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二嗪类

中文名称 英文名称 CAS号 化学式 结构式图片
—— 2-[4-(4-fluorophenyl)phthalazin-1-yl]sulfanyl-1-[(2R)-2-methylpiperidin-1-yl]ethanone —— C22H22FN3OS
2-[4-(4-fluorophenyl)phthalazin-1-yl]sulfanyl-1-[(2R)-2-methylpiperidin-1-yl]ethanone
—— (3S)-3-[4-(4-fluorophenyl)phthalazin-1-yl]sulfanyloxolan-2-one —— C18H13FN2O2S
(3S)-3-[4-(4-fluorophenyl)phthalazin-1-yl]sulfanyloxolan-2-one
—— (2R)-2-[4-(4-fluorophenyl)phthalazin-1-yl]sulfanylpropanenitrile —— C17H12FN3S
(2R)-2-[4-(4-fluorophenyl)phthalazin-1-yl]sulfanylpropanenitrile
—— 2-[4-(4-fluorophenyl)phthalazin-1-yl]sulfanyl-N-[(2R)-pentan-2-yl]acetamide —— C21H22FN3OS
2-[4-(4-fluorophenyl)phthalazin-1-yl]sulfanyl-N-[(2R)-pentan-2-yl]acetamide
—— piperidin-1-yl-[3-[(3S)-3-(1H-pyrazol-5-yl)piperidine-1-carbonyl]pyrazin-2-yl]methanone —— C19H24N6O2
piperidin-1-yl-[3-[(3S)-3-(1H-pyrazol-5-yl)piperidine-1-carbonyl]pyrazin-2-yl]methanone
—— propyl (4R)-4-(2-ethoxyphenyl)-6-methyl-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C17H22N2O4
propyl (4R)-4-(2-ethoxyphenyl)-6-methyl-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— (2R)-1-[(2R,6R)-2,6-dimethylpiperidin-1-yl]-2-[4-(4-fluorophenyl)phthalazin-1-yl]sulfanylpropan-1-one —— C24H26FN3OS
(2R)-1-[(2R,6R)-2,6-dimethylpiperidin-1-yl]-2-[4-(4-fluorophenyl)phthalazin-1-yl]sulfanylpropan-1-one
—— (2S)-N-cyclopropyl-2-[4-(4-fluorophenyl)phthalazin-1-yl]sulfanylpropanamide —— C20H18FN3OS
(2S)-N-cyclopropyl-2-[4-(4-fluorophenyl)phthalazin-1-yl]sulfanylpropanamide
—— N-[[(3R)-1-methylpyrrolidin-3-yl]methyl]-2-(propan-2-ylamino)pyrimidine-5-carboxamide —— C14H23N5O
N-[[(3R)-1-methylpyrrolidin-3-yl]methyl]-2-(propan-2-ylamino)pyrimidine-5-carboxamide
—— N-[[(3S)-1-methylpyrrolidin-3-yl]methyl]-2-(propan-2-ylamino)pyrimidine-5-carboxamide —— C14H23N5O
N-[[(3S)-1-methylpyrrolidin-3-yl]methyl]-2-(propan-2-ylamino)pyrimidine-5-carboxamide
—— 2,4-dimethyl-N-[[(3S)-1-(pyridin-2-ylmethyl)pyrrolidin-3-yl]methyl]pyrimidine-5-carboxamide —— C18H23N5O
2,4-dimethyl-N-[[(3S)-1-(pyridin-2-ylmethyl)pyrrolidin-3-yl]methyl]pyrimidine-5-carboxamide
—— 5-methyl-N-[2-[(3R)-1-(2-methylpropyl)piperidin-3-yl]ethyl]pyrazine-2-carboxamide —— C17H28N4O
5-methyl-N-[2-[(3R)-1-(2-methylpropyl)piperidin-3-yl]ethyl]pyrazine-2-carboxamide
—— (4R)-6-methyl-N-[[3-(2-methylpropyl)imidazol-4-yl]methyl]-2-oxo-4-pyridin-3-yl-3,4-dihydro-1H-pyrimidine-5-carboxamide —— C19H24N6O2
(4R)-6-methyl-N-[[3-(2-methylpropyl)imidazol-4-yl]methyl]-2-oxo-4-pyridin-3-yl-3,4-dihydro-1H-pyrimidine-5-carboxamide
—— (4S)-6-methyl-N-[[3-(2-methylpropyl)imidazol-4-yl]methyl]-2-oxo-4-pyridin-3-yl-3,4-dihydro-1H-pyrimidine-5-carboxamide —— C19H24N6O2
