimidine-5-carbonyl)piperidin-3-yl]-4-ethyl-2-methyl-1,2,4-triazol-3-one —— C19H26N6O2
5-[(3S)-1-(2-cyclopropyl-4-methylpyrimidine-5-carbonyl)piperidin-3-yl]-4-ethyl-2-methyl-1,2,4-triazol-3-one
—— (2S)-1-[[6-(2-methoxyphenyl)pyridazin-3-yl]amino]propan-2-ol —— C14H17N3O2
(2S)-1-[[6-(2-methoxyphenyl)pyridazin-3-yl]amino]propan-2-ol
—— 5-[4-[(3S)-3-(pyrrolidine-1-carbonyl)piperidin-1-yl]piperidine-1-carbonyl]-1H-pyrazin-2-one —— C20H29N5O3
5-[4-[(3S)-3-(pyrrolidine-1-carbonyl)piperidin-1-yl]piperidine-1-carbonyl]-1H-pyrazin-2-one
—— N-[[(2S)-1,4-dioxan-2-yl]methyl]-6-(2-methoxyphenyl)pyridazin-3-amine —— C16H19N3O3
N-[[(2S)-1,4-dioxan-2-yl]methyl]-6-(2-methoxyphenyl)pyridazin-3-amine
—— N-[[(2R)-1,4-dioxan-2-yl]methyl]-6-(2-methoxyphenyl)pyridazin-3-amine —— C16H19N3O3
N-[[(2R)-1,4-dioxan-2-yl]methyl]-6-(2-methoxyphenyl)pyridazin-3-amine
—— (4S)-4,6-dimethyl-N-[(2-methylimidazo[2,1-b][1,3,4]thiadiazol-6-yl)methyl]-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxamide —— C13H16N6O2S
(4S)-4,6-dimethyl-N-[(2-methylimidazo[2,1-b][1,3,4]thiadiazol-6-yl)methyl]-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxamide
—— 2-methyl-6-[(3R)-piperidin-3-yl]-N-[(5-thiophen-2-yl-1H-pyrazol-4-yl)methyl]pyrimidin-4-amine —— C18H22N6S
2-methyl-6-[(3R)-piperidin-3-yl]-N-[(5-thiophen-2-yl-1H-pyrazol-4-yl)methyl]pyrimidin-4-amine
—— 2-phenyl-N-[(3R)-piperidin-3-yl]-6,7-dihydro-5H-cyclopenta[d]pyrimidin-4-amine —— C18H22N4
2-phenyl-N-[(3R)-piperidin-3-yl]-6,7-dihydro-5H-cyclopenta[d]pyrimidin-4-amine
—— 3-methyl-6-[methyl-[(Z)-[(Z)-2-methyl-3-phenylprop-2-enylidene]amino]amino]-1H-pyrimidine-2,4-dione —— C16H18N4O2
3-methyl-6-[methyl-[(Z)-[(Z)-2-methyl-3-phenylprop-2-enylidene]amino]amino]-1H-pyrimidine-2,4-dione
—— (4R)-6-methyl-N-[(5-methylpyrazin-2-yl)methyl]-2-oxo-4-thiophen-2-yl-3,4-dihydro-1H-pyrimidine-5-carboxamide —— C16H17N5O2S
(4R)-6-methyl-N-[(5-methylpyrazin-2-yl)methyl]-2-oxo-4-thiophen-2-yl-3,4-dihydro-1H-pyrimidine-5-carboxamide
—— (4S)-6-methyl-N-[(5-methylpyrazin-2-yl)methyl]-2-oxo-4-thiophen-2-yl-3,4-dihydro-1H-pyrimidine-5-carboxamide —— C16H17N5O2S
(4S)-6-methyl-N-[(5-methylpyrazin-2-yl)methyl]-2-oxo-4-thiophen-2-yl-3,4-dihydro-1H-pyrimidine-5-carboxamide
—— 2-phenyl-N-[(3S)-piperidin-3-yl]-6,7-dihydro-5H-cyclopenta[d]pyrimidin-4-amine —— C18H22N4
2-phenyl-N-[(3S)-piperidin-3-yl]-6,7-dihydro-5H-cyclopenta[d]pyrimidin-4-amine
—— (4R)-4,6-dimethyl-N-[(2-methylimidazo[2,1-b][1,3,4]thiadiazol-6-yl)methyl]-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxamide —— C13H16N6O2S
