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二嗪类

中文名称 英文名称 CAS号 化学式 结构式图片
—— (2R)-1-(2-tert-butyl-5,7-dihydropyrrolo[3,4-d]pyrimidin-6-yl)-2-pyrazol-1-ylpropan-1-one —— C16H21N5O
(2R)-1-(2-tert-butyl-5,7-dihydropyrrolo[3,4-d]pyrimidin-6-yl)-2-pyrazol-1-ylpropan-1-one
—— (4R)-N-[(4-ethyl-1,3-thiazol-2-yl)methyl]-4,6-dimethyl-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxamide —— C13H18N4O2S
(4R)-N-[(4-ethyl-1,3-thiazol-2-yl)methyl]-4,6-dimethyl-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxamide
—— N-[(2S)-1-pyrazin-2-ylpropan-2-yl]-2-pyridin-4-yl-5,6,7,8-tetrahydropyrido[3,4-d]pyrimidin-4-amine —— C19H21N7
N-[(2S)-1-pyrazin-2-ylpropan-2-yl]-2-pyridin-4-yl-5,6,7,8-tetrahydropyrido[3,4-d]pyrimidin-4-amine
—— (3R)-3-(2-methoxyethyl)-1-(6-phenylpyridazin-3-yl)piperidine-3-carboxylic acid —— C19H23N3O3
(3R)-3-(2-methoxyethyl)-1-(6-phenylpyridazin-3-yl)piperidine-3-carboxylic acid
—— 2,4-dimethyl-N-[[(3R)-1-[(5-methyl-1H-pyrazol-3-yl)methyl]pyrrolidin-3-yl]methyl]pyrimidine-5-carboxamide —— C17H24N6O
2,4-dimethyl-N-[[(3R)-1-[(5-methyl-1H-pyrazol-3-yl)methyl]pyrrolidin-3-yl]methyl]pyrimidine-5-carboxamide
—— (3S)-3-(2-methoxyethyl)-1-(6-phenylpyridazin-3-yl)piperidine-3-carboxylic acid —— C19H23N3O3
(3S)-3-(2-methoxyethyl)-1-(6-phenylpyridazin-3-yl)piperidine-3-carboxylic acid
—— N-[(1S)-1-(1-methylimidazol-2-yl)butyl]-2-pyridin-3-yl-5,6,7,8-tetrahydropyrido[3,4-d]pyrimidin-4-amine —— C20H25N7
N-[(1S)-1-(1-methylimidazol-2-yl)butyl]-2-pyridin-3-yl-5,6,7,8-tetrahydropyrido[3,4-d]pyrimidin-4-amine
—— N-[(1R)-1-(1-methylimidazol-2-yl)butyl]-2-pyridin-3-yl-5,6,7,8-tetrahydropyrido[3,4-d]pyrimidin-4-amine —— C20H25N7
N-[(1R)-1-(1-methylimidazol-2-yl)butyl]-2-pyridin-3-yl-5,6,7,8-tetrahydropyrido[3,4-d]pyrimidin-4-amine
—— N-methyl-N-[(1S,2S)-2-methylcyclohexyl]-3-(3-pyrimidin-2-yl-1,2,4-oxadiazol-5-yl)propanamide —— C17H23N5O2
N-methyl-N-[(1S,2S)-2-methylcyclohexyl]-3-(3-pyrimidin-2-yl-1,2,4-oxadiazol-5-yl)propanamide
—— (4S)-4,6-dimethyl-N-[2-(2-methylimidazo[2,1-b][1,3,4]thiadiazol-6-yl)ethyl]-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxamide —— C14H18N6O2S
(4S)-4,6-dimethyl-N-[2-(2-methylimidazo[2,1-b][1,3,4]thiadiazol-6-yl)ethyl]-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxamide
—— (4R)-4,6-dimethyl-N-[2-(2-methylimidazo[2,1-b][1,3,4]thiadiazol-6-yl)ethyl]-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxamide —— C14H18N6O2S
(4R)-4,6-dimethyl-N-[2-(2-methylimidazo[2,1-b][1,3,4]thiadiazol-6-yl)ethyl]-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxamide
—— N-[(2R,6S)-2,6-dimethylcyclohexyl]-3-(3-pyrimidin-2-yl-1,2,4-oxadiazol-5-yl)propanamide —— C17H23N5O2
N-[(2R,6S)-2,6-dimethylcyclohexyl]-3-(3-pyrimidin-2-yl-1,2,4-oxadiazol-5-yl)propanamide
