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二嗪类

中文名称 英文名称 CAS号 化学式 结构式图片
—— 1-[2-(2-methylpropyl)-5,7-dihydropyrrolo[3,4-d]pyrimidin-6-yl]-2-[[(2R)-oxan-2-yl]methoxy]ethanone —— C18H27N3O3
1-[2-(2-methylpropyl)-5,7-dihydropyrrolo[3,4-d]pyrimidin-6-yl]-2-[[(2R)-oxan-2-yl]methoxy]ethanone
—— N-methyl-2-pyridin-4-yl-N-[(1S)-1-pyridin-3-ylethyl]pyrimidine-5-carboxamide —— C18H17N5O
N-methyl-2-pyridin-4-yl-N-[(1S)-1-pyridin-3-ylethyl]pyrimidine-5-carboxamide
—— 4-[(7S)-2-amino-7-methyl-4-(3-methylphenyl)-5,7-dihydropyrrolo[3,4-d]pyrimidin-6-yl]-N,N-dimethyl-4-oxobutanamide —— C20H25N5O2
4-[(7S)-2-amino-7-methyl-4-(3-methylphenyl)-5,7-dihydropyrrolo[3,4-d]pyrimidin-6-yl]-N,N-dimethyl-4-oxobutanamide
—— 4-(3,4-Difluorophenyl)-6-(4-methoxyphenyl)-2-thiophen-2-ylpyrimidine —— C21H14F2N2OS
4-(3,4-Difluorophenyl)-6-(4-methoxyphenyl)-2-thiophen-2-ylpyrimidine
—— N-[(1R)-2-methoxy-1-pyridin-2-ylethyl]-N-methyl-6-oxo-1H-pyrazine-3-carboxamide —— C14H16N4O3
N-[(1R)-2-methoxy-1-pyridin-2-ylethyl]-N-methyl-6-oxo-1H-pyrazine-3-carboxamide
—— N-[(1S)-1-(cyclohexen-1-yl)ethyl]-3-(2,4-dioxopyrimidin-1-yl)propanamide —— C15H21N3O3
N-[(1S)-1-(cyclohexen-1-yl)ethyl]-3-(2,4-dioxopyrimidin-1-yl)propanamide
—— 4-[(7R)-2-amino-7-methyl-4-(3-methylphenyl)-5,7-dihydropyrrolo[3,4-d]pyrimidin-6-yl]-N,N-dimethyl-4-oxobutanamide —— C20H25N5O2
4-[(7R)-2-amino-7-methyl-4-(3-methylphenyl)-5,7-dihydropyrrolo[3,4-d]pyrimidin-6-yl]-N,N-dimethyl-4-oxobutanamide
—— (1S)-2-[[6-(aminomethyl)-2-methylpyrimidin-4-yl]amino]-1-pyridin-3-ylethanol —— C13H17N5O
(1S)-2-[[6-(aminomethyl)-2-methylpyrimidin-4-yl]amino]-1-pyridin-3-ylethanol
—— N-methyl-2-pyridin-4-yl-N-[(1R)-1-pyridin-3-ylethyl]pyrimidine-5-carboxamide —— C18H17N5O
N-methyl-2-pyridin-4-yl-N-[(1R)-1-pyridin-3-ylethyl]pyrimidine-5-carboxamide
—— (1S)-2,2-dimethyl-N-[2-(6-oxo-2-phenyl-1H-pyrimidin-4-yl)ethyl]-1-thiophen-2-ylcyclopropane-1-carboxamide —— C22H23N3O2S
(1S)-2,2-dimethyl-N-[2-(6-oxo-2-phenyl-1H-pyrimidin-4-yl)ethyl]-1-thiophen-2-ylcyclopropane-1-carboxamide
—— (1R)-2-[[6-(aminomethyl)-2-methylpyrimidin-4-yl]amino]-1-pyridin-3-ylethanol —— C13H17N5O
(1R)-2-[[6-(aminomethyl)-2-methylpyrimidin-4-yl]amino]-1-pyridin-3-ylethanol
—— N-[(1R)-1-(cyclohexen-1-yl)ethyl]-3-(2,4-dioxopyrimidin-1-yl)propanamide —— C15H21N3O3
N-[(1R)-1-(cyclohexen-1-yl)ethyl]-3-(2,4-dioxopyrimidin-1-yl)propanamide
—— N-[[(3S)-1-(2-methylpropyl)pyrrolidin-3-yl]methyl]-6-oxo-2-propan-2-yl-1H-pyrimidine-5-carboxamide —— C17H28N4O2
N-[[(3S)-1-(2-methylpropyl)pyrrolidin-3-yl]methyl]-6-oxo-2-propan-2-yl-1H-pyrimidine-5-carboxamide
