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二嗪类

中文名称 英文名称 CAS号 化学式 结构式图片
—— 7-oxo-6-[2-oxo-2-[[(2R)-4-phenylbutan-2-yl]amino]ethyl]-[1,2]thiazolo[4,5-d]pyrimidine-3-carboxamide —— C18H19N5O3S
7-oxo-6-[2-oxo-2-[[(2R)-4-phenylbutan-2-yl]amino]ethyl]-[1,2]thiazolo[4,5-d]pyrimidine-3-carboxamide
—— 3-fluoro-N-(4-(3-methyl-[1,2,4]triazolo[4,3-b]pyridazin-6-yl)phenyl)benzenesulfonamide —— C18H14FN5O2S
3-fluoro-N-(4-(3-methyl-[1,2,4]triazolo[4,3-b]pyridazin-6-yl)phenyl)benzenesulfonamide
—— N-(3-([1,2,4]triazolo[4,3-b]pyridazin-6-yl)phenyl)-5,6,7,8-tetrahydronaphthalene-2-sulfonamide —— C21H19N5O2S
N-(3-([1,2,4]triazolo[4,3-b]pyridazin-6-yl)phenyl)-5,6,7,8-tetrahydronaphthalene-2-sulfonamide
—— N-(4-(N-(3-([1,2,4]triazolo[4,3-b]pyridazin-6-yl)phenyl)sulfamoyl)phenyl)acetamide —— C19H16N6O3S
N-(4-(N-(3-([1,2,4]triazolo[4,3-b]pyridazin-6-yl)phenyl)sulfamoyl)phenyl)acetamide
—— N-(3-([1,2,4]triazolo[4,3-b]pyridazin-6-yl)phenyl)ethanesulfonamide —— C13H13N5O2S
N-(3-([1,2,4]triazolo[4,3-b]pyridazin-6-yl)phenyl)ethanesulfonamide
—— methyl (6S)-6-(2,4-dichlorophenyl)-3,4-dimethyl-2-oxo-1,6-dihydropyrimidine-5-carboxylate —— C14H14Cl2N2O3
methyl (6S)-6-(2,4-dichlorophenyl)-3,4-dimethyl-2-oxo-1,6-dihydropyrimidine-5-carboxylate
—— 4-ethoxy-N-[3-([1,2,4]triazolo[4,3-b]pyridazin-6-yl)phenyl]benzenesulfonamide —— C19H17N5O3S
4-ethoxy-N-[3-([1,2,4]triazolo[4,3-b]pyridazin-6-yl)phenyl]benzenesulfonamide
—— 7-oxo-6-[2-oxo-2-[[(2S)-4-phenylbutan-2-yl]amino]ethyl]-[1,2]thiazolo[4,5-d]pyrimidine-3-carboxamide —— C18H19N5O3S
7-oxo-6-[2-oxo-2-[[(2S)-4-phenylbutan-2-yl]amino]ethyl]-[1,2]thiazolo[4,5-d]pyrimidine-3-carboxamide
—— N-(3-([1,2,4]triazolo[4,3-b]pyridazin-6-yl)phenyl)propane-1-sulfonamide —— C14H15N5O2S
N-(3-([1,2,4]triazolo[4,3-b]pyridazin-6-yl)phenyl)propane-1-sulfonamide
—— methyl (6R)-6-(2,4-dichlorophenyl)-3,4-dimethyl-2-oxo-1,6-dihydropyrimidine-5-carboxylate —— C14H14Cl2N2O3
methyl (6R)-6-(2,4-dichlorophenyl)-3,4-dimethyl-2-oxo-1,6-dihydropyrimidine-5-carboxylate
—— N-(3-([1,2,4]triazolo[4,3-b]pyridazin-6-yl)phenyl)-2,3-dihydrobenzo[b][1,4]dioxine-6-sulfonamide —— C19H15N5O4S
