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二氮杂萘

中文名称 英文名称 CAS号 化学式 结构式图片
—— N-[[4-[(2S,4S,5R,6R)-4-[[benzyl(methyl)amino]methyl]-6-[4-(hydroxymethyl)phenyl]-5-methyl-1,3-dioxan-2-yl]phenyl]methyl]quinoxaline-2-carboxamide —— C37H38N4O4
N-[[4-[(2S,4S,5R,6R)-4-[[benzyl(methyl)amino]methyl]-6-[4-(hydroxymethyl)phenyl]-5-methyl-1,3-dioxan-2-yl]phenyl]methyl]quinoxaline-2-carboxamide
—— 2-(8-methyl-4-oxoquinazolin-3-yl)-N-[4-[(3S)-3-methylpiperidin-1-yl]butyl]acetamide —— C21H30N4O2
2-(8-methyl-4-oxoquinazolin-3-yl)-N-[4-[(3S)-3-methylpiperidin-1-yl]butyl]acetamide
—— 2-(8-methyl-4-oxoquinazolin-3-yl)-N-[4-[(2R)-2-methylpiperidin-1-yl]butyl]acetamide —— C21H30N4O2
2-(8-methyl-4-oxoquinazolin-3-yl)-N-[4-[(2R)-2-methylpiperidin-1-yl]butyl]acetamide
—— 2-(8-methyl-4-oxoquinazolin-3-yl)-N-[(2R)-2-[(3S)-3-methylpiperidin-1-yl]propyl]acetamide —— C20H28N4O2
2-(8-methyl-4-oxoquinazolin-3-yl)-N-[(2R)-2-[(3S)-3-methylpiperidin-1-yl]propyl]acetamide
—— N-[[4-[(2S,4S,5R,6R)-4-(benzimidazol-1-ylmethyl)-6-[4-(hydroxymethyl)phenyl]-5-methyl-1,3-dioxan-2-yl]phenyl]methyl]quinoxaline-2-carboxamide —— C36H33N5O4
N-[[4-[(2S,4S,5R,6R)-4-(benzimidazol-1-ylmethyl)-6-[4-(hydroxymethyl)phenyl]-5-methyl-1,3-dioxan-2-yl]phenyl]methyl]quinoxaline-2-carboxamide
—— N-[[4-[(2S,4R,5R,6S)-4-[4-(hydroxymethyl)phenyl]-5-methyl-6-[(1-methyltetrazol-5-yl)sulfanylmethyl]-1,3-dioxan-2-yl]phenyl]methyl]quinoxaline-2-carboxamide —— C31H31N7O4S
N-[[4-[(2S,4R,5R,6S)-4-[4-(hydroxymethyl)phenyl]-5-methyl-6-[(1-methyltetrazol-5-yl)sulfanylmethyl]-1,3-dioxan-2-yl]phenyl]methyl]quinoxaline-2-carboxamide
—— N-[[4-[(2S,4R,5R,6S)-4-[4-(hydroxymethyl)phenyl]-5-methyl-6-[(4-methyl-1,2,4-triazol-3-yl)sulfanylmethyl]-1,3-dioxan-2-yl]phenyl]methyl]quinoxaline-2-carboxamide —— C32H32N6O4S
N-[[4-[(2S,4R,5R,6S)-4-[4-(hydroxymethyl)phenyl]-5-methyl-6-[(4-methyl-1,2,4-triazol-3-yl)sulfanylmethyl]-1,3-dioxan-2-yl]phenyl]methyl]quinoxaline-2-carboxamide
—— 3-ethyl-2,4-dioxo-N-[(2S)-4-phenylbutan-2-yl]-1H-quinazoline-7-carboxamide —— C21H23N3O3
3-ethyl-2,4-dioxo-N-[(2S)-4-phenylbutan-2-yl]-1H-quinazoline-7-carboxamide
—— 3-ethyl-2,4-dioxo-N-[(S)-phenyl(thiophen-2-yl)methyl]-1H-quinazoline-7-carboxamide —— C22H19N3O3S
3-ethyl-2,4-dioxo-N-[(S)-phenyl(thiophen-2-yl)methyl]-1H-quinazoline-7-carboxamide
