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中文名称 英文名称 CAS号 化学式 结构式图片
—— 1-{1-[3-(3-phenylisoxazol-5-yl)propyl]-4-piperidyl}-3-hydrobenzimidazol-2-on 457660-15-0 C24H26N4O2
1-{1-[3-(3-phenylisoxazol-5-yl)propyl]-4-piperidyl}-3-hydrobenzimidazol-2-on
—— 1-[[3-[4,8-dihydro-5-hydroxy-8-[(4-methoxyphenyl)methyl]-4-oxo-1H-pyrazolo[4',3':5,6]pyrido[4,3-d]pyrimidin-2-yl]-4-propoxyphenyl]sulfonyl]-4-ethylpiperazine 459124-64-2 C31H35N7O6S
1-[[3-[4,8-dihydro-5-hydroxy-8-[(4-methoxyphenyl)methyl]-4-oxo-1H-pyrazolo[4',3':5,6]pyrido[4,3-d]pyrimidin-2-yl]-4-propoxyphenyl]sulfonyl]-4-ethylpiperazine
—— 1'-(1-methylethyl)-4'-[(2-fluoro-4-methoxyphenyl)methyl]-5'-methyl-1H-pyrazol-3'-O-β-D-glucopyranoside 421592-30-5 C21H29FN2O7
1'-(1-methylethyl)-4'-[(2-fluoro-4-methoxyphenyl)methyl]-5'-methyl-1H-pyrazol-3'-O-β-D-glucopyranoside
—— 3-[1-(3,5-Difluorophenyl)piperidin-4-yl]-1-methyl-1-(1-methylsulfonylpiperidin-4-yl)urea 494860-56-9 C19H28F2N4O3S
3-[1-(3,5-Difluorophenyl)piperidin-4-yl]-1-methyl-1-(1-methylsulfonylpiperidin-4-yl)urea
—— 4-(2-Chloro-5-methoxyanilino)-2-(3-pyridinyl)-6-(trifluoromethyl)pyrimidine 438247-85-9 C17H12ClF3N4O
4-(2-Chloro-5-methoxyanilino)-2-(3-pyridinyl)-6-(trifluoromethyl)pyrimidine
—— 2-(dimethylamino)-N-{(2-(2,6-dioxo(3-piperidyl))-1,3-dioxoisoindolin-4-yl)methyl}-acetamide 444287-51-8 C18H20N4O5
2-(dimethylamino)-N-{(2-(2,6-dioxo(3-piperidyl))-1,3-dioxoisoindolin-4-yl)methyl}-acetamide
—— 8-{3-[1-(4-Chloro-phenyl)-2-pyridin-4-yl-ethyl]-phenyl}-6-isopropyl-quinoline 481680-46-0 C31H27ClN2
8-{3-[1-(4-Chloro-phenyl)-2-pyridin-4-yl-ethyl]-phenyl}-6-isopropyl-quinoline
—— 4-ethyl-N-[1-[2-fluoro-4-(2-methylsulfonylphenyl)phenyl]-2-oxopiperidin-3-yl]benzenesulfonamide 477738-85-5 C26H27FN2O5S2
4-ethyl-N-[1-[2-fluoro-4-(2-methylsulfonylphenyl)phenyl]-2-oxopiperidin-3-yl]benzenesulfonamide
—— N-ethyl-4-(5-methyl-3-phenylisoxazol-4-yl)-N-propionylbenzenesulfonamide 473465-00-8 C21H22N2O4S
N-ethyl-4-(5-methyl-3-phenylisoxazol-4-yl)-N-propionylbenzenesulfonamide
—— 3-(5-Bromo-7-methoxy-2,3-dihydro-4H-1,4-benzoxazin-4-yl)-5-chloro-1-[(1S)-2-methoxy-1-methylethyl]-2 (1H)-pyrazinone 475159-50-3 C17H19BrClN3O4