N-(3-([1,2,4]triazolo[4,3-b]pyridazin-6-yl)phenyl)-2,3-dihydrobenzo[b][1,4]dioxine-6-sulfonamide
—— methyl (6S)-6-[2-(difluoromethoxy)phenyl]-3,4-dimethyl-2-oxo-1,6-dihydropyrimidine-5-carboxylate —— C15H16F2N2O4
methyl (6S)-6-[2-(difluoromethoxy)phenyl]-3,4-dimethyl-2-oxo-1,6-dihydropyrimidine-5-carboxylate
—— N-[(1S)-1-(4-methoxyphenyl)ethyl]-2-(5-methyl-3-oxo-7-phenyl-[1,2,4]triazolo[4,3-c]pyrimidin-2-yl)acetamide —— C23H23N5O3
N-[(1S)-1-(4-methoxyphenyl)ethyl]-2-(5-methyl-3-oxo-7-phenyl-[1,2,4]triazolo[4,3-c]pyrimidin-2-yl)acetamide
—— N-[(2R)-butan-2-yl]-2-[6-oxo-3-(3-pyridin-3-yl-1,2,4-oxadiazol-5-yl)pyridazin-1-yl]acetamide —— C17H18N6O3
N-[(2R)-butan-2-yl]-2-[6-oxo-3-(3-pyridin-3-yl-1,2,4-oxadiazol-5-yl)pyridazin-1-yl]acetamide
—— N-[(1R)-1-(4-methoxyphenyl)ethyl]-2-(5-methyl-3-oxo-7-phenyl-[1,2,4]triazolo[4,3-c]pyrimidin-2-yl)acetamide —— C23H23N5O3
N-[(1R)-1-(4-methoxyphenyl)ethyl]-2-(5-methyl-3-oxo-7-phenyl-[1,2,4]triazolo[4,3-c]pyrimidin-2-yl)acetamide
—— 7-(4-methoxyphenyl)-5-methyl-2-[2-[(3S)-3-methylpiperidin-1-yl]-2-oxoethyl]-[1,2,4]triazolo[4,3-c]pyrimidin-3-one —— C21H25N5O3
7-(4-methoxyphenyl)-5-methyl-2-[2-[(3S)-3-methylpiperidin-1-yl]-2-oxoethyl]-[1,2,4]triazolo[4,3-c]pyrimidin-3-one
—— 2-(5-methyl-3-oxo-7-phenyl-[1,2,4]triazolo[4,3-c]pyrimidin-2-yl)-N-[(2R)-4-phenylbutan-2-yl]acetamide —— C24H25N5O2
2-(5-methyl-3-oxo-7-phenyl-[1,2,4]triazolo[4,3-c]pyrimidin-2-yl)-N-[(2R)-4-phenylbutan-2-yl]acetamide
—— N-[(2S)-butan-2-yl]-2-[6-oxo-3-(3-pyridin-3-yl-1,2,4-oxadiazol-5-yl)pyridazin-1-yl]acetamide —— C17H18N6O3
N-[(2S)-butan-2-yl]-2-[6-oxo-3-(3-pyridin-3-yl-1,2,4-oxadiazol-5-yl)pyridazin-1-yl]acetamide
—— 2-(5-methyl-3-oxo-7-phenyl-[1,2,4]triazolo[4,3-c]pyrimidin-2-yl)-N-[(2S)-4-phenylbutan-2-yl]acetamide —— C24H25N5O2
2-(5-methyl-3-oxo-7-phenyl-[1,2,4]triazolo[4,3-c]pyrimidin-2-yl)-N-[(2S)-4-phenylbutan-2-yl]acetamide
—— 5-methyl-2-[2-[(3R)-3-methylpiperidin-1-yl]-2-oxoethyl]-7-phenyl-[1,2,4]triazolo[4,3-c]pyrimidin-3-one —— C20H23N5O2
5-methyl-2-[2-[(3R)-3-methylpiperidin-1-yl]-2-oxoethyl]-7-phenyl-[1,2,4]triazolo[4,3-c]pyrimidin-3-one