(4R)-4,6-dimethyl-N-[(2-methylimidazo[2,1-b][1,3,4]thiadiazol-6-yl)methyl]-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxamide
—— N-(1,1-dioxothian-4-yl)-2-methyl-6-[(3R)-piperidin-3-yl]pyrimidin-4-amine —— C15H24N4O2S
N-(1,1-dioxothian-4-yl)-2-methyl-6-[(3R)-piperidin-3-yl]pyrimidin-4-amine
—— (3R)-1-[3-[[(6-phenylpyridazin-3-yl)amino]methyl]pyridin-2-yl]piperidin-3-ol —— C21H23N5O
(3R)-1-[3-[[(6-phenylpyridazin-3-yl)amino]methyl]pyridin-2-yl]piperidin-3-ol
—— 2-methyl-6-[(3S)-piperidin-3-yl]-N-[(5-thiophen-2-yl-1H-pyrazol-4-yl)methyl]pyrimidin-4-amine —— C18H22N6S
2-methyl-6-[(3S)-piperidin-3-yl]-N-[(5-thiophen-2-yl-1H-pyrazol-4-yl)methyl]pyrimidin-4-amine
—— (2S)-1-[2-amino-4-(4-methoxyphenyl)-5,7-dihydropyrrolo[3,4-d]pyrimidin-6-yl]-2-pyrrolidin-1-ylpropan-1-one —— C20H25N5O2
(2S)-1-[2-amino-4-(4-methoxyphenyl)-5,7-dihydropyrrolo[3,4-d]pyrimidin-6-yl]-2-pyrrolidin-1-ylpropan-1-one
—— N-[2-[(4R)-2,2-dimethyl-4-phenyloxan-4-yl]ethyl]-6-oxo-4,5-dihydro-1H-pyridazine-3-carboxamide —— C20H27N3O3
N-[2-[(4R)-2,2-dimethyl-4-phenyloxan-4-yl]ethyl]-6-oxo-4,5-dihydro-1H-pyridazine-3-carboxamide
—— (7R)-6-[(2-ethyl-5-methyl-1H-imidazol-4-yl)methyl]-7-methyl-4-(3-methylphenyl)-5,7-dihydropyrrolo[3,4-d]pyrimidin-2-amine —— C21H26N6
(7R)-6-[(2-ethyl-5-methyl-1H-imidazol-4-yl)methyl]-7-methyl-4-(3-methylphenyl)-5,7-dihydropyrrolo[3,4-d]pyrimidin-2-amine
—— (4S)-4,6-dimethyl-N-[2-(2-methyl-6-oxo-1H-pyrimidin-4-yl)ethyl]-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxamide —— C14H19N5O3
(4S)-4,6-dimethyl-N-[2-(2-methyl-6-oxo-1H-pyrimidin-4-yl)ethyl]-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxamide
—— N-[2-[(4S)-2,2-dimethyl-4-phenyloxan-4-yl]ethyl]-6-oxo-4,5-dihydro-1H-pyridazine-3-carboxamide —— C20H27N3O3
N-[2-[(4S)-2,2-dimethyl-4-phenyloxan-4-yl]ethyl]-6-oxo-4,5-dihydro-1H-pyridazine-3-carboxamide
—— N-[[(3R)-1-butylpyrrolidin-3-yl]methyl]-2-methylimidazo[1,2-a]pyrimidine-3-carboxamide —— C17H25N5O
N-[[(3R)-1-butylpyrrolidin-3-yl]methyl]-2-methylimidazo[1,2-a]pyrimidine-3-carboxamide
—— (2R)-1-[2-amino-4-(4-methoxyphenyl)-5,7-dihydropyrrolo[3,4-d]pyrimidin-6-yl]-2-pyrrolidin-1-ylpropan-1-one —— C20H25N5O2
(2R)-1-[2-amino-4-(4-methoxyphenyl)-5,7-dihydropyrrolo[3,4-d]pyrimidin-6-yl]-2-pyrrolidin-1-ylpropan-1-one
—— (E)-[amino-[(4,6-dimethylpyrimidin-2-yl)amino]methylidene]-(2,2,6,6-tetramethylpiperidin-1-ium-4-yl)azanium —— C16H30N6+2
