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二嗪类

中文名称 英文名称 CAS号 化学式 结构式图片
—— (4R)-3-tert-butyl-1-methyl-4-(2-pyridin-2-ylpyrimidin-5-yl)-4,5-dihydro-2H-pyrazolo[3,4-b]pyridin-6-one —— C20H22N6O
(4R)-3-tert-butyl-1-methyl-4-(2-pyridin-2-ylpyrimidin-5-yl)-4,5-dihydro-2H-pyrazolo[3,4-b]pyridin-6-one
—— (4S)-3-tert-butyl-1-methyl-4-(2-pyridin-2-ylpyrimidin-5-yl)-4,5-dihydro-2H-pyrazolo[3,4-b]pyridin-6-one —— C20H22N6O
(4S)-3-tert-butyl-1-methyl-4-(2-pyridin-2-ylpyrimidin-5-yl)-4,5-dihydro-2H-pyrazolo[3,4-b]pyridin-6-one
—— (3S)-3-methyl-1-(2-pyridin-3-yl-6,7,8,9-tetrahydro-5H-pyrimido[4,5-d]azepin-4-yl)piperidin-3-ol —— C19H25N5O
(3S)-3-methyl-1-(2-pyridin-3-yl-6,7,8,9-tetrahydro-5H-pyrimido[4,5-d]azepin-4-yl)piperidin-3-ol
—— 5-ethyl-2-methyl-N-[(1S)-1-(1-methylpyrazol-4-yl)propyl]pyrimidin-4-amine —— C14H21N5
5-ethyl-2-methyl-N-[(1S)-1-(1-methylpyrazol-4-yl)propyl]pyrimidin-4-amine
—— N-[(2S,4R,6S)-2-(2-methylpropyl)-6-[2-[[(2S)-oxolan-2-yl]methylamino]pyrimidin-5-yl]oxan-4-yl]acetamide —— C20H32N4O3
N-[(2S,4R,6S)-2-(2-methylpropyl)-6-[2-[[(2S)-oxolan-2-yl]methylamino]pyrimidin-5-yl]oxan-4-yl]acetamide
—— (3R)-3-methyl-1-(2-pyridin-3-yl-6,7,8,9-tetrahydro-5H-pyrimido[4,5-d]azepin-4-yl)piperidin-3-ol —— C19H25N5O
(3R)-3-methyl-1-(2-pyridin-3-yl-6,7,8,9-tetrahydro-5H-pyrimido[4,5-d]azepin-4-yl)piperidin-3-ol
—— [2-[[(1S)-1-(4-chlorophenyl)ethyl]amino]-2-oxoethyl] 6-oxo-4,5-dihydro-1H-pyridazine-3-carboxylate —— C15H16ClN3O4
[2-[[(1S)-1-(4-chlorophenyl)ethyl]amino]-2-oxoethyl] 6-oxo-4,5-dihydro-1H-pyridazine-3-carboxylate
—— [2-[(1-cyanocyclohexyl)-methylamino]-2-oxoethyl] 6-oxo-4,5-dihydro-1H-pyridazine-3-carboxylate —— C15H20N4O4
[2-[(1-cyanocyclohexyl)-methylamino]-2-oxoethyl] 6-oxo-4,5-dihydro-1H-pyridazine-3-carboxylate
—— (3R)-N-methyl-1-(2-pyridin-2-yl-6,7,8,9-tetrahydro-5H-pyrimido[4,5-d]azepin-4-yl)piperidine-3-carboxamide —— C20H26N6O
(3R)-N-methyl-1-(2-pyridin-2-yl-6,7,8,9-tetrahydro-5H-pyrimido[4,5-d]azepin-4-yl)piperidine-3-carboxamide
—— [2-oxo-2-(5-phenyl-3,4-dihydropyrazol-2-yl)ethyl] 6-oxo-4,5-dihydro-1H-pyridazine-3-carboxylate —— C16H16N4O4
[2-oxo-2-(5-phenyl-3,4-dihydropyrazol-2-yl)ethyl] 6-oxo-4,5-dihydro-1H-pyridazine-3-carboxylate
—— (3S)-N-methyl-1-(2-pyridin-2-yl-6,7,8,9-tetrahydro-5H-pyrimido[4,5-d]azepin-4-yl)piperidine-3-carboxamide —— C20H26N6O
(3S)-N-methyl-1-(2-pyridin-2-yl-6,7,8,9-tetrahydro-5H-pyrimido[4,5-d]azepin-4-yl)piperidine-3-carboxamide
—— 5-ethyl-2-methyl-N-[(1R)-1-(1-methylpyrazol-4-yl)propyl]pyrimidin-4-amine —— C14H21N5