—— 7-(4-methoxyphenyl)-5-methyl-2-[2-[(3R)-3-methylpiperidin-1-yl]-2-oxoethyl]-[1,2,4]triazolo[4,3-c]pyrimidin-3-one —— C21H25N5O3
7-(4-methoxyphenyl)-5-methyl-2-[2-[(3R)-3-methylpiperidin-1-yl]-2-oxoethyl]-[1,2,4]triazolo[4,3-c]pyrimidin-3-one
—— 5-methyl-2-[2-[(3S)-3-methylpiperidin-1-yl]-2-oxoethyl]-7-phenyl-[1,2,4]triazolo[4,3-c]pyrimidin-3-one —— C20H23N5O2
5-methyl-2-[2-[(3S)-3-methylpiperidin-1-yl]-2-oxoethyl]-7-phenyl-[1,2,4]triazolo[4,3-c]pyrimidin-3-one
—— 4-(4-Methylpiperazin-4-ium-1-yl)-2-pyridin-3-ylquinazoline —— C18H20N5+
4-(4-Methylpiperazin-4-ium-1-yl)-2-pyridin-3-ylquinazoline
—— (2R)-N-[3-(6-ethylsulfanylpyridazin-3-yl)phenyl]oxolane-2-carboxamide —— C17H19N3O2S
(2R)-N-[3-(6-ethylsulfanylpyridazin-3-yl)phenyl]oxolane-2-carboxamide
—— N-[(2S)-butan-2-yl]-2-[6-[(3-methylphenyl)methyl]-5,7-dioxo-[1,2]thiazolo[4,3-d]pyrimidin-4-yl]acetamide —— C19H22N4O3S
N-[(2S)-butan-2-yl]-2-[6-[(3-methylphenyl)methyl]-5,7-dioxo-[1,2]thiazolo[4,3-d]pyrimidin-4-yl]acetamide
—— N-[(2S)-butan-2-yl]-2-[6-[(2-fluorophenyl)methyl]-5,7-dioxo-[1,2]thiazolo[4,3-d]pyrimidin-4-yl]acetamide —— C18H19FN4O3S
N-[(2S)-butan-2-yl]-2-[6-[(2-fluorophenyl)methyl]-5,7-dioxo-[1,2]thiazolo[4,3-d]pyrimidin-4-yl]acetamide
—— 2-[6-[(2-fluorophenyl)methyl]-5,7-dioxo-[1,2]thiazolo[4,3-d]pyrimidin-4-yl]-N-[[(2S)-oxolan-2-yl]methyl]acetamide —— C19H19FN4O4S
2-[6-[(2-fluorophenyl)methyl]-5,7-dioxo-[1,2]thiazolo[4,3-d]pyrimidin-4-yl]-N-[[(2S)-oxolan-2-yl]methyl]acetamide
—— 2-(6-benzyl-5,7-dioxo-[1,2]thiazolo[4,3-d]pyrimidin-4-yl)-N-[(2R)-butan-2-yl]acetamide —— C18H20N4O3S
2-(6-benzyl-5,7-dioxo-[1,2]thiazolo[4,3-d]pyrimidin-4-yl)-N-[(2R)-butan-2-yl]acetamide
—— 2-[6-[(4-methylphenyl)methyl]-5,7-dioxo-[1,2]thiazolo[4,3-d]pyrimidin-4-yl]-N-[[(2R)-oxolan-2-yl]methyl]acetamide —— C20H22N4O4S
2-[6-[(4-methylphenyl)methyl]-5,7-dioxo-[1,2]thiazolo[4,3-d]pyrimidin-4-yl]-N-[[(2R)-oxolan-2-yl]methyl]acetamide
—— N-[(2R)-butan-2-yl]-2-[6-[(2-fluorophenyl)methyl]-5,7-dioxo-[1,2]thiazolo[4,3-d]pyrimidin-4-yl]acetamide —— C18H19FN4O3S
