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二嗪类

中文名称 英文名称 CAS号 化学式 结构式图片
—— 5-[(1R)-1-[2-(2-cyclohexylpyrimidin-5-yl)imidazol-1-yl]propyl]-3-methyl-1,2,4-oxadiazole —— C19H24N6O
5-[(1R)-1-[2-(2-cyclohexylpyrimidin-5-yl)imidazol-1-yl]propyl]-3-methyl-1,2,4-oxadiazole
—— [6-[(6R)-6-hydroxy-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-4-yl]pyrazin-2-yl]-pyrrolidin-1-ylmethanone —— C19H29N5O3
[6-[(6R)-6-hydroxy-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-4-yl]pyrazin-2-yl]-pyrrolidin-1-ylmethanone
—— [6-[(6S)-6-hydroxy-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-4-yl]pyrazin-2-yl]-pyrrolidin-1-ylmethanone —— C19H29N5O3
[6-[(6S)-6-hydroxy-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-4-yl]pyrazin-2-yl]-pyrrolidin-1-ylmethanone
—— ethyl 2-[(2S)-1-(2-phenylpyrimidine-5-carbonyl)piperidin-2-yl]acetate —— C20H23N3O3
ethyl 2-[(2S)-1-(2-phenylpyrimidine-5-carbonyl)piperidin-2-yl]acetate
—— 5-[(1S)-1-[2-(2-cyclohexylpyrimidin-5-yl)imidazol-1-yl]propyl]-3-methyl-1,2,4-oxadiazole —— C19H24N6O
5-[(1S)-1-[2-(2-cyclohexylpyrimidin-5-yl)imidazol-1-yl]propyl]-3-methyl-1,2,4-oxadiazole
—— 2-ethoxy-5-[2-[[(3R)-thiolan-3-yl]amino]pyrimidin-4-yl]benzoic acid —— C17H19N3O3S
2-ethoxy-5-[2-[[(3R)-thiolan-3-yl]amino]pyrimidin-4-yl]benzoic acid
—— [2-(dimethylamino)-4-methylpyrimidin-5-yl]-[4-[(1R)-1-hydroxy-2-phenylethyl]piperidin-1-yl]methanone —— C21H28N4O2
[2-(dimethylamino)-4-methylpyrimidin-5-yl]-[4-[(1R)-1-hydroxy-2-phenylethyl]piperidin-1-yl]methanone
—— 2-ethoxy-5-[2-[[(3R)-1-methylpyrrolidin-3-yl]methylamino]pyrimidin-4-yl]benzoic acid —— C19H24N4O3
2-ethoxy-5-[2-[[(3R)-1-methylpyrrolidin-3-yl]methylamino]pyrimidin-4-yl]benzoic acid
—— 2-ethoxy-5-[2-[(2S)-2-methylbutyl]pyrimidin-4-yl]benzoic acid —— C18H22N2O3
2-ethoxy-5-[2-[(2S)-2-methylbutyl]pyrimidin-4-yl]benzoic acid
—— methyl (6S)-6-[4-(cyanomethoxy)phenyl]-3-(3-ethoxypropyl)-4-methyl-2-sulfanylidene-1,6-dihydropyrimidine-5-carboxylate —— C20H25N3O4S
methyl (6S)-6-[4-(cyanomethoxy)phenyl]-3-(3-ethoxypropyl)-4-methyl-2-sulfanylidene-1,6-dihydropyrimidine-5-carboxylate
—— 2-ethoxy-5-[2-[[(3S)-1-methylpyrrolidin-3-yl]methylamino]pyrimidin-4-yl]benzoic acid —— C19H24N4O3
2-ethoxy-5-[2-[[(3S)-1-methylpyrrolidin-3-yl]methylamino]pyrimidin-4-yl]benzoic acid
—— [2-(dimethylamino)-4-methylpyrimidin-5-yl]-[4-[(1S)-1-hydroxy-2-phenylethyl]piperidin-1-yl]methanone —— C21H28N4O2
