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二嗪类

中文名称 英文名称 CAS号 化学式 结构式图片
—— N-methyl-N-[[5-[(1S,2S)-2-methylcyclopropyl]furan-2-yl]methyl]-2-phenylpyrimidine-5-carboxamide —— C21H21N3O2
N-methyl-N-[[5-[(1S,2S)-2-methylcyclopropyl]furan-2-yl]methyl]-2-phenylpyrimidine-5-carboxamide
—— (1R)-N-(5-ethyl-2-methylpyrimidin-4-yl)-N',N'-dimethyl-1-phenylethane-1,2-diamine —— C17H24N4
(1R)-N-(5-ethyl-2-methylpyrimidin-4-yl)-N',N'-dimethyl-1-phenylethane-1,2-diamine
—— [(2R)-2-(4-methoxyphenyl)azepan-1-yl]-(2-methylpyrimidin-4-yl)methanone —— C19H23N3O2
[(2R)-2-(4-methoxyphenyl)azepan-1-yl]-(2-methylpyrimidin-4-yl)methanone
—— [(2S)-2-(4-methoxyphenyl)azepan-1-yl]-(2-methylpyrimidin-4-yl)methanone —— C19H23N3O2
[(2S)-2-(4-methoxyphenyl)azepan-1-yl]-(2-methylpyrimidin-4-yl)methanone
—— (9aR)-8-methyl-2-(2-pyridin-2-ylpyrimidine-5-carbonyl)-1,3,4,6,7,9a-hexahydropyrazino[1,2-a]pyrazin-9-one —— C18H20N6O2
(9aR)-8-methyl-2-(2-pyridin-2-ylpyrimidine-5-carbonyl)-1,3,4,6,7,9a-hexahydropyrazino[1,2-a]pyrazin-9-one
—— (9aS)-8-methyl-2-(2-pyridin-2-ylpyrimidine-5-carbonyl)-1,3,4,6,7,9a-hexahydropyrazino[1,2-a]pyrazin-9-one —— C18H20N6O2
(9aS)-8-methyl-2-(2-pyridin-2-ylpyrimidine-5-carbonyl)-1,3,4,6,7,9a-hexahydropyrazino[1,2-a]pyrazin-9-one
—— [(4R)-5-ethoxycarbonyl-4-methyl-2-oxo-3,4-dihydro-1H-pyrimidin-6-yl]methyl 5-methyl-3-phenyl-1,2-oxazole-4-carboxylate —— C20H21N3O6
[(4R)-5-ethoxycarbonyl-4-methyl-2-oxo-3,4-dihydro-1H-pyrimidin-6-yl]methyl 5-methyl-3-phenyl-1,2-oxazole-4-carboxylate
—— prop-2-enyl 4-[(3S)-4-benzoyl-3-methylpiperazine-1-carbonyl]-2,6-dimethylpyrimidine-5-carboxylate —— C23H26N4O4
prop-2-enyl 4-[(3S)-4-benzoyl-3-methylpiperazine-1-carbonyl]-2,6-dimethylpyrimidine-5-carboxylate
—— prop-2-enyl 4-[(3R)-4-benzoyl-3-methylpiperazine-1-carbonyl]-2,6-dimethylpyrimidine-5-carboxylate —— C23H26N4O4
prop-2-enyl 4-[(3R)-4-benzoyl-3-methylpiperazine-1-carbonyl]-2,6-dimethylpyrimidine-5-carboxylate
—— 5-(6-aminopyridin-3-yl)-4-(4-methylphenyl)-N-[(1S)-1-pyrimidin-4-ylethyl]pyrimidin-2-amine —— C22H21N7
5-(6-aminopyridin-3-yl)-4-(4-methylphenyl)-N-[(1S)-1-pyrimidin-4-ylethyl]pyrimidin-2-amine
—— 5-(6-aminopyridin-3-yl)-4-(4-methylphenyl)-N-[(1R)-1-pyrimidin-4-ylethyl]pyrimidin-2-amine —— C22H21N7
5-(6-aminopyridin-3-yl)-4-(4-methylphenyl)-N-[(1R)-1-pyrimidin-4-ylethyl]pyrimidin-2-amine
—— 2-ethyl-6-methyl-N-[(2S)-1-(5-methyl-1H-pyrazol-3-yl)propan-2-yl]pyrimidin-4-amine —— C14H21N5
2-ethyl-6-methyl-N-[(2S)-1-(5-methyl-1H-pyrazol-3-yl)propan-2-yl]pyrimidin-4-amine
—— 2-ethyl-6-methyl-N-[(2R)-1-(5-methyl-1H-pyrazol-3-yl)propan-2-yl]pyrimidin-4-amine —— C14H21N5
2-ethyl-6-methyl-N-[(2R)-1-(5-methyl-1H-pyrazol-3-yl)propan-2-yl]pyrimidin-4-amine
—— N-(cyclobutylmethyl)-N-[[(2S)-oxolan-2-yl]methyl]-2-pyridin-3-ylpyrimidine-5-carboxamide —— C20H24N4O2
