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中文名称 英文名称 CAS号 化学式 结构式图片
—— N-[1-[2-fluoro-4-(2-methylsulfonylphenyl)phenyl]-2-oxopiperidin-3-yl]benzenesulfonamide 477739-39-2 C24H23FN2O5S2
N-[1-[2-fluoro-4-(2-methylsulfonylphenyl)phenyl]-2-oxopiperidin-3-yl]benzenesulfonamide
—— (3R)-3-[2-benzyl-4-((3R,4S)-3,4-dimethoxypyrrolidin-1-yl)phenyl]ethynyl-3-quinuclidinol 464174-21-8 C28H34N2O3
(3R)-3-[2-benzyl-4-((3R,4S)-3,4-dimethoxypyrrolidin-1-yl)phenyl]ethynyl-3-quinuclidinol
—— 2-(2-cyanophenyl)-4-(2-methoxyphenyl)-6-(2-pyridyl)-4,5-dihydro-1,2,4-triazin-3-(2H)-one 404932-58-7 C22H17N5O2
2-(2-cyanophenyl)-4-(2-methoxyphenyl)-6-(2-pyridyl)-4,5-dihydro-1,2,4-triazin-3-(2H)-one
—— 6-[[1-phenyl-2-phenylamino-1H-benzimidazol-6-yl]oxy]hexanoic acid methyl ester 488141-29-3 C26H27N3O3
6-[[1-phenyl-2-phenylamino-1H-benzimidazol-6-yl]oxy]hexanoic acid methyl ester
—— N-Isopropyl-1-[3-(5-Carboethoxy-1-oxidopyridin-3-yl)phenyl]-1,4-dihydro[1,8]naphthyridin-4-one-3-carboxamide 477252-46-3 C26H24N4O5
N-Isopropyl-1-[3-(5-Carboethoxy-1-oxidopyridin-3-yl)phenyl]-1,4-dihydro[1,8]naphthyridin-4-one-3-carboxamide
—— 3-[1-(3-Chlorophenyl)piperidin-4-yl]-1-methyl-1-(1-methylsulfonylpiperidin-4-yl)urea 494860-64-9 C19H29ClN4O3S
3-[1-(3-Chlorophenyl)piperidin-4-yl]-1-methyl-1-(1-methylsulfonylpiperidin-4-yl)urea
—— (3S)-3-amino-3-(5-bromopyridin-3-yl)propanoic Acid 444806-05-7 C8H9BrN2O2
(3S)-3-amino-3-(5-bromopyridin-3-yl)propanoic Acid
—— N-[2-[[(1R)-2-[[(2,4-dimethylphenyl)methyl]amino]-1-(hydroxymethyl)ethyl]amino]-2-oxoethyl]-3-(trifluoromethyl)benzamide 439148-94-4 C22H26F3N3O3
N-[2-[[(1R)-2-[[(2,4-dimethylphenyl)methyl]amino]-1-(hydroxymethyl)ethyl]amino]-2-oxoethyl]-3-(trifluoromethyl)benzamide
—— 7-dimethylamino-4-(3-imidazol-1-yl-phenyl)-8-trifluoromethyl-1,3-dihydro-benzo[b][1,4]diazepin-2-one 473550-75-3 C21H18F3N5O
7-dimethylamino-4-(3-imidazol-1-yl-phenyl)-8-trifluoromethyl-1,3-dihydro-benzo[b][1,4]diazepin-2-one
—— 2-(N-Ethyl-N-2,4,6-trichlorophenylamino)-5-(N-cyclopropylmethyl-N-n-propyl)aminocarbonyl-4-methylthiazole 405878-74-2 C20H24Cl3N3OS
2-(N-Ethyl-N-2,4,6-trichlorophenylamino)-5-(N-cyclopropylmethyl-N-n-propyl)aminocarbonyl-4-methylthiazole
—— methyl 2-(4-{[4-[(carboxycarbonyl)(2-carboxyphenyl)amino]-N-(methoxycarbonyl)-L-phenylalanyl]amino}butoxy)-6-hydroxy-4-pentylbenzoate 436864-24-3 C37H43N3O12