—— N-[[4-[(2S,4R,5R,6S)-4-[4-(hydroxymethyl)phenyl]-6-[[(2S)-2-(methoxymethyl)pyrrolidin-1-yl]methyl]-5-methyl-1,3-dioxan-2-yl]phenyl]methyl]quinoxaline-2-carboxamide —— C35H40N4O5
N-[[4-[(2S,4R,5R,6S)-4-[4-(hydroxymethyl)phenyl]-6-[[(2S)-2-(methoxymethyl)pyrrolidin-1-yl]methyl]-5-methyl-1,3-dioxan-2-yl]phenyl]methyl]quinoxaline-2-carboxamide
—— 3-ethyl-N-[(S)-(1-methylimidazol-2-yl)-phenylmethyl]-2,4-dioxo-1H-quinazoline-7-carboxamide —— C22H21N5O3
3-ethyl-N-[(S)-(1-methylimidazol-2-yl)-phenylmethyl]-2,4-dioxo-1H-quinazoline-7-carboxamide
—— N-[(1S)-1-(3-chlorophenyl)ethyl]-3-ethyl-2,4-dioxo-1H-quinazoline-7-carboxamide —— C19H18ClN3O3
N-[(1S)-1-(3-chlorophenyl)ethyl]-3-ethyl-2,4-dioxo-1H-quinazoline-7-carboxamide
—— 3-ethyl-2,4-dioxo-N-[(2R)-pentan-2-yl]-1H-quinazoline-7-carboxamide —— C16H21N3O3
3-ethyl-2,4-dioxo-N-[(2R)-pentan-2-yl]-1H-quinazoline-7-carboxamide
—— 4-(2-methyl-4-oxoquinazolin-3-yl)-N-[2-(trifluoromethylsulfanyl)ethyl]benzamide —— C19H16F3N3O2S
4-(2-methyl-4-oxoquinazolin-3-yl)-N-[2-(trifluoromethylsulfanyl)ethyl]benzamide
—— 2-(6-fluoro-4-oxoquinazolin-3-yl)-N-[2-[(1R,2S)-2-methylcyclohexyl]oxyethyl]acetamide —— C19H24FN3O3
2-(6-fluoro-4-oxoquinazolin-3-yl)-N-[2-[(1R,2S)-2-methylcyclohexyl]oxyethyl]acetamide
—— N-[[4-[(2S,4R,5R,6S)-4-[4-(hydroxymethyl)phenyl]-5-methyl-6-[(1-methylimidazol-2-yl)sulfanylmethyl]-1,3-dioxan-2-yl]phenyl]methyl]quinoxaline-2-carboxamide —— C33H33N5O4S
N-[[4-[(2S,4R,5R,6S)-4-[4-(hydroxymethyl)phenyl]-5-methyl-6-[(1-methylimidazol-2-yl)sulfanylmethyl]-1,3-dioxan-2-yl]phenyl]methyl]quinoxaline-2-carboxamide
—— 2-(6-fluoro-4-oxoquinazolin-3-yl)-N-[4-[(3R)-3-methylpiperidin-1-yl]butyl]acetamide —— C20H27FN4O2
2-(6-fluoro-4-oxoquinazolin-3-yl)-N-[4-[(3R)-3-methylpiperidin-1-yl]butyl]acetamide
—— N-[4-[(2S)-2-methylpiperidin-1-yl]butyl]-4-oxo-3-phenylphthalazine-1-carboxamide —— C25H30N4O2
N-[4-[(2S)-2-methylpiperidin-1-yl]butyl]-4-oxo-3-phenylphthalazine-1-carboxamide
—— 2-(6-fluoro-4-oxoquinazolin-3-yl)-N-[4-[(3S)-3-methylpiperidin-1-yl]butyl]acetamide —— C20H27FN4O2
2-(6-fluoro-4-oxoquinazolin-3-yl)-N-[4-[(3S)-3-methylpiperidin-1-yl]butyl]acetamide
—— N-[4-[(3R)-3-methylpiperidin-1-yl]butyl]-4-oxo-3-prop-2-enyl-2-sulfanylidene-1H-quinazoline-7-carboxamide —— C22H30N4O2S