(4S)-6-methyl-N-[[3-(2-methylpropyl)imidazol-4-yl]methyl]-2-oxo-4-pyridin-3-yl-3,4-dihydro-1H-pyrimidine-5-carboxamide
—— N-(2-cyanoethyl)-2-[4-(4-fluorophenyl)phthalazin-1-yl]sulfanyl-N-methylacetamide —— C20H17FN4OS
N-(2-cyanoethyl)-2-[4-(4-fluorophenyl)phthalazin-1-yl]sulfanyl-N-methylacetamide
—— 5-[(3S)-1-(2,6-dimethoxypyrimidine-4-carbonyl)piperidin-3-yl]-4-ethyl-2-methyl-1,2,4-triazol-3-one —— C17H24N6O4
5-[(3S)-1-(2,6-dimethoxypyrimidine-4-carbonyl)piperidin-3-yl]-4-ethyl-2-methyl-1,2,4-triazol-3-one
—— N-[[(3S)-1-cyclopentylpiperidin-3-yl]methyl]-3-(6-oxo-4,5-dihydro-1H-pyridazin-3-yl)propanamide —— C18H30N4O2
N-[[(3S)-1-cyclopentylpiperidin-3-yl]methyl]-3-(6-oxo-4,5-dihydro-1H-pyridazin-3-yl)propanamide
—— propan-2-yl (6R)-6-[3-(cyclobutanecarbonylamino)phenyl]-3-ethyl-4-methyl-2-oxo-1,6-dihydropyrimidine-5-carboxylate —— C22H29N3O4
propan-2-yl (6R)-6-[3-(cyclobutanecarbonylamino)phenyl]-3-ethyl-4-methyl-2-oxo-1,6-dihydropyrimidine-5-carboxylate
—— 2,4-dimethyl-N-[[(3R)-1-(pyridin-2-ylmethyl)pyrrolidin-3-yl]methyl]pyrimidine-5-carboxamide —— C18H23N5O
2,4-dimethyl-N-[[(3R)-1-(pyridin-2-ylmethyl)pyrrolidin-3-yl]methyl]pyrimidine-5-carboxamide
—— 5-[(3R)-1-(2,6-dimethoxypyrimidine-4-carbonyl)piperidin-3-yl]-4-ethyl-2-methyl-1,2,4-triazol-3-one —— C17H24N6O4
5-[(3R)-1-(2,6-dimethoxypyrimidine-4-carbonyl)piperidin-3-yl]-4-ethyl-2-methyl-1,2,4-triazol-3-one
—— 5-methyl-N-[2-[(3S)-1-(2-methylpropyl)piperidin-3-yl]ethyl]pyrazine-2-carboxamide —— C17H28N4O
5-methyl-N-[2-[(3S)-1-(2-methylpropyl)piperidin-3-yl]ethyl]pyrazine-2-carboxamide
—— propan-2-yl (6R)-3,4-dimethyl-2-oxo-6-[4-(pentanoylamino)phenyl]-1,6-dihydropyrimidine-5-carboxylate —— C21H29N3O4
propan-2-yl (6R)-3,4-dimethyl-2-oxo-6-[4-(pentanoylamino)phenyl]-1,6-dihydropyrimidine-5-carboxylate
—— (6Z)-2-(2-chlorophenyl)-5-imino-6-(thien-2-ylmethylene)-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C16H9ClN4OS2
(6Z)-2-(2-chlorophenyl)-5-imino-6-(thien-2-ylmethylene)-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— propan-2-yl (6S)-3,4-dimethyl-2-oxo-6-[4-(pentanoylamino)phenyl]-1,6-dihydropyrimidine-5-carboxylate —— C21H29N3O4
propan-2-yl (6S)-3,4-dimethyl-2-oxo-6-[4-(pentanoylamino)phenyl]-1,6-dihydropyrimidine-5-carboxylate
—— N-[(1S)-2,3-dihydro-1H-inden-1-yl]-2-pyridin-3-yl-5,6,7,8-tetrahydropyrido[3,4-d]pyrimidin-4-amine —— C21H21N5
N-[(1S)-2,3-dihydro-1H-inden-1-yl]-2-pyridin-3-yl-5,6,7,8-tetrahydropyrido[3,4-d]pyrimidin-4-amine
—— N-[(1R)-2,3-dihydro-1H-inden-1-yl]-2-pyridin-3-yl-5,6,7,8-tetrahydropyrido[3,4-d]pyrimidin-4-amine —— C21H21N5