[2-(dimethylamino)-4-methylpyrimidin-5-yl]-[4-[(1S)-1-hydroxy-2-phenylethyl]piperidin-1-yl]methanone
—— 1-[4-[[(2R)-4-pyrazol-1-ylbutan-2-yl]amino]-2-pyridin-2-yl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-7-yl]ethanone —— C21H25N7O
1-[4-[[(2R)-4-pyrazol-1-ylbutan-2-yl]amino]-2-pyridin-2-yl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-7-yl]ethanone
—— 1-[4-[[(2S)-4-pyrazol-1-ylbutan-2-yl]amino]-2-pyridin-2-yl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-7-yl]ethanone —— C21H25N7O
1-[4-[[(2S)-4-pyrazol-1-ylbutan-2-yl]amino]-2-pyridin-2-yl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-7-yl]ethanone
—— [4-[(1R)-1-hydroxy-2-phenylethyl]piperidin-1-yl]-(2-methylpyrimidin-5-yl)methanone —— C19H23N3O2
[4-[(1R)-1-hydroxy-2-phenylethyl]piperidin-1-yl]-(2-methylpyrimidin-5-yl)methanone
—— [4-[(1S)-1-hydroxy-2-phenylethyl]piperidin-1-yl]-(2-methylpyrimidin-5-yl)methanone —— C19H23N3O2
[4-[(1S)-1-hydroxy-2-phenylethyl]piperidin-1-yl]-(2-methylpyrimidin-5-yl)methanone
—— 6-[(3R)-3-[(3-methylphenoxy)methyl]piperidine-1-carbonyl]-[1,3]thiazolo[3,2-a]pyrimidin-5-one —— C20H21N3O3S
6-[(3R)-3-[(3-methylphenoxy)methyl]piperidine-1-carbonyl]-[1,3]thiazolo[3,2-a]pyrimidin-5-one
—— 6-[(3S)-3-[(3-methylphenoxy)methyl]piperidine-1-carbonyl]-[1,3]thiazolo[3,2-a]pyrimidin-5-one —— C20H21N3O3S
6-[(3S)-3-[(3-methylphenoxy)methyl]piperidine-1-carbonyl]-[1,3]thiazolo[3,2-a]pyrimidin-5-one
—— N-[(3R)-1,1-dioxothiolan-3-yl]-N-ethyl-2-(2-ethyl-4-methyl-6-oxo-1H-pyrimidin-5-yl)acetamide —— C15H23N3O4S
N-[(3R)-1,1-dioxothiolan-3-yl]-N-ethyl-2-(2-ethyl-4-methyl-6-oxo-1H-pyrimidin-5-yl)acetamide
—— N-[(3S)-1,1-dioxothiolan-3-yl]-N-ethyl-2-(2-ethyl-4-methyl-6-oxo-1H-pyrimidin-5-yl)acetamide —— C15H23N3O4S
N-[(3S)-1,1-dioxothiolan-3-yl]-N-ethyl-2-(2-ethyl-4-methyl-6-oxo-1H-pyrimidin-5-yl)acetamide
—— 5-[[(2S)-2-(2-pyrazol-1-ylethyl)piperidin-1-yl]methyl]-2-pyridin-2-ylpyrimidine —— C20H24N6
5-[[(2S)-2-(2-pyrazol-1-ylethyl)piperidin-1-yl]methyl]-2-pyridin-2-ylpyrimidine
—— 5-[[(2R)-2-(2-pyrazol-1-ylethyl)piperidin-1-yl]methyl]-2-pyridin-2-ylpyrimidine —— C20H24N6
5-[[(2R)-2-(2-pyrazol-1-ylethyl)piperidin-1-yl]methyl]-2-pyridin-2-ylpyrimidine
—— [2-amino-6-(2-methylpropyl)pyrimidin-4-yl]-[(3R)-3-(1H-imidazol-2-yl)piperidin-1-yl]methanone —— C17H24N6O
[2-amino-6-(2-methylpropyl)pyrimidin-4-yl]-[(3R)-3-(1H-imidazol-2-yl)piperidin-1-yl]methanone