N-[4-[(3R)-3-methylpiperidin-1-yl]butyl]-4-oxo-3-prop-2-enyl-2-sulfanylidene-1H-quinazoline-7-carboxamide
—— 2-(2,4-dioxo-1H-quinazolin-3-yl)-N-[(1S)-1-(3,4,5-trimethoxyphenyl)ethyl]acetamide —— C21H23N3O6
2-(2,4-dioxo-1H-quinazolin-3-yl)-N-[(1S)-1-(3,4,5-trimethoxyphenyl)ethyl]acetamide
—— N-[(1R,2R)-1-(1H-benzimidazol-2-yl)-2-methylbutyl]-3-(4-oxoquinazolin-3-yl)propanamide —— C23H25N5O2
N-[(1R,2R)-1-(1H-benzimidazol-2-yl)-2-methylbutyl]-3-(4-oxoquinazolin-3-yl)propanamide
—— N-[[4-[(2S,4R,5R,6S)-4-[4-(hydroxymethyl)phenyl]-5-methyl-6-(pyrimidin-2-ylsulfanylmethyl)-1,3-dioxan-2-yl]phenyl]methyl]quinoxaline-2-carboxamide —— C33H31N5O4S
N-[[4-[(2S,4R,5R,6S)-4-[4-(hydroxymethyl)phenyl]-5-methyl-6-(pyrimidin-2-ylsulfanylmethyl)-1,3-dioxan-2-yl]phenyl]methyl]quinoxaline-2-carboxamide
—— N-[(1R,2R)-1-(1H-benzimidazol-2-yl)-2-methylbutyl]-2-(1-oxophthalazin-2-yl)acetamide —— C22H23N5O2
N-[(1R,2R)-1-(1H-benzimidazol-2-yl)-2-methylbutyl]-2-(1-oxophthalazin-2-yl)acetamide
—— N-[4-(furan-2-yl)-1,3-thiazol-2-yl]-3-(4-oxo-2-sulfanylidene-1H-quinazolin-3-yl)propanamide —— C18H14N4O3S2
N-[4-(furan-2-yl)-1,3-thiazol-2-yl]-3-(4-oxo-2-sulfanylidene-1H-quinazolin-3-yl)propanamide
—— 3-propan-2-yl-7-[(2S)-2-thiophen-3-ylpyrrolidine-1-carbonyl]-1H-quinazoline-2,4-dione —— C20H21N3O3S
3-propan-2-yl-7-[(2S)-2-thiophen-3-ylpyrrolidine-1-carbonyl]-1H-quinazoline-2,4-dione
—— N-[[4-[(2S,4R,5R,6S)-4-[4-(hydroxymethyl)phenyl]-5-methyl-6-(phenylsulfanylmethyl)-1,3-dioxan-2-yl]phenyl]methyl]quinoxaline-2-carboxamide —— C35H33N3O4S
N-[[4-[(2S,4R,5R,6S)-4-[4-(hydroxymethyl)phenyl]-5-methyl-6-(phenylsulfanylmethyl)-1,3-dioxan-2-yl]phenyl]methyl]quinoxaline-2-carboxamide
—— N-[[4-[(2S,4R,5R,6S)-4-[4-(hydroxymethyl)phenyl]-5-methyl-6-(1H-1,2,4-triazol-5-ylsulfanylmethyl)-1,3-dioxan-2-yl]phenyl]methyl]quinoxaline-2-carboxamide —— C31H30N6O4S
N-[[4-[(2S,4R,5R,6S)-4-[4-(hydroxymethyl)phenyl]-5-methyl-6-(1H-1,2,4-triazol-5-ylsulfanylmethyl)-1,3-dioxan-2-yl]phenyl]methyl]quinoxaline-2-carboxamide
—— N-[[4-[(2S,4R,5R,6S)-4-[4-(hydroxymethyl)phenyl]-5-methyl-6-(pyridin-2-ylsulfanylmethyl)-1,3-dioxan-2-yl]phenyl]methyl]quinoxaline-2-carboxamide —— C34H32N4O4S
N-[[4-[(2S,4R,5R,6S)-4-[4-(hydroxymethyl)phenyl]-5-methyl-6-(pyridin-2-ylsulfanylmethyl)-1,3-dioxan-2-yl]phenyl]methyl]quinoxaline-2-carboxamide