N-(cyclobutylmethyl)-N-[[(2S)-oxolan-2-yl]methyl]-2-pyridin-3-ylpyrimidine-5-carboxamide
—— N-(cyclobutylmethyl)-N-[[(2R)-oxolan-2-yl]methyl]-2-pyridin-3-ylpyrimidine-5-carboxamide —— C20H24N4O2
N-(cyclobutylmethyl)-N-[[(2R)-oxolan-2-yl]methyl]-2-pyridin-3-ylpyrimidine-5-carboxamide
—— methyl (4R)-4-(2,4-dimethylphenyl)-6-[(1-methyltetrazol-5-yl)sulfanylmethyl]-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C17H20N6O3S
methyl (4R)-4-(2,4-dimethylphenyl)-6-[(1-methyltetrazol-5-yl)sulfanylmethyl]-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— methyl (4S)-4-(2,4-dimethylphenyl)-6-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanylmethyl]-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C18H20N4O3S2
methyl (4S)-4-(2,4-dimethylphenyl)-6-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanylmethyl]-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— methyl (4R)-4-(2,4-dimethylphenyl)-2-oxo-6-(pyrrolidin-1-ylmethyl)-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C19H25N3O3
methyl (4R)-4-(2,4-dimethylphenyl)-2-oxo-6-(pyrrolidin-1-ylmethyl)-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— 2-[2-[(2R,6R)-2,6-dimethylpiperidin-1-yl]-2-oxoethyl]-6-(2-fluorophenyl)pyridazin-3-one —— C19H22FN3O2
2-[2-[(2R,6R)-2,6-dimethylpiperidin-1-yl]-2-oxoethyl]-6-(2-fluorophenyl)pyridazin-3-one
—— 2-[2-[(2S,6S)-2,6-dimethylpiperidin-1-yl]-2-oxoethyl]-6-(2-fluorophenyl)pyridazin-3-one —— C19H22FN3O2
2-[2-[(2S,6S)-2,6-dimethylpiperidin-1-yl]-2-oxoethyl]-6-(2-fluorophenyl)pyridazin-3-one
—— methyl (4S)-6-[(5-amino-1,3,4-thiadiazol-2-yl)sulfanylmethyl]-4-(2,5-dimethylphenyl)-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C17H19N5O3S2
methyl (4S)-6-[(5-amino-1,3,4-thiadiazol-2-yl)sulfanylmethyl]-4-(2,5-dimethylphenyl)-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— methyl (4R)-4-(2,5-dimethylphenyl)-6-[(2-morpholin-4-ylethylamino)methyl]-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C21H30N4O4
methyl (4R)-4-(2,5-dimethylphenyl)-6-[(2-morpholin-4-ylethylamino)methyl]-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— methyl (4S)-4-(2,5-dimethylphenyl)-6-[(2-morpholin-4-ylethylamino)methyl]-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C21H30N4O4
methyl (4S)-4-(2,5-dimethylphenyl)-6-[(2-morpholin-4-ylethylamino)methyl]-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— methyl (4S)-6-[(5-amino-1,3,4-thiadiazol-2-yl)sulfanylmethyl]-4-(2,4-dimethylphenyl)-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C17H19N5O3S2
methyl (4S)-6-[(5-amino-1,3,4-thiadiazol-2-yl)sulfanylmethyl]-4-(2,4-dimethylphenyl)-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— methyl (4R)-4-(2,4-dimethylphenyl)-6-[(4-methylpiperazin-1-yl)methyl]-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C20H28N4O3