N-[(1R)-2,3-dihydro-1H-inden-1-yl]-2-pyridin-3-yl-5,6,7,8-tetrahydropyrido[3,4-d]pyrimidin-4-amine
—— 6-[(3S)-3-(4-ethyl-5-oxo-1H-1,2,4-triazol-3-yl)piperidine-1-carbonyl]-[1,3]thiazolo[3,2-a]pyrimidin-5-one —— C16H18N6O3S
6-[(3S)-3-(4-ethyl-5-oxo-1H-1,2,4-triazol-3-yl)piperidine-1-carbonyl]-[1,3]thiazolo[3,2-a]pyrimidin-5-one
—— 6-[(3R)-3-(4-ethyl-5-oxo-1H-1,2,4-triazol-3-yl)piperidine-1-carbonyl]-[1,3]thiazolo[3,2-a]pyrimidin-5-one —— C16H18N6O3S
6-[(3R)-3-(4-ethyl-5-oxo-1H-1,2,4-triazol-3-yl)piperidine-1-carbonyl]-[1,3]thiazolo[3,2-a]pyrimidin-5-one
—— ethyl (6R)-3,4-dimethyl-2-oxo-6-[3-[[(3R)-3,5,5-trimethylhexanoyl]amino]phenyl]-1,6-dihydropyrimidine-5-carboxylate —— C24H35N3O4
ethyl (6R)-3,4-dimethyl-2-oxo-6-[3-[[(3R)-3,5,5-trimethylhexanoyl]amino]phenyl]-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (6R)-3,4-dimethyl-2-oxo-6-[3-[[(3S)-3,5,5-trimethylhexanoyl]amino]phenyl]-1,6-dihydropyrimidine-5-carboxylate —— C24H35N3O4
ethyl (6R)-3,4-dimethyl-2-oxo-6-[3-[[(3S)-3,5,5-trimethylhexanoyl]amino]phenyl]-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (6S)-3,4-dimethyl-2-oxo-6-[3-[[(3S)-3,5,5-trimethylhexanoyl]amino]phenyl]-1,6-dihydropyrimidine-5-carboxylate —— C24H35N3O4
ethyl (6S)-3,4-dimethyl-2-oxo-6-[3-[[(3S)-3,5,5-trimethylhexanoyl]amino]phenyl]-1,6-dihydropyrimidine-5-carboxylate
—— (3S)-3-[[(2-aminopyrimidin-5-yl)methyl-methylamino]methyl]-1-(2-cyclohexylethyl)-3-hydroxypiperidin-2-one —— C20H33N5O2
(3S)-3-[[(2-aminopyrimidin-5-yl)methyl-methylamino]methyl]-1-(2-cyclohexylethyl)-3-hydroxypiperidin-2-one
—— 4-[3-[(1S)-1-methoxyethyl]phenyl]-5,6-dimethyl-2-(trifluoromethyl)pyrimidine —— C16H17F3N2O
4-[3-[(1S)-1-methoxyethyl]phenyl]-5,6-dimethyl-2-(trifluoromethyl)pyrimidine
—— N-[[(3S)-1-[(2,4,5-trimethylphenyl)methyl]pyrrolidin-3-yl]methyl]pyrimidine-5-carboxamide —— C20H26N4O
N-[[(3S)-1-[(2,4,5-trimethylphenyl)methyl]pyrrolidin-3-yl]methyl]pyrimidine-5-carboxamide
—— N-[[(3R)-1-[(2,4,5-trimethylphenyl)methyl]pyrrolidin-3-yl]methyl]pyrimidine-5-carboxamide —— C20H26N4O
N-[[(3R)-1-[(2,4,5-trimethylphenyl)methyl]pyrrolidin-3-yl]methyl]pyrimidine-5-carboxamide
—— (2S)-2-methyl-1-(2-phenyl-5,7-dihydropyrrolo[3,4-d]pyrimidin-6-yl)-3-(1,2,4-triazol-1-yl)propan-1-one —— C18H18N6O
(2S)-2-methyl-1-(2-phenyl-5,7-dihydropyrrolo[3,4-d]pyrimidin-6-yl)-3-(1,2,4-triazol-1-yl)propan-1-one
—— 6-(aminomethyl)-N-[(2S)-1-(3,5-dimethylpyrazol-1-yl)propan-2-yl]-2-methylpyrimidin-4-amine —— C14H22N6
6-(aminomethyl)-N-[(2S)-1-(3,5-dimethylpyrazol-1-yl)propan-2-yl]-2-methylpyrimidin-4-amine
—— 2-[(3S)-1,1-dioxothiolan-3-yl]-1-[2-(2-methylpropyl)-5,7-dihydropyrrolo[3,4-d]pyrimidin-6-yl]ethanone —— C16H23N3O3S