3-(5-Bromo-7-methoxy-2,3-dihydro-4H-1,4-benzoxazin-4-yl)-5-chloro-1-[(1S)-2-methoxy-1-methylethyl]-2 (1H)-pyrazinone
—— 5-Chloro-1-[(1S)-1-cyclopropylpropyl]-3-(5-methoxy-7-methyl-2,3-dihydro-1H-indol-1-yl)-2 (1H)-pyrazinone 475158-90-8 C20H24ClN3O2
5-Chloro-1-[(1S)-1-cyclopropylpropyl]-3-(5-methoxy-7-methyl-2,3-dihydro-1H-indol-1-yl)-2 (1H)-pyrazinone
—— beta-L-Tagatopyranose 41847-58-9 C6H12O6
beta-L-Tagatopyranose
—— 4-(5,7-dichloro-2,3-dihydro-1H-indol-1-yl)-6-(1-ethylpropylamino)-5-formyl-2-methylpyrimidine 475158-36-2 C19H22Cl2N4O
4-(5,7-dichloro-2,3-dihydro-1H-indol-1-yl)-6-(1-ethylpropylamino)-5-formyl-2-methylpyrimidine
—— 6-(2-hydroxyethoxy)-3,3,14-trimethyl-3,14-dihydro-7H-benzo[b]pyrano[3,2-h]-acridin-7-one 498545-79-2 C25H23NO4
6-(2-hydroxyethoxy)-3,3,14-trimethyl-3,14-dihydro-7H-benzo[b]pyrano[3,2-h]-acridin-7-one
—— 5-(3-amino-propylamino)-6-fluoro-3-(1H-pyrrol-2-yl)-1H-benzo[cd]indol-2-one acetic acid salt 444099-80-3 C2H4O2*C18H17FN4O
5-(3-amino-propylamino)-6-fluoro-3-(1H-pyrrol-2-yl)-1H-benzo[cd]indol-2-one acetic acid salt
—— (2S,4S)-1-((2R)-2-amino-3-[(4-methoxybenzyl)sulfonyl]-3-methyl-butanoyl)-4-fluoropyrrolidine-2-carbonitrile hydrochloride 483367-72-2 C18H24FN3O4S*ClH
(2S,4S)-1-((2R)-2-amino-3-[(4-methoxybenzyl)sulfonyl]-3-methyl-butanoyl)-4-fluoropyrrolidine-2-carbonitrile hydrochloride
—— (2S,4S)-1-((R)-2-amino-3-methyl-3-(3-phenylpropylsulfonyl)butanoyl)-4-fluoropyrrolidine-2-carbonitrile 483367-77-7 C19H26FN3O3S
(2S,4S)-1-((R)-2-amino-3-methyl-3-(3-phenylpropylsulfonyl)butanoyl)-4-fluoropyrrolidine-2-carbonitrile
—— ethyl 2-[[2-[(E)-2-(3-carbamimidoylphenyl)ethenyl]-5-(1-ethanimidoylpiperidin-4-yl)oxy-6-(trifluoromethyl)-2,3-dihydroindol-1-yl]sulfonyl]acetate 405886-91-1 C29H34F3N5O5S
ethyl 2-[[2-[(E)-2-(3-carbamimidoylphenyl)ethenyl]-5-(1-ethanimidoylpiperidin-4-yl)oxy-6-(trifluoromethyl)-2,3-dihydroindol-1-yl]sulfonyl]acetate
—— TIE-2/VEGFR-2 kinase-IN-3 433224-09-0 C23H17F4N5O3S
TIE-2/VEGFR-2 kinase-IN-3
—— (+/-)-4-(3-chlorophenyl)-α-(4chlorophenyl)-2-methyl-α-(1-methyl-1H-imidazol-5-yl)-6-quinazolinemethanol 405548-93-8 C26H20Cl2N4O
(+/-)-4-(3-chlorophenyl)-α-(4chlorophenyl)-2-methyl-α-(1-methyl-1H-imidazol-5-yl)-6-quinazolinemethanol