methyl 2-(4-{[4-[(carboxycarbonyl)(2-carboxyphenyl)amino]-N-(methoxycarbonyl)-L-phenylalanyl]amino}butoxy)-6-hydroxy-4-pentylbenzoate
—— N-cyclopropyl-1-[3-(pyridin-4-yl)phenyl]-1,4-dihydro[1,8]naphthyridin-4-one-3-carboxamide 477252-00-9 C23H18N4O2
N-cyclopropyl-1-[3-(pyridin-4-yl)phenyl]-1,4-dihydro[1,8]naphthyridin-4-one-3-carboxamide
—— 3-(7-Bromo-5-methoxy-2,3-dihydro-1H-indol-1-yl)-5-chloro-1-(1-ethylpropyl)-2 (1H)-pyrazinone 475158-64-6 C18H21BrClN3O2
3-(7-Bromo-5-methoxy-2,3-dihydro-1H-indol-1-yl)-5-chloro-1-(1-ethylpropyl)-2 (1H)-pyrazinone
—— (R)-1-(6-Methoxyquinolin-4-yl)-2-{4-[(5,6,7,8-tetrahydro-[1,8]naphthyridin-2-ylmethyl)amino]piperidin-1-yl}ethanol 443955-92-8 C26H33N5O2
(R)-1-(6-Methoxyquinolin-4-yl)-2-{4-[(5,6,7,8-tetrahydro-[1,8]naphthyridin-2-ylmethyl)amino]piperidin-1-yl}ethanol
—— (S)-2-[[6-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-1,2,3,4-tetrahydro-3-methyl-1-(1-methylethyl)-2,4-dioxothieno[2,3-d]pyrimidin-5-yl]carbonyl]-4-isoxazolidinol 496792-57-5 C20H25N5O5S
(S)-2-[[6-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-1,2,3,4-tetrahydro-3-methyl-1-(1-methylethyl)-2,4-dioxothieno[2,3-d]pyrimidin-5-yl]carbonyl]-4-isoxazolidinol
—— 4-{(E)-2-[5,5,8,8-tetramethyl-3-(thiophen-3-yl)-5,6,7,8-tetrahydro-naphthalen-2-yl]vinyl}benzoic acid 410528-44-8 C27H28O2S
4-{(E)-2-[5,5,8,8-tetramethyl-3-(thiophen-3-yl)-5,6,7,8-tetrahydro-naphthalen-2-yl]vinyl}benzoic acid
—— 5-(4-acetylphenyl)-N-[1-(3,4-dichlorobenzyl)piperidin-4-yl]valeramide 474969-99-8 C25H30Cl2N2O2
5-(4-acetylphenyl)-N-[1-(3,4-dichlorobenzyl)piperidin-4-yl]valeramide
—— N-Cyclopropyl-1-[3-(1-Oxidopyridin-3-yl)Phenyl]-1,4-Dihydro[1,8]Naphthyridin-4-One-3-Carboxamide 477252-50-9 C23H18N4O3
N-Cyclopropyl-1-[3-(1-Oxidopyridin-3-yl)Phenyl]-1,4-Dihydro[1,8]Naphthyridin-4-One-3-Carboxamide
—— 7-(methyl-propyl-amino)-4-(3-[1,2,3]triazol-1-yl-phenyl)-8-trifluoromethyl-1,3-dihydro-benzo[b][1,4]diazepin-2-one 473551-70-1 C22H21F3N6O
7-(methyl-propyl-amino)-4-(3-[1,2,3]triazol-1-yl-phenyl)-8-trifluoromethyl-1,3-dihydro-benzo[b][1,4]diazepin-2-one
—— 5-Chloro-3-(5,7-dichloro-2,3-dihydro-1H-indol-1-yl)-1-[(1R)-2-methoxy-1-methylethyl]-2 (1H)-pyrazinone 475158-94-2 C16H16Cl3N3O2
5-Chloro-3-(5,7-dichloro-2,3-dihydro-1H-indol-1-yl)-1-[(1R)-2-methoxy-1-methylethyl]-2 (1H)-pyrazinone
