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二氮杂萘

中文名称 英文名称 CAS号 化学式 结构式图片
—— N-[(2S)-butan-2-yl]-1-[(4-fluorophenyl)methylsulfanyl]-4-(2-methylpropyl)-5-oxo-[1,2,4]triazolo[4,3-a]quinazoline-8-carboxamide —— C25H28FN5O2S
N-[(2S)-butan-2-yl]-1-[(4-fluorophenyl)methylsulfanyl]-4-(2-methylpropyl)-5-oxo-[1,2,4]triazolo[4,3-a]quinazoline-8-carboxamide
—— N-[(2S)-butan-2-yl]-1-(cyanomethylsulfanyl)-4-(2-methylpropyl)-5-oxo-[1,2,4]triazolo[4,3-a]quinazoline-8-carboxamide —— C20H24N6O2S
N-[(2S)-butan-2-yl]-1-(cyanomethylsulfanyl)-4-(2-methylpropyl)-5-oxo-[1,2,4]triazolo[4,3-a]quinazoline-8-carboxamide
—— N-[(2R)-butan-2-yl]-1-[(2-fluorophenyl)methylsulfanyl]-4-(2-methylpropyl)-5-oxo-[1,2,4]triazolo[4,3-a]quinazoline-8-carboxamide —— C25H28FN5O2S
N-[(2R)-butan-2-yl]-1-[(2-fluorophenyl)methylsulfanyl]-4-(2-methylpropyl)-5-oxo-[1,2,4]triazolo[4,3-a]quinazoline-8-carboxamide
—— N-[(2R)-butan-2-yl]-1-[(2-fluorophenyl)methylsulfanyl]-5-oxo-4-propyl-[1,2,4]triazolo[4,3-a]quinazoline-8-carboxamide —— C24H26FN5O2S
N-[(2R)-butan-2-yl]-1-[(2-fluorophenyl)methylsulfanyl]-5-oxo-4-propyl-[1,2,4]triazolo[4,3-a]quinazoline-8-carboxamide
—— N-[(2R)-butan-2-yl]-1-[(2-methylphenyl)methylsulfanyl]-4-(2-methylpropyl)-5-oxo-[1,2,4]triazolo[4,3-a]quinazoline-8-carboxamide —— C26H31N5O2S
N-[(2R)-butan-2-yl]-1-[(2-methylphenyl)methylsulfanyl]-4-(2-methylpropyl)-5-oxo-[1,2,4]triazolo[4,3-a]quinazoline-8-carboxamide
—— N-[(2S)-butan-2-yl]-1-[(2,5-dimethylphenyl)methylsulfanyl]-4-(2-methylpropyl)-5-oxo-[1,2,4]triazolo[4,3-a]quinazoline-8-carboxamide —— C27H33N5O2S
N-[(2S)-butan-2-yl]-1-[(2,5-dimethylphenyl)methylsulfanyl]-4-(2-methylpropyl)-5-oxo-[1,2,4]triazolo[4,3-a]quinazoline-8-carboxamide
—— N-[(2S)-butan-2-yl]-1-[(4-methylphenyl)methylsulfanyl]-5-oxo-4-propyl-[1,2,4]triazolo[4,3-a]quinazoline-8-carboxamide —— C25H29N5O2S
N-[(2S)-butan-2-yl]-1-[(4-methylphenyl)methylsulfanyl]-5-oxo-4-propyl-[1,2,4]triazolo[4,3-a]quinazoline-8-carboxamide
—— N-[(2S)-butan-2-yl]-1-[(2-methylphenyl)methylsulfanyl]-4-(2-methylpropyl)-5-oxo-[1,2,4]triazolo[4,3-a]quinazoline-8-carboxamide —— C26H31N5O2S
N-[(2S)-butan-2-yl]-1-[(2-methylphenyl)methylsulfanyl]-4-(2-methylpropyl)-5-oxo-[1,2,4]triazolo[4,3-a]quinazoline-8-carboxamide
—— N-[(2S)-butan-2-yl]-1-[(4-fluorophenyl)methylsulfanyl]-5-oxo-4-propyl-[1,2,4]triazolo[4,3-a]quinazoline-8-carboxamide —— C24H26FN5O2S