—— 2,6-dimethoxy-N-[2-[(2S)-4-methylmorpholin-2-yl]ethyl]pyrimidine-4-carboxamide —— C14H22N4O4
2,6-dimethoxy-N-[2-[(2S)-4-methylmorpholin-2-yl]ethyl]pyrimidine-4-carboxamide
—— N-[(2R)-1-pyrazin-2-ylpropan-2-yl]-2-pyridin-4-yl-5,6,7,8-tetrahydropyrido[3,4-d]pyrimidin-4-amine —— C19H21N7
N-[(2R)-1-pyrazin-2-ylpropan-2-yl]-2-pyridin-4-yl-5,6,7,8-tetrahydropyrido[3,4-d]pyrimidin-4-amine
—— 6-(1-methylimidazol-2-yl)-N-[(1S)-1-phenylethyl]pyridazin-3-amine —— C16H17N5
6-(1-methylimidazol-2-yl)-N-[(1S)-1-phenylethyl]pyridazin-3-amine
—— 2,6-dimethoxy-N-[2-[(2R)-4-methylmorpholin-2-yl]ethyl]pyrimidine-4-carboxamide —— C14H22N4O4
2,6-dimethoxy-N-[2-[(2R)-4-methylmorpholin-2-yl]ethyl]pyrimidine-4-carboxamide
—— N-[(2S,6S)-2,6-dimethylcyclohexyl]-3-(3-pyrimidin-2-yl-1,2,4-oxadiazol-5-yl)propanamide —— C17H23N5O2
N-[(2S,6S)-2,6-dimethylcyclohexyl]-3-(3-pyrimidin-2-yl-1,2,4-oxadiazol-5-yl)propanamide
—— ethyl (4R)-4-methyl-2-oxo-6-[(4-propan-2-yl-1,2,4-triazol-3-yl)sulfanylmethyl]-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C14H21N5O3S
ethyl (4R)-4-methyl-2-oxo-6-[(4-propan-2-yl-1,2,4-triazol-3-yl)sulfanylmethyl]-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— N-methyl-N-[(1R,2R)-2-methylcyclohexyl]-3-(3-pyrimidin-2-yl-1,2,4-oxadiazol-5-yl)propanamide —— C17H23N5O2
N-methyl-N-[(1R,2R)-2-methylcyclohexyl]-3-(3-pyrimidin-2-yl-1,2,4-oxadiazol-5-yl)propanamide
—— [(3R)-3-(4-ethyl-1H-pyrazol-5-yl)piperidin-1-yl]-(4-methyl-2-propan-2-ylpyrimidin-5-yl)methanone —— C19H27N5O
[(3R)-3-(4-ethyl-1H-pyrazol-5-yl)piperidin-1-yl]-(4-methyl-2-propan-2-ylpyrimidin-5-yl)methanone
—— N-[(2R,6R)-2,6-dimethylcyclohexyl]-3-(3-pyrimidin-2-yl-1,2,4-oxadiazol-5-yl)propanamide —— C17H23N5O2
N-[(2R,6R)-2,6-dimethylcyclohexyl]-3-(3-pyrimidin-2-yl-1,2,4-oxadiazol-5-yl)propanamide
—— ethyl (4S)-6-[[2-(3,4-dimethylphenyl)sulfanylacetyl]oxymethyl]-4-methyl-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C19H24N2O5S
ethyl (4S)-6-[[2-(3,4-dimethylphenyl)sulfanylacetyl]oxymethyl]-4-methyl-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— [(3S)-3-(4-ethyl-1H-pyrazol-5-yl)piperidin-1-yl]-(4-methyl-2-propan-2-ylpyrimidin-5-yl)methanone —— C19H27N5O
[(3S)-3-(4-ethyl-1H-pyrazol-5-yl)piperidin-1-yl]-(4-methyl-2-propan-2-ylpyrimidin-5-yl)methanone
—— N-methyl-N-[(1R,2S)-2-methylcyclohexyl]-3-(3-pyrimidin-2-yl-1,2,4-oxadiazol-5-yl)propanamide —— C17H23N5O2
N-methyl-N-[(1R,2S)-2-methylcyclohexyl]-3-(3-pyrimidin-2-yl-1,2,4-oxadiazol-5-yl)propanamide
—— N-methyl-N-[(1S,2R)-2-methylcyclohexyl]-3-(3-pyrimidin-2-yl-1,2,4-oxadiazol-5-yl)propanamide —— C17H23N5O2
N-methyl-N-[(1S,2R)-2-methylcyclohexyl]-3-(3-pyrimidin-2-yl-1,2,4-oxadiazol-5-yl)propanamide