—— 5-Chloro-3-(7-chloro-5-methoxy-2,3-dihydro-1H-indol-1-yl)-1-(1-cyclobutylpropyl)-2 (1H)-pyrazinone 475159-43-4 C20H23Cl2N3O2
5-Chloro-3-(7-chloro-5-methoxy-2,3-dihydro-1H-indol-1-yl)-1-(1-cyclobutylpropyl)-2 (1H)-pyrazinone
—— Dimethyl 1-(4-(methylsulfonyl)phenyl)-2-(3-(6-(2-(methylsulfonyl)propan-2-yl)quinolin-8-yl)phenyl)ethylphosphonate 481680-39-1 C30H34NO7PS2
Dimethyl 1-(4-(methylsulfonyl)phenyl)-2-(3-(6-(2-(methylsulfonyl)propan-2-yl)quinolin-8-yl)phenyl)ethylphosphonate
—— Palmitoyl 3-carbacyclic Phosphatidic Acid 476310-22-2 C20H39O5P
Palmitoyl 3-carbacyclic Phosphatidic Acid
—— 3-(5-(2-(2-(4-methylphenyl)-5-methyloxazol-4-yl)ethoxy)-3,4-dihydronaphthalen-1-yl)propanoic acid ethyl ester 439801-95-3 C28H31NO4
3-(5-(2-(2-(4-methylphenyl)-5-methyloxazol-4-yl)ethoxy)-3,4-dihydronaphthalen-1-yl)propanoic acid ethyl ester
—— 5-Chloro-1-[(1S)-1-cyclopropylpropyl]-3-(5,7-dibromo-2,3-dihydro-1H-indol-1-yl)-2 (1H)-pyrazinone 475158-92-0 C18H18Br2ClN3O
5-Chloro-1-[(1S)-1-cyclopropylpropyl]-3-(5,7-dibromo-2,3-dihydro-1H-indol-1-yl)-2 (1H)-pyrazinone
—— (2S)-3-[[(2,4-dimethylphenyl)methyl]amino]-2-[[[[3-(trifluoromethyl)benzoyl]amino]acetyl]amino]-propanamide 439148-65-9 C22H25F3N4O3
(2S)-3-[[(2,4-dimethylphenyl)methyl]amino]-2-[[[[3-(trifluoromethyl)benzoyl]amino]acetyl]amino]-propanamide
—— 2-{4-[({4-(4-tert-butylbenzyl)-2-[4-(trifluoromethyl)phenyl]-1,3-thiazol-5-yl}methyl)sulfanyl]-2-methylphenoxy}-2-methylpropanoic acid 444610-29-1 C33H34F3NO3S2
2-{4-[({4-(4-tert-butylbenzyl)-2-[4-(trifluoromethyl)phenyl]-1,3-thiazol-5-yl}methyl)sulfanyl]-2-methylphenoxy}-2-methylpropanoic acid
—— 4-[2-(3-chlorophenyl)ethyl]-6-[(4-chlorophenyl)hydroxy(1-methyl-1H-imidazol-5-yl)methyl]-1-methyl-2(1H)-quinolinone 439906-16-8 C29H25Cl2N3O2
4-[2-(3-chlorophenyl)ethyl]-6-[(4-chlorophenyl)hydroxy(1-methyl-1H-imidazol-5-yl)methyl]-1-methyl-2(1H)-quinolinone
—— 2-{[6-(3-Pentanoyl-1-benzofuran-2-yl)-2-naphthyl]oxy}-3-phenylpropanoic acid 481070-66-0 C32H28O5
2-{[6-(3-Pentanoyl-1-benzofuran-2-yl)-2-naphthyl]oxy}-3-phenylpropanoic acid
—— ethyl N-{3,5-dichloro-4-[(3-isopropyl-1H-indol-5-yl)oxy]phenyl}glycinate 439612-21-2 C21H22Cl2N2O3
ethyl N-{3,5-dichloro-4-[(3-isopropyl-1H-indol-5-yl)oxy]phenyl}glycinate
—— ethyl 8,9-dimethoxy-3-methyl-2-(3-nitrophenyl)-5,6-dihydropyrrolo[2,1-a]isoquinoline-1-carboxylate 438037-97-9 C24H24N2O6
ethyl 8,9-dimethoxy-3-methyl-2-(3-nitrophenyl)-5,6-dihydropyrrolo[2,1-a]isoquinoline-1-carboxylate
—— 1-(5-cyclohexyl-2-oxo-1-propyl-3H-1,4-benzodiazepin-3-yl)-3-[4-(4-piperidin-1-ylpiperidin-1-yl)phenyl]urea 478055-54-8 C35H48N6O2
1-(5-cyclohexyl-2-oxo-1-propyl-3H-1,4-benzodiazepin-3-yl)-3-[4-(4-piperidin-1-ylpiperidin-1-yl)phenyl]urea
—— 2-{2-methyl-4-[({4-(3-thienylmethyl)-2-[4-(trifluoromethyl)phenyl]-1,3-thiazol-5-yl}methyl)sulfanyl]phenoxy)propanoic acid 444612-48-0 C26H22F3NO3S3
2-{2-methyl-4-[({4-(3-thienylmethyl)-2-[4-(trifluoromethyl)phenyl]-1,3-thiazol-5-yl}methyl)sulfanyl]phenoxy)propanoic acid
—— (3R)-3-Amino-4-(2,5-difluorophenyl)-1-[5,6-dihydro-2-(trifluoromethyl)imidazo[1,2-a]pyrazin-7(8H)-yl]-1-butanone 486460-28-0 C17H17F5N4O
(3R)-3-Amino-4-(2,5-difluorophenyl)-1-[5,6-dihydro-2-(trifluoromethyl)imidazo[1,2-a]pyrazin-7(8H)-yl]-1-butanone
—— L-Threonine, L-threonyl-L-prolyl-L-lysyl-L-threonyl-L-seryl-L-valyl- 404334-08-3 C31H56N8O12
L-Threonine, L-threonyl-L-prolyl-L-lysyl-L-threonyl-L-seryl-L-valyl-
—— N,N1-(tricyclo[3.3.1.1<sup>3,7</sup>]dec-1-yl)imidodisulfamide monophosphate 446038-35-3 C20H34N3O7PS2
N,N1-(tricyclo[3.3.1.1<sup>3,7</sup>]dec-1-yl)imidodisulfamide monophosphate
—— H-Ala-Val-Pro-Ile-Ala-Gln-Lys-Ser-OH 402594-20-1 C36H64N10O11
H-Ala-Val-Pro-Ile-Ala-Gln-Lys-Ser-OH
—— 2-(2-bromophenyl)-4-(2-hydroxyphenyl)-6-(2-pyridyl)-4,5-dihydro-1,2,4-triazin-3-(2H)-one 404932-56-5 C20H15BrN4O2
2-(2-bromophenyl)-4-(2-hydroxyphenyl)-6-(2-pyridyl)-4,5-dihydro-1,2,4-triazin-3-(2H)-one
—— N-(4-(6-Cyano-7-(2-methoxyethoxy)-4-quinolyl)oxyphenyl)-N'-(3-(methylsulfonyl)phenyl)urea 417713-05-4 C27H24N4O6S
N-(4-(6-Cyano-7-(2-methoxyethoxy)-4-quinolyl)oxyphenyl)-N'-(3-(methylsulfonyl)phenyl)urea
—— 1-(1-{3-[3-(2-thienyl)isoxazol-5-yl]propyl}-4-piperidyl)-3-hydrobenzimidazol-2-on 457660-31-0 C22H24N4O2S
1-(1-{3-[3-(2-thienyl)isoxazol-5-yl]propyl}-4-piperidyl)-3-hydrobenzimidazol-2-on