N-[(2S)-butan-2-yl]-1-[(4-fluorophenyl)methylsulfanyl]-5-oxo-4-propyl-[1,2,4]triazolo[4,3-a]quinazoline-8-carboxamide
—— N-[(2S)-butan-2-yl]-1-[(2-chloro-6-fluorophenyl)methylsulfanyl]-4-(2-methylpropyl)-5-oxo-[1,2,4]triazolo[4,3-a]quinazoline-8-carboxamide —— C25H27ClFN5O2S
N-[(2S)-butan-2-yl]-1-[(2-chloro-6-fluorophenyl)methylsulfanyl]-4-(2-methylpropyl)-5-oxo-[1,2,4]triazolo[4,3-a]quinazoline-8-carboxamide
—— N-[(2R)-butan-2-yl]-1-[(4-fluorophenyl)methylsulfanyl]-5-oxo-4-propyl-[1,2,4]triazolo[4,3-a]quinazoline-8-carboxamide —— C24H26FN5O2S
N-[(2R)-butan-2-yl]-1-[(4-fluorophenyl)methylsulfanyl]-5-oxo-4-propyl-[1,2,4]triazolo[4,3-a]quinazoline-8-carboxamide
—— N-[(2R)-butan-2-yl]-1-[(4-chlorophenyl)methylsulfanyl]-4-(2-methylpropyl)-5-oxo-[1,2,4]triazolo[4,3-a]quinazoline-8-carboxamide —— C25H28ClN5O2S
N-[(2R)-butan-2-yl]-1-[(4-chlorophenyl)methylsulfanyl]-4-(2-methylpropyl)-5-oxo-[1,2,4]triazolo[4,3-a]quinazoline-8-carboxamide
—— N-[(2R)-butan-2-yl]-1-[(2-chlorophenyl)methylsulfanyl]-5-oxo-4-propyl-[1,2,4]triazolo[4,3-a]quinazoline-8-carboxamide —— C24H26ClN5O2S
N-[(2R)-butan-2-yl]-1-[(2-chlorophenyl)methylsulfanyl]-5-oxo-4-propyl-[1,2,4]triazolo[4,3-a]quinazoline-8-carboxamide
—— N-[(2R)-butan-2-yl]-1-[(4-methylphenyl)methylsulfanyl]-4-(2-methylpropyl)-5-oxo-[1,2,4]triazolo[4,3-a]quinazoline-8-carboxamide —— C26H31N5O2S
N-[(2R)-butan-2-yl]-1-[(4-methylphenyl)methylsulfanyl]-4-(2-methylpropyl)-5-oxo-[1,2,4]triazolo[4,3-a]quinazoline-8-carboxamide
—— N-[(2S)-butan-2-yl]-1-[(2-chlorophenyl)methylsulfanyl]-4-(2-methylpropyl)-5-oxo-[1,2,4]triazolo[4,3-a]quinazoline-8-carboxamide —— C25H28ClN5O2S
N-[(2S)-butan-2-yl]-1-[(2-chlorophenyl)methylsulfanyl]-4-(2-methylpropyl)-5-oxo-[1,2,4]triazolo[4,3-a]quinazoline-8-carboxamide
—— N-[(2R)-butan-2-yl]-1-[(3-fluorophenyl)methylsulfanyl]-5-oxo-4-propyl-[1,2,4]triazolo[4,3-a]quinazoline-8-carboxamide —— C24H26FN5O2S
N-[(2R)-butan-2-yl]-1-[(3-fluorophenyl)methylsulfanyl]-5-oxo-4-propyl-[1,2,4]triazolo[4,3-a]quinazoline-8-carboxamide
—— N-[(2R)-butan-2-yl]-1-(cyanomethylsulfanyl)-5-oxo-4-propyl-[1,2,4]triazolo[4,3-a]quinazoline-8-carboxamide —— C19H22N6O2S
N-[(2R)-butan-2-yl]-1-(cyanomethylsulfanyl)-5-oxo-4-propyl-[1,2,4]triazolo[4,3-a]quinazoline-8-carboxamide