—— 5-Chloro-3-(7-chloro-5-methoxy-2,3-dihydro-1H-indol-1-yl)-1-[1-(methoxymethyl)propyl]-2 (1H)-pyrazinone 475158-58-8 C18H21Cl2N3O3
5-Chloro-3-(7-chloro-5-methoxy-2,3-dihydro-1H-indol-1-yl)-1-[1-(methoxymethyl)propyl]-2 (1H)-pyrazinone
—— 4-[[5-[(Methoxyamino)carbonyl]-2-methylphenyl]amino]-5-methyl-N-[2-(4-morpholinyl)ethyl]pyrrolo[2,1-f][1,2,4]triazine-6-carboxamide 427877-82-5 C23H29N7O4
4-[[5-[(Methoxyamino)carbonyl]-2-methylphenyl]amino]-5-methyl-N-[2-(4-morpholinyl)ethyl]pyrrolo[2,1-f][1,2,4]triazine-6-carboxamide
—— [2-Methyl-4-[[[3-methyl-5-[4-(trifluoromethyl)phenyl]-2-thienyl]methyl]thio]phenoxy]acetic acid 476154-13-9 C22H19F3O3S2
[2-Methyl-4-[[[3-methyl-5-[4-(trifluoromethyl)phenyl]-2-thienyl]methyl]thio]phenoxy]acetic acid
—— N-[[1-(dimethylamino)cyclopentyl]methyl]-3,5-dimethoxy-4-[(4-methylphenyl)methoxy]benzamide 495077-04-8 C25H34N2O4
N-[[1-(dimethylamino)cyclopentyl]methyl]-3,5-dimethoxy-4-[(4-methylphenyl)methoxy]benzamide
—— N-{3-[2-(Dimethylamino)ethoxy]phenyl}[2-(1H-indazol-6-ylamino)(3-pyridyl)]carboxamide 454481-02-8 C23H24N6O2
N-{3-[2-(Dimethylamino)ethoxy]phenyl}[2-(1H-indazol-6-ylamino)(3-pyridyl)]carboxamide
—— 5-(1-Benzyl-pyrrolidin-3-yloxy)-2-methyl-1H-indole-3-carboxylic acid benzyl ester 459449-55-9 C28H28N2O3
5-(1-Benzyl-pyrrolidin-3-yloxy)-2-methyl-1H-indole-3-carboxylic acid benzyl ester
—— N-{3-[4-(7-chloro-3,4-dihydro-2H-quinolin-1-yl)-[1,3,5]triazin-2-ylamino]-phenyl}-acrylamide 473430-75-0 C21H19ClN6O
N-{3-[4-(7-chloro-3,4-dihydro-2H-quinolin-1-yl)-[1,3,5]triazin-2-ylamino]-phenyl}-acrylamide
—— 8-[3-[2-Dimethoxyphosphoryl-2-fluoro-2-(4-methylsulfonylphenyl)ethyl]phenyl]-6-(2-methylsulfonylpropan-2-yl)quinoline 481680-41-5 C30H33FNO7PS2
8-[3-[2-Dimethoxyphosphoryl-2-fluoro-2-(4-methylsulfonylphenyl)ethyl]phenyl]-6-(2-methylsulfonylpropan-2-yl)quinoline
—— 3-{4-[2-(2-Biphenyl-4-yl-5-methyl-oxazol-4-yl)-ethoxy]-phenyl}-2-(2-methoxy-phenoxy)-2-methyl-propionic Acid 401469-58-7 C35H33NO6
3-{4-[2-(2-Biphenyl-4-yl-5-methyl-oxazol-4-yl)-ethoxy]-phenyl}-2-(2-methoxy-phenoxy)-2-methyl-propionic Acid
—— 6-[(2-Benzylmercapto-1-phenyl-1H-benzimidazol-6-yl]oxy]Hexanoic Acid 488141-43-1 C26H26N2O3S
6-[(2-Benzylmercapto-1-phenyl-1H-benzimidazol-6-yl]oxy]Hexanoic Acid
—— 7-dimethylamino-4-[3-(3-methyl-isoxazol-5-yl)-phenyl]-8-trifluoromethyl-1,3-dihydro-benzo[b][1,4]diazepin-2-one 473550-33-3 C22H19F3N4O2
