3-Diethoxyphosphinothioyloxy-2,6-dimethylbenzenesulfonamide

• 分子结构分类: 有机化合物 - 有机酸及其衍生物 - 有机硫代磷酸及其衍生物
• 英文名称: 3-Diethoxyphosphinothioyloxy-2,6-dimethylbenzenesulfonamide
• 英文别名: 3-diethoxyphosphinothioyloxy-2,6-dimethylbenzenesulfonamide
• 化学式: C₁₂H₂₀NO₅PS₂
• 分子量: 353.4
• InChiKey: NAXPDGOGBNQZCU-UHFFFAOYSA-N

计算性质

• 辛醇/水分配系数(LogP)：
  3.1
• 重原子数：
  21
• 可旋转键数：
  7
• 环数：
  1.0
• sp3杂化的碳原子比例：
  0.5
• 拓扑面积：
  128
• 氢给体数：
  1
• 氢受体数：
  7

文献信息

• HYDRAZONYL GROUP-CONTAINING CONDENSED HETEROCYCLIC COMPOUND OR SALT THEREOF, AGRICULTURAL AND HORTICULTURAL INSECTICIDE COMPRISING THE COMPOUND, AND METHOD FOR USING THE INSECTICIDE
  申请人：Nihon Nohyaku Co., Ltd.

  公开号：US20190177319A1

  公开（公告）日：2019-06-13

  An object of the present invention is to develop and provide a novel agricultural and horticultural insecticide in view of the still immense damage caused by insect pests etc. and the emergence of insect pests resistant to existing insecticides in crop production in the fields of agriculture, horticulture and the like. Provided is a hydrazonyl group-containing condensed heterocyclic compound or a salt thereof, preferably a condensed heterocyclic compound represented by the general formula (1): wherein R 1 represents, for example, an alkyl group, R 2 represents, for example, a hydrogen atom, R 3 and R 4 each represent, for example, an alkyl group, a haloalkyl group or an acyl group, A 1 represents, for example, a nitrogen atom, A 2 represents, for example, N-Me or an oxygen atom, A 3 represents, for example, a carbon atom or a nitrogen atom, A 4 represents, for example, C—H, m represents, for example, 2, and n represents, for example, 1}, or a salt thereof; an agricultural and horticultural insecticide comprising the compound or a salt thereof as an active ingredient; and a method for using the insecticide.

  本发明的一个目的是开发并提供一种新型农艺和园艺杀虫剂，鉴于昆虫害虫等造成的损害仍然巨大，以及在农业、园艺等领域作物生产中出现的对现有杀虫剂具有抗性的昆虫害虫。 提供了一种含有肼酰基的稠合杂环化合物或其盐，优选为通式(1)表示的稠合杂环化合物： 其中R1代表例如烷基，R2代表例如氢原子，R3和R4各自代表例如烷基、卤代烷基或酰基，A1代表例如氮原子，A2代表例如N-Me或氧原子，A3代表例如碳原子或氮原子，A4代表例如C—H，m代表例如2，n代表例如1}，或其盐；一种包含该化合物或其盐作为活性成分的农艺和园艺杀虫剂；以及使用该杀虫剂的方法。
• OXIME GROUP-CONTAINING CONDENSED HETEROCYCLIC COMPOUND OR SALT THEREOF, AGRICULTURAL AND HORTICULTURAL INSECTICIDE COMPRISING THE COMPOUND, AND METHOD FOR USING THE INSECTICIDE
  申请人：NIHON NOHYAKU CO., LTD.

  公开号：US20210371424A1

  公开（公告）日：2021-12-02

  Provided are an oxime group-containing condensed heterocyclic compound or a salt thereof, preferably a condensed heterocyclic compound represented by general formula (1): (wherein the symbols are defined in the specification); an agricultural and horticultural insecticide comprising the compound or a salt thereof as an active ingredient; and a method for using the insecticide.

  提供的是含有肟基的缩合杂环化合物或其盐，优选是由通式（1）表示的缩合杂环化合物： （其中符号在规范中定义）；包括该化合物或其盐作为活性成分的农业和园艺杀虫剂；以及使用该杀虫剂的方法。
• 3H-PYRROLOPYRIDINE COMPOUND, N-OXIDE THEREOF OR SALT THEREOF, AGRICULTURAL AND HORTICULTURAL INSECTICIDE COMPRISING THE COMPOUND AND METHOD FOR USING THE SAME
  申请人：Nihon Nohyaku Co., Ltd.