—— N-[(2S)-butan-2-yl]-1-[(2-chloro-6-fluorophenyl)methylsulfanyl]-5-oxo-4-propyl-[1,2,4]triazolo[4,3-a]quinazoline-8-carboxamide —— C24H25ClFN5O2S
N-[(2S)-butan-2-yl]-1-[(2-chloro-6-fluorophenyl)methylsulfanyl]-5-oxo-4-propyl-[1,2,4]triazolo[4,3-a]quinazoline-8-carboxamide
—— N-[(2R)-butan-2-yl]-1-[(4-chlorophenyl)methylsulfanyl]-4-(3-methylbutyl)-5-oxo-[1,2,4]triazolo[4,3-a]quinazoline-8-carboxamide —— C26H30ClN5O2S
N-[(2R)-butan-2-yl]-1-[(4-chlorophenyl)methylsulfanyl]-4-(3-methylbutyl)-5-oxo-[1,2,4]triazolo[4,3-a]quinazoline-8-carboxamide
—— N-[(2S)-butan-2-yl]-1-[(2-methylphenyl)methylsulfanyl]-5-oxo-4-propyl-[1,2,4]triazolo[4,3-a]quinazoline-8-carboxamide —— C25H29N5O2S
N-[(2S)-butan-2-yl]-1-[(2-methylphenyl)methylsulfanyl]-5-oxo-4-propyl-[1,2,4]triazolo[4,3-a]quinazoline-8-carboxamide
—— 4-[(2,3-dioxo-4-prop-2-enylquinoxalin-1-yl)methyl]-N-[(2S)-4-phenylbutan-2-yl]benzamide —— C29H29N3O3
4-[(2,3-dioxo-4-prop-2-enylquinoxalin-1-yl)methyl]-N-[(2S)-4-phenylbutan-2-yl]benzamide
—— 1-ethyl-4-[2-[(3S)-3-methylpiperidin-1-yl]-2-oxoethyl]quinoxaline-2,3-dione —— C18H23N3O3
1-ethyl-4-[2-[(3S)-3-methylpiperidin-1-yl]-2-oxoethyl]quinoxaline-2,3-dione
—— 1-methyl-4-[2-[(3R)-3-methylpiperidin-1-yl]-2-oxoethyl]quinoxaline-2,3-dione —— C17H21N3O3
1-methyl-4-[2-[(3R)-3-methylpiperidin-1-yl]-2-oxoethyl]quinoxaline-2,3-dione
—— 1-methyl-4-[2-[(3S)-3-methylpiperidin-1-yl]-2-oxoethyl]quinoxaline-2,3-dione —— C17H21N3O3
1-methyl-4-[2-[(3S)-3-methylpiperidin-1-yl]-2-oxoethyl]quinoxaline-2,3-dione
—— 7-bromo-5-[4-[(3R)-3-methylpiperidin-1-yl]-4-oxobutyl]pyrrolo[1,2-a]quinoxalin-4-one —— C21H24BrN3O2
7-bromo-5-[4-[(3R)-3-methylpiperidin-1-yl]-4-oxobutyl]pyrrolo[1,2-a]quinoxalin-4-one
—— 4-[(2,3-dioxo-4-prop-2-enylquinoxalin-1-yl)methyl]-N-[(2R)-2-phenylpropyl]benzamide —— C28H27N3O3
4-[(2,3-dioxo-4-prop-2-enylquinoxalin-1-yl)methyl]-N-[(2R)-2-phenylpropyl]benzamide
—— 7-bromo-5-[4-[(3S)-3-methylpiperidin-1-yl]-4-oxobutyl]pyrrolo[1,2-a]quinoxalin-4-one —— C21H24BrN3O2
7-bromo-5-[4-[(3S)-3-methylpiperidin-1-yl]-4-oxobutyl]pyrrolo[1,2-a]quinoxalin-4-one
—— 1-[(4-chlorophenyl)methyl]-4-[2-[(3S)-3-methylpiperidin-1-yl]-2-oxoethyl]quinoxaline-2,3-dione —— C23H24ClN3O3
1-[(4-chlorophenyl)methyl]-4-[2-[(3S)-3-methylpiperidin-1-yl]-2-oxoethyl]quinoxaline-2,3-dione
—— N-[[(3S)-1-[(4-methylphenyl)methyl]pyrrolidin-3-yl]methyl]-2-(3,6,7-trimethyl-2-oxoquinoxalin-1-yl)acetamide —— C26H32N4O2
