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二嗪类

中文名称 英文名称 CAS号 化学式 结构式图片
—— ethyl (4S)-6-[[(2S)-1,4-dithiane-2-carbonyl]oxymethyl]-4-(4-methoxyphenyl)-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C20H24N2O6S2
ethyl (4S)-6-[[(2S)-1,4-dithiane-2-carbonyl]oxymethyl]-4-(4-methoxyphenyl)-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— [(2R,4aR,8aR)-1,2,3,4,4a,5,6,7,8,8a-decahydronaphthalen-2-yl] 5-oxo-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C17H20N2O3S
[(2R,4aR,8aR)-1,2,3,4,4a,5,6,7,8,8a-decahydronaphthalen-2-yl] 5-oxo-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— [(2S,4aR,8aR)-1,2,3,4,4a,5,6,7,8,8a-decahydronaphthalen-2-yl] 5-oxo-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C17H20N2O3S
[(2S,4aR,8aR)-1,2,3,4,4a,5,6,7,8,8a-decahydronaphthalen-2-yl] 5-oxo-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— [(2S,4aS,8aR)-1,2,3,4,4a,5,6,7,8,8a-decahydronaphthalen-2-yl] 5-oxo-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C17H20N2O3S
[(2S,4aS,8aR)-1,2,3,4,4a,5,6,7,8,8a-decahydronaphthalen-2-yl] 5-oxo-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— [(2R,4aS,8aR)-1,2,3,4,4a,5,6,7,8,8a-decahydronaphthalen-2-yl] 5-oxo-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C17H20N2O3S
[(2R,4aS,8aR)-1,2,3,4,4a,5,6,7,8,8a-decahydronaphthalen-2-yl] 5-oxo-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— N-[(1R)-1-phenyl-2-pyrazol-1-ylethyl]pyrazine-2-carboxamide —— C16H15N5O
N-[(1R)-1-phenyl-2-pyrazol-1-ylethyl]pyrazine-2-carboxamide
—— N-[(1S)-1-phenyl-2-pyrazol-1-ylethyl]pyrazine-2-carboxamide —— C16H15N5O
N-[(1S)-1-phenyl-2-pyrazol-1-ylethyl]pyrazine-2-carboxamide
—— N-[(2R)-2-phenoxybutyl]-2-pyrimidin-5-ylbenzamide —— C21H21N3O2
N-[(2R)-2-phenoxybutyl]-2-pyrimidin-5-ylbenzamide
—— 2-pyrimidin-5-yl-N-[(5R)-2,3,4,5-tetrahydro-1-benzoxepin-5-yl]benzamide —— C21H19N3O2
2-pyrimidin-5-yl-N-[(5R)-2,3,4,5-tetrahydro-1-benzoxepin-5-yl]benzamide
—— [(3S)-3-(2-methylphenyl)pyrrolidin-1-yl]-(2-pyrimidin-5-ylphenyl)methanone —— C22H21N3O
[(3S)-3-(2-methylphenyl)pyrrolidin-1-yl]-(2-pyrimidin-5-ylphenyl)methanone
—— N-[(3S)-6,7-dimethyl-2,3-dihydro-1-benzofuran-3-yl]-2-pyrimidin-5-ylbenzamide —— C21H19N3O2
N-[(3S)-6,7-dimethyl-2,3-dihydro-1-benzofuran-3-yl]-2-pyrimidin-5-ylbenzamide
—— 2-pyrimidin-5-yl-N-[(5S)-2,3,4,5-tetrahydro-1-benzoxepin-5-yl]benzamide —— C21H19N3O2
2-pyrimidin-5-yl-N-[(5S)-2,3,4,5-tetrahydro-1-benzoxepin-5-yl]benzamide
—— N-[(3R)-6,7-dimethyl-2,3-dihydro-1-benzofuran-3-yl]-2-pyrimidin-5-ylbenzamide —— C21H19N3O2
N-[(3R)-6,7-dimethyl-2,3-dihydro-1-benzofuran-3-yl]-2-pyrimidin-5-ylbenzamide
—— N-[(2S)-2-phenoxybutyl]-2-pyrimidin-5-ylbenzamide —— C21H21N3O2
N-[(2S)-2-phenoxybutyl]-2-pyrimidin-5-ylbenzamide
—— N-[(2R)-1-(2-methylpropoxy)propan-2-yl]-2-pyrimidin-5-ylbenzamide —— C18H23N3O2
N-[(2R)-1-(2-methylpropoxy)propan-2-yl]-2-pyrimidin-5-ylbenzamide
—— [(3R)-3-(2-methylphenyl)pyrrolidin-1-yl]-(2-pyrimidin-5-ylphenyl)methanone —— C22H21N3O
[(3R)-3-(2-methylphenyl)pyrrolidin-1-yl]-(2-pyrimidin-5-ylphenyl)methanone
—— N-[(3R)-oxan-3-yl]-2-pyrimidin-5-ylbenzamide —— C16H17N3O2
N-[(3R)-oxan-3-yl]-2-pyrimidin-5-ylbenzamide