methyl (4R)-4-(2,4-dimethylphenyl)-6-[(4-methylpiperazin-1-yl)methyl]-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— methyl (4R)-6-[(5-amino-1,3,4-thiadiazol-2-yl)sulfanylmethyl]-4-(2,5-dimethylphenyl)-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C17H19N5O3S2
methyl (4R)-6-[(5-amino-1,3,4-thiadiazol-2-yl)sulfanylmethyl]-4-(2,5-dimethylphenyl)-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— methyl (4R)-6-[(5-amino-1,3,4-thiadiazol-2-yl)sulfanylmethyl]-4-(2,4-dimethylphenyl)-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C17H19N5O3S2
methyl (4R)-6-[(5-amino-1,3,4-thiadiazol-2-yl)sulfanylmethyl]-4-(2,4-dimethylphenyl)-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— methyl (4S)-4-(2,5-dimethylphenyl)-6-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanylmethyl]-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C18H20N4O3S2
methyl (4S)-4-(2,5-dimethylphenyl)-6-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanylmethyl]-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— 2-[2-[(2S,6R)-2,6-dimethylpiperidin-1-yl]-2-oxoethyl]-6-(2-fluorophenyl)pyridazin-3-one —— C19H22FN3O2
2-[2-[(2S,6R)-2,6-dimethylpiperidin-1-yl]-2-oxoethyl]-6-(2-fluorophenyl)pyridazin-3-one
—— methyl (4R)-4-(2,4-dimethylphenyl)-6-[(4-ethylpiperazin-1-yl)methyl]-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C21H30N4O3
methyl (4R)-4-(2,4-dimethylphenyl)-6-[(4-ethylpiperazin-1-yl)methyl]-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— methyl (4R)-4-(2,5-dimethylphenyl)-6-[(4-ethylpiperazin-1-yl)methyl]-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C21H30N4O3
methyl (4R)-4-(2,5-dimethylphenyl)-6-[(4-ethylpiperazin-1-yl)methyl]-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— methyl (4R)-4-(2,4-dimethylphenyl)-6-[(2-morpholin-4-ylethylamino)methyl]-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C21H30N4O4
methyl (4R)-4-(2,4-dimethylphenyl)-6-[(2-morpholin-4-ylethylamino)methyl]-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— 5-[(9aS)-8-methyl-3,4,6,7,9,9a-hexahydro-1H-pyrazino[1,2-a]pyrazine-2-carbonyl]-2-methylsulfanyl-1H-pyrimidin-6-one —— C14H21N5O2S
5-[(9aS)-8-methyl-3,4,6,7,9,9a-hexahydro-1H-pyrazino[1,2-a]pyrazine-2-carbonyl]-2-methylsulfanyl-1H-pyrimidin-6-one
—— 5-[[(3R)-3-[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl]methyl]pyrimidin-2-amine —— C16H24N6O
5-[[(3R)-3-[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl]methyl]pyrimidin-2-amine
—— methyl (4S)-4-(2,4-dimethylphenyl)-6-[(4-ethylpiperazin-1-yl)methyl]-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C21H30N4O3
methyl (4S)-4-(2,4-dimethylphenyl)-6-[(4-ethylpiperazin-1-yl)methyl]-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— N,2,6-trimethyl-N-[(1S)-1-(1,3-thiazol-2-yl)ethyl]pyrimidine-4-carboxamide —— C13H16N4OS