—— N-[2-[(3S)-1-[(2-aminopyrimidin-5-yl)methyl]piperidin-3-yl]ethyl]-3-methylbut-2-enamide —— C17H27N5O
N-[2-[(3S)-1-[(2-aminopyrimidin-5-yl)methyl]piperidin-3-yl]ethyl]-3-methylbut-2-enamide
—— N-[[(3R)-1-(2-methylpropyl)pyrrolidin-3-yl]methyl]-6-oxo-2-propan-2-yl-1H-pyrimidine-5-carboxamide —— C17H28N4O2
N-[[(3R)-1-(2-methylpropyl)pyrrolidin-3-yl]methyl]-6-oxo-2-propan-2-yl-1H-pyrimidine-5-carboxamide
—— N-[(1R)-1-(2-ethyl-1,2,4-triazol-3-yl)ethyl]-2-methylimidazo[1,2-a]pyrimidine-3-carboxamide —— C14H17N7O
N-[(1R)-1-(2-ethyl-1,2,4-triazol-3-yl)ethyl]-2-methylimidazo[1,2-a]pyrimidine-3-carboxamide
—— N-[2-[(3R)-1-[(2-aminopyrimidin-5-yl)methyl]piperidin-3-yl]ethyl]-3-methylbut-2-enamide —— C17H27N5O
N-[2-[(3R)-1-[(2-aminopyrimidin-5-yl)methyl]piperidin-3-yl]ethyl]-3-methylbut-2-enamide
—— N-[(1S)-1-(2-ethyl-1,2,4-triazol-3-yl)ethyl]-2-methylimidazo[1,2-a]pyrimidine-3-carboxamide —— C14H17N7O
N-[(1S)-1-(2-ethyl-1,2,4-triazol-3-yl)ethyl]-2-methylimidazo[1,2-a]pyrimidine-3-carboxamide
—— 3-[3-[(1R)-1-methyl-3,4-dihydro-1H-pyrrolo[1,2-a]pyrazin-2-yl]-3-oxopropyl]-4,5-dihydro-1H-pyridazin-6-one —— C15H20N4O2
3-[3-[(1R)-1-methyl-3,4-dihydro-1H-pyrrolo[1,2-a]pyrazin-2-yl]-3-oxopropyl]-4,5-dihydro-1H-pyridazin-6-one
—— 6-(1-methylimidazol-2-yl)-N-[(2S)-1-thiophen-2-ylpropan-2-yl]pyridazin-3-amine —— C15H17N5S
6-(1-methylimidazol-2-yl)-N-[(2S)-1-thiophen-2-ylpropan-2-yl]pyridazin-3-amine
—— 3-[3-[(1S)-1-methyl-3,4-dihydro-1H-pyrrolo[1,2-a]pyrazin-2-yl]-3-oxopropyl]-4,5-dihydro-1H-pyridazin-6-one —— C15H20N4O2
3-[3-[(1S)-1-methyl-3,4-dihydro-1H-pyrrolo[1,2-a]pyrazin-2-yl]-3-oxopropyl]-4,5-dihydro-1H-pyridazin-6-one
—— 6-(1-methylimidazol-2-yl)-N-[(2R)-1-thiophen-2-ylpropan-2-yl]pyridazin-3-amine —— C15H17N5S
6-(1-methylimidazol-2-yl)-N-[(2R)-1-thiophen-2-ylpropan-2-yl]pyridazin-3-amine
—— 2-(3,6-dioxo-1H-pyridazin-2-yl)-N-[(1S)-2-methyl-1-(1-methylimidazol-2-yl)propyl]acetamide —— C14H19N5O3
2-(3,6-dioxo-1H-pyridazin-2-yl)-N-[(1S)-2-methyl-1-(1-methylimidazol-2-yl)propyl]acetamide
—— (4S)-4,6-dimethyl-2-oxo-N-[(5R,7S)-3-(tetrazol-2-yl)-1-adamantyl]-3,4-dihydro-1H-pyrimidine-5-carboxamide —— C18H25N7O2
(4S)-4,6-dimethyl-2-oxo-N-[(5R,7S)-3-(tetrazol-2-yl)-1-adamantyl]-3,4-dihydro-1H-pyrimidine-5-carboxamide
—— N-[(1R)-1-(2-ethyl-1,2,4-triazol-3-yl)ethyl]-2-pyridin-3-ylpyrimidine-5-carboxamide —— C16H17N7O
N-[(1R)-1-(2-ethyl-1,2,4-triazol-3-yl)ethyl]-2-pyridin-3-ylpyrimidine-5-carboxamide
—— N-[(1S)-1-(2-ethyl-1,2,4-triazol-3-yl)ethyl]-2-pyridin-3-ylpyrimidine-5-carboxamide —— C16H17N7O
N-[(1S)-1-(2-ethyl-1,2,4-triazol-3-yl)ethyl]-2-pyridin-3-ylpyrimidine-5-carboxamide