—— N-[[4-[(2S,4R,5R,6S)-4-[4-(hydroxymethyl)phenyl]-6-[[(2S)-2-(hydroxymethyl)pyrrolidin-1-yl]methyl]-5-methyl-1,3-dioxan-2-yl]phenyl]methyl]quinoxaline-2-carboxamide —— C34H38N4O5
N-[[4-[(2S,4R,5R,6S)-4-[4-(hydroxymethyl)phenyl]-6-[[(2S)-2-(hydroxymethyl)pyrrolidin-1-yl]methyl]-5-methyl-1,3-dioxan-2-yl]phenyl]methyl]quinoxaline-2-carboxamide
—— N-[(2S)-1-morpholin-4-ylpropan-2-yl]-2-(2-oxoquinoxalin-1-yl)acetamide —— C17H22N4O3
N-[(2S)-1-morpholin-4-ylpropan-2-yl]-2-(2-oxoquinoxalin-1-yl)acetamide
—— N-[2-[(3S)-3-methylpiperidin-1-yl]ethyl]-2-(4-oxoquinazolin-3-yl)acetamide —— C18H24N4O2
N-[2-[(3S)-3-methylpiperidin-1-yl]ethyl]-2-(4-oxoquinazolin-3-yl)acetamide
—— 2-(6-bromo-4-oxoquinazolin-3-yl)-N-[2-[(2S)-2-methylpiperidin-1-yl]ethyl]acetamide —— C18H23BrN4O2
2-(6-bromo-4-oxoquinazolin-3-yl)-N-[2-[(2S)-2-methylpiperidin-1-yl]ethyl]acetamide
—— N-[[4-[(2S,4R,5R,6S)-4-[4-(hydroxymethyl)phenyl]-6-[[(3S)-3-hydroxypyrrolidin-1-yl]methyl]-5-methyl-1,3-dioxan-2-yl]phenyl]methyl]quinoxaline-2-carboxamide —— C33H36N4O5
N-[[4-[(2S,4R,5R,6S)-4-[4-(hydroxymethyl)phenyl]-6-[[(3S)-3-hydroxypyrrolidin-1-yl]methyl]-5-methyl-1,3-dioxan-2-yl]phenyl]methyl]quinoxaline-2-carboxamide
—— ethyl 4-[4-[[(2S)-butan-2-yl]sulfamoyl]anilino]-7-methyl-1,8-naphthyridine-3-carboxylate —— C22H26N4O4S
ethyl 4-[4-[[(2S)-butan-2-yl]sulfamoyl]anilino]-7-methyl-1,8-naphthyridine-3-carboxylate
—— N-[[4-[(2S,4R,5R,6S)-4-[4-(hydroxymethyl)phenyl]-5-methyl-6-(piperidin-1-ylmethyl)-1,3-dioxan-2-yl]phenyl]methyl]quinoxaline-2-carboxamide —— C34H38N4O4
N-[[4-[(2S,4R,5R,6S)-4-[4-(hydroxymethyl)phenyl]-5-methyl-6-(piperidin-1-ylmethyl)-1,3-dioxan-2-yl]phenyl]methyl]quinoxaline-2-carboxamide
—— 2-(8-methyl-4-oxoquinazolin-3-yl)-N-[3-[(3R)-3-methylpiperidin-1-yl]propyl]acetamide —— C20H28N4O2
2-(8-methyl-4-oxoquinazolin-3-yl)-N-[3-[(3R)-3-methylpiperidin-1-yl]propyl]acetamide
—— N-[(2R)-2-(N-methylanilino)propyl]-2-(4-oxocinnolin-1-yl)acetamide —— C20H22N4O2
N-[(2R)-2-(N-methylanilino)propyl]-2-(4-oxocinnolin-1-yl)acetamide
—— N-[(4R)-3,4-dihydro-2H-thiochromen-4-yl]-4-oxo-2-sulfanylidene-1H-quinazoline-7-carboxamide —— C18H15N3O2S2
N-[(4R)-3,4-dihydro-2H-thiochromen-4-yl]-4-oxo-2-sulfanylidene-1H-quinazoline-7-carboxamide