N-[[(3S)-1-[(4-methylphenyl)methyl]pyrrolidin-3-yl]methyl]-2-(3,6,7-trimethyl-2-oxoquinoxalin-1-yl)acetamide
—— 2-(3-methyl-2-oxoquinoxalin-1-yl)-N-[(2R)-4-phenylbutan-2-yl]acetamide —— C21H23N3O2
2-(3-methyl-2-oxoquinoxalin-1-yl)-N-[(2R)-4-phenylbutan-2-yl]acetamide
—— 3-(3-chlorophenyl)-4-[2-[(3S)-3-methylpiperidin-1-yl]-2-oxoethyl]-1-sulfanylidene-[1,3]thiazolo[3,4-a]quinazolin-5-one —— C24H22ClN3O2S2
3-(3-chlorophenyl)-4-[2-[(3S)-3-methylpiperidin-1-yl]-2-oxoethyl]-1-sulfanylidene-[1,3]thiazolo[3,4-a]quinazolin-5-one
—— N-[3-[(2R)-2-methylpiperidin-1-yl]propyl]-2-(3,6,7-trimethyl-2-oxoquinoxalin-1-yl)acetamide —— C22H32N4O2
N-[3-[(2R)-2-methylpiperidin-1-yl]propyl]-2-(3,6,7-trimethyl-2-oxoquinoxalin-1-yl)acetamide
—— methyl 3-[4-[[(2S)-butan-2-yl]carbamoyl]phenyl]-4-oxo-2-sulfanylidene-1H-quinazoline-7-carboxylate —— C21H21N3O4S
methyl 3-[4-[[(2S)-butan-2-yl]carbamoyl]phenyl]-4-oxo-2-sulfanylidene-1H-quinazoline-7-carboxylate
—— methyl 4-oxo-3-[4-oxo-4-[[(2S)-2-phenylpropyl]amino]butyl]-2-sulfanylidene-1H-quinazoline-7-carboxylate —— C23H25N3O4S
methyl 4-oxo-3-[4-oxo-4-[[(2S)-2-phenylpropyl]amino]butyl]-2-sulfanylidene-1H-quinazoline-7-carboxylate
—— N-[[(2S)-1-ethylpyrrolidin-2-yl]methyl]-2-(3-methyl-2-oxoquinoxalin-1-yl)acetamide —— C18H24N4O2
N-[[(2S)-1-ethylpyrrolidin-2-yl]methyl]-2-(3-methyl-2-oxoquinoxalin-1-yl)acetamide
—— methyl 3-[[4-[[(2S)-butan-2-yl]carbamoyl]phenyl]methyl]-4-oxo-2-sulfanylidene-1H-quinazoline-7-carboxylate —— C22H23N3O4S
methyl 3-[[4-[[(2S)-butan-2-yl]carbamoyl]phenyl]methyl]-4-oxo-2-sulfanylidene-1H-quinazoline-7-carboxylate
—— N-[[(2R)-1-ethylpyrrolidin-2-yl]methyl]-2-(3-methyl-2-oxoquinoxalin-1-yl)acetamide —— C18H24N4O2
N-[[(2R)-1-ethylpyrrolidin-2-yl]methyl]-2-(3-methyl-2-oxoquinoxalin-1-yl)acetamide
—— 2-(3-methyl-2-oxoquinoxalin-1-yl)-N-[[(3S)-1-[(4-methylphenyl)methyl]pyrrolidin-3-yl]methyl]acetamide —— C24H28N4O2
2-(3-methyl-2-oxoquinoxalin-1-yl)-N-[[(3S)-1-[(4-methylphenyl)methyl]pyrrolidin-3-yl]methyl]acetamide
—— 2-(3-methyl-2-oxoquinoxalin-1-yl)-N-[(1R)-1-thiophen-2-ylbutyl]acetamide —— C19H21N3O2S
2-(3-methyl-2-oxoquinoxalin-1-yl)-N-[(1R)-1-thiophen-2-ylbutyl]acetamide
—— methyl 4-oxo-3-[[4-[[(2R)-oxolan-2-yl]methylcarbamoyl]phenyl]methyl]-2-sulfanylidene-1H-quinazoline-7-carboxylate —— C23H23N3O5S