—— N-[[(3S)-1-[(E)-3-(furan-2-yl)prop-2-enyl]piperidin-3-yl]methyl]-5-methylpyrazine-2-carboxamide —— C19H24N4O2
N-[[(3S)-1-[(E)-3-(furan-2-yl)prop-2-enyl]piperidin-3-yl]methyl]-5-methylpyrazine-2-carboxamide
—— ethyl (4R)-6-[[2-(3,4-dimethylphenyl)sulfanylacetyl]oxymethyl]-4-methyl-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C19H24N2O5S
ethyl (4R)-6-[[2-(3,4-dimethylphenyl)sulfanylacetyl]oxymethyl]-4-methyl-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— ethyl (4S)-4-methyl-2-oxo-6-[(4-propan-2-yl-1,2,4-triazol-3-yl)sulfanylmethyl]-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C14H21N5O3S
ethyl (4S)-4-methyl-2-oxo-6-[(4-propan-2-yl-1,2,4-triazol-3-yl)sulfanylmethyl]-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— (4R)-6-methyl-N-[3-(4-methyl-1,3-thiazol-5-yl)propyl]-2-oxo-4-thiophen-3-yl-3,4-dihydro-1H-pyrimidine-5-carboxamide —— C17H20N4O2S2
(4R)-6-methyl-N-[3-(4-methyl-1,3-thiazol-5-yl)propyl]-2-oxo-4-thiophen-3-yl-3,4-dihydro-1H-pyrimidine-5-carboxamide
—— N-[[(3R)-1-[(E)-3-(furan-2-yl)prop-2-enyl]piperidin-3-yl]methyl]-5-methylpyrazine-2-carboxamide —— C19H24N4O2
N-[[(3R)-1-[(E)-3-(furan-2-yl)prop-2-enyl]piperidin-3-yl]methyl]-5-methylpyrazine-2-carboxamide
—— (4S)-6-methyl-N-[3-(4-methyl-1,3-thiazol-5-yl)propyl]-2-oxo-4-thiophen-3-yl-3,4-dihydro-1H-pyrimidine-5-carboxamide —— C17H20N4O2S2
(4S)-6-methyl-N-[3-(4-methyl-1,3-thiazol-5-yl)propyl]-2-oxo-4-thiophen-3-yl-3,4-dihydro-1H-pyrimidine-5-carboxamide
—— (2-anilinopyrimidin-5-yl)-[(3R)-3-(1H-pyrazol-5-yl)piperidin-1-yl]methanone —— C19H20N6O
(2-anilinopyrimidin-5-yl)-[(3R)-3-(1H-pyrazol-5-yl)piperidin-1-yl]methanone
—— 4-[(3S)-1-(furan-2-ylmethyl)piperidin-3-yl]-2-pyrazin-2-yl-1H-pyrimidin-6-one —— C18H19N5O2
4-[(3S)-1-(furan-2-ylmethyl)piperidin-3-yl]-2-pyrazin-2-yl-1H-pyrimidin-6-one
—— (1R)-N-[2-(3,6-dioxo-1H-pyridazin-2-yl)ethyl]-2,2-dimethyl-1-thiophen-2-ylcyclopropane-1-carboxamide —— C16H19N3O3S
(1R)-N-[2-(3,6-dioxo-1H-pyridazin-2-yl)ethyl]-2,2-dimethyl-1-thiophen-2-ylcyclopropane-1-carboxamide
—— (1S)-N-[2-(3,6-dioxo-1H-pyridazin-2-yl)ethyl]-2,2-dimethyl-1-thiophen-2-ylcyclopropane-1-carboxamide —— C16H19N3O3S
(1S)-N-[2-(3,6-dioxo-1H-pyridazin-2-yl)ethyl]-2,2-dimethyl-1-thiophen-2-ylcyclopropane-1-carboxamide
—— (2-anilinopyrimidin-5-yl)-[(3S)-3-(1H-pyrazol-5-yl)piperidin-1-yl]methanone —— C19H20N6O
(2-anilinopyrimidin-5-yl)-[(3S)-3-(1H-pyrazol-5-yl)piperidin-1-yl]methanone
—— 4-[(3R)-1-(furan-2-ylmethyl)piperidin-3-yl]-2-pyrazin-2-yl-1H-pyrimidin-6-one —— C18H19N5O2
4-[(3R)-1-(furan-2-ylmethyl)piperidin-3-yl]-2-pyrazin-2-yl-1H-pyrimidin-6-one
—— 6-(1-methylimidazol-2-yl)-N-[(1S)-1-(5-methyl-1H-1,2,4-triazol-3-yl)ethyl]pyridazin-3-amine —— C13H16N8
6-(1-methylimidazol-2-yl)-N-[(1S)-1-(5-methyl-1H-1,2,4-triazol-3-yl)ethyl]pyridazin-3-amine