—— N-[(2S)-1-(2-methylpropoxy)propan-2-yl]-2-pyrimidin-5-ylbenzamide —— C18H23N3O2
N-[(2S)-1-(2-methylpropoxy)propan-2-yl]-2-pyrimidin-5-ylbenzamide
—— N-[(3S)-oxan-3-yl]-2-pyrimidin-5-ylbenzamide —— C16H17N3O2
N-[(3S)-oxan-3-yl]-2-pyrimidin-5-ylbenzamide
—— N-[(2S)-1-(3-fluorophenoxy)propan-2-yl]imidazo[1,2-a]pyrazine-8-carboxamide —— C16H15FN4O2
N-[(2S)-1-(3-fluorophenoxy)propan-2-yl]imidazo[1,2-a]pyrazine-8-carboxamide
—— N-[(2S)-3-ethyl-2-morpholin-4-ylpentyl]imidazo[1,2-a]pyrazine-8-carboxamide —— C18H27N5O2
N-[(2S)-3-ethyl-2-morpholin-4-ylpentyl]imidazo[1,2-a]pyrazine-8-carboxamide
—— N-[(2R)-1-(3-fluorophenoxy)propan-2-yl]imidazo[1,2-a]pyrazine-8-carboxamide —— C16H15FN4O2
N-[(2R)-1-(3-fluorophenoxy)propan-2-yl]imidazo[1,2-a]pyrazine-8-carboxamide
—— (3S)-1-methyl-3-[(2-pyridin-4-yl-6,7-dihydro-5H-cyclopenta[d]pyrimidin-4-yl)amino]pyrrolidin-2-one —— C17H19N5O
(3S)-1-methyl-3-[(2-pyridin-4-yl-6,7-dihydro-5H-cyclopenta[d]pyrimidin-4-yl)amino]pyrrolidin-2-one
—— (3R)-1-methyl-3-[(2-pyridin-2-yl-6,7-dihydro-5H-cyclopenta[d]pyrimidin-4-yl)amino]pyrrolidin-2-one —— C17H19N5O
(3R)-1-methyl-3-[(2-pyridin-2-yl-6,7-dihydro-5H-cyclopenta[d]pyrimidin-4-yl)amino]pyrrolidin-2-one
—— (5R)-5-[[6-(3,5-dimethylpyrazol-1-yl)pyridazin-3-yl]amino]-1-methylpiperidin-2-one —— C15H20N6O
(5R)-5-[[6-(3,5-dimethylpyrazol-1-yl)pyridazin-3-yl]amino]-1-methylpiperidin-2-one
—— 4-chloro-2-methyl-5-[[(3R)-1-methyl-6-oxopiperidin-3-yl]amino]pyridazin-3-one —— C11H15ClN4O2
4-chloro-2-methyl-5-[[(3R)-1-methyl-6-oxopiperidin-3-yl]amino]pyridazin-3-one
—— (2S)-2-methyl-1-methylsulfanyl-3-[[4-(trifluoromethyl)pyrimidin-2-yl]amino]propan-2-ol —— C10H14F3N3OS
(2S)-2-methyl-1-methylsulfanyl-3-[[4-(trifluoromethyl)pyrimidin-2-yl]amino]propan-2-ol
—— (2R)-2-methyl-1-methylsulfanyl-3-[[4-(trifluoromethyl)pyrimidin-2-yl]amino]propan-2-ol —— C10H14F3N3OS
(2R)-2-methyl-1-methylsulfanyl-3-[[4-(trifluoromethyl)pyrimidin-2-yl]amino]propan-2-ol
—— (3S)-1-methyl-3-[(2-pyridin-2-yl-6,7-dihydro-5H-cyclopenta[d]pyrimidin-4-yl)amino]pyrrolidin-2-one —— C17H19N5O
(3S)-1-methyl-3-[(2-pyridin-2-yl-6,7-dihydro-5H-cyclopenta[d]pyrimidin-4-yl)amino]pyrrolidin-2-one
—— (3R)-1-methyl-3-[(2-pyridin-4-yl-6,7-dihydro-5H-cyclopenta[d]pyrimidin-4-yl)amino]pyrrolidin-2-one —— C17H19N5O
(3R)-1-methyl-3-[(2-pyridin-4-yl-6,7-dihydro-5H-cyclopenta[d]pyrimidin-4-yl)amino]pyrrolidin-2-one
—— N-[(2R)-3-ethyl-2-morpholin-4-ylpentyl]imidazo[1,2-a]pyrazine-8-carboxamide —— C18H27N5O2
N-[(2R)-3-ethyl-2-morpholin-4-ylpentyl]imidazo[1,2-a]pyrazine-8-carboxamide
—— 4-bromo-2-methyl-5-[[(3S)-1-methyl-6-oxopiperidin-3-yl]amino]pyridazin-3-one —— C11H15BrN4O2
4-bromo-2-methyl-5-[[(3S)-1-methyl-6-oxopiperidin-3-yl]amino]pyridazin-3-one
—— (5S)-5-[[6-(3,5-dimethylpyrazol-1-yl)pyridazin-3-yl]amino]-1-methylpiperidin-2-one —— C15H20N6O
(5S)-5-[[6-(3,5-dimethylpyrazol-1-yl)pyridazin-3-yl]amino]-1-methylpiperidin-2-one
—— (5R)-1-methyl-5-[(2-pyridin-4-yl-6,7-dihydro-5H-cyclopenta[d]pyrimidin-4-yl)amino]piperidin-2-one —— C18H21N5O
(5R)-1-methyl-5-[(2-pyridin-4-yl-6,7-dihydro-5H-cyclopenta[d]pyrimidin-4-yl)amino]piperidin-2-one