—— [2-amino-6-(2-methylpropyl)pyrimidin-4-yl]-[(3S)-3-(1H-imidazol-2-yl)piperidin-1-yl]methanone —— C17H24N6O
[2-amino-6-(2-methylpropyl)pyrimidin-4-yl]-[(3S)-3-(1H-imidazol-2-yl)piperidin-1-yl]methanone
—— 2-amino-N-[(4R)-1,9-dioxaspiro[5.5]undecan-4-yl]-4-phenylpyrimidine-5-carboxamide —— C20H24N4O3
2-amino-N-[(4R)-1,9-dioxaspiro[5.5]undecan-4-yl]-4-phenylpyrimidine-5-carboxamide
—— 2-amino-N-[(4S)-1,9-dioxaspiro[5.5]undecan-4-yl]-4-phenylpyrimidine-5-carboxamide —— C20H24N4O3
2-amino-N-[(4S)-1,9-dioxaspiro[5.5]undecan-4-yl]-4-phenylpyrimidine-5-carboxamide
—— 2-(2-Cycloheptyloxyethyl)-6-cyclopropyl-4-(trifluoromethyl)pyridazin-3-one —— C17H23F3N2O2
2-(2-Cycloheptyloxyethyl)-6-cyclopropyl-4-(trifluoromethyl)pyridazin-3-one
—— N-[(3S,4R)-4-methoxypyrrolidin-3-yl]-6-methylpyridazin-3-amine —— C10H16N4O
N-[(3S,4R)-4-methoxypyrrolidin-3-yl]-6-methylpyridazin-3-amine
—— N-[(3R,4R)-4-methoxypyrrolidin-3-yl]-6-methylpyridazin-3-amine —— C10H16N4O
N-[(3R,4R)-4-methoxypyrrolidin-3-yl]-6-methylpyridazin-3-amine
—— N-[(4S)-1,9-dioxaspiro[5.5]undecan-4-yl]-2-pyrazin-2-ylacetamide —— C15H21N3O3
N-[(4S)-1,9-dioxaspiro[5.5]undecan-4-yl]-2-pyrazin-2-ylacetamide
—— N-[(4R)-1,9-dioxaspiro[5.5]undecan-4-yl]-2-pyrazin-2-ylacetamide —— C15H21N3O3
N-[(4R)-1,9-dioxaspiro[5.5]undecan-4-yl]-2-pyrazin-2-ylacetamide
—— 1-[4-[[(3R)-oxolan-3-yl]amino]-2-pyridin-2-yl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-7-yl]ethanone —— C18H21N5O2
1-[4-[[(3R)-oxolan-3-yl]amino]-2-pyridin-2-yl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-7-yl]ethanone
—— 1-[4-[[(3S)-oxolan-3-yl]amino]-2-pyridin-2-yl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-7-yl]ethanone —— C18H21N5O2
1-[4-[[(3S)-oxolan-3-yl]amino]-2-pyridin-2-yl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-7-yl]ethanone
—— N-[(3R,4R)-4-methoxypyrrolidin-3-yl]pyrimidin-4-amine —— C9H14N4O
N-[(3R,4R)-4-methoxypyrrolidin-3-yl]pyrimidin-4-amine
—— N-[(3S,4R)-4-methoxypyrrolidin-3-yl]pyrimidin-4-amine —— C9H14N4O
N-[(3S,4R)-4-methoxypyrrolidin-3-yl]pyrimidin-4-amine
—— N-[(3R,4R)-4-methoxypyrrolidin-3-yl]-6-methylpyrimidin-4-amine —— C10H16N4O
N-[(3R,4R)-4-methoxypyrrolidin-3-yl]-6-methylpyrimidin-4-amine
—— N-[(3S,4R)-4-methoxypyrrolidin-3-yl]-6-methylpyrimidin-4-amine —— C10H16N4O
N-[(3S,4R)-4-methoxypyrrolidin-3-yl]-6-methylpyrimidin-4-amine