—— 6-[(2S)-2-(aminomethyl)-5-fluoro-2,3-dihydro-1-benzofuran-7-yl]-N,N-dimethylpyrazine-2-carboxamide —— C16H17FN4O2
6-[(2S)-2-(aminomethyl)-5-fluoro-2,3-dihydro-1-benzofuran-7-yl]-N,N-dimethylpyrazine-2-carboxamide
—— (7S)-7-[4-(dimethylamino)phenyl]-N-(2,4-dimethylphenyl)-5-methyl-4,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide —— C22H25N7O
(7S)-7-[4-(dimethylamino)phenyl]-N-(2,4-dimethylphenyl)-5-methyl-4,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide
—— 2-[2-[[(2R)-1-morpholin-4-ylpropan-2-yl]amino]ethyl]-1H-pyridazine-3,6-dione —— C13H22N4O3
2-[2-[[(2R)-1-morpholin-4-ylpropan-2-yl]amino]ethyl]-1H-pyridazine-3,6-dione
—— 6-(1-methylimidazol-2-yl)-N-[(1R)-1-(5-methyl-1H-1,2,4-triazol-3-yl)ethyl]pyridazin-3-amine —— C13H16N8
6-(1-methylimidazol-2-yl)-N-[(1R)-1-(5-methyl-1H-1,2,4-triazol-3-yl)ethyl]pyridazin-3-amine
—— N-[(1R)-1-[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]ethyl]-2-pyridin-3-yl-5,6,7,8-tetrahydropyrido[3,4-d]pyrimidin-4-amine —— C20H25N7O
N-[(1R)-1-[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]ethyl]-2-pyridin-3-yl-5,6,7,8-tetrahydropyrido[3,4-d]pyrimidin-4-amine
—— N-[(1S)-1-[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]ethyl]-2-pyridin-3-yl-5,6,7,8-tetrahydropyrido[3,4-d]pyrimidin-4-amine —— C20H25N7O
N-[(1S)-1-[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]ethyl]-2-pyridin-3-yl-5,6,7,8-tetrahydropyrido[3,4-d]pyrimidin-4-amine
—— N-[[(3S)-1-(2,2,6,6-tetramethylpiperidin-4-yl)pyrrolidin-3-yl]methyl]pyrazine-2-carboxamide —— C19H31N5O
N-[[(3S)-1-(2,2,6,6-tetramethylpiperidin-4-yl)pyrrolidin-3-yl]methyl]pyrazine-2-carboxamide
—— N-[[(3R)-1-(2,2,6,6-tetramethylpiperidin-4-yl)pyrrolidin-3-yl]methyl]pyrazine-2-carboxamide —— C19H31N5O
N-[[(3R)-1-(2,2,6,6-tetramethylpiperidin-4-yl)pyrrolidin-3-yl]methyl]pyrazine-2-carboxamide
—— [2-amino-4-(4-methoxyphenyl)-5,7-dihydropyrrolo[3,4-d]pyrimidin-6-yl]-[(3R)-1-methylpiperidin-3-yl]methanone —— C20H25N5O2
[2-amino-4-(4-methoxyphenyl)-5,7-dihydropyrrolo[3,4-d]pyrimidin-6-yl]-[(3R)-1-methylpiperidin-3-yl]methanone
—— 6-(aminomethyl)-N-[(1S)-1-(1,3-dimethylpyrazol-4-yl)ethyl]pyrimidin-4-amine —— C12H18N6
6-(aminomethyl)-N-[(1S)-1-(1,3-dimethylpyrazol-4-yl)ethyl]pyrimidin-4-amine
—— [2-amino-4-(4-methoxyphenyl)-5,7-dihydropyrrolo[3,4-d]pyrimidin-6-yl]-[(3S)-1-methylpiperidin-3-yl]methanone —— C20H25N5O2
[2-amino-4-(4-methoxyphenyl)-5,7-dihydropyrrolo[3,4-d]pyrimidin-6-yl]-[(3S)-1-methylpiperidin-3-yl]methanone
—— (4R)-4,6-dimethyl-N,N-bis(2-methylpropyl)-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxamide —— C15H27N3O2
(4R)-4,6-dimethyl-N,N-bis(2-methylpropyl)-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxamide