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二氮杂萘

中文名称 英文名称 CAS号 化学式 结构式图片
—— N-[[4-[(2R,4R,5S,6S)-4-[(dioctylamino)methyl]-6-[4-(hydroxymethyl)phenyl]-5-methyl-1,3-dioxan-2-yl]phenyl]methyl]quinoxaline-2-carboxamide —— C45H62N4O4
N-[[4-[(2R,4R,5S,6S)-4-[(dioctylamino)methyl]-6-[4-(hydroxymethyl)phenyl]-5-methyl-1,3-dioxan-2-yl]phenyl]methyl]quinoxaline-2-carboxamide
—— 1-[(7-chloro-4-oxo-1H-quinazolin-2-yl)methyl]-3-(2-ethoxypyridin-3-yl)-1-propylurea —— C20H22ClN5O3
1-[(7-chloro-4-oxo-1H-quinazolin-2-yl)methyl]-3-(2-ethoxypyridin-3-yl)-1-propylurea
—— 4-(2-methyl-4-oxoquinazolin-3-yl)-N-[(1R)-1-(4-methylsulfanylphenyl)ethyl]butanamide —— C22H25N3O2S
4-(2-methyl-4-oxoquinazolin-3-yl)-N-[(1R)-1-(4-methylsulfanylphenyl)ethyl]butanamide
—— 2-methyl-5-[(1S)-1-quinazolin-4-ylsulfanylethyl]-1,3,4-oxadiazole —— C13H12N4OS
2-methyl-5-[(1S)-1-quinazolin-4-ylsulfanylethyl]-1,3,4-oxadiazole
—— 4-(2-methyl-4-oxoquinazolin-3-yl)-N-[(1S)-1-(4-methylsulfanylphenyl)ethyl]butanamide —— C22H25N3O2S
4-(2-methyl-4-oxoquinazolin-3-yl)-N-[(1S)-1-(4-methylsulfanylphenyl)ethyl]butanamide
—— N-[[4-[(2S,4R,6S)-4-[4-(hydroxymethyl)phenyl]-6-[[methyl(prop-2-enyl)amino]methyl]-1,3-dioxan-2-yl]phenyl]methyl]quinoxaline-2-carboxamide —— C32H34N4O4
N-[[4-[(2S,4R,6S)-4-[4-(hydroxymethyl)phenyl]-6-[[methyl(prop-2-enyl)amino]methyl]-1,3-dioxan-2-yl]phenyl]methyl]quinoxaline-2-carboxamide
—— 3-(2,5-dimethylphenyl)-2-[(1R)-1-(5-methyl-1,3,4-oxadiazol-2-yl)ethyl]sulfanylquinazolin-4-one —— C21H20N4O2S
3-(2,5-dimethylphenyl)-2-[(1R)-1-(5-methyl-1,3,4-oxadiazol-2-yl)ethyl]sulfanylquinazolin-4-one
—— 2-[(1R)-1-(5-methyl-1,3,4-oxadiazol-2-yl)ethyl]sulfanyl-3-(4-methylpyridin-2-yl)quinazolin-4-one —— C19H17N5O2S
2-[(1R)-1-(5-methyl-1,3,4-oxadiazol-2-yl)ethyl]sulfanyl-3-(4-methylpyridin-2-yl)quinazolin-4-one
—— N-[[4-[(2R,4R,5S,6S)-4-[(dibenzylamino)methyl]-6-[4-(hydroxymethyl)phenyl]-5-methyl-1,3-dioxan-2-yl]phenyl]methyl]quinoxaline-2-carboxamide —— C43H42N4O4
N-[[4-[(2R,4R,5S,6S)-4-[(dibenzylamino)methyl]-6-[4-(hydroxymethyl)phenyl]-5-methyl-1,3-dioxan-2-yl]phenyl]methyl]quinoxaline-2-carboxamide
—— methyl (2S)-2-quinazolin-4-ylsulfanylpropanoate —— C12H12N2O2S
methyl (2S)-2-quinazolin-4-ylsulfanylpropanoate
—— N-[[4-[(2R,4R,5S,6S)-4-[[[(2S)-2-hydroxy-2-(3-hydroxyphenyl)ethyl]-methylamino]methyl]-6-[4-(hydroxymethyl)phenyl]-5-methyl-1,3-dioxan-2-yl]phenyl]methyl]quinoxaline-2-carboxamide —— C38H40N4O6
N-[[4-[(2R,4R,5S,6S)-4-[[[(2S)-2-hydroxy-2-(3-hydroxyphenyl)ethyl]-methylamino]methyl]-6-[4-(hydroxymethyl)phenyl]-5-methyl-1,3-dioxan-2-yl]phenyl]methyl]quinoxaline-2-carboxamide
—— N-[[4-[(2R,4S,5S,6R)-4-[4-(hydroxymethyl)phenyl]-5-methyl-6-[[methyl-[(1R)-1-naphthalen-2-ylethyl]amino]methyl]-1,3-dioxan-2-yl]phenyl]methyl]quinoxaline-2-carboxamide —— C42H42N4O4
N-[[4-[(2R,4S,5S,6R)-4-[4-(hydroxymethyl)phenyl]-5-methyl-6-[[methyl-[(1R)-1-naphthalen-2-ylethyl]amino]methyl]-1,3-dioxan-2-yl]phenyl]methyl]quinoxaline-2-carboxamide
—— N-[[4-[(2R,4R,5S,6S)-4-[(4-benzylpiperazin-1-yl)methyl]-6-[4-(hydroxymethyl)phenyl]-5-methyl-1,3-dioxan-2-yl]phenyl]methyl]quinoxaline-2-carboxamide —— C40H43N5O4
N-[[4-[(2R,4R,5S,6S)-4-[(4-benzylpiperazin-1-yl)methyl]-6-[4-(hydroxymethyl)phenyl]-5-methyl-1,3-dioxan-2-yl]phenyl]methyl]quinoxaline-2-carboxamide
—— N-[[4-[(2R,4R,5S,6S)-4-(1,3-benzothiazol-2-ylsulfanylmethyl)-6-[4-(hydroxymethyl)phenyl]-5-methyl-1,3-dioxan-2-yl]phenyl]methyl]quinoxaline-2-carboxamide —— C36H32N4O4S2
N-[[4-[(2R,4R,5S,6S)-4-(1,3-benzothiazol-2-ylsulfanylmethyl)-6-[4-(hydroxymethyl)phenyl]-5-methyl-1,3-dioxan-2-yl]phenyl]methyl]quinoxaline-2-carboxamide
—— N-[[4-[(2R,4R,5S,6S)-4-[(4-acetamidophenyl)sulfanylmethyl]-6-[4-(hydroxymethyl)phenyl]-5-methyl-1,3-dioxan-2-yl]phenyl]methyl]quinoxaline-2-carboxamide —— C37H36N4O5S
N-[[4-[(2R,4R,5S,6S)-4-[(4-acetamidophenyl)sulfanylmethyl]-6-[4-(hydroxymethyl)phenyl]-5-methyl-1,3-dioxan-2-yl]phenyl]methyl]quinoxaline-2-carboxamide
—— N-[[4-[(2R,4S,5S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[[[(1S,2R)-1-hydroxy-1-phenylpropan-2-yl]-methylamino]methyl]-5-methyl-1,3-dioxan-2-yl]phenyl]methyl]quinoxaline-2-carboxamide —— C39H42N4O5
N-[[4-[(2R,4S,5S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[[[(1S,2R)-1-hydroxy-1-phenylpropan-2-yl]-methylamino]methyl]-5-methyl-1,3-dioxan-2-yl]phenyl]methyl]quinoxaline-2-carboxamide
—— N-[[4-[(2R,4S,5S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[[[(1R,2S)-1-hydroxy-1-phenylpropan-2-yl]-methylamino]methyl]-5-methyl-1,3-dioxan-2-yl]phenyl]methyl]quinoxaline-2-carboxamide —— C39H42N4O5
N-[[4-[(2R,4S,5S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[[[(1R,2S)-1-hydroxy-1-phenylpropan-2-yl]-methylamino]methyl]-5-methyl-1,3-dioxan-2-yl]phenyl]methyl]quinoxaline-2-carboxamide
—— (4-aminoquinazolin-2-yl)methyl (5R)-3-(3-fluorophenyl)-4,5-dihydro-1,2-oxazole-5-carboxylate —— C19H15FN4O3
(4-aminoquinazolin-2-yl)methyl (5R)-3-(3-fluorophenyl)-4,5-dihydro-1,2-oxazole-5-carboxylate
—— N-[(1R)-2,3-dihydro-1H-inden-1-yl]-4-oxo-2-sulfanylidene-1H-quinazoline-7-carboxamide —— C18H15N3O2S
N-[(1R)-2,3-dihydro-1H-inden-1-yl]-4-oxo-2-sulfanylidene-1H-quinazoline-7-carboxamide
—— N-[[4-[(2R,4S,5S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[(2-methoxyphenyl)sulfanylmethyl]-5-methyl-1,3-dioxan-2-yl]phenyl]methyl]quinoxaline-2-carboxamide —— C36H35N3O5S
N-[[4-[(2R,4S,5S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[(2-methoxyphenyl)sulfanylmethyl]-5-methyl-1,3-dioxan-2-yl]phenyl]methyl]quinoxaline-2-carboxamide
—— N-[(2S)-2-cyclopropyl-2-(dimethylamino)ethyl]quinoxaline-2-carboxamide —— C16H20N4O
N-[(2S)-2-cyclopropyl-2-(dimethylamino)ethyl]quinoxaline-2-carboxamide
—— 3-benzyl-N-[(2R)-1-imidazol-1-ylpropan-2-yl]-4-oxophthalazine-1-carboxamide —— C22H21N5O2
3-benzyl-N-[(2R)-1-imidazol-1-ylpropan-2-yl]-4-oxophthalazine-1-carboxamide
—— 4-methyl-3-nitro-N-(9-oxo-2,3-dihydro-1H-pyrrolo[2,1-b]quinazolin-7-yl)benzenesulfonamide —— C18H16N4O5S
4-methyl-3-nitro-N-(9-oxo-2,3-dihydro-1H-pyrrolo[2,1-b]quinazolin-7-yl)benzenesulfonamide
—— N-[(1R)-2,2-dimethyl-1-phenylpropyl]-2-(3-ethyl-2,4-dioxoquinazolin-1-yl)acetamide —— C23H27N3O3
N-[(1R)-2,2-dimethyl-1-phenylpropyl]-2-(3-ethyl-2,4-dioxoquinazolin-1-yl)acetamide
—— 2-(2-methoxy-5-methylphenyl)-N-(9-oxo-2,3-dihydro-1H-pyrrolo[2,1-b]quinazolin-7-yl)acetamide —— C21H21N3O3
2-(2-methoxy-5-methylphenyl)-N-(9-oxo-2,3-dihydro-1H-pyrrolo[2,1-b]quinazolin-7-yl)acetamide
—— N-(9-oxo-2,3-dihydro-1H-pyrrolo[2,1-b]quinazolin-7-yl)-3-(5-phenyl-1,3-oxazol-2-yl)propanamide —— C23H20N4O3
N-(9-oxo-2,3-dihydro-1H-pyrrolo[2,1-b]quinazolin-7-yl)-3-(5-phenyl-1,3-oxazol-2-yl)propanamide
—— N-[[4-[(2R,4S,5S,6R)-4-[4-(hydroxymethyl)phenyl]-5-methyl-6-[(1-oxidopyridin-1-ium-2-yl)sulfanylmethyl]-1,3-dioxan-2-yl]phenyl]methyl]quinoxaline-2-carboxamide —— C34H32N4O5S
N-[[4-[(2R,4S,5S,6R)-4-[4-(hydroxymethyl)phenyl]-5-methyl-6-[(1-oxidopyridin-1-ium-2-yl)sulfanylmethyl]-1,3-dioxan-2-yl]phenyl]methyl]quinoxaline-2-carboxamide
—— N-[(2S)-1-pyrazol-1-ylpropan-2-yl]phthalazin-1-amine —— C14H15N5
N-[(2S)-1-pyrazol-1-ylpropan-2-yl]phthalazin-1-amine
—— N-[[4-[(2R,4R,5S,6S)-4-(benzimidazol-1-ylmethyl)-6-[4-(hydroxymethyl)phenyl]-5-methyl-1,3-dioxan-2-yl]phenyl]methyl]quinoxaline-2-carboxamide —— C36H33N5O4
N-[[4-[(2R,4R,5S,6S)-4-(benzimidazol-1-ylmethyl)-6-[4-(hydroxymethyl)phenyl]-5-methyl-1,3-dioxan-2-yl]phenyl]methyl]quinoxaline-2-carboxamide
—— N-[[4-[(2R,4R,5S,6S)-4-[[cyclopentyl(prop-2-enyl)amino]methyl]-6-[4-(hydroxymethyl)phenyl]-5-methyl-1,3-dioxan-2-yl]phenyl]methyl]quinoxaline-2-carboxamide —— C37H42N4O4
N-[[4-[(2R,4R,5S,6S)-4-[[cyclopentyl(prop-2-enyl)amino]methyl]-6-[4-(hydroxymethyl)phenyl]-5-methyl-1,3-dioxan-2-yl]phenyl]methyl]quinoxaline-2-carboxamide
—— N-[2-[(2S)-oxolan-2-yl]ethyl]quinoxalin-2-amine —— C14H17N3O
N-[2-[(2S)-oxolan-2-yl]ethyl]quinoxalin-2-amine
—— N-[[4-[(2R,4S,5S,6R)-4-[4-(hydroxymethyl)phenyl]-5-methyl-6-[(1-methyltetrazol-5-yl)sulfanylmethyl]-1,3-dioxan-2-yl]phenyl]methyl]quinoxaline-2-carboxamide —— C31H31N7O4S
N-[[4-[(2R,4S,5S,6R)-4-[4-(hydroxymethyl)phenyl]-5-methyl-6-[(1-methyltetrazol-5-yl)sulfanylmethyl]-1,3-dioxan-2-yl]phenyl]methyl]quinoxaline-2-carboxamide
—— N-[[4-[(2R,4S,5S,6R)-4-[4-(hydroxymethyl)phenyl]-5-methyl-6-[(4-methyl-1,2,4-triazol-3-yl)sulfanylmethyl]-1,3-dioxan-2-yl]phenyl]methyl]quinoxaline-2-carboxamide —— C32H32N6O4S
N-[[4-[(2R,4S,5S,6R)-4-[4-(hydroxymethyl)phenyl]-5-methyl-6-[(4-methyl-1,2,4-triazol-3-yl)sulfanylmethyl]-1,3-dioxan-2-yl]phenyl]methyl]quinoxaline-2-carboxamide
—— N-[[4-[(2R,4S,5S,6R)-4-[4-(hydroxymethyl)phenyl]-5-methyl-6-[(1-methylimidazol-2-yl)sulfanylmethyl]-1,3-dioxan-2-yl]phenyl]methyl]quinoxaline-2-carboxamide —— C33H33N5O4S
N-[[4-[(2R,4S,5S,6R)-4-[4-(hydroxymethyl)phenyl]-5-methyl-6-[(1-methylimidazol-2-yl)sulfanylmethyl]-1,3-dioxan-2-yl]phenyl]methyl]quinoxaline-2-carboxamide
—— N-[[4-[(2R,4R,5S,6S)-4-(azocan-1-ylmethyl)-6-[4-(hydroxymethyl)phenyl]-5-methyl-1,3-dioxan-2-yl]phenyl]methyl]quinoxaline-2-carboxamide —— C36H42N4O4
N-[[4-[(2R,4R,5S,6S)-4-(azocan-1-ylmethyl)-6-[4-(hydroxymethyl)phenyl]-5-methyl-1,3-dioxan-2-yl]phenyl]methyl]quinoxaline-2-carboxamide
—— N-[[4-[(2R,4S,5S,6R)-4-[4-(hydroxymethyl)phenyl]-5-methyl-6-(pyrimidin-2-ylsulfanylmethyl)-1,3-dioxan-2-yl]phenyl]methyl]quinoxaline-2-carboxamide —— C33H31N5O4S
N-[[4-[(2R,4S,5S,6R)-4-[4-(hydroxymethyl)phenyl]-5-methyl-6-(pyrimidin-2-ylsulfanylmethyl)-1,3-dioxan-2-yl]phenyl]methyl]quinoxaline-2-carboxamide
—— N-[[4-[(2R,4S,5S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[[(2S)-2-(hydroxymethyl)pyrrolidin-1-yl]methyl]-5-methyl-1,3-dioxan-2-yl]phenyl]methyl]quinoxaline-2-carboxamide —— C34H38N4O5
N-[[4-[(2R,4S,5S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[[(2S)-2-(hydroxymethyl)pyrrolidin-1-yl]methyl]-5-methyl-1,3-dioxan-2-yl]phenyl]methyl]quinoxaline-2-carboxamide
—— N-[[4-[(2R,4S,5S,6R)-4-[4-(hydroxymethyl)phenyl]-5-methyl-6-(phenylsulfanylmethyl)-1,3-dioxan-2-yl]phenyl]methyl]quinoxaline-2-carboxamide —— C35H33N3O4S
N-[[4-[(2R,4S,5S,6R)-4-[4-(hydroxymethyl)phenyl]-5-methyl-6-(phenylsulfanylmethyl)-1,3-dioxan-2-yl]phenyl]methyl]quinoxaline-2-carboxamide
—— N-[[4-[(2R,4S,5S,6R)-4-[4-(hydroxymethyl)phenyl]-5-methyl-6-(morpholin-4-ylmethyl)-1,3-dioxan-2-yl]phenyl]methyl]quinoxaline-2-carboxamide —— C33H36N4O5
N-[[4-[(2R,4S,5S,6R)-4-[4-(hydroxymethyl)phenyl]-5-methyl-6-(morpholin-4-ylmethyl)-1,3-dioxan-2-yl]phenyl]methyl]quinoxaline-2-carboxamide
—— 3-butyl-N-[(2R)-4-(furan-2-yl)butan-2-yl]-4-oxophthalazine-1-carboxamide —— C21H25N3O3
3-butyl-N-[(2R)-4-(furan-2-yl)butan-2-yl]-4-oxophthalazine-1-carboxamide
—— 3-butyl-N-[(2S)-4-(furan-2-yl)butan-2-yl]-4-oxophthalazine-1-carboxamide —— C21H25N3O3
3-butyl-N-[(2S)-4-(furan-2-yl)butan-2-yl]-4-oxophthalazine-1-carboxamide
—— N-[[4-[(2R,4S,5S,6R)-4-[4-(hydroxymethyl)phenyl]-5-methyl-6-(1H-1,2,4-triazol-5-ylsulfanylmethyl)-1,3-dioxan-2-yl]phenyl]methyl]quinoxaline-2-carboxamide —— C31H30N6O4S
N-[[4-[(2R,4S,5S,6R)-4-[4-(hydroxymethyl)phenyl]-5-methyl-6-(1H-1,2,4-triazol-5-ylsulfanylmethyl)-1,3-dioxan-2-yl]phenyl]methyl]quinoxaline-2-carboxamide
—— N-[[4-[(2R,4R,5S,6S)-4-(2-hydroxyethylsulfanylmethyl)-6-[4-(hydroxymethyl)phenyl]-5-methyl-1,3-dioxan-2-yl]phenyl]methyl]quinoxaline-2-carboxamide —— C31H33N3O5S
N-[[4-[(2R,4R,5S,6S)-4-(2-hydroxyethylsulfanylmethyl)-6-[4-(hydroxymethyl)phenyl]-5-methyl-1,3-dioxan-2-yl]phenyl]methyl]quinoxaline-2-carboxamide
—— N-[[3-[2-(dimethylamino)ethoxy]phenyl]methyl]-2-(4-oxo-3H-phthalazin-1-yl)acetamide —— C21H24N4O3
N-[[3-[2-(dimethylamino)ethoxy]phenyl]methyl]-2-(4-oxo-3H-phthalazin-1-yl)acetamide
—— N-[[4-[(2R,4S,5S,6R)-4-[4-(hydroxymethyl)phenyl]-5-methyl-6-[[methyl(prop-2-enyl)amino]methyl]-1,3-dioxan-2-yl]phenyl]methyl]quinoxaline-2-carboxamide —— C33H36N4O4
N-[[4-[(2R,4S,5S,6R)-4-[4-(hydroxymethyl)phenyl]-5-methyl-6-[[methyl(prop-2-enyl)amino]methyl]-1,3-dioxan-2-yl]phenyl]methyl]quinoxaline-2-carboxamide
—— 2-(6-fluoro-4-oxoquinazolin-3-yl)-N-[(1S)-1-(2-oxo-1,3-dihydrobenzimidazol-5-yl)ethyl]acetamide —— C19H16FN5O3
2-(6-fluoro-4-oxoquinazolin-3-yl)-N-[(1S)-1-(2-oxo-1,3-dihydrobenzimidazol-5-yl)ethyl]acetamide
—— N-[[4-[(2S,4R,5R,6S)-4-[4-(hydroxymethyl)phenyl]-5-methyl-6-[[4-(2-oxo-3H-benzimidazol-1-yl)piperidin-1-yl]methyl]-1,3-dioxan-2-yl]phenyl]methyl]quinoxaline-2-carboxamide —— C41H42N6O5
N-[[4-[(2S,4R,5R,6S)-4-[4-(hydroxymethyl)phenyl]-5-methyl-6-[[4-(2-oxo-3H-benzimidazol-1-yl)piperidin-1-yl]methyl]-1,3-dioxan-2-yl]phenyl]methyl]quinoxaline-2-carboxamide
—— 2,3-dimethyl-N-[(1S)-1-(2-oxo-1,3-dihydrobenzimidazol-5-yl)ethyl]quinoxaline-6-carboxamide —— C20H19N5O2
2,3-dimethyl-N-[(1S)-1-(2-oxo-1,3-dihydrobenzimidazol-5-yl)ethyl]quinoxaline-6-carboxamide
—— 2-(1-oxophthalazin-2-yl)-N-(5-phenyl-1,3-thiazol-2-yl)acetamide —— C19H14N4O2S
2-(1-oxophthalazin-2-yl)-N-(5-phenyl-1,3-thiazol-2-yl)acetamide
—— N-[(2R)-2-(diethylamino)-3-phenylpropyl]-2-(2-methyl-4-oxoquinazolin-3-yl)acetamide —— C24H30N4O2
N-[(2R)-2-(diethylamino)-3-phenylpropyl]-2-(2-methyl-4-oxoquinazolin-3-yl)acetamide