—— (4S)-N-[[1-[(3,5-dimethylpyrazol-1-yl)methyl]cyclopropyl]methyl]-4-(furan-3-yl)-6-methyl-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxamide —— C20H25N5O3
(4S)-N-[[1-[(3,5-dimethylpyrazol-1-yl)methyl]cyclopropyl]methyl]-4-(furan-3-yl)-6-methyl-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxamide
—— 2-(3,6-dioxo-1H-pyridazin-2-yl)-N-[(1R)-2-methyl-1-(1-methylimidazol-2-yl)propyl]acetamide —— C14H19N5O3
2-(3,6-dioxo-1H-pyridazin-2-yl)-N-[(1R)-2-methyl-1-(1-methylimidazol-2-yl)propyl]acetamide
—— ethyl (6R)-6-[4-[(3-chloro-2,2-dimethylpropanoyl)amino]phenyl]-3,4-dimethyl-2-sulfanylidene-1,6-dihydropyrimidine-5-carboxylate —— C20H26ClN3O3S
ethyl (6R)-6-[4-[(3-chloro-2,2-dimethylpropanoyl)amino]phenyl]-3,4-dimethyl-2-sulfanylidene-1,6-dihydropyrimidine-5-carboxylate
—— (4R)-N-[[1-[(3,5-dimethylpyrazol-1-yl)methyl]cyclopropyl]methyl]-4-(furan-3-yl)-6-methyl-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxamide —— C20H25N5O3
(4R)-N-[[1-[(3,5-dimethylpyrazol-1-yl)methyl]cyclopropyl]methyl]-4-(furan-3-yl)-6-methyl-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxamide
—— (4R)-4,6-dimethyl-2-oxo-N-[(5R,7S)-3-(tetrazol-2-yl)-1-adamantyl]-3,4-dihydro-1H-pyrimidine-5-carboxamide —— C18H25N7O2
(4R)-4,6-dimethyl-2-oxo-N-[(5R,7S)-3-(tetrazol-2-yl)-1-adamantyl]-3,4-dihydro-1H-pyrimidine-5-carboxamide
—— (2-phenylpyrimidin-5-yl)-[(2R)-2-pyridin-4-ylazepan-1-yl]methanone —— C22H22N4O
(2-phenylpyrimidin-5-yl)-[(2R)-2-pyridin-4-ylazepan-1-yl]methanone
—— (2-phenylpyrimidin-5-yl)-[(2S)-2-pyridin-4-ylazepan-1-yl]methanone —— C22H22N4O
(2-phenylpyrimidin-5-yl)-[(2S)-2-pyridin-4-ylazepan-1-yl]methanone
—— (2R)-2-(2,5-dioxopyrrolidin-1-yl)-N-[3-(6-oxo-1H-pyridazin-3-yl)phenyl]propanamide —— C17H16N4O4
(2R)-2-(2,5-dioxopyrrolidin-1-yl)-N-[3-(6-oxo-1H-pyridazin-3-yl)phenyl]propanamide
—— (2S)-2-(2,5-dioxopyrrolidin-1-yl)-N-[3-(6-oxo-1H-pyridazin-3-yl)phenyl]propanamide —— C17H16N4O4
(2S)-2-(2,5-dioxopyrrolidin-1-yl)-N-[3-(6-oxo-1H-pyridazin-3-yl)phenyl]propanamide
—— (2S)-1-(2-phenyl-5,7-dihydropyrrolo[3,4-d]pyrimidin-6-yl)-2-pyrazol-1-ylbutan-1-one —— C19H19N5O
(2S)-1-(2-phenyl-5,7-dihydropyrrolo[3,4-d]pyrimidin-6-yl)-2-pyrazol-1-ylbutan-1-one
—— (4R)-N-(1-adamantyl)-6-methyl-2-oxo-4-pyridin-3-yl-3,4-dihydro-1H-pyrimidine-5-carboxamide —— C21H26N4O2
(4R)-N-(1-adamantyl)-6-methyl-2-oxo-4-pyridin-3-yl-3,4-dihydro-1H-pyrimidine-5-carboxamide
—— (4S)-N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-4,6-dimethyl-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxamide —— C14H21N5O2