  公开号：US20180352811A1

  公开（公告）日：2018-12-13

  In crop production in the fields of agriculture, horticulture and the like, the damage caused by insect pests etc. is still immense, and insect pests resistant to existing insecticides have emerged. Under such circumstances, the development of novel agricultural and horticultural insecticides is desired. The present invention provides an agricultural and horticultural insecticide comprising, as an active ingredient, a 3H-pyrrolopyridine compound represented by the general formula (1): (wherein A 1 , A 2 , and A 3 each represent a nitrogen atom or a CH group, R 1 represents an ethyl group, R 2 and R 4 each represent a hydrogen atom, R 3 and R 7 each represent a haloalkyl group, R 5 and R 6 each represent a fluorine atom, and m represents 0 or 2), an N-oxide thereof or a salt thereof; and a method for using the agricultural and horticultural insecticide.

  在农业、园艺等领域的作物生产中，由昆虫害等造成的损害仍然巨大，并且出现了对现有杀虫剂产生抗药性的昆虫害。在这种情况下，需要开发新型的农业和园艺杀虫剂。本发明提供了一种农业和园艺杀虫剂，其活性成分为一种由通式（1）表示的3H-吡咯吡啶化合物（其中A1、A2和A3分别表示氮原子或CH基团，R1表示乙基基团，R2和R4分别表示氢原子，R3和R7分别表示卤代烷基基团，R5和R6分别表示氟原子，m表示0或2），其N-氧化物或盐；以及使用该农业和园艺杀虫剂的方法。
• 1H-PYRROLOPYRIDINE COMPOUND, N-OXIDE THEREOF OR SALT THEREOF, AGRICULTURAL AND HORTICULTURAL INSECTICIDE COMPRISING THE COMPOUND, AND METHOD FOR USING THE INSECTICIDE
  申请人：Nihon Nohyaku Co., Ltd.

  公开号：US20200045975A1

  公开（公告）日：2020-02-13

  In crop production in the fields of agriculture, horticulture and the like, the damage caused by insect pests etc. is still immense, and insect pests resistant to existing insecticides have emerged. Under such circumstances, the development of novel agricultural and horticultural insecticides is desired. The present invention provides an agricultural and horticultural insecticide comprising a 1H-pyrrolo-condensed heterocyclic compound represented by the general formula (1): wherein A and A 1 each represent a nitrogen atom, R 3 and R 4 each represent a haloalkyl group, R 2 represents a hydrogen atom or an acetyl group, R 1 represents a halogen atom, and m represents 0 or 2}, an N-oxide thereof or a salt thereof as an active ingredient, and a method for using the insecticide.

  在农业、园艺等领域的作物生产中，由昆虫害等造成的损害仍然是巨大的，而对现有杀虫剂产生抗性的昆虫害也已经出现。在这种情况下，需要开发新型的农业和园艺杀虫剂。本发明提供了一种农业和园艺杀虫剂，其包括一种由一般式（1）表示的1H-吡咯并杂环化合物：其中A和A1分别表示氮原子，R3和R4分别表示卤代烷基，R2表示氢原子或乙酰基，R1表示卤原子，m表示0或2}，其N-氧化物或盐作为活性成分，以及使用该杀虫剂的方法。
• 4H-PYRROLOPYRIDINE COMPOUND OR SALT THEREOF, AGRICULTURAL AND HORTICULTURAL INSECTICIDE COMPRISING THE COMPOUND OR THE SALT, AND METHOD FOR USING THE INSECTICIDE
  申请人：Nihon Nohyaku Co., Ltd.

  公开号：US20200085056A1

  公开（公告）日：2020-03-19

  In crop production in the fields of agriculture, horticulture and the like, the damage caused by insect pests etc. is still immense, and insect pests resistant to existing insecticides have emerged. Under such circumstances, the development of novel agricultural and horticultural insecticides is desired. The present invention provides an agricultural and horticultural insecticide comprising a 4H-pyrrolopyridine compound represented by the general formula (1): wherein R 1 represents a halogen atom, R 2 and R 3 each represent a haloalkyl group, Q represents Q-A, Q-B or Q-C, X represents a nitrogen atom, R 4 and R 7 each represent a hydrogen atom, R 2 and R 3 each represent a halogen atom, a haloalkyl group or a substituted phenyl group, and m represents 2} or a salt thereof as an active ingredient; and a method for using the insecticide.

  在农业、园艺等领域的作物生产中，由昆虫害等造成的损害仍然巨大，而对现有杀虫剂产生抗性的昆虫害已经出现。在这种情况下，需要开发新型的农业和园艺杀虫剂。本发明提供了一种农业和园艺杀虫剂，包括一种由通式(1)表示的4H-吡咯吡啶化合物：其中R1代表卤素原子，R2和R3各代表卤代烷基，Q代表Q-A、Q-B或Q-C，X代表氮原子，R4和R7各代表氢原子，R2和R3各代表卤素原子、卤代烷基或取代苯基，m代表2}或其盐作为活性成分；以及使用该杀虫剂的方法。