—— N-[3-[(3S)-3-methylpiperidin-1-yl]propyl]-4-(4-oxoquinazolin-3-yl)benzamide —— C24H28N4O2
N-[3-[(3S)-3-methylpiperidin-1-yl]propyl]-4-(4-oxoquinazolin-3-yl)benzamide
—— N-[[4-[(2S,4R,5R,6S)-4-[4-(hydroxymethyl)phenyl]-5-methyl-6-[[methyl(prop-2-enyl)amino]methyl]-1,3-dioxan-2-yl]phenyl]methyl]quinoxaline-2-carboxamide —— C33H36N4O4
N-[[4-[(2S,4R,5R,6S)-4-[4-(hydroxymethyl)phenyl]-5-methyl-6-[[methyl(prop-2-enyl)amino]methyl]-1,3-dioxan-2-yl]phenyl]methyl]quinoxaline-2-carboxamide
—— N-[(2S)-2-(3,4-difluorophenyl)-2-hydroxyethyl]-4-oxo-2-sulfanylidene-1H-quinazoline-7-carboxamide —— C17H13F2N3O3S
N-[(2S)-2-(3,4-difluorophenyl)-2-hydroxyethyl]-4-oxo-2-sulfanylidene-1H-quinazoline-7-carboxamide
—— N-[(1S)-1-(4-methylsulfanylphenyl)ethyl]-4-oxo-2-sulfanylidene-1H-quinazoline-7-carboxamide —— C18H17N3O2S2
N-[(1S)-1-(4-methylsulfanylphenyl)ethyl]-4-oxo-2-sulfanylidene-1H-quinazoline-7-carboxamide
—— N-[4-[(3R,5R)-3,5-dimethylpiperidin-1-yl]butyl]-3-(4-oxoquinazolin-3-yl)propanamide —— C22H32N4O2
N-[4-[(3R,5R)-3,5-dimethylpiperidin-1-yl]butyl]-3-(4-oxoquinazolin-3-yl)propanamide
—— N-[(1R)-1-(2,5-dimethylthiophen-3-yl)ethyl]-4-oxo-2-sulfanylidene-1H-quinazoline-7-carboxamide —— C17H17N3O2S2
N-[(1R)-1-(2,5-dimethylthiophen-3-yl)ethyl]-4-oxo-2-sulfanylidene-1H-quinazoline-7-carboxamide
—— 2-(6-bromo-4-oxoquinazolin-3-yl)-N-[(4S)-1-methyl-4,5,6,7-tetrahydroindazol-4-yl]acetamide —— C18H18BrN5O2
2-(6-bromo-4-oxoquinazolin-3-yl)-N-[(4S)-1-methyl-4,5,6,7-tetrahydroindazol-4-yl]acetamide
—— N-[(1S)-1-(2,5-dimethylthiophen-3-yl)ethyl]-4-oxo-2-sulfanylidene-1H-quinazoline-7-carboxamide —— C17H17N3O2S2
N-[(1S)-1-(2,5-dimethylthiophen-3-yl)ethyl]-4-oxo-2-sulfanylidene-1H-quinazoline-7-carboxamide
—— N-[(1S)-1-naphthalen-2-ylethyl]-4-oxo-2-sulfanylidene-1H-quinazoline-7-carboxamide —— C21H17N3O2S
N-[(1S)-1-naphthalen-2-ylethyl]-4-oxo-2-sulfanylidene-1H-quinazoline-7-carboxamide
—— N-[[(2R)-1-ethylpyrrolidin-2-yl]methyl]-4-oxo-2-sulfanylidene-1H-quinazoline-7-carboxamide —— C16H20N4O2S
N-[[(2R)-1-ethylpyrrolidin-2-yl]methyl]-4-oxo-2-sulfanylidene-1H-quinazoline-7-carboxamide
—— N-[4-[(2S)-2-methylpiperidin-1-yl]butyl]-3-(2-methylpropyl)-4-oxophthalazine-1-carboxamide —— C23H34N4O2
N-[4-[(2S)-2-methylpiperidin-1-yl]butyl]-3-(2-methylpropyl)-4-oxophthalazine-1-carboxamide