5-ethyl-2-methyl-N-[(1R)-1-(1-methylpyrazol-4-yl)propyl]pyrimidin-4-amine
—— [2-oxo-2-(3-phenylpropylamino)ethyl] 6-oxo-4,5-dihydro-1H-pyridazine-3-carboxylate —— C16H19N3O4
[2-oxo-2-(3-phenylpropylamino)ethyl] 6-oxo-4,5-dihydro-1H-pyridazine-3-carboxylate
—— [2-oxo-2-[(4-phenyl-1,3-thiazol-2-yl)-prop-2-enylamino]ethyl] 6-oxo-4,5-dihydro-1H-pyridazine-3-carboxylate —— C19H18N4O4S
[2-oxo-2-[(4-phenyl-1,3-thiazol-2-yl)-prop-2-enylamino]ethyl] 6-oxo-4,5-dihydro-1H-pyridazine-3-carboxylate
—— 6-methyl-2-propyl-N-[(2R)-2-(1,2,4-triazol-1-yl)propyl]pyrimidin-4-amine —— C13H20N6
6-methyl-2-propyl-N-[(2R)-2-(1,2,4-triazol-1-yl)propyl]pyrimidin-4-amine
—— [2-(dibenzylamino)-2-oxoethyl] 6-oxo-4,5-dihydro-1H-pyridazine-3-carboxylate —— C21H21N3O4
[2-(dibenzylamino)-2-oxoethyl] 6-oxo-4,5-dihydro-1H-pyridazine-3-carboxylate
—— [2-[[(1R)-1-(2-chlorophenyl)ethyl]amino]-2-oxoethyl] 6-oxo-4,5-dihydro-1H-pyridazine-3-carboxylate —— C15H16ClN3O4
[2-[[(1R)-1-(2-chlorophenyl)ethyl]amino]-2-oxoethyl] 6-oxo-4,5-dihydro-1H-pyridazine-3-carboxylate
—— [2-[benzyl(ethyl)amino]-2-oxoethyl] 6-oxo-4,5-dihydro-1H-pyridazine-3-carboxylate —— C16H19N3O4
[2-[benzyl(ethyl)amino]-2-oxoethyl] 6-oxo-4,5-dihydro-1H-pyridazine-3-carboxylate
—— [2-[(3R)-3-(furan-2-yl)-5-(4-methylphenyl)-3,4-dihydropyrazol-2-yl]-2-oxoethyl] 6-oxo-4,5-dihydro-1H-pyridazine-3-carboxylate —— C21H20N4O5
[2-[(3R)-3-(furan-2-yl)-5-(4-methylphenyl)-3,4-dihydropyrazol-2-yl]-2-oxoethyl] 6-oxo-4,5-dihydro-1H-pyridazine-3-carboxylate
—— [2-oxo-2-[[(1R)-1-phenylethyl]amino]ethyl] 6-oxo-4,5-dihydro-1H-pyridazine-3-carboxylate —— C15H17N3O4
[2-oxo-2-[[(1R)-1-phenylethyl]amino]ethyl] 6-oxo-4,5-dihydro-1H-pyridazine-3-carboxylate
—— [2-[(2-chlorophenyl)methylamino]-2-oxoethyl] 6-oxo-4,5-dihydro-1H-pyridazine-3-carboxylate —— C14H14ClN3O4
[2-[(2-chlorophenyl)methylamino]-2-oxoethyl] 6-oxo-4,5-dihydro-1H-pyridazine-3-carboxylate
—— (3,3-dimethyl-2-oxobutyl) 6-oxo-4,5-dihydro-1H-pyridazine-3-carboxylate —— C11H16N2O4
(3,3-dimethyl-2-oxobutyl) 6-oxo-4,5-dihydro-1H-pyridazine-3-carboxylate
—— [(2R)-4-(2-pyridin-3-yl-6,7,8,9-tetrahydro-5H-pyrimido[4,5-d]azepin-4-yl)morpholin-2-yl]methanamine —— C18H24N6O
[(2R)-4-(2-pyridin-3-yl-6,7,8,9-tetrahydro-5H-pyrimido[4,5-d]azepin-4-yl)morpholin-2-yl]methanamine
—— [2-[(1-cyanocyclohexyl)amino]-2-oxoethyl] 6-oxo-4,5-dihydro-1H-pyridazine-3-carboxylate —— C14H18N4O4
[2-[(1-cyanocyclohexyl)amino]-2-oxoethyl] 6-oxo-4,5-dihydro-1H-pyridazine-3-carboxylate