N,2,6-trimethyl-N-[(1S)-1-(1,3-thiazol-2-yl)ethyl]pyrimidine-4-carboxamide
—— 5-[[(3S)-3-[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl]methyl]pyrimidin-2-amine —— C16H24N6O
5-[[(3S)-3-[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl]methyl]pyrimidin-2-amine
—— 6-methyl-N-[[(3S)-1-methylsulfonylpiperidin-3-yl]methyl]-2-propylpyrimidin-4-amine —— C15H26N4O2S
6-methyl-N-[[(3S)-1-methylsulfonylpiperidin-3-yl]methyl]-2-propylpyrimidin-4-amine
—— 5-ethyl-2-methyl-N-[(1S)-2-methyl-1-pyridin-2-ylpropyl]pyrimidin-4-amine —— C16H22N4
5-ethyl-2-methyl-N-[(1S)-2-methyl-1-pyridin-2-ylpropyl]pyrimidin-4-amine
—— methyl (4S)-4-(2,5-dimethylphenyl)-6-[(4-ethylpiperazin-1-yl)methyl]-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C21H30N4O3
methyl (4S)-4-(2,5-dimethylphenyl)-6-[(4-ethylpiperazin-1-yl)methyl]-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— N,2,6-trimethyl-N-[(1R)-1-(1,3-thiazol-2-yl)ethyl]pyrimidine-4-carboxamide —— C13H16N4OS
N,2,6-trimethyl-N-[(1R)-1-(1,3-thiazol-2-yl)ethyl]pyrimidine-4-carboxamide
—— 6-methyl-N-[[(3R)-1-methylsulfonylpiperidin-3-yl]methyl]-2-propylpyrimidin-4-amine —— C15H26N4O2S
6-methyl-N-[[(3R)-1-methylsulfonylpiperidin-3-yl]methyl]-2-propylpyrimidin-4-amine
—— (5R)-1-methyl-5-[(2-pyridin-2-yl-6,7,8,9-tetrahydro-5H-pyrimido[4,5-d]azepin-4-yl)amino]piperidin-2-one —— C19H24N6O
(5R)-1-methyl-5-[(2-pyridin-2-yl-6,7,8,9-tetrahydro-5H-pyrimido[4,5-d]azepin-4-yl)amino]piperidin-2-one
—— 6-methyl-N-[[(2S)-4-methylsulfonylmorpholin-2-yl]methyl]-2-propylpyrimidin-4-amine —— C14H24N4O3S
6-methyl-N-[[(2S)-4-methylsulfonylmorpholin-2-yl]methyl]-2-propylpyrimidin-4-amine
—— 3-amino-N-[(1S)-1-[4-(trifluoromethoxy)phenyl]ethyl]pyrazine-2-carboxamide —— C14H13F3N4O2
3-amino-N-[(1S)-1-[4-(trifluoromethoxy)phenyl]ethyl]pyrazine-2-carboxamide
—— 6-methoxy-N-[(2R)-2-pyridin-3-yloxypropyl]pyrimidin-4-amine —— C13H16N4O2
6-methoxy-N-[(2R)-2-pyridin-3-yloxypropyl]pyrimidin-4-amine
—— 6-methoxy-N-[(2S)-2-pyridin-3-yloxypropyl]pyrimidin-4-amine —— C13H16N4O2
6-methoxy-N-[(2S)-2-pyridin-3-yloxypropyl]pyrimidin-4-amine
—— N-[(3S)-1,1-dioxothiolan-3-yl]-6-methoxypyrimidin-4-amine —— C9H13N3O3S
N-[(3S)-1,1-dioxothiolan-3-yl]-6-methoxypyrimidin-4-amine
—— N-[[(3R)-3-(dimethylamino)thiolan-3-yl]methyl]-3-(4,6-dimethyl-2-oxo-1H-pyrimidin-5-yl)propanamide —— C16H26N4O2S
N-[[(3R)-3-(dimethylamino)thiolan-3-yl]methyl]-3-(4,6-dimethyl-2-oxo-1H-pyrimidin-5-yl)propanamide
—— (5S)-1-methyl-5-[(2-pyridin-2-yl-6,7,8,9-tetrahydro-5H-pyrimido[4,5-d]azepin-4-yl)amino]piperidin-2-one —— C19H24N6O
(5S)-1-methyl-5-[(2-pyridin-2-yl-6,7,8,9-tetrahydro-5H-pyrimido[4,5-d]azepin-4-yl)amino]piperidin-2-one