2-[(3S)-1,1-dioxothiolan-3-yl]-1-[2-(2-methylpropyl)-5,7-dihydropyrrolo[3,4-d]pyrimidin-6-yl]ethanone
—— (2R)-1-(2-tert-butyl-5,7-dihydropyrrolo[3,4-d]pyrimidin-6-yl)-3-(1H-imidazol-5-yl)-2-pyrrol-1-ylpropan-1-one —— C20H24N6O
(2R)-1-(2-tert-butyl-5,7-dihydropyrrolo[3,4-d]pyrimidin-6-yl)-3-(1H-imidazol-5-yl)-2-pyrrol-1-ylpropan-1-one
—— (2S)-1-(2-tert-butyl-5,7-dihydropyrrolo[3,4-d]pyrimidin-6-yl)-3-(1H-imidazol-5-yl)-2-pyrrol-1-ylpropan-1-one —— C20H24N6O
(2S)-1-(2-tert-butyl-5,7-dihydropyrrolo[3,4-d]pyrimidin-6-yl)-3-(1H-imidazol-5-yl)-2-pyrrol-1-ylpropan-1-one
—— 2-[(3R)-1,1-dioxothiolan-3-yl]-1-[2-(2-methylpropyl)-5,7-dihydropyrrolo[3,4-d]pyrimidin-6-yl]ethanone —— C16H23N3O3S
2-[(3R)-1,1-dioxothiolan-3-yl]-1-[2-(2-methylpropyl)-5,7-dihydropyrrolo[3,4-d]pyrimidin-6-yl]ethanone
—— 4-[3-[(1R)-1-methoxyethyl]phenyl]-5,6-dimethyl-2-(trifluoromethyl)pyrimidine —— C16H17F3N2O
4-[3-[(1R)-1-methoxyethyl]phenyl]-5,6-dimethyl-2-(trifluoromethyl)pyrimidine
—— (2R)-2-methyl-1-(2-phenyl-5,7-dihydropyrrolo[3,4-d]pyrimidin-6-yl)-3-(1,2,4-triazol-1-yl)propan-1-one —— C18H18N6O
(2R)-2-methyl-1-(2-phenyl-5,7-dihydropyrrolo[3,4-d]pyrimidin-6-yl)-3-(1,2,4-triazol-1-yl)propan-1-one
—— 6-(aminomethyl)-N-[(2R)-1-(3,5-dimethylpyrazol-1-yl)propan-2-yl]-2-methylpyrimidin-4-amine —— C14H22N6
6-(aminomethyl)-N-[(2R)-1-(3,5-dimethylpyrazol-1-yl)propan-2-yl]-2-methylpyrimidin-4-amine
—— ethyl (6R)-3,4-dimethyl-2-oxo-6-[3-[(2-phenoxyacetyl)amino]phenyl]-1,6-dihydropyrimidine-5-carboxylate —— C23H25N3O5
ethyl (6R)-3,4-dimethyl-2-oxo-6-[3-[(2-phenoxyacetyl)amino]phenyl]-1,6-dihydropyrimidine-5-carboxylate
—— (4R)-1-(2-tert-butyl-5,7-dihydropyrrolo[3,4-d]pyrimidin-6-yl)-4-piperidin-1-ylpentan-1-one —— C20H32N4O
(4R)-1-(2-tert-butyl-5,7-dihydropyrrolo[3,4-d]pyrimidin-6-yl)-4-piperidin-1-ylpentan-1-one
—— 2,6-dimethoxy-N-[2-[(3S)-1-methylpiperidin-3-yl]ethyl]pyrimidine-4-carboxamide —— C15H24N4O3
2,6-dimethoxy-N-[2-[(3S)-1-methylpiperidin-3-yl]ethyl]pyrimidine-4-carboxamide
—— (4S)-4,6-dimethyl-N-[2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl]-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxamide —— C12H17N5O4
(4S)-4,6-dimethyl-N-[2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl]-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxamide
—— ethyl (6S)-3,4-dimethyl-2-oxo-6-[3-[(2-phenoxyacetyl)amino]phenyl]-1,6-dihydropyrimidine-5-carboxylate —— C23H25N3O5
ethyl (6S)-3,4-dimethyl-2-oxo-6-[3-[(2-phenoxyacetyl)amino]phenyl]-1,6-dihydropyrimidine-5-carboxylate
—— 2,6-dimethoxy-N-[2-[(3R)-1-methylpiperidin-3-yl]ethyl]pyrimidine-4-carboxamide —— C15H24N4O3
2,6-dimethoxy-N-[2-[(3R)-1-methylpiperidin-3-yl]ethyl]pyrimidine-4-carboxamide