(4S)-N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-4,6-dimethyl-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxamide
—— N-[(1R)-2-methyl-1-(6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)propyl]-2-pyridin-3-ylpyrimidine-5-carboxamide —— C20H24N8O
N-[(1R)-2-methyl-1-(6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)propyl]-2-pyridin-3-ylpyrimidine-5-carboxamide
—— ethyl (6S)-6-[3-(butanoylamino)phenyl]-3-ethyl-4-methyl-2-sulfanylidene-1,6-dihydropyrimidine-5-carboxylate —— C20H27N3O3S
ethyl (6S)-6-[3-(butanoylamino)phenyl]-3-ethyl-4-methyl-2-sulfanylidene-1,6-dihydropyrimidine-5-carboxylate
—— (4S)-N-(1-adamantyl)-6-methyl-2-oxo-4-pyridin-3-yl-3,4-dihydro-1H-pyrimidine-5-carboxamide —— C21H26N4O2
(4S)-N-(1-adamantyl)-6-methyl-2-oxo-4-pyridin-3-yl-3,4-dihydro-1H-pyrimidine-5-carboxamide
—— (4R)-N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-4,6-dimethyl-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxamide —— C14H21N5O2
(4R)-N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-4,6-dimethyl-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxamide
—— 6-(1-methylimidazol-2-yl)-N-[(2S)-2-morpholin-4-yl-2-pyridin-2-ylethyl]pyridazin-3-amine —— C19H23N7O
6-(1-methylimidazol-2-yl)-N-[(2S)-2-morpholin-4-yl-2-pyridin-2-ylethyl]pyridazin-3-amine
—— (1S)-N-methyl-1-pyridin-3-yl-N-[(2-pyridin-2-ylpyrimidin-5-yl)methyl]ethanamine —— C18H19N5
(1S)-N-methyl-1-pyridin-3-yl-N-[(2-pyridin-2-ylpyrimidin-5-yl)methyl]ethanamine
—— (4S)-4,6-dimethyl-2-oxo-N-(2-propoxyethyl)-3,4-dihydro-1H-pyrimidine-5-carboxamide —— C12H21N3O3
(4S)-4,6-dimethyl-2-oxo-N-(2-propoxyethyl)-3,4-dihydro-1H-pyrimidine-5-carboxamide
—— (4R)-5-(3-ethyl-1,4,6,7-tetrahydropyrazolo[4,3-c]pyridine-5-carbonyl)-6-methyl-4-thiophen-2-yl-3,4-dihydro-1H-pyrimidin-2-one —— C18H21N5O2S
(4R)-5-(3-ethyl-1,4,6,7-tetrahydropyrazolo[4,3-c]pyridine-5-carbonyl)-6-methyl-4-thiophen-2-yl-3,4-dihydro-1H-pyrimidin-2-one
—— (4R)-4,6-dimethyl-2-oxo-N-(2-propoxyethyl)-3,4-dihydro-1H-pyrimidine-5-carboxamide —— C12H21N3O3
(4R)-4,6-dimethyl-2-oxo-N-(2-propoxyethyl)-3,4-dihydro-1H-pyrimidine-5-carboxamide
—— N-[[(3S)-1-[(E)-2-methylpent-2-enyl]pyrrolidin-3-yl]methyl]pyrimidine-4-carboxamide —— C16H24N4O
N-[[(3S)-1-[(E)-2-methylpent-2-enyl]pyrrolidin-3-yl]methyl]pyrimidine-4-carboxamide
—— 6-(2-methoxyphenyl)-N-[(1S)-1-(4-methyl-1,3-thiazol-2-yl)ethyl]pyridazin-3-amine —— C17H18N4OS
6-(2-methoxyphenyl)-N-[(1S)-1-(4-methyl-1,3-thiazol-2-yl)ethyl]pyridazin-3-amine
—— 6-(2-methoxyphenyl)-N-[(1R)-1-(4-methyl-1,3-thiazol-2-yl)ethyl]pyridazin-3-amine —— C17H18N4OS
6-(2-methoxyphenyl)-N-[(1R)-1-(4-methyl-1,3-thiazol-2-yl)ethyl]pyridazin-3-amine