—— 2-ethoxy-5-[2-[(3R)-3-hydroxypiperidin-1-yl]pyrimidin-4-yl]benzoic acid —— C18H21N3O4
2-ethoxy-5-[2-[(3R)-3-hydroxypiperidin-1-yl]pyrimidin-4-yl]benzoic acid
—— (3R)-4-(2-amino-4-phenylpyrimidine-5-carbonyl)-3-methyl-1-(2-methylpropyl)piperazin-2-one —— C20H25N5O2
(3R)-4-(2-amino-4-phenylpyrimidine-5-carbonyl)-3-methyl-1-(2-methylpropyl)piperazin-2-one
—— (3S)-4-(2-amino-4-phenylpyrimidine-5-carbonyl)-3-methyl-1-(2-methylpropyl)piperazin-2-one —— C20H25N5O2
(3S)-4-(2-amino-4-phenylpyrimidine-5-carbonyl)-3-methyl-1-(2-methylpropyl)piperazin-2-one
—— 6-[(2S)-2-(2-pyrazol-1-ylethyl)piperidine-1-carbonyl]-1H-pyrimidine-2,4-dione —— C15H19N5O3
6-[(2S)-2-(2-pyrazol-1-ylethyl)piperidine-1-carbonyl]-1H-pyrimidine-2,4-dione
—— 6-[(2R)-2-(2-pyrazol-1-ylethyl)piperidine-1-carbonyl]-1H-pyrimidine-2,4-dione —— C15H19N5O3
6-[(2R)-2-(2-pyrazol-1-ylethyl)piperidine-1-carbonyl]-1H-pyrimidine-2,4-dione
—— 3-phenyl-6-[(3R)-3-(pyridin-2-ylmethoxy)piperidin-1-yl]pyridazine —— C21H22N4O
3-phenyl-6-[(3R)-3-(pyridin-2-ylmethoxy)piperidin-1-yl]pyridazine
—— 6-[(1S)-1-ethyl-3,4-dihydro-1H-pyrrolo[1,2-a]pyrazine-2-carbonyl]-2,3-dimethyl-[1,3]thiazolo[3,2-a]pyrimidin-5-one —— C18H20N4O2S
6-[(1S)-1-ethyl-3,4-dihydro-1H-pyrrolo[1,2-a]pyrazine-2-carbonyl]-2,3-dimethyl-[1,3]thiazolo[3,2-a]pyrimidin-5-one
—— 3-phenyl-6-[(3S)-3-(pyridin-2-ylmethoxy)piperidin-1-yl]pyridazine —— C21H22N4O
3-phenyl-6-[(3S)-3-(pyridin-2-ylmethoxy)piperidin-1-yl]pyridazine
—— N-methyl-5-methylsulfonyl-4-[(3S)-piperidin-3-yl]pyrimidin-2-amine —— C11H18N4O2S
N-methyl-5-methylsulfonyl-4-[(3S)-piperidin-3-yl]pyrimidin-2-amine
—— [(3S)-3-(4-ethyl-1H-pyrazol-5-yl)piperidin-1-yl]-(4-methyl-2-pyridin-3-ylpyrimidin-5-yl)methanone —— C21H24N6O
[(3S)-3-(4-ethyl-1H-pyrazol-5-yl)piperidin-1-yl]-(4-methyl-2-pyridin-3-ylpyrimidin-5-yl)methanone
—— [(3R)-3-(4-ethyl-1H-pyrazol-5-yl)piperidin-1-yl]-(4-methyl-2-pyridin-3-ylpyrimidin-5-yl)methanone —— C21H24N6O
[(3R)-3-(4-ethyl-1H-pyrazol-5-yl)piperidin-1-yl]-(4-methyl-2-pyridin-3-ylpyrimidin-5-yl)methanone
—— (2-ethylpyrimidin-5-yl)-[4-[(1S)-1-hydroxy-3-phenylpropyl]piperidin-1-yl]methanone —— C21H27N3O2
(2-ethylpyrimidin-5-yl)-[4-[(1S)-1-hydroxy-3-phenylpropyl]piperidin-1-yl]methanone
—— N-[(3R,4R)-4-methoxypyrrolidin-3-yl]-2,6-dimethylpyrimidin-4-amine —— C11H18N4O
N-[(3R,4R)-4-methoxypyrrolidin-3-yl]-2,6-dimethylpyrimidin-4-amine