—— (1R)-1-cyclopentyl-2-[[6-(3,5-dimethylpyrazol-1-yl)pyridazin-3-yl]amino]ethanol —— C16H23N5O
(1R)-1-cyclopentyl-2-[[6-(3,5-dimethylpyrazol-1-yl)pyridazin-3-yl]amino]ethanol
—— 4-bromo-2-methyl-5-[[(3R)-1-methyl-6-oxopiperidin-3-yl]amino]pyridazin-3-one —— C11H15BrN4O2
4-bromo-2-methyl-5-[[(3R)-1-methyl-6-oxopiperidin-3-yl]amino]pyridazin-3-one
—— (1S)-1-cyclopentyl-2-[[6-(3,5-dimethylpyrazol-1-yl)pyridazin-3-yl]amino]ethanol —— C16H23N5O
(1S)-1-cyclopentyl-2-[[6-(3,5-dimethylpyrazol-1-yl)pyridazin-3-yl]amino]ethanol
—— 4-chloro-2-methyl-5-[[(3S)-1-methyl-6-oxopiperidin-3-yl]amino]pyridazin-3-one —— C11H15ClN4O2
4-chloro-2-methyl-5-[[(3S)-1-methyl-6-oxopiperidin-3-yl]amino]pyridazin-3-one
—— ethyl (4R)-4-ethyl-6-[[(2-fluorophenyl)methyl-methylamino]methyl]-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C18H24FN3O3
ethyl (4R)-4-ethyl-6-[[(2-fluorophenyl)methyl-methylamino]methyl]-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— N-[(1S)-cyclohex-3-en-1-yl]-6-(3-methylpyrazol-1-yl)pyridazin-3-amine —— C14H17N5
N-[(1S)-cyclohex-3-en-1-yl]-6-(3-methylpyrazol-1-yl)pyridazin-3-amine
—— (5S)-1-methyl-5-[(2-pyridin-4-yl-6,7-dihydro-5H-cyclopenta[d]pyrimidin-4-yl)amino]piperidin-2-one —— C18H21N5O
(5S)-1-methyl-5-[(2-pyridin-4-yl-6,7-dihydro-5H-cyclopenta[d]pyrimidin-4-yl)amino]piperidin-2-one
—— N-[(1R)-cyclohex-3-en-1-yl]-6-(3-methylpyrazol-1-yl)pyridazin-3-amine —— C14H17N5
N-[(1R)-cyclohex-3-en-1-yl]-6-(3-methylpyrazol-1-yl)pyridazin-3-amine
—— Imidazo[1,2-a]pyrazin-8-yl-[4-[2-(4-methylphenyl)ethyl]piperidin-1-yl]methanone —— C21H24N4O
Imidazo[1,2-a]pyrazin-8-yl-[4-[2-(4-methylphenyl)ethyl]piperidin-1-yl]methanone
—— cyclopropyl-(4-phenyl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-7-yl)methanone —— C17H17N3O
cyclopropyl-(4-phenyl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-7-yl)methanone
—— (4-phenyl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-7-yl)-pyridin-4-ylmethanone —— C19H16N4O
(4-phenyl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-7-yl)-pyridin-4-ylmethanone
—— N-tert-butyl-4-phenyl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidine-7-carboxamide —— C18H22N4O
N-tert-butyl-4-phenyl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidine-7-carboxamide
—— (4-phenyl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-7-yl)-[3-(pyrrolidin-1-ylmethyl)phenyl]methanone —— C25H26N4O
(4-phenyl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-7-yl)-[3-(pyrrolidin-1-ylmethyl)phenyl]methanone
—— (4-phenyl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-7-yl)-[(2S)-1-(thiophene-3-carbonyl)pyrrolidin-2-yl]methanone —— C23H22N4O2S
(4-phenyl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-7-yl)-[(2S)-1-(thiophene-3-carbonyl)pyrrolidin-2-yl]methanone
—— N-(2-chlorophenyl)-4-phenyl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidine-7-carboxamide —— C20H17ClN4O
N-(2-chlorophenyl)-4-phenyl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidine-7-carboxamide
—— 2-methyl-1-(4-phenyl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-7-yl)propan-1-one —— C17H19N3O
2-methyl-1-(4-phenyl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-7-yl)propan-1-one