N-[(2R)-butan-2-yl]-2-[6-[(2-fluorophenyl)methyl]-5,7-dioxo-[1,2]thiazolo[4,3-d]pyrimidin-4-yl]acetamide
—— 2-[6-[(3-methylphenyl)methyl]-5,7-dioxo-[1,2]thiazolo[4,3-d]pyrimidin-4-yl]-N-[[(2S)-oxolan-2-yl]methyl]acetamide —— C20H22N4O4S
2-[6-[(3-methylphenyl)methyl]-5,7-dioxo-[1,2]thiazolo[4,3-d]pyrimidin-4-yl]-N-[[(2S)-oxolan-2-yl]methyl]acetamide
—— N-[(2R)-butan-2-yl]-2-(5,7-dioxo-6-propyl-[1,2]thiazolo[4,3-d]pyrimidin-4-yl)acetamide —— C14H20N4O3S
N-[(2R)-butan-2-yl]-2-(5,7-dioxo-6-propyl-[1,2]thiazolo[4,3-d]pyrimidin-4-yl)acetamide
—— 2-[6-[(2-fluorophenyl)methyl]-5,7-dioxo-[1,2]thiazolo[4,3-d]pyrimidin-4-yl]-N-[[(2R)-oxolan-2-yl]methyl]acetamide —— C19H19FN4O4S
2-[6-[(2-fluorophenyl)methyl]-5,7-dioxo-[1,2]thiazolo[4,3-d]pyrimidin-4-yl]-N-[[(2R)-oxolan-2-yl]methyl]acetamide
—— 2-[6-[(4-methylphenyl)methyl]-5,7-dioxo-[1,2]thiazolo[4,3-d]pyrimidin-4-yl]-N-[[(2S)-oxolan-2-yl]methyl]acetamide —— C20H22N4O4S
2-[6-[(4-methylphenyl)methyl]-5,7-dioxo-[1,2]thiazolo[4,3-d]pyrimidin-4-yl]-N-[[(2S)-oxolan-2-yl]methyl]acetamide
—— N-[(2S)-butan-2-yl]-2-[6-[(4-fluorophenyl)methyl]-5,7-dioxo-[1,2]thiazolo[4,3-d]pyrimidin-4-yl]acetamide —— C18H19FN4O3S
N-[(2S)-butan-2-yl]-2-[6-[(4-fluorophenyl)methyl]-5,7-dioxo-[1,2]thiazolo[4,3-d]pyrimidin-4-yl]acetamide
—— N-[(2R)-butan-2-yl]-2-[6-[(3-methylphenyl)methyl]-5,7-dioxo-[1,2]thiazolo[4,3-d]pyrimidin-4-yl]acetamide —— C19H22N4O3S
N-[(2R)-butan-2-yl]-2-[6-[(3-methylphenyl)methyl]-5,7-dioxo-[1,2]thiazolo[4,3-d]pyrimidin-4-yl]acetamide
—— (2S)-N-[3-(6-ethylsulfanylpyridazin-3-yl)phenyl]oxolane-2-carboxamide —— C17H19N3O2S
(2S)-N-[3-(6-ethylsulfanylpyridazin-3-yl)phenyl]oxolane-2-carboxamide
—— 2-[6-[(3-methylphenyl)methyl]-5,7-dioxo-[1,2]thiazolo[4,3-d]pyrimidin-4-yl]-N-[[(2R)-oxolan-2-yl]methyl]acetamide —— C20H22N4O4S
2-[6-[(3-methylphenyl)methyl]-5,7-dioxo-[1,2]thiazolo[4,3-d]pyrimidin-4-yl]-N-[[(2R)-oxolan-2-yl]methyl]acetamide
—— 2-(6-benzyl-5,7-dioxo-[1,2]thiazolo[4,3-d]pyrimidin-4-yl)-N-[(2S)-butan-2-yl]acetamide —— C18H20N4O3S
2-(6-benzyl-5,7-dioxo-[1,2]thiazolo[4,3-d]pyrimidin-4-yl)-N-[(2S)-butan-2-yl]acetamide