methyl 4-oxo-3-[[4-[[(2R)-oxolan-2-yl]methylcarbamoyl]phenyl]methyl]-2-sulfanylidene-1H-quinazoline-7-carboxylate
—— 6,7-dimethyl-1-[(2R)-1-(4-methylpiperidin-1-yl)-1-oxopropan-2-yl]-3-(trifluoromethyl)quinoxalin-2-one —— C20H24F3N3O2
6,7-dimethyl-1-[(2R)-1-(4-methylpiperidin-1-yl)-1-oxopropan-2-yl]-3-(trifluoromethyl)quinoxalin-2-one
—— (2S)-2-[6,7-dimethyl-2-oxo-3-(trifluoromethyl)quinoxalin-1-yl]-N-[(4-propan-2-yloxyphenyl)methyl]propanamide —— C24H26F3N3O3
(2S)-2-[6,7-dimethyl-2-oxo-3-(trifluoromethyl)quinoxalin-1-yl]-N-[(4-propan-2-yloxyphenyl)methyl]propanamide
—— (2R)-2-[6,7-dimethyl-2-oxo-3-(trifluoromethyl)quinoxalin-1-yl]-N-[(2-methylphenyl)methyl]propanamide —— C22H22F3N3O2
(2R)-2-[6,7-dimethyl-2-oxo-3-(trifluoromethyl)quinoxalin-1-yl]-N-[(2-methylphenyl)methyl]propanamide
—— (2R)-N-[(2-chlorophenyl)methyl]-2-[6,7-dimethyl-2-oxo-3-(trifluoromethyl)quinoxalin-1-yl]butanamide —— C22H21ClF3N3O2
(2R)-N-[(2-chlorophenyl)methyl]-2-[6,7-dimethyl-2-oxo-3-(trifluoromethyl)quinoxalin-1-yl]butanamide
—— 3-[(5-oxo-[1,3,4]thiadiazolo[2,3-b]quinazolin-2-yl)amino]-N-[(2R)-2-phenylpropyl]benzamide —— C25H21N5O2S
3-[(5-oxo-[1,3,4]thiadiazolo[2,3-b]quinazolin-2-yl)amino]-N-[(2R)-2-phenylpropyl]benzamide
—— 4-[(5-oxo-[1,3,4]thiadiazolo[2,3-b]quinazolin-2-yl)amino]-N-[(2S)-2-phenylpropyl]benzamide —— C25H21N5O2S
4-[(5-oxo-[1,3,4]thiadiazolo[2,3-b]quinazolin-2-yl)amino]-N-[(2S)-2-phenylpropyl]benzamide
—— 1-[(2R)-1-(4-cyclohexylpiperazin-1-yl)-1-oxopropan-2-yl]-6,7-dimethyl-3-(trifluoromethyl)quinoxalin-2-one —— C24H31F3N4O2
1-[(2R)-1-(4-cyclohexylpiperazin-1-yl)-1-oxopropan-2-yl]-6,7-dimethyl-3-(trifluoromethyl)quinoxalin-2-one
—— 1-[(2R)-1-(4-ethylpiperazin-1-yl)-1-oxopropan-2-yl]-6,7-dimethyl-3-(trifluoromethyl)quinoxalin-2-one —— C20H25F3N4O2
1-[(2R)-1-(4-ethylpiperazin-1-yl)-1-oxopropan-2-yl]-6,7-dimethyl-3-(trifluoromethyl)quinoxalin-2-one
—— (2S)-N-[[4-(dimethylamino)phenyl]methyl]-2-[2-oxo-3-(trifluoromethyl)quinoxalin-1-yl]propanamide —— C21H21F3N4O2
(2S)-N-[[4-(dimethylamino)phenyl]methyl]-2-[2-oxo-3-(trifluoromethyl)quinoxalin-1-yl]propanamide
—— 6,7-dimethyl-1-[(2R)-1-oxo-1-pyrrolidin-1-ylpropan-2-yl]-3-(trifluoromethyl)quinoxalin-2-one —— C18H20F3N3O2
6,7-dimethyl-1-[(2R)-1-oxo-1-pyrrolidin-1-ylpropan-2-yl]-3-(trifluoromethyl)quinoxalin-2-one