—— N-(2,6-dimethylphenyl)-2-{4-[2-hydroxy-3-(isoquinolin-5-yloxy)-propyl]-piperazin-1-yl}acetamide 449756-53-0 C26H32N4O3
N-(2,6-dimethylphenyl)-2-{4-[2-hydroxy-3-(isoquinolin-5-yloxy)-propyl]-piperazin-1-yl}acetamide
—— 4-(5-Methoxy-2-nitroanilino)-2-(2-pyrazinyl)-6-trifluoromethylpyrimidine 438249-18-4 C16H11F3N6O3
4-(5-Methoxy-2-nitroanilino)-2-(2-pyrazinyl)-6-trifluoromethylpyrimidine
—— 5-chloro-1-(1-cyclobutylpropyl)-3-(7-methoxy-2,3-dihydro-4H-1,4-benzoxazin-4-yl)-2 (1H)-pyrazinone 475159-52-5 C20H24ClN3O3
5-chloro-1-(1-cyclobutylpropyl)-3-(7-methoxy-2,3-dihydro-4H-1,4-benzoxazin-4-yl)-2 (1H)-pyrazinone
—— 4-[[4-[3-(2-benzoxazolylthio)propoxy]phenyl]sulfonyl]tetrahydro-N-N-hydroxy-2H-pyran-4-carboxamide 476182-92-0 C22H24N2O7S2
4-[[4-[3-(2-benzoxazolylthio)propoxy]phenyl]sulfonyl]tetrahydro-N-N-hydroxy-2H-pyran-4-carboxamide
—— 3-(7-Bromo-5-methoxy-2,3-dihydro-1H-indol-1-yl)-5-chloro-1-[2-(methylthio)ethyl]-2 (1H)-pyrazinone 475159-13-8 C16H17BrClN3O2S
3-(7-Bromo-5-methoxy-2,3-dihydro-1H-indol-1-yl)-5-chloro-1-[2-(methylthio)ethyl]-2 (1H)-pyrazinone
—— 5-(2-ethoxy-5-(methylsulfonyl)phenyl)-1-methyl-3-propyl-1H-pyrazolo[4,3-d]pyrimidin-7(6H)-one 459834-16-3 C18H22N4O4S
5-(2-ethoxy-5-(methylsulfonyl)phenyl)-1-methyl-3-propyl-1H-pyrazolo[4,3-d]pyrimidin-7(6H)-one
—— 2-(2-Methoxy-phenoxy)-2-methyl-3-{4-[2-(5-methyl-2-thiophen-2-yl-oxazol-4-yl)-ethoxy]-phenyl}-propionic Acid 401790-42-9 C27H27NO6S
2-(2-Methoxy-phenoxy)-2-methyl-3-{4-[2-(5-methyl-2-thiophen-2-yl-oxazol-4-yl)-ethoxy]-phenyl}-propionic Acid
—— N-{2-[4-(3,5-Dichlorophenoxy)-3,5-diethyl-1H-pyrazol-1-yl]ethyl}-2-methoxyacetamide 473919-61-8 C18H23Cl2N3O3
N-{2-[4-(3,5-Dichlorophenoxy)-3,5-diethyl-1H-pyrazol-1-yl]ethyl}-2-methoxyacetamide
—— 3-(5-Bromo-7-chloro-2,3-dihydro-1H-indol-1-yl)-5-chloro-1-[(1S)-1-(methoxymethyl)propyl]-2 (1H)-pyrazinone 475159-32-1 C17H18BrCl2N3O2
3-(5-Bromo-7-chloro-2,3-dihydro-1H-indol-1-yl)-5-chloro-1-[(1S)-1-(methoxymethyl)propyl]-2 (1H)-pyrazinone
—— 3-Benzyl-6-[3-(4-methoxy-phenyl)-prop-1-ynyl]-1-methyl-1H-thieno[2,3-d]pyrimidine-2,4-dione 448969-11-7 C24H20N2O3S
3-Benzyl-6-[3-(4-methoxy-phenyl)-prop-1-ynyl]-1-methyl-1H-thieno[2,3-d]pyrimidine-2,4-dione