7-dimethylamino-4-[3-(3-methyl-isoxazol-5-yl)-phenyl]-8-trifluoromethyl-1,3-dihydro-benzo[b][1,4]diazepin-2-one
—— 4-benzyloxymethyl-5-(3,5-dichlorophenylthio)-3-methyl-1-phenyl-1H-pyrazole 412326-10-4 C24H20Cl2N2OS
4-benzyloxymethyl-5-(3,5-dichlorophenylthio)-3-methyl-1-phenyl-1H-pyrazole
—— 2-(2-bromophenyl)-N-cyclopentyl-3-[2-(cyclopentylamino)pyrimidin-4-yl]pyrazolo[1,5-a]pyridin-7-amine 460078-45-9 C27H29BrN6
2-(2-bromophenyl)-N-cyclopentyl-3-[2-(cyclopentylamino)pyrimidin-4-yl]pyrazolo[1,5-a]pyridin-7-amine
—— N-(4-(6-Cyano-7-(2-methoxyethoxy)-4-quinolyl)oxyphenyl)-N'-(2,4-difluorophenyl)urea 417713-02-1 C26H20F2N4O4
N-(4-(6-Cyano-7-(2-methoxyethoxy)-4-quinolyl)oxyphenyl)-N'-(2,4-difluorophenyl)urea
—— N-[1-[2-fluoro-4-(2-methylsulfonylphenyl)phenyl]-2-oxopiperidin-3-yl]quinoline-6-sulfonamide 477739-43-8 C27H24FN3O5S2
N-[1-[2-fluoro-4-(2-methylsulfonylphenyl)phenyl]-2-oxopiperidin-3-yl]quinoline-6-sulfonamide
—— 1-(2-methoxy-ethyl)-3-{1-[(R)-3-(5-methoxy-2-methyl-phenoxy)-4-methyl-pentyl]-piperidin-4-yl}-1,3-dihydro-benzimidazol-2-one 478613-79-5 C29H41N3O4
1-(2-methoxy-ethyl)-3-{1-[(R)-3-(5-methoxy-2-methyl-phenoxy)-4-methyl-pentyl]-piperidin-4-yl}-1,3-dihydro-benzimidazol-2-one
—— 1-Methyl-2,4-dioxo-3-[4-(1H-tetrazol-5-yl)-benzyl]-1,2,3,4-tetrahydro-thieno[2,3-d]pyrimidine-6-carboxylic acid 3-methoxy-benzylamide 448965-12-6 C24H21N7O4S
1-Methyl-2,4-dioxo-3-[4-(1H-tetrazol-5-yl)-benzyl]-1,2,3,4-tetrahydro-thieno[2,3-d]pyrimidine-6-carboxylic acid 3-methoxy-benzylamide
—— 6-Methoxy-2-(4-methoxy-phenyl)-1-[4-(2-pyrrolidin-1-yl-ethoxy)-benzyl]-1,2,3,4-tetrahydro-quinoline 476304-49-1 C30H36N2O3
6-Methoxy-2-(4-methoxy-phenyl)-1-[4-(2-pyrrolidin-1-yl-ethoxy)-benzyl]-1,2,3,4-tetrahydro-quinoline
—— N-[3,3-Dimethyl-1-(1-methyl(4-piperidyl))indolin-6-yl][2-(1H-indazol-6-ylamino)(3-pyridyl)]carboxamide 454481-15-3 C29H33N7O
N-[3,3-Dimethyl-1-(1-methyl(4-piperidyl))indolin-6-yl][2-(1H-indazol-6-ylamino)(3-pyridyl)]carboxamide
—— N-[3,3-Dimethyl-1-(1-methyl-piperidin-4-ylmethyl)-2,3-dihydro-1H-indol-6-yl]-2-(1H-indazol-6-ylamino)-nicotinamide 454481-09-5 C30H35N7O
N-[3,3-Dimethyl-1-(1-methyl-piperidin-4-ylmethyl)-2,3-dihydro-1H-indol-6-yl]-2-(1H-indazol-6-ylamino)-nicotinamide