—— cyclohexylmethyl 6-oxo-4,5-dihydro-1H-pyridazine-3-carboxylate —— C12H18N2O3
cyclohexylmethyl 6-oxo-4,5-dihydro-1H-pyridazine-3-carboxylate
—— [(2S)-4-(2-pyridin-3-yl-6,7,8,9-tetrahydro-5H-pyrimido[4,5-d]azepin-4-yl)morpholin-2-yl]methanamine —— C18H24N6O
[(2S)-4-(2-pyridin-3-yl-6,7,8,9-tetrahydro-5H-pyrimido[4,5-d]azepin-4-yl)morpholin-2-yl]methanamine
—— 6-methyl-2-propyl-N-[(2S)-2-(1,2,4-triazol-1-yl)propyl]pyrimidin-4-amine —— C13H20N6
6-methyl-2-propyl-N-[(2S)-2-(1,2,4-triazol-1-yl)propyl]pyrimidin-4-amine
—— [2-[benzyl(2-phenylethyl)amino]-2-oxoethyl] 6-oxo-4,5-dihydro-1H-pyridazine-3-carboxylate —— C22H23N3O4
[2-[benzyl(2-phenylethyl)amino]-2-oxoethyl] 6-oxo-4,5-dihydro-1H-pyridazine-3-carboxylate
—— [2-oxo-2-(2-phenylethylamino)ethyl] 6-oxo-4,5-dihydro-1H-pyridazine-3-carboxylate —— C15H17N3O4
[2-oxo-2-(2-phenylethylamino)ethyl] 6-oxo-4,5-dihydro-1H-pyridazine-3-carboxylate
—— [2-[[(1S)-1-(3-chlorophenyl)ethyl]amino]-2-oxoethyl] 6-oxo-4,5-dihydro-1H-pyridazine-3-carboxylate —— C15H16ClN3O4
[2-[[(1S)-1-(3-chlorophenyl)ethyl]amino]-2-oxoethyl] 6-oxo-4,5-dihydro-1H-pyridazine-3-carboxylate
—— [2-[[3-[(4-methylphenyl)methyl]-1,3-thiazol-2-ylidene]amino]-2-oxoethyl] 6-oxo-4,5-dihydro-1H-pyridazine-3-carboxylate —— C18H18N4O4S
[2-[[3-[(4-methylphenyl)methyl]-1,3-thiazol-2-ylidene]amino]-2-oxoethyl] 6-oxo-4,5-dihydro-1H-pyridazine-3-carboxylate
—— (4R)-4-[2-(ethylamino)pyrimidin-5-yl]-1-(pyridin-4-ylmethyl)-4,5-dihydro-2H-pyrazolo[3,4-b]pyridin-6-one —— C18H19N7O
(4R)-4-[2-(ethylamino)pyrimidin-5-yl]-1-(pyridin-4-ylmethyl)-4,5-dihydro-2H-pyrazolo[3,4-b]pyridin-6-one
—— (3S)-1-[5-(4-hydroxyphenyl)-4-(4-methylphenyl)pyrimidin-2-yl]piperidine-3-carboxamide —— C23H24N4O2
(3S)-1-[5-(4-hydroxyphenyl)-4-(4-methylphenyl)pyrimidin-2-yl]piperidine-3-carboxamide
—— 2-ethyl-N-[(S)-furan-2-yl(phenyl)methyl]pyrimidine-5-carboxamide —— C18H17N3O2
2-ethyl-N-[(S)-furan-2-yl(phenyl)methyl]pyrimidine-5-carboxamide
—— [(2R)-1-[(1-cyanocyclohexyl)amino]-1-oxopropan-2-yl] 6-oxo-4,5-dihydro-1H-pyridazine-3-carboxylate —— C15H20N4O4
[(2R)-1-[(1-cyanocyclohexyl)amino]-1-oxopropan-2-yl] 6-oxo-4,5-dihydro-1H-pyridazine-3-carboxylate
—— (4S)-4-[2-(ethylamino)pyrimidin-5-yl]-1-(pyridin-4-ylmethyl)-4,5-dihydro-2H-pyrazolo[3,4-b]pyridin-6-one —— C18H19N7O
(4S)-4-[2-(ethylamino)pyrimidin-5-yl]-1-(pyridin-4-ylmethyl)-4,5-dihydro-2H-pyrazolo[3,4-b]pyridin-6-one
—— 5-ethyl-2-methyl-N-[(2S)-2-morpholin-4-yl-2-pyridin-4-ylethyl]pyrimidin-4-amine —— C18H25N5O