—— N-[(2R)-butan-2-yl]-2-[6-(2-methylpropyl)-5,7-dioxo-[1,2]thiazolo[4,3-d]pyrimidin-4-yl]acetamide —— C15H22N4O3S
N-[(2R)-butan-2-yl]-2-[6-(2-methylpropyl)-5,7-dioxo-[1,2]thiazolo[4,3-d]pyrimidin-4-yl]acetamide
—— N-[(2R)-butan-2-yl]-2-[6-[(4-fluorophenyl)methyl]-5,7-dioxo-[1,2]thiazolo[4,3-d]pyrimidin-4-yl]acetamide —— C18H19FN4O3S
N-[(2R)-butan-2-yl]-2-[6-[(4-fluorophenyl)methyl]-5,7-dioxo-[1,2]thiazolo[4,3-d]pyrimidin-4-yl]acetamide
—— N-[(2S)-butan-2-yl]-2-[6-(2-methylpropyl)-5,7-dioxo-[1,2]thiazolo[4,3-d]pyrimidin-4-yl]acetamide —— C15H22N4O3S
N-[(2S)-butan-2-yl]-2-[6-(2-methylpropyl)-5,7-dioxo-[1,2]thiazolo[4,3-d]pyrimidin-4-yl]acetamide
—— 2-(6-benzyl-5,7-dioxo-[1,2]thiazolo[4,3-d]pyrimidin-4-yl)-N-[[(2S)-oxolan-2-yl]methyl]acetamide —— C19H20N4O4S
2-(6-benzyl-5,7-dioxo-[1,2]thiazolo[4,3-d]pyrimidin-4-yl)-N-[[(2S)-oxolan-2-yl]methyl]acetamide
—— N-[(1R)-1-(4-fluorophenyl)ethyl]-2-methoxypyrimidine-5-carboxamide —— C14H14FN3O2
N-[(1R)-1-(4-fluorophenyl)ethyl]-2-methoxypyrimidine-5-carboxamide
—— N-[(2S)-butan-2-yl]-2-(5,7-dioxo-6-propyl-[1,2]thiazolo[4,3-d]pyrimidin-4-yl)acetamide —— C14H20N4O3S
N-[(2S)-butan-2-yl]-2-(5,7-dioxo-6-propyl-[1,2]thiazolo[4,3-d]pyrimidin-4-yl)acetamide
—— prop-2-enyl (4R)-4-(4-chlorophenyl)-6-methyl-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C15H15ClN2O3
prop-2-enyl (4R)-4-(4-chlorophenyl)-6-methyl-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— N-[(1S)-1-(4-fluorophenyl)ethyl]-2-methoxypyrimidine-5-carboxamide —— C14H14FN3O2
N-[(1S)-1-(4-fluorophenyl)ethyl]-2-methoxypyrimidine-5-carboxamide
—— N-[(1R)-1-pyridin-3-ylethyl]-4-(2-pyrrolidin-1-ylpyrimidin-4-yl)benzamide —— C22H23N5O
N-[(1R)-1-pyridin-3-ylethyl]-4-(2-pyrrolidin-1-ylpyrimidin-4-yl)benzamide
—— 4-(2-pyrrolidin-1-ylpyrimidin-4-yl)-N-[(1R)-1-thiophen-2-ylpropyl]benzamide —— C22H24N4OS
4-(2-pyrrolidin-1-ylpyrimidin-4-yl)-N-[(1R)-1-thiophen-2-ylpropyl]benzamide
—— 2-[(2S)-3-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-2-hydroxypropyl]-4-phenylphthalazin-1-one —— C23H27N3O3
2-[(2S)-3-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-2-hydroxypropyl]-4-phenylphthalazin-1-one