(E)-[amino-[(4,6-dimethylpyrimidin-2-yl)amino]methylidene]-(2,2,6,6-tetramethylpiperidin-1-ium-4-yl)azanium
—— N-(1,1-dioxothian-4-yl)-2-methyl-6-[(3S)-piperidin-3-yl]pyrimidin-4-amine —— C15H24N4O2S
N-(1,1-dioxothian-4-yl)-2-methyl-6-[(3S)-piperidin-3-yl]pyrimidin-4-amine
—— 6-(aminomethyl)-N-[(2S)-1-pyrazol-1-ylpropan-2-yl]pyrimidin-4-amine —— C11H16N6
6-(aminomethyl)-N-[(2S)-1-pyrazol-1-ylpropan-2-yl]pyrimidin-4-amine
—— 1-[[(3S)-1-(3-methoxypyrazin-2-yl)piperidin-3-yl]methyl]triazole-4-carboxylic acid —— C14H18N6O3
1-[[(3S)-1-(3-methoxypyrazin-2-yl)piperidin-3-yl]methyl]triazole-4-carboxylic acid
—— N-[2-(4-ethyl-1,2,4-triazol-3-yl)ethyl]-2-methyl-6-[(3R)-piperidin-3-yl]pyrimidin-4-amine —— C16H25N7
N-[2-(4-ethyl-1,2,4-triazol-3-yl)ethyl]-2-methyl-6-[(3R)-piperidin-3-yl]pyrimidin-4-amine
—— (4R)-4,6-dimethyl-N-[2-(2-methyl-6-oxo-1H-pyrimidin-4-yl)ethyl]-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxamide —— C14H19N5O3
(4R)-4,6-dimethyl-N-[2-(2-methyl-6-oxo-1H-pyrimidin-4-yl)ethyl]-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxamide
—— 6-(aminomethyl)-N-[(2R)-1-pyrazol-1-ylpropan-2-yl]pyrimidin-4-amine —— C11H16N6
6-(aminomethyl)-N-[(2R)-1-pyrazol-1-ylpropan-2-yl]pyrimidin-4-amine
—— N-[2-(4-ethyl-1,2,4-triazol-3-yl)ethyl]-2-methyl-6-[(3S)-piperidin-3-yl]pyrimidin-4-amine —— C16H25N7
N-[2-(4-ethyl-1,2,4-triazol-3-yl)ethyl]-2-methyl-6-[(3S)-piperidin-3-yl]pyrimidin-4-amine
—— 1-[[(3R)-1-(3-methoxypyrazin-2-yl)piperidin-3-yl]methyl]triazole-4-carboxylic acid —— C14H18N6O3
1-[[(3R)-1-(3-methoxypyrazin-2-yl)piperidin-3-yl]methyl]triazole-4-carboxylic acid
—— 2-methoxyethyl (4R)-4-(2,3-dichlorophenyl)-6-methyl-2-sulfanylidene-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C15H16Cl2N2O3S
2-methoxyethyl (4R)-4-(2,3-dichlorophenyl)-6-methyl-2-sulfanylidene-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— (3S)-1-[2-[2-(2-methylpropyl)-5,7-dihydropyrrolo[3,4-d]pyrimidin-6-yl]pyrimidin-4-yl]pyrrolidin-3-ol —— C18H24N6O
(3S)-1-[2-[2-(2-methylpropyl)-5,7-dihydropyrrolo[3,4-d]pyrimidin-6-yl]pyrimidin-4-yl]pyrrolidin-3-ol
—— (4S)-4,6-dimethyl-2-oxo-N-[[2-[(2-oxopyrrolidin-1-yl)methyl]phenyl]methyl]-3,4-dihydro-1H-pyrimidine-5-carboxamide —— C19H24N4O3
(4S)-4,6-dimethyl-2-oxo-N-[[2-[(2-oxopyrrolidin-1-yl)methyl]phenyl]methyl]-3,4-dihydro-1H-pyrimidine-5-carboxamide
—— (4R)-4,6-dimethyl-2-oxo-N-[[2-[(2-oxopyrrolidin-1-yl)methyl]phenyl]methyl]-3,4-dihydro-1H-pyrimidine-5-carboxamide —— C19H24N4O3
(4R)-4,6-dimethyl-2-oxo-N-[[2-[(2-oxopyrrolidin-1-yl)methyl]phenyl]methyl]-3,4-dihydro-1H-pyrimidine-5-carboxamide