—— N-[3-(4-isopropylphenyl)-prop-2-ynyl]-4-(4'-trifluoromethyl-biphenyl-2-carbonylamino)-1-methyl-pyrrole-2-carboxylic acid amide 486435-30-7 C32H28F3N3O2
N-[3-(4-isopropylphenyl)-prop-2-ynyl]-4-(4'-trifluoromethyl-biphenyl-2-carbonylamino)-1-methyl-pyrrole-2-carboxylic acid amide
—— 2-phenylethanesulfonic acid [6-(2-hydroxy-ethoxy)-5-(2-methoxy-phenoxy)-2-(2-pyrimidinyl)-4-pyrimidinyl]-amide 405307-47-3 C25H25N5O6S
2-phenylethanesulfonic acid [6-(2-hydroxy-ethoxy)-5-(2-methoxy-phenoxy)-2-(2-pyrimidinyl)-4-pyrimidinyl]-amide
—— N-[N-(4-aminobutyl)-N-methylpyrrole-4-(N-methylpyrrole-2-carboxamido)-2-carboxamido]-N-[5-(4-(2-chloroethyl)phenol-3-yl)benzofuran-2-carboxamido]glutarodiamide hydrochloride 413577-08-9 C38H43ClN8O7*ClH
N-[N-(4-aminobutyl)-N-methylpyrrole-4-(N-methylpyrrole-2-carboxamido)-2-carboxamido]-N-[5-(4-(2-chloroethyl)phenol-3-yl)benzofuran-2-carboxamido]glutarodiamide hydrochloride
—— 4-[4-oxo-8-(2,2,2-trifluoro-ethoxy)-7-trifluoromethyl-4,5-dihydro-3H-benzo[b][1,4]diazepin-2-yl]-pyridine-2-carbonitrile 473546-94-0 C18H10F6N4O2
4-[4-oxo-8-(2,2,2-trifluoro-ethoxy)-7-trifluoromethyl-4,5-dihydro-3H-benzo[b][1,4]diazepin-2-yl]-pyridine-2-carbonitrile
—— N-[3-(3-butyl-7-dimethylamino-3-ethyl-4-hydroxy-1,1-dioxo-2,3,4,5-tetrahydro-1H-benzo[b]thiepin-5-yl)-phenyl]-5-{4-[3-(3-hydroxy-3-phenylpropyl)-2-(4-methoxy-phenyl)-4-oxoazetidin-1-yl]benzylamino}pentanamide 439113-82-3 C55H68N4O7S
N-[3-(3-butyl-7-dimethylamino-3-ethyl-4-hydroxy-1,1-dioxo-2,3,4,5-tetrahydro-1H-benzo[b]thiepin-5-yl)-phenyl]-5-{4-[3-(3-hydroxy-3-phenylpropyl)-2-(4-methoxy-phenyl)-4-oxoazetidin-1-yl]benzylamino}pentanamide
—— palmitoyl-Val-Gly-Val-Ala-Pro-Gly-NH2 478798-23-1 C38H69N7O7
palmitoyl-Val-Gly-Val-Ala-Pro-Gly-NH2
—— L-Threonine, L-seryl-L-cysteinyl-L-asparaginyl-L-threonyl-L-alanyl- 401844-67-5 C21H37N7O11S
L-Threonine, L-seryl-L-cysteinyl-L-asparaginyl-L-threonyl-L-alanyl-
—— 3,7,9-trimethoxy-5,11-dioxa-benzo[b]fluoren-10-one 406214-64-0 C18H14O6
3,7,9-trimethoxy-5,11-dioxa-benzo[b]fluoren-10-one
—— 6-Methyl-5-phenyl-4-thioxo-4,5-dihydro-3H-pyrrolo[3,2-d]pyrimidine-7-carbonitrile 473997-03-4 C14H10N4S
6-Methyl-5-phenyl-4-thioxo-4,5-dihydro-3H-pyrrolo[3,2-d]pyrimidine-7-carbonitrile
—— 1-Methyl-3-[1-(3-methylphenyl)piperidin-4-yl]-1-(1-methylsulfonylpiperidin-4-yl)urea 494860-76-3 C20H32N4O3S
1-Methyl-3-[1-(3-methylphenyl)piperidin-4-yl]-1-(1-methylsulfonylpiperidin-4-yl)urea