5-ethyl-2-methyl-N-[(2S)-2-morpholin-4-yl-2-pyridin-4-ylethyl]pyrimidin-4-amine
—— 2-ethyl-N-[(R)-furan-2-yl(phenyl)methyl]pyrimidine-5-carboxamide —— C18H17N3O2
2-ethyl-N-[(R)-furan-2-yl(phenyl)methyl]pyrimidine-5-carboxamide
—— N-[(2R)-2-(dimethylamino)-2-(3-methylthiophen-2-yl)ethyl]-2-ethylpyrimidine-5-carboxamide —— C16H22N4OS
N-[(2R)-2-(dimethylamino)-2-(3-methylthiophen-2-yl)ethyl]-2-ethylpyrimidine-5-carboxamide
—— (3R)-1-[5-(4-hydroxyphenyl)-4-(4-methylphenyl)pyrimidin-2-yl]piperidine-3-carboxamide —— C23H24N4O2
(3R)-1-[5-(4-hydroxyphenyl)-4-(4-methylphenyl)pyrimidin-2-yl]piperidine-3-carboxamide
—— [(2R)-1-(cyclohexylamino)-1-oxopropan-2-yl] 6-oxo-4,5-dihydro-1H-pyridazine-3-carboxylate —— C14H21N3O4
[(2R)-1-(cyclohexylamino)-1-oxopropan-2-yl] 6-oxo-4,5-dihydro-1H-pyridazine-3-carboxylate
—— N-[(2S)-2-(dimethylamino)-2-(3-methylthiophen-2-yl)ethyl]-2-ethylpyrimidine-5-carboxamide —— C16H22N4OS
N-[(2S)-2-(dimethylamino)-2-(3-methylthiophen-2-yl)ethyl]-2-ethylpyrimidine-5-carboxamide
—— [(2S)-1-(cyclohexylamino)-1-oxopropan-2-yl] 6-oxo-4,5-dihydro-1H-pyridazine-3-carboxylate —— C14H21N3O4
[(2S)-1-(cyclohexylamino)-1-oxopropan-2-yl] 6-oxo-4,5-dihydro-1H-pyridazine-3-carboxylate
—— (2-pyridin-3-ylpyrimidin-5-yl)-[(2S)-2-pyridin-2-ylpyrrolidin-1-yl]methanone —— C19H17N5O
(2-pyridin-3-ylpyrimidin-5-yl)-[(2S)-2-pyridin-2-ylpyrrolidin-1-yl]methanone
—— [amino-(2,4,6-trimethylanilino)methylidene]-(4-methyl-6-oxo-1H-pyrimidin-2-yl)azanium —— C15H20N5O+
[amino-(2,4,6-trimethylanilino)methylidene]-(4-methyl-6-oxo-1H-pyrimidin-2-yl)azanium
—— 5-ethyl-2-methyl-N-[(2R)-2-morpholin-4-yl-2-pyridin-4-ylethyl]pyrimidin-4-amine —— C18H25N5O
5-ethyl-2-methyl-N-[(2R)-2-morpholin-4-yl-2-pyridin-4-ylethyl]pyrimidin-4-amine
—— (2-pyridin-3-ylpyrimidin-5-yl)-[(2R)-2-pyridin-2-ylpyrrolidin-1-yl]methanone —— C19H17N5O
(2-pyridin-3-ylpyrimidin-5-yl)-[(2R)-2-pyridin-2-ylpyrrolidin-1-yl]methanone
—— 2,6-dimethyl-N-[(2S)-2-morpholin-4-yl-2-pyridin-4-ylethyl]pyrimidine-4-carboxamide —— C18H23N5O2
2,6-dimethyl-N-[(2S)-2-morpholin-4-yl-2-pyridin-4-ylethyl]pyrimidine-4-carboxamide
—— 2,6-dimethyl-N-[(2R)-2-morpholin-4-yl-2-pyridin-4-ylethyl]pyrimidine-4-carboxamide —— C18H23N5O2
2,6-dimethyl-N-[(2R)-2-morpholin-4-yl-2-pyridin-4-ylethyl]pyrimidine-4-carboxamide
—— [(3S)-3-(3,5-dimethylpyrazol-1-yl)pyrrolidin-1-yl]-(2,4-dimethylpyrimidin-5-yl)methanone —— C16H21N5O
[(3S)-3-(3,5-dimethylpyrazol-1-yl)pyrrolidin-1-yl]-(2,4-dimethylpyrimidin-5-yl)methanone