—— 2-methyl-N-[(2S)-2-(4-methylpyrazol-1-yl)propyl]-6-piperidin-4-ylpyrimidin-4-amine —— C17H26N6
2-methyl-N-[(2S)-2-(4-methylpyrazol-1-yl)propyl]-6-piperidin-4-ylpyrimidin-4-amine
—— N-[(2S)-2-(dimethylamino)-2-(2-methylphenyl)ethyl]imidazo[1,2-a]pyrimidine-2-carboxamide —— C18H21N5O
N-[(2S)-2-(dimethylamino)-2-(2-methylphenyl)ethyl]imidazo[1,2-a]pyrimidine-2-carboxamide
—— (4S)-4-(4-methylphenyl)-5-[(2-pyridin-2-ylpyrimidin-5-yl)methyl]-1,4,6,7-tetrahydroimidazo[4,5-c]pyridine —— C23H22N6
(4S)-4-(4-methylphenyl)-5-[(2-pyridin-2-ylpyrimidin-5-yl)methyl]-1,4,6,7-tetrahydroimidazo[4,5-c]pyridine
—— propan-2-yl (4R)-4-(2-ethoxyphenyl)-6-methyl-2-sulfanylidene-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C17H22N2O3S
propan-2-yl (4R)-4-(2-ethoxyphenyl)-6-methyl-2-sulfanylidene-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— N-[(1S)-1-(3-methylpyridin-2-yl)propyl]-6-oxo-4,5-dihydro-1H-pyridazine-3-carboxamide —— C14H18N4O2
N-[(1S)-1-(3-methylpyridin-2-yl)propyl]-6-oxo-4,5-dihydro-1H-pyridazine-3-carboxamide
—— (4R)-N-(imidazo[2,1-b][1,3]thiazol-6-ylmethyl)-6-methyl-2-oxo-4-thiophen-2-yl-3,4-dihydro-1H-pyrimidine-5-carboxamide —— C16H15N5O2S2
(4R)-N-(imidazo[2,1-b][1,3]thiazol-6-ylmethyl)-6-methyl-2-oxo-4-thiophen-2-yl-3,4-dihydro-1H-pyrimidine-5-carboxamide
—— (4R)-4-(4-methylphenyl)-5-[(2-pyridin-2-ylpyrimidin-5-yl)methyl]-1,4,6,7-tetrahydroimidazo[4,5-c]pyridine —— C23H22N6
(4R)-4-(4-methylphenyl)-5-[(2-pyridin-2-ylpyrimidin-5-yl)methyl]-1,4,6,7-tetrahydroimidazo[4,5-c]pyridine
—— 6-oxo-N-[2-[(2S)-4-propylmorpholin-2-yl]ethyl]-1H-pyrazine-3-carboxamide —— C14H22N4O3
6-oxo-N-[2-[(2S)-4-propylmorpholin-2-yl]ethyl]-1H-pyrazine-3-carboxamide
—— N-[(2R)-2-(dimethylamino)-2-(2-methylphenyl)ethyl]imidazo[1,2-a]pyrimidine-2-carboxamide —— C18H21N5O
N-[(2R)-2-(dimethylamino)-2-(2-methylphenyl)ethyl]imidazo[1,2-a]pyrimidine-2-carboxamide
—— (4S)-N-(imidazo[2,1-b][1,3]thiazol-6-ylmethyl)-6-methyl-2-oxo-4-thiophen-2-yl-3,4-dihydro-1H-pyrimidine-5-carboxamide —— C16H15N5O2S2
(4S)-N-(imidazo[2,1-b][1,3]thiazol-6-ylmethyl)-6-methyl-2-oxo-4-thiophen-2-yl-3,4-dihydro-1H-pyrimidine-5-carboxamide
—— 2-(Tetrazolo[1,5-b]pyridazin-6-ylamino)ethylazanium —— C6H10N7+
2-(Tetrazolo[1,5-b]pyridazin-6-ylamino)ethylazanium
—— N-[[(3R)-1-[(2-fluorophenyl)methyl]pyrrolidin-3-yl]methyl]-6-oxo-1H-pyrazine-3-carboxamide —— C17H19FN4O2
N-[[(3R)-1-[(2-fluorophenyl)methyl]pyrrolidin-3-yl]methyl]-6-oxo-1H-